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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 89 / 252
Darifenacin Approved DB00496
small molecule | CAS: 133099-04-4

Darifenacin (Enablex®, Novartis) is a medication used to treat urinary incontinence. Darifenacin blocks M3 muscarinic acetylcholine receptors, which mediate bladder muscle contractions. This block reduces the urgency to urinate and so it should not be used…

Kategori:
Agents producing tachycardiaAnticholinergic AgentsCholinergic Agents +15
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +2
Waktu ParuhThe elimination hal…
Vol. Distribusi* 163 L
Klirens* 40 L/h [extensive…
Genetik -
Darigabat DB18966
small molecule | CAS: 1614245-70-3

Darigabat is under investigation in clinical trial NCT05941442 (A Study to Evaluate Efficacy, Safety, and Tolerability of Darigabat in Participants With Panic Disorder).

Kategori:
GABA AgentsGABA ModulatorsNeurotransmitter Agents
Waktu Paruh-
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Genetik -
Darleukin DB17157
biotech

Deskripsi belum tersedia.

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Darolutamide Approved DB12941
small molecule | CAS: 1297538-32-9

Darolutamide is a nonsteroidal androgen receptor antagonist for the treatment of castrate-resistant, non-metastatic prostate cancer (nmCRPC). This condition occurs in the majority of patients with advanced prostate cancer who have been treated with androgen r…

Kategori:
Androgen Receptor InhibitorsAntiandrogensAntiandrogens, non-steroidal +14
Target Protein:
Androgen receptorProgesterone receptor
Waktu ParuhThe half-life of da…
Vol. DistribusiAfter intravenous a…
KlirensThe clearance of da…
Genetik -
Darovasertib DB16059
small molecule | CAS: 1874276-76-2

IDE-196 is under investigation in clinical trial NCT03947385 (Study of IDE196 in Patients With Solid Tumors Harboring GNAQ/11 Mutations or PRKC Fusions).

Waktu Paruh-
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Darunavir Approved DB01264
small molecule | CAS: 206361-99-1

Darunavir is a protease inhibitor used with other HIV protease inhibitor drugs as well as [ritonavir] for the effective management of HIV-1 infection.[L9227] As a second-generation protease inhibitor, darunavir is designed to combat resistance to standard HIV…

Kategori:
AmidesAnti-HIV AgentsAnti-Infective Agents +33
Target Protein:
Pol polyproteinGag-Pol polyprotein
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensDarunavir has a low…
Genetik -
Darvadstrocel Approved DB16581
biotech

Darvadstrocel is a suspension of expanded human allogeneic adipose-derived mesenchymal stem cells extracted from the subdermal adipose tissue of healthy donors via liposuction.[A244524] Darvadstrocel was first approved by the European Commission on March 23, …

Kategori:
Antineoplastic and Immunomodulating AgentsImmunomodulatory AgentsImmunosuppressive Agents +1
Waktu ParuhPharmacokinetic inf…
Vol. DistribusiIn preclinical tria…
KlirensPharmacokinetic inf…
Genetik -
DAS-181 DB15313
biotech | CAS: 946032-08-2

DAS-181 is under investigation in clinical trial NCT00527865 (Single Dose Escalating Study of DAS181 in Adults).

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
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DAS-431 IV DB05432
small molecule

DAS-431 IV is a dopamine D1 receptor agonist developed by DrugAbuse Sciences for the treatment of Addictions, Schizophrenia, Schizoaffective Disorders, Dementia, Parkinson's Disease, Strokes etc.

Target Protein:
Neuron-specific vesicular protein calcyon
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DAS869 DB02850
small molecule

Deskripsi belum tersedia.

Target Protein:
4-hydroxyphenylpyruvate dioxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dasabuvir Approved DB09183
small molecule | CAS: 1132935-63-7

Dasabuvir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine …

Kategori:
AmidesAminesAntiinfectives for Systemic Use +20
Target Protein:
Genome polyproteinNonstructural protein 5b
Waktu ParuhThe half-life of el…
Vol. DistribusiDasabuvir has a vol…
KlirensClearance of Dasabu…
Genetik -
Dasatinib Approved DB01254
small molecule | CAS: 302962-49-8

Dasatinib is an orally available multikinase inhibitor indicated for the treatment of Philadelphia chromosome (Ph)-positive leukemias.[A2224,L45171] Ph is a chromosomal abnormality found in patients with chronic myelogenous leukemia (CML) and acute lymphocyti…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBcr-Abl Tyrosine Kinase Inhibitors +31
Target Protein:
Tyrosine-protein kinase ABL1Proto-oncogene tyrosine-protein kinase SrcEphrin type-A receptor 2 +20
Waktu ParuhThe terminal half-l…
Vol. DistribusiDasatinib has an ap…
KlirensThe clearance of da…
Genetik -
Dasiglucagon Approved DB15226
biotech | CAS: 1544300-84-6

Dasiglucagon is a glucagon analog that acts to increase blood sugar levels.[L39190] It consists of 29 amino acids similar to endogenous glucagon; however, it contains seven substituted amino acids for improved physical and chemical stability in its drug formu…

Kategori:
Amino Acids, Peptides, and ProteinsAntihypertensive AgentsAntihypoglycemic Agent +10
Target Protein:
Glucagon receptor
Waktu ParuhThe half-life was a…
Vol. DistribusiThe mean apparent v…
Klirens-
Genetik -
Dasiprotimut-T DB17287
biotech

Dasiprotimut-T is a personalized therapeutic vaccine against B-cell lymphomas.[A254701] It has been investigated in clinical trials.

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating Agents
Waktu Paruh-
Vol. Distribusi-
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small molecule | CAS: 503291-52-9

Dasolampanel etibutil has been used in trials studying the treatment of Diabetic Neuropathy, Painful.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
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Dasotraline DB12305
small molecule | CAS: 675126-05-3

Dasotraline is a serotonin, norepinephrine and dopamine reuptake inhibitor (SNDRI) that is under investigation for the treatment of Binge Eating Disorder, Adult Attention Hyperactivity Disorder, Attention Deficit Hyperactivity Disorder, and Adult Attention De…

Kategori:
AminesCycloparaffinsNaphthalenes
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2238831-60-0

Datopotamab deruxtecan is under investigation in clinical trial NCT04656652 (Study of DS-1062A Versus Docetaxel in Previously Treated Advanced or Metastatic Non-small Cell Lung Cancer Without Actionable Genomic Alterations (TROPION-LUNG01)).

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dATP DB03222
small molecule | CAS: 1927-31-7

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesDeoxyribonucleotidesHeterocyclic Compounds, Fused-Ring +4
Target Protein:
P2Y purinoceptor 11Anaerobic ribonucleoside-triphosphate reductaseProtein RecA +4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Daunorubicin Approved DB00694
small molecule | CAS: 20830-81-3

A very toxic anthracycline aminoglycoside antineoplastic isolated from Streptomyces peucetius and others, used in treatment of leukemia and other neoplasms.

Kategori:
Anthracycline Topoisomerase InhibitorAnthracyclinesAnthracyclines and Related Substances +30
Target Protein:
DNADNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Gen Terkait:
CYP1B1 HNRNPD SEC14L3 +4
Waktu ParuhDaunorubicin has be…
Vol. DistribusiDaunorubicin has a …
KlirensDaunorubicin has a …
Genetik 7 Varian
Davalintide DB14956
biotech | CAS: 863919-85-1

Davalintide is under investigation in clinical trial NCT00785408 (Study to Examine Safety, Tolerability and Effect on Body Weight of Subcutaneous AC2307 in Obese or Overweight Subjects).

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Davanat DB15311
small molecule | CAS: 916851-14-4

Davanat is under investigation in clinical trial NCT00054977 (Safety of GM-CT-01 With and Without 5-Fluorouracil in Patients With Solid Tumors).

Kategori:
CarbohydratesHexosesMonosaccharides +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Davesomeran Approved DB17091
biotech | CAS: 2798905-80-1

Davesomeran is a mRNA vaccine used in conjunction with [elasomeran] as part of the Moderna Bivalent COVID-19 vaccine. Similar to the previous Moderna COVID-19 vaccine, Moderna Bivalent vaccine encodes the full-length pre-fusion stabilized spike (S) protein to…

Kategori:
COVID-19 VaccinesVaccinesViral Vaccines
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
Daxdilimab DB16391
biotech | CAS: 2245966-28-1

Daxdilimab is under investigation in clinical trial NCT04526912 (Treatment and Prevention of Acute Lung Injury (ALI) in Patients With COVID-19 Infection).

Waktu Paruh-
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DaxibotulinumtoxinA Approved DB17929
biotech | CAS: 93384-43-1

DaxibotulinumtoxinA is an acetylcholine release inhibitor and neuromuscular blocking agent. It is a botulinum toxin without accessory proteins purified from the bacterium _Clostridium botulinum_ type A,[L47840] the gram-positive anaerobic bacterium primarily …

Kategori:
Acetylcholine Release InhibitorsBotulinum ToxinsBotulinum Toxins, Type A +6
Target Protein:
Synaptosomal-associated protein 25
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Dazcapistat DB18301
small molecule | CAS: 2221010-42-8

Deskripsi belum tersedia.

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Dazodalibep DB19025
biotech | CAS: 2245953-10-8

Dazodalibep is under investigation in clinical trial NCT06104124 (A Study to Evaluate the Efficacy and Safety of Dazodalibep in Participants With Sjögren's Syndrome (SS) With Moderate-to-severe Systemic Disease Activity).

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Dazostinag DB18889
small molecule | CAS: 2553413-86-6

Dazostinag is under investigation in clinical trial NCT04420884 (A Study of Dazostinag as Single Agent and Dazostinag in Combination With Pembrolizumab in Adults With Advanced or Metastatic Solid Tumors).

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Dazoxiben DB03052
small molecule | CAS: 78218-09-4

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsThromboxane-A Synthase, antagonists & inhibitors
Target Protein:
Thromboxane-A synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dazucorilant DB18025
small molecule | CAS: 1496508-34-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Dazukibart DB18429
biotech | CAS: 2639474-65-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
DCFBC DB07754
small molecule | CAS: 564482-79-7

Deskripsi belum tersedia.

Target Protein:
Glutamate carboxypeptidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DCLL-9718S DB17392
biotech

DCLL9718S is an antibody-drug conjugate targeting C-type lectin-like molecule-1 (CLL-1). DCLL9718S is under investigation in clinical trial NCT03298516 (A Study of DCLL9718S in Participants With Relapsed or Refractory Acute Myeloid Leukemia (AML) or DCLL9718S…

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DCVAC/OvCa DB18571
biotech

DCVAC/OvCa is a therapy comprising autologous dendritic cells pulsed with killed ovarian cancer cells and matured by TLR3 ligand _ex vivo_. It is under investigation for the treatment of ovarian cancer.

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DCVax-L DB17580
biotech

DCVax-L is a personalized immunotherapy comprising an autologous vaccine with dendritic cells loaded _in vitro_ with autologous tumour lysate.

Waktu Paruh-
Vol. Distribusi-
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DDP-200 DB05919
small molecule

DDP200 is developed by Dynogen for the treatment of non-incontinent form of overactive bladder (OAB) with particular focus on both male and female patients with urinary frequency, urinary urgency and nocturia.

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DDP-225 DB05642
small molecule | CAS: 476148-82-0

DDP225 is both a noradrenaline reuptake inhibitor and a serotonin type 3 receptor (5-HT3) antagonist. Noradrenaline and serotonin are neurotransmitters that are known to be involved in the control of the gastrointestinal system. The unique combination of nor…

Target Protein:
5-hydroxytryptamine receptor 3ASodium-dependent noradrenaline transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 99487-25-9

Deskripsi belum tersedia.

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Genetik -
DDP733 DB05049
small molecule

DDP733 is an oral prokinetic drug which Dynogen is developing as a treatment for both Irritable Bowel Syndrome with constipation (IBS-c) and nocturnal gastroesophageal reflux disease (NGERD). It is a partial agonist of the serotonin type 3 receptor (5-HT3). S…

Target Protein:
5-hydroxytryptamine receptor 3A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 165659-77-8

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntineoplastic AgentsHeterocyclic Compounds, Fused-Ring +6
Target Protein:
Calmodulin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deanol DB13352
small molecule | CAS: 108-01-0

Deanol is commonly referred to as 2-(dimethylamino)ethanol, dimethylaminoethanol (DMAE) or dimethylethanolamine (DMEA). It holds tertiary amine and primary alcohol groups as functional groups. Deanol has been used in the treatment of attention deficit-hyperac…

Kategori:
AlcoholsAminesAmino Alcohols +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DEBIO-1347 DB12903
small molecule | CAS: 1265229-25-1

Ch5183284 has been used in trials studying the treatment of Solid Tumours.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Debrisoquine Approved DB04840
small molecule | CAS: 1131-64-2

An adrenergic neuron-blocking drug similar in effects to guanethidine. It is also noteworthy in being a substrate for a polymorphic cytochrome P-450 enzyme. Persons with certain isoforms of this enzyme are unable to properly metabolize this and many other cli…

Kategori:
Adrenergic AgentsAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +12
Target Protein:
Sodium-dependent noradrenaline transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 125118-55-0

Deskripsi belum tersedia.

Kategori:
Protein Kinase C, antagonists & inhibitors
Target Protein:
Serine/threonine-protein kinase Chk2Serine/threonine-protein kinase Chk1Dual specificity mitogen-activated protein kinase kinase 1 +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Decamethonium Approved DB01245
small molecule | CAS: 156-74-1

Decamethonium is used in anesthesia to cause paralysis. It is a short acting depolarizing muscle relaxant. It is similar to acetylcholine and acts as a partial agonist of the nicotinic acetylcholine receptor.

Kategori:
AminesBis-Trimethylammonium CompoundsCentral Nervous System Depressants +8
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Acetylcholine receptor subunit alphaNeuronal acetylcholine receptor subunit alpha-4 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Decamethoxine DB13705
small molecule | CAS: 38146-42-8

Deskripsi belum tersedia.

Kategori:
AminesAnti-Bacterial AgentsAnti-Infective Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Decernotinib DB12566
small molecule | CAS: 944842-54-0

Decernotinib has been used in trials studying the treatment of Drug Interactions and Rheumatoid Arthritis.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins +1
Target Protein:
Tyrosine-protein kinase JAK3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Decitabine Approved DB01262
small molecule | CAS: 2353-33-5

Myelodysplastic syndromes (MDS) are a heterogeneous group of hematopoietic neoplasms with variable underlying etiology and presentation, including neutropenia and thrombocytopenia. Further mutations leading to increased proliferation of cancerous cells can ev…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
DNADNA (cytosine-5)-methyltransferase 1DNA (cytosine-5)-methyltransferase 3A +2
Waktu ParuhDecitabine has a ha…
Vol. DistribusiDecitabine as an ap…
KlirensDecitabine has a cl…
Genetik -
Decoglurant DB11923
small molecule | CAS: 911115-16-7

Decoglurant has been used in trials studying the treatment of Major Depressive Disorder.

Target Protein:
Metabotropic glutamate receptor 3Metabotropic glutamate receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Decoquinate DB11394
small molecule | CAS: 18507-89-6

Decoquinate is used in veterinary to delay the growth and reproduction of coccidian parasites.

Kategori:
Anti-Infective AgentsAntiparasitic AgentsAntiprotozoals +4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Dectrekumab DB14789
biotech | CAS: 1528523-94-5

Dectrekumab is under investigation in clinical trial NCT00987545 (Efficacy 2 Part Study of Identification of Keloid Biomarkers and Effect of QAX576 on Keloid Recurrence).

Waktu Paruh-
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Menampilkan 4401–4450 dari 12560
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