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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 89 / 236
Diphenylguanidine Approved DB14191
small molecule | CAS: 102-06-7

Diphenylguanidine is a complexing agent used in the detection of metals and organic bases and used as an accelerator in the vulcanization of rubber. It is found in some rubber products. It is also a dermatological sensitizer and allergen. Sensitivity to di…

Kategori:
AmidinesCell-mediated ImmunityIncreased Histamine Release +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diphenylpyraline Approved DB01146
small molecule | CAS: 147-20-6

Diphenylpyraline is an antihistamine. Antihistamines used in the treatment of allergy act by competing with histamine for H 1-receptor sites on effector cells. Antihistamines prevent, but do not reverse, responses mediated by histamine alone. Antihistamines a…

Kategori:
Aminoalkyl EthersAntihistamines for Systemic UseHistamine Antagonists +1
Target Protein:
Histamine H1 receptorSodium-dependent dopamine transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diphthamide DB03223
small molecule | CAS: 75645-22-6

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins
Target Protein:
Elongation factor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 499-83-2

Deskripsi belum tersedia.

Kategori:
Chelating AgentsCompounds used in a research, industrial, or household settingEnzyme Inhibitors +3
Target Protein:
4-hydroxy-tetrahydrodipicolinate reductase4-hydroxy-tetrahydrodipicolinate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dipipanone DB01491
small molecule | CAS: 467-83-4

Deskripsi belum tersedia.

Kategori:
Ketones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dipotassium phosphate Approved DB09414
small molecule | CAS: 7758-11-4

Dipotassium phosphate (K2HPO4) is a highly water-soluble salt often used as a fertilizer and food additive as a source of phosphorus and potassium as well as a buffering agent.

Kategori:
AcidsAcids, NoncarboxylicAnions +14
Waktu ParuhIn healthy children…
Vol. DistribusiDistribution is lar…
KlirensPhosphates are rapi…
Genetik -
Dipraglurant DB12733
small molecule | CAS: 872363-17-2

Dipraglurant has been used in trials studying the treatment of Parkinson's Disease. It is a metabotropic glutamate receptor 5 (mGluR5) negative allosteric modulator (NAM).

Target Protein:
Metabotropic glutamate receptor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diprenorphine DB01548
small molecule | CAS: 14357-78-9

A narcotic antagonist similar in action to naloxone. It is used to remobilize animals after etorphine neuroleptanalgesia and is considered a specific antagonist to etorphine. [PubChem]

Kategori:
AlkaloidsCentral Nervous System AgentsHeterocyclic Compounds, Fused-Ring +6
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 25265-71-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Dipyridamole Approved DB00975
small molecule | CAS: 58-32-2

A phosphodiesterase inhibitor that blocks uptake and metabolism of adenosine by erythrocytes and vascular endothelial cells. Dipyridamole also potentiates the antiaggregating action of prostacyclin. (From AMA Drug Evaluations Annual, 1994, p752)

Kategori:
AnticoagulantsAntiplatelet agentsBlood and Blood Forming Organs +17
Target Protein:
cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10AcGMP-specific 3',5'-cyclic phosphodiesterase3',5'-cyclic-AMP phosphodiesterase 4A +3
Waktu Paruh40 minutes
Vol. Distribusi* 1 to 2.5 L/kg
Klirens* 2.3-3.5 mL/min/kg
Genetik -
Dipyrithione Approved DB11327
small molecule | CAS: 3696-28-4

Dipyrithione, a bactericidal and fungicidal pyrithione derivate, was formulated as Crimanex anti-dandruff shampoo, but is no longer available.[L2611] It is currently used as a pesticide, and not used in any FDA approved drug products.[A32829] Interestingl…

Target Protein:
Nitric oxide synthase, inducibleProstaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dipyrocetyl DB13839
small molecule | CAS: 486-79-3

Deskripsi belum tersedia.

Kategori:
AnalgesicsAntiinflammatory and Antirheumatic ProductsMusculo-Skeletal System +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
CoenzymesEnzymes and Coenzymes
Target Protein:
Porphobilinogen deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diridavumab DB12607
biotech | CAS: 1393659-46-5

Cr6261 is under investigation in clinical trial NCT02016066 (A Study to Assess the Safety, Pharmacokinetics and Immunogenicity of Diridavumab in Japanese Healthy Participants).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2163074-23-3

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dirocaftor DB16143
small molecule | CAS: 2137932-23-9

Dirocaftor is under investigation in clinical trial NCT03251092 (Study Designed to Assess the Safety, Tolerability and PK of PTI-808 in Healthy Volunteers and in Adults With Cystic Fibrosis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diroximel fumarate Approved DB14783
small molecule | CAS: 1577222-14-0

Multiple Sclerosis (MS) is a chronic, debilitating neurological disease that can lead to profound cognitive and physical symptoms, severely affecting quality of life.[A176474] It is the main cause of neurological disability not caused by trauma in the young a…

Kategori:
Acids, AcyclicAntineoplastic and Immunomodulating AgentsDicarboxylic Acids +3
Target Protein:
Neuronal acetylcholine receptor subunit alpha-10
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe apparent volume…
KlirensNo clearance inform…
Genetik -
Dirucotide DB04921
biotech | CAS: 152074-97-0

Dirucotide is a synthetically prepared peptide. In particular, the sequence prepared is a 17 amino acid chain that is identical to a section of myelin basic protein (MBP) that is found in humans. Dirucotide has been developed for the treatment of multiple scl…

Kategori:
Amino Acids, Peptides, and ProteinsMembrane ProteinsMyelin Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 130114-83-9

Disaccharide tripeptide glycerol dipalmitoyl is under investigation in clinical trial NCT00003667 (Combination Chemotherapy and Biological Therapy in Treating Patients With High-Risk Ewing's Sarcoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2136633-23-1

Disitamab vedotin is an antibody-drug conjugate drug targeting human epidermal growth factor receptor 2 (HER2). It is currently being investigated for cancers.[A254721]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibody-drug Conjugates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disitertide DB12953
biotech | CAS: 272105-42-7

Disitertide has been used in trials studying the treatment of Skin Fibrosis.

Target Protein:
Transforming growth factor beta-1 proprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disomotide DB17469
biotech | CAS: 181477-43-0

Disomotide is a synthetic peptide cancer vaccine.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disopyramide Approved DB00280
small molecule | CAS: 3737-09-5

A class I anti-arrhythmic agent (one that interferes directly with the depolarization of the cardiac membrane and thus serves as a membrane-stabilizing agent) with a depressant action on the heart similar to that of guanidine. It also possesses some anticholi…

Kategori:
Agents producing tachycardiaAntiarrhythmic agentsAntiarrhythmics, Class I +21
Target Protein:
Sodium channel protein type 5 subunit alphaMuscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +5
Waktu Paruh6.7 hours (range 4-…
Vol. Distribusi-
Klirens-
Genetik -
Disperse Blue 106 Approved DB14203
small molecule | CAS: 68516-81-4

Disperse Blue 106 is used in allergenic testing.

Kategori:
AllergensAntigensBiological Factors +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Distearyldimonium Approved DB14143
small molecule | CAS: 14357-21-2

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAminesAmmonium Compounds +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Distigmine DB13694
small molecule | CAS: 17299-00-2

Distigmine is a parasympathomimetic agent with a longer duration of action and enhanced drug accumulation compared to [DB00545] and [DB01400]. It is an anticholinergic drug and long-acting reversible carbamate cholinesterase inhibitor that binds directly and …

Kategori:
Cholinergic AgentsCholinesterase InhibitorsEnzyme Inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disufenton DB17298
small molecule | CAS: 168021-77-0

Deskripsi belum tersedia.

Kategori:
AntioxidantsArylsulfonatesArylsulfonic Acids +9
Target Protein:
Extracellular sulfatase Sulf-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disulfiram Approved DB00822
small molecule | CAS: 97-77-8

A carbamate derivative used as an alcohol deterrent. It is a relatively nontoxic substance when administered alone, but markedly alters the intermediary metabolism of alcohol. When alcohol is ingested after administration of disulfiram, blood acetaldehyde con…

Kategori:
Acetyl Aldehyde Dehydrogenase InhibitorsAcids, AcyclicAgents that reduce seizure threshold +26
Target Protein:
Dopamine beta-hydroxylaseAldehyde dehydrogenase family 3 member A2Aldehyde dehydrogenase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ditazole DB08994
small molecule | CAS: 18471-20-0

Ditazole is a non-steroidal anti-inflammatory drug (NSAID). Ditazole's analgesic and antipyretic effects are similar to phenylbutazone. Additionally, ditazole is a platelet aggregation inhibitor marketed in Spain and Portugal with trade name Ageroplas.

Kategori:
AnticoagulantsBlood and Blood Forming OrgansPlatelet Aggregation Inhibitors Excl. Heparin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dithiazanine DB11516
small molecule | CAS: 7187-55-5

Dithiazanine is a highly potent anthelmintic, introduced in 1959 for the treatment of strongyloid worms and whipworms. However, its use is severely limited due to its toxicity. Dithiazanine iodide was associated with eight fatal cases of severe acidosis and s…

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dithiopyr DB15230
small molecule | CAS: 97886-45-8

Dithiopyr is under investigation in clinical trial NCT01236781 (Comparison of Full-Field Digital Mammography With Digital Breast Tomography for Screening Call-Back Rates).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ditiocarb DB02520
small molecule | CAS: 147-84-2

A chelating agent that has been used to mobilize toxic metals from the tissues of man and experimental animals. It is the main metabolite of DISULFIRAM.

Kategori:
Acids, AcyclicAdjuvants, ImmunologicAnti-Infective Agents +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Divarasib DB17488
small molecule | CAS: 2417987-45-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Divozilimab DB18878
biotech | CAS: 2254061-60-2

Divozilimab is under investigation in clinical trial NCT05730699 (Efficacy and Safety of Divozilimab in Patients With Neuromyelitis Optica Spectrum Disorders (AQUARELLE)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic and Immunomodulating Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dixanthogen DB13712
small molecule | CAS: 502-55-6

Deskripsi belum tersedia.

Kategori:
AnionsAntiparasitic Products, Insecticides and RepellentsEctoparasiticides, Incl. Scabicides +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dixyrazine DB13784
small molecule | CAS: 2470-73-7

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAntiemetics +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-alpha tocopheryl acetate Approved DB14477
small molecule | CAS: 52225-20-4

Deskripsi belum tersedia.

Kategori:
Vitamin EVitaminsVitamins (Fat Soluble)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-alpha-Tocopherol Approved DB14476
small molecule | CAS: 10191-41-0

Deskripsi belum tersedia.

Kategori:
Vitamin EVitaminsVitamins (Fat Soluble)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 18656-38-7

A synthetic phospholipid used in liposomes and lipid bilayers for the study of biological membranes. It is used in commercial drug preparations to solubilize drugs for injection [A32711]

Kategori:
Compounds used in a research, industrial, or household settingGlycerophosphatesGlycerophospholipids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61361-72-6

DL-dimyristoylphosphatidylglycerol is a phospholipid used in commercially available pharmaceutical preparations to solubilize drugs for injection.

Kategori:
GlycerophosphatesGlycerophospholipidsLipids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-Methylephedrine Approved DB11278
small molecule | CAS: 1201-56-5

Methylephedrine is a sympathomimetic amine that appears in various over-the-counter cough and cold medications throughout the world [L2838], [L2839], [L2840]. The abuse of methylephedrine-containing medications has been reported in Japan. Methylephedrine is n…

Kategori:
Adrenergic AgonistsAdrenergic alpha-2 Receptor AgonistsAdrenergic alpha-Agonists +10
Target Protein:
Beta-1 adrenergic receptorAlpha-2A adrenergic receptorAlpha adrenergic receptor +1
Waktu Paruh3-6 hours (Ephedrin…
Vol. DistribusiEphedrine: 2.5-3.0 …
Klirens-
Genetik -
DLO6001 DB05178
small molecule

DL6001 is developed by DanioLabs using proprietary zebrafish technology to treat Parkinson’s disease symptoms including sialorrhoea and hyperhidrosis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DLO6002 DB05179
small molecule

DLO6002 is developed by Summit Corporation and is in phase I of clinical trials for the treatment of Parkinson's disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DM-1157 DB18600
small molecule | CAS: 1239953-66-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DMP-777 DB18488
small molecule | CAS: 157341-41-8

DMP-777 is a selective inhibitor of polymorphonuclear leukocyte (PMN) elastase.

Kategori:
AzetinesEnzyme InhibitorsPancreatic Elastase, antagonists & inhibitors
Target Protein:
Neutrophil elastase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DNB-001 DB05757
small molecule

DNB-001 is a first-in-class oral therapy with dual mechanism of action, which is initially being developed for the treatment of glaucoma. In preclinical animal models, DNB-001 has demonstrated potent IOP- lowering effects as well as neuroprotective effects on…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DNL343 DB18678
small molecule | CAS: 2278265-85-1

DNL343 is under investigation in clinical trial NCT05842941 (HEALEY ALS Platform Trial - Regimen G DNL343).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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Klirens-
Genetik -
Docaravimab DB17802
biotech | CAS: 2247196-23-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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