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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 89 / 282
Certoparin Approved DB09261
small molecule

Certoparin is part of the heparins of low molecular weight that presents high activity against the coagulation factor Xa. It is normally used to prevent deep venous thrombosis.

Kategori:
Agents causing hyperkalemiaAnticoagulantsCarbohydrates +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerulenin DB01034
small molecule | CAS: 17397-89-6

Cerulenin is an antifungal agent whose activity interferes with or otherwise acts to prevent the formation of fatty acids and sterols. In fatty acid synthesis, reported to bind in equimolar ratio to b-keto-acyl-ACP synthase. In sterol synthesis, inhibits HMG-…

Kategori:
AmidesAnti-Infective AgentsAntifungal Agents +3
Target Protein:
3-oxoacyl-[acyl-carrier-protein] synthase 13-oxoacyl-[acyl-carrier-protein] synthase 23-oxoacyl-[acyl-carrier-protein] synthase 3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cesium DB15392
small molecule | CAS: 7440-46-2

Cesium is under investigation in clinical trial NCT02794675 (Intraoperative Placement of Cesium-131 Permanent Interstitial Brachytherapy in Head and Neck Cancer).

Kategori:
ElementsMetalsMetals, Alkali +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cesium Cs-131 DB19250
small molecule | CAS: 14914-76-2

Cesium Cs-131 is under investigation in clinical trial NCT04340258 (Trial Combining Pembrolizumab and Cesium 131 Brachytherapy With Salvage Surgery in HNSCC).

Kategori:
Cesium IsotopesElementsIsotopes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetalkonium Approved DB11583
small molecule | CAS: 10328-34-4

Cetalkonium is a C16 alkyl benzalkonium chloride derivative with an amphipathic property which allows it to be used in different types of formulations.[A27143] It is a quaternary ammonium salt that acts as an antiseptic against a variety of bacteria and fungi…

Kategori:
AlcoholsAminesAmmonium Compounds +7
Waktu ParuhAs cetalkonium is n…
Vol. DistribusiAs cetalkonium is n…
KlirensAs cetalkonium is n…
Genetik -
Cethromycin DB06419
small molecule | CAS: 205110-48-1

Cethromycin is a 3-keto (ketolide) derivative of erythromycin A with an 11,12-carbamate group and an O-6-linked aromatic ring system.[A203369] Cethromycin represents a joint development effort by Abbott Laboratories, Taisho Pharmaceuticals, and Advanced Life …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCytochrome P-450 CYP3A Inhibitors +15
Target Protein:
23S ribosomal RNA
Waktu ParuhCethromycin given i…
Vol. DistribusiCethromycin given i…
KlirensCethromycin clearan…
Genetik -
Cetilistat DB06586
small molecule | CAS: 282526-98-1

Cetilistat is a novel inhibitor of pancreatic lipase being developed by Alizyme for the treatment of obesity and associated co-morbidities, including type 2 diabetes.

Kategori:
Anti-Obesity AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Endothelial lipaseGastric triacylglycerol lipasePancreatic triacylglycerol lipase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetrelimab DB15421
biotech | CAS: 2050478-92-5

Cetrelimab is under investigation in clinical trial NCT03547037 (A Study to Evaluate the Safety, Pharmacokinetics, Pharmacodynamics, and Immunogenicity of JNJ-63723283, an Anti-Programmed Cell Death (PD)-1 Monoclonal Antibody, as Monotherapy or in Combination…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetrorelix Approved DB00050
small molecule | CAS: 120287-85-6

Cetrorelix is a man-made hormone that blocks the effects of Gonadotropin Releasing Hormone (GnRH). GnRH controls another hormone that is called luteinizing hormone (LH), which is the hormone that starts ovulation during the menstrual cycle. When undergoing ho…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Gonadotropin-Releasing HormonesDecreased GnRH Secretion +18
Target Protein:
Gonadotropin-releasing hormone receptorLutropin-choriogonadotropic hormone receptor
Waktu Paruh~62.8 hours
Vol. Distribusi* 1.16 L/kg
Klirens* 1.28 ml/min·kg [a…
Genetik -
Cetuximab Approved DB00002
biotech | CAS: 205923-56-4

Cetuximab is a recombinant chimeric human/mouse IgG1 monoclonal antibody that competitively binds to epidermal growth factor receptor (EGFR) and competitively inhibits the binding of epidermal growth factor (EGF).[A227973] EGFR is a member of the ErbB family …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Epidermal growth factor receptorLow affinity immunoglobulin gamma Fc region receptor III-BComplement C1q subcomponent subunit A +5
Gen Terkait:
FCGR2A FCGR3A
Waktu ParuhAfter administratio…
Vol. DistribusiThe volume of the d…
KlirensIn patients with re…
Genetik 2 Varian
biotech | CAS: 2166339-33-7

Cetuximab sarotalocan is under investigation in clinical trial NCT03769506 (ASP-1929 Photoimmunotherapy (PIT) Study in Recurrent Head/Neck Cancer for Patients Who Have Failed at Least Two Lines of Therapy) for the treatment of Recurrent Head/Neck Cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetyl alcohol Approved DB09494
small molecule | CAS: 36653-82-4

Cetyl alcohol, also known as 1-hexadecanol or n-hexadecyl alcohol, is a 16-C fatty alcohol with the chemical formula CH3(CH2)15OH. It can be produced from the reduction of palmitic acid. Cetyl alcohol is present in a waxy white powder or flake form at room te…

Kategori:
AlcoholsDrugs that are Mainly Renally ExcretedLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 59130-69-7

Cetyl ethylhexanoate is an ester of cetyl alcohol and 2-ethylhexanoic acid. It is present in cosmetic products as a skin conditioning agent and emollient.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetyl oleate DB19454
small molecule | CAS: 22393-86-8

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetyl palmitate DB15782
small molecule | CAS: 540-10-3

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipidsPalmitic Acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 22393-83-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetylpyridinium Approved DB11073
small molecule | CAS: 7773-52-6

Cetylpyridinium is a quaternary ammonium with broad-spectrum antiseptic properties. Its salt form, cetylpyridinium chloride, is typically found as an active ingredient in mouthwashes, toothpastes, lozenges, throat sprays, breath sprays, and nasal sprays. In t…

Kategori:
Alimentary Tract and MetabolismAnti-Infective AgentsAnti-Infective Agents, Local +19
Waktu ParuhNo readily availabl…
Vol. DistribusiNo readily availabl…
KlirensNo readily availabl…
Genetik -
small molecule | CAS: 102580-74-5

Deskripsi belum tersedia.

Kategori:
AminesAnti-Infective AgentsAnti-Infective Agents, Local +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2247971-00-0

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cevidoplenib DB18725
small molecule | CAS: 1703788-21-9

Deskripsi belum tersedia.

Kategori:
Oxazoles
Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cevimeline Approved DB00185
small molecule | CAS: 107233-08-9

Cevimeline is a parasympathomimetic agent that act as an agonist at the muscarinic acetylcholine receptors M1 and M3. It is indicated by the Food and Drug Administration for the treatment of dry mouth associated with Sjögren's syndrome.

Kategori:
Autonomic AgentsCholinergic AgentsCholinergic Agonists +12
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1
Waktu Paruh5 ± 1 hours
Vol. Distribusi* 6 L/kg
Klirens-
Genetik -
Cevipabulin DB12533
small molecule | CAS: 849550-05-6

Cevipabulin has been used in trials studying the treatment and educational/counseling/training of Tumors and Neoplasms.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cevostamab DB18374
biotech | CAS: 2249888-53-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CFG-920 DB19193
small molecule | CAS: 1260006-20-9

CFG-920 is under investigation in clinical trial NCT04060394 (Dose-escalation and Efficacy Study of Lae001/prednisone Plus Afuresertib Patients With M-crpc).

Target Protein:
Steroid 17-alpha-hydroxylase/17,20 lyase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CFT-8634 DB18443
small molecule | CAS: 2704617-96-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CG-200745 DB12259
small molecule | CAS: 936221-33-9

Cg200745 has been used in trials studying the treatment of Solid Tumour.

Kategori:
AminesAntineoplastic AgentsHistone Deacetylase Inhibitors +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CG-400549 DB12347
small molecule | CAS: 934628-27-0

CG400549 has been used in trials studying the treatment of Skin Infection.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CGC-11047 DB05722
small molecule | CAS: 206991-64-2

CGC-11047 is a polyamine analog designed to halt cell growth and induce apoptosis.

Kategori:
AminesBiogenic AminesBiogenic Polyamines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CGI-1842 DB12744
small molecule | CAS: 900573-88-8

JI-101 has been used in trials studying the treatment of Cancer, Colon Cancer, Neuroendocrine, Ovarian Cancer, and Advanced Solid Tumors.

Kategori:
AmidesBenzene DerivativesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Receptor tyrosine-protein kinase erbB-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CGP 4832 DB04220
small molecule | CAS: 113303-81-4

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingLactams, Macrocyclic
Target Protein:
Ferrichrome-iron receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CGS-27023 DB07556
small molecule | CAS: 161314-70-1

Deskripsi belum tersedia.

Kategori:
AmidesAminesEnzyme Inhibitors +8
Target Protein:
Neutrophil collagenaseA disintegrin and metalloproteinase with thrombospondin motifs 472 kDa type IV collagenase +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CGX-1321 DB17491
small molecule

CGX-1321 is a porcupine inhibitor that affects Wnt production and can block Wnt downstream signaling.[A257038]

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 227016-66-2

CH-1504 L-isomer is under investigation in clinical trial NCT01116141 (A Study of CH-4051 in Patients With Rheumatoid Arthritis (RA)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CH-5132799 DB13051
small molecule | CAS: 1007207-67-1

CH5132799 has been used in trials studying the treatment of Solid Tumors.

Kategori:
AmidesClass I Phosphatidylinositol 3-Kinases, antagonists & inhibitorsSulfones +1
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Chamaemelum nobile flower is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAsteraceaeBiological Products +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chamazulene DB15931
small molecule | CAS: 529-05-5

Deskripsi belum tersedia.

Kategori:
CycloheptanesCycloparaffins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chelerythrine DB17024
small molecule | CAS: 34316-15-9

A benzophenanthridine alkaloid evaluated as a kinase-inhibitor.[A252982]

Kategori:
AlkaloidsAnti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
P2X purinoceptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chenodeoxycholic acid Approved DB06777
small molecule | CAS: 474-25-9

Chenodeoxycholic acid (or Chenodiol) is an epimer of ursodeoxycholic acid (DB01586). Chenodeoxycholic acid is a bile acid naturally found in the body. It works by dissolving the cholesterol that makes gallstones and inhibiting production of cholesterol in the…

Kategori:
Alimentary Tract and MetabolismBile Acid PreparationsBile acids and derivatives +12
Target Protein:
Bile acid receptorNuclear receptor subfamily 1 group I member 2G-protein coupled bile acid receptor 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CHF 4227 DB05882
small molecule

CHF 4227 is a new selective estrogen receptor modulator (SERM). The compound has a high receptor affinity and has shown promising efficacy in the prevention of bone loss in animal models of osteoporosis. Additionally, the compound has shown no uterotrophic ac…

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CHF-6001 DB12800
small molecule | CAS: 1239278-59-1

CHF6001 has been used in trials studying the treatment of Asthma and Chronic Obstructive Pulmonary Disease.

Kategori:
Acids, CarbocyclicAmidesAminobenzoates +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CHF-6333 DB17815
small molecule | CAS: 1613621-54-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CHGN111 DB06376
small molecule

CHGN111 is an inhibitor of the mitochondrial enzyme CLK-1 which is a demethoxyubiquinone hydroxylase. Numerous parameters of mitochondrial function are altered when the activity of CLK-1 is reduced, which results in a decrease of ROS at critical cellular site…

Target Protein:
Dual specificity protein kinase CLK1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chiauranib DB16124
small molecule | CAS: 1256349-48-0

Chiauranib is under investigation in clinical trial NCT03974243 (Chiauranib in Combination With Chidamide in Patients With Relapsed/refractory Non-hodgkin's Lymphoma).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chickpea Approved DB10662
biotech

Chickpea allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chiglitazar DB19023
small molecule | CAS: 743438-45-1

Chiglitazar is under investigation in clinical trial NCT06125587 (Chiglitazar/metformin in Non-obese Women With PCOS).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +3
Target Protein:
Peroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Chikungunya virus (CHIKV) is a member of the Alphavirus genus that was first identified in Tanzania in 1952.[A262051] It is spread primarily by the bite of infected mosquitos of the _Aedes_ genus. Infection with CHIKV causes chikungunya fever, an illness char…

Kategori:
Live vaccinesVaccinesViral Vaccines
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
Chiniofon DB13379
small molecule | CAS: 8002-90-2

Deskripsi belum tersedia.

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CHIR-124 DB06852
small molecule | CAS: 405168-58-3

CHIR-124 is a potent inhibitor of Chk1 that potentiates the cytotoxicity of topoisomerase I poisons in vitro and in vivo.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chitin DB15142
small molecule | CAS: 1398-61-4

Shrimp shell chitin is under investigation in clinical trial NCT00863356 (Trial of a Novel Chitosan Hemostatic Sealant in the Management of Complicated Epistaxis).

Kategori:
BiopolymersCarbohydratesChitin, antagonists & inhibitors +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4401–4450 dari 14063
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