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14361

Total database: 17430
Struktur (SMILES)
9916 (69.0%)
Target
7893 (55.0%)
Genomik
112 (0.8%)
Referensi
14361 (100.0%)

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Hasil Pencarian (14361)

Halaman 88 / 288
CFG-920 DB19193
small molecule | CAS: 1260006-20-9

CFG-920 is under investigation in clinical trial NCT04060394 (Dose-escalation and Efficacy Study of Lae001/prednisone Plus Afuresertib Patients With M-crpc).

Target Protein:
Steroid 17-alpha-hydroxylase/17,20 lyase
Waktu Paruh-
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CFT-8634 DB18443
small molecule | CAS: 2704617-96-7

Deskripsi belum tersedia.

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CG0070 DB05148
small molecule

CG0070 is investigated in clinical trials for treating bladder cancer. CG0070 is a solid. CG0070 can potentially destroy cancer cells by two different mechanisms: direct cell killing by the virus and immune-mediated cell killing stimulated by GM-CSF. CG0070, …

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CG7870 DB04981
biotech

CG7870 is an oncolytic virus therapy for prostate cancer. It is a replication-selective, prostate-specific antigen-targeted oncolytic adenovirus, for the treatment of hormone-refractory, metastatic prostate cancer.

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CGC-11047 DB05722
small molecule | CAS: 206991-64-2

CGC-11047 is a polyamine analog designed to halt cell growth and induce apoptosis.

Kategori:
AminesBiogenic AminesBiogenic Polyamines +1
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CGP 4832 DB04220
small molecule | CAS: 113303-81-4

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingLactams, Macrocyclic
Target Protein:
Ferrichrome-iron receptor
Waktu Paruh-
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CGX-1321 DB17491
small molecule

CGX-1321 is a porcupine inhibitor that affects Wnt production and can block Wnt downstream signaling.[A257038]

Kategori:
Heterocyclic Compounds, Fused-Ring
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small molecule | CAS: 227016-66-2

CH-1504 L-isomer is under investigation in clinical trial NCT01116141 (A Study of CH-4051 in Patients With Rheumatoid Arthritis (RA)).

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Chaetomium globosum Approved DB10430
biotech

Chaetomium globosum is a fungus which can provoke allergic reactions. Chaetomium globosum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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biotech

Deskripsi belum tersedia.

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biotech

Deskripsi belum tersedia.

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biotech

Chamaecyparis obtusa wood oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Genetik -
biotech

Chamaemelum nobile flower is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAsteraceaeBiological Products +8
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Chamomile Approved DB14357
biotech

Chamomile is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAsteraceaeBiological Products +8
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Channel catfish Approved DB15548
biotech

Channel catfish allergenic extract is used in allergenic testing.

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Chelerythrine DB17024
small molecule | CAS: 34316-15-9

A benzophenanthridine alkaloid evaluated as a kinase-inhibitor.[A252982]

Kategori:
AlkaloidsAnti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
P2X purinoceptor 7
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Chenodeoxycholic acid Approved DB06777
small molecule | CAS: 474-25-9

Chenodeoxycholic acid (or Chenodiol) is an epimer of ursodeoxycholic acid (DB01586). Chenodeoxycholic acid is a bile acid naturally found in the body. It works by dissolving the cholesterol that makes gallstones and inhibiting production of cholesterol in the…

Kategori:
Alimentary Tract and MetabolismBile Acid PreparationsBile acids and derivatives +12
Target Protein:
Bile acid receptorNuclear receptor subfamily 1 group I member 2G-protein coupled bile acid receptor 1 +1
Waktu Paruh-
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Chenopodium album pollen Approved DB10368
biotech

Chenopodium album pollen is the pollen of the Chenopodium album plant. Chenopodium album pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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biotech

Chenopodium ambrosioides pollen is the pollen of the Chenopodium ambrosioides plant. Chenopodium ambrosioides pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Chenopodium botrys pollen Approved DB10838
biotech

Chenopodium botrys pollen is the pollen of the Chenopodium botrys plant. Chenopodium botrys pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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CHF 4227 DB05882
small molecule

CHF 4227 is a new selective estrogen receptor modulator (SERM). The compound has a high receptor affinity and has shown promising efficacy in the prevention of bone loss in animal models of osteoporosis. Additionally, the compound has shown no uterotrophic ac…

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
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CHF-6001 DB12800
small molecule | CAS: 1239278-59-1

CHF6001 has been used in trials studying the treatment of Asthma and Chronic Obstructive Pulmonary Disease.

Kategori:
Acids, CarbocyclicAmidesAminobenzoates +4
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CHF-6333 DB17815
small molecule | CAS: 1613621-54-7

Deskripsi belum tersedia.

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CHF5633 DB18696
biotech

CHF5633 is a fully synthetic pulmonary surfactant preparation comprising DPPC (dipalmitoylphosphatidylcholine), POPG Na (palmitoyl?oleoyl?phosphatidylglycerol sodium), a synthetic SP-C analogue, and a synthetic SP-B analogue.

Kategori:
Amino Acids, Peptides, and ProteinsGlycerophosphatesGlycerophospholipids +9
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CHGN111 DB06376
small molecule

CHGN111 is an inhibitor of the mitochondrial enzyme CLK-1 which is a demethoxyubiquinone hydroxylase. Numerous parameters of mitochondrial function are altered when the activity of CLK-1 is reduced, which results in a decrease of ROS at critical cellular site…

Target Protein:
Dual specificity protein kinase CLK1
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Chiauranib DB16124
small molecule | CAS: 1256349-48-0

Chiauranib is under investigation in clinical trial NCT03974243 (Chiauranib in Combination With Chidamide in Patients With Relapsed/refractory Non-hodgkin's Lymphoma).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +1
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Chickpea Approved DB10662
biotech

Chickpea allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
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Chicory leaf DB14376
biotech

Chicory leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Chiglitazar DB19023
small molecule | CAS: 743438-45-1

Chiglitazar is under investigation in clinical trial NCT06125587 (Chiglitazar/metformin in Non-obese Women With PCOS).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +3
Target Protein:
Peroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha
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biotech

Chikungunya virus (CHIKV) is a member of the Alphavirus genus that was first identified in Tanzania in 1952.[A262051] It is spread primarily by the bite of infected mosquitos of the _Aedes_ genus. Infection with CHIKV causes chikungunya fever, an illness char…

Kategori:
Live vaccinesVaccinesViral Vaccines
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
biotech

Deskripsi belum tersedia.

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CHIR-124 DB06852
small molecule | CAS: 405168-58-3

CHIR-124 is a potent inhibitor of Chk1 that potentiates the cytotoxicity of topoisomerase I poisons in vitro and in vivo.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase Chk1
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Chitin DB15142
small molecule | CAS: 1398-61-4

Shrimp shell chitin is under investigation in clinical trial NCT00863356 (Trial of a Novel Chitosan Hemostatic Sealant in the Management of Complicated Epistaxis).

Kategori:
BiopolymersCarbohydratesChitin, antagonists & inhibitors +3
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small molecule | CAS: 9012-76-4

Deskripsi belum tersedia.

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Chloral hydrate Approved DB01563
small molecule | CAS: 302-17-0

A hypnotic and sedative used in the treatment of insomnia. The safety margin is too narrow for chloral hydrate to be used as a general anesthetic in humans, but it is commonly used for that purpose in animal experiments. It is no longer considered useful as a…

Kategori:
AlcoholsCentral Nervous System AgentsCentral Nervous System Depressants +7
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Chlorambucil Approved DB00291
small molecule | CAS: 305-03-3

A nitrogen mustard alkylating agent used as antineoplastic agent for the treatment of various malignant and nonmalignant diseases. Although it is less toxic than most other nitrogen mustards, it has been listed as a known carcinogen in the Fourth Annual Repor…

Kategori:
Agents that reduce seizure thresholdAlkylating ActivityAlkylating Drugs +12
Target Protein:
DNA
Waktu Paruh1.5 hours
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Chloramphenicol Approved DB00446
small molecule | CAS: 56-75-7

An antibiotic first isolated from cultures of _Streptomyces venezuelae_ in 1947 but now produced synthetically. It has a relatively simple structure and was the first broad-spectrum antibiotic to be discovered. It acts by interfering with bacterial protein sy…

Kategori:
AlcoholsAmphenicolsAnti-Acne Preparations +34
Target Protein:
50S ribosomal protein L16Dr hemagglutinin structural subunitComplement decay-accelerating factor
Waktu ParuhHalf-life in adults…
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Chloramphenicol palmitate Approved DB14658
small molecule | CAS: 530-43-8

Deskripsi belum tersedia.

Kategori:
AlcoholsBenzene DerivativesGlycols +3
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Chloramphenicol succinate Approved DB07565
small molecule | CAS: 3544-94-3

Chloramphenicol succinate is an ester prodrug of [chloramphenicol].[A192987] Chloramphenicol is a bacteriostatic antibiotic.[A204065] Use of chloramphenicol succinate and chloramphenicol has decreased due to the risk of potentially fatal blood dyscrasias.[L14…

Kategori:
AlcoholsAnti-Bacterial AgentsAnti-Infective Agents +8
Target Protein:
Dr hemagglutinin structural subunit
Waktu ParuhThe half life of ch…
Vol. DistribusiChloramphenicol suc…
KlirensChloramphenicol suc…
Genetik -
Chlorcyclizine Approved DB08936
small molecule | CAS: 82-93-9

Chlorcyclizine is a first generation phenylpiperazine class antihistamine used to treat urticaria, rhinitis, pruritus, and other allergy symptoms. Chlorcyclizine also has some local anesthetic, anticholinergic, and antiserotonergic properties, and can be used…

Kategori:
Antihistamines for Systemic UseHistamine AntagonistsHistamine H1 Antagonists +3
Target Protein:
Histamine H1 receptor
Waktu Paruhabout 12 h.
Vol. DistribusiAfter a single oral…
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Chlordiazepoxide Approved DB00475
small molecule | CAS: 58-25-3

An anxiolytic benzodiazepine derivative with anticonvulsant, sedative, and amnesic properties. It has also been used in the symptomatic treatment of alcohol withdrawal.

Kategori:
Adjuvants, AnesthesiaAnti-Anxiety AgentsBenzazepines +22
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh24-48 hours
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Chlorfenson DB05377
small molecule | CAS: 80-33-1

Chlorfenson is developed by Moberg Derma for the treatment of onychomycosis (nail fungus) as the primary indication.

Kategori:
ArylsulfonatesArylsulfonic AcidsBenzene Derivatives +3
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Chlorhexadol DB01534
small molecule | CAS: 3563-58-4

Chlorhexadol is a sedative and hypnotic which is regulated in the United States as a Schedule III controlled substance. It is a derivative of chloral hydrate.

Kategori:
AldehydesCentral Nervous System DepressantsHypnotics and Sedatives +2
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Chlorhexidine Approved DB00878
small molecule | CAS: 55-56-1

Chlorhexidine is a broad-spectrum antimicrobial biguanide used as a topical antiseptic and in dental practice for the treatment of inflammatory dental conditions caused by microorganisms.[L11512] It is one of the most common skin and mucous membrane antisepti…

Kategori:
Alimentary Tract and MetabolismAmidinesAnti-Infective Agents +25
Target Protein:
Bacterial outer membrane
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Chlorine DB11109
small molecule | CAS: 7782-50-5

Chlorine is a stongly oxidizing agent and the third most electronegative element which belongs to the group of halogens with the atomic number 17 and symbol Cl. Being a yellow-green gas at room temperature, chlorine is the second most abundant halogen on Eart…

Kategori:
Compounds used in a research, industrial, or household settingElementsGases +4
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small molecule | CAS: 302-22-7

Chlormadinone acetate is a progesterone derivative first synthesized in 1961. In the US, chlormadinone acetate was formerly marketed as a component of the combination drug products Estalor-21 and C-Quens. However, the use of these drugs was associated with th…

Kategori:
Adrenal Cortex HormonesAntiandrogensContraceptive Agents, Female +13
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Chlormerodrin Approved DB00534
small molecule | CAS: 62-37-3

Chlormerodrin is a mercurial compound with toxic side effects that was previously used as a diuretic. The radiolabeled form has been used as a diagnostic and research tool. It is no longer used and has been replaced with new classes of diuretic drugs.

Kategori:
Alkylmercury CompoundsOrganomercury CompoundsOrganometallic Compounds
Target Protein:
Solute carrier family 12 member 1Succinate-semialdehyde dehydrogenase, mitochondrial
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Chlormerodrin Hg-197 Approved DB09406
small molecule | CAS: 64461-80-9

Chlormerodrin Hg-197 is a radiolabelled form of chlormerodrin, an organomercury compound that was previously used as a diuretic. Its radiolabelled form was used as diagnostics in brain scans.

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Chlormezanone Approved DB01178
small molecule | CAS: 80-77-3

A non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.

Kategori:
Anti-Anxiety AgentsCentral Nervous System AgentsCentral Nervous System Depressants +10
Target Protein:
Translocator protein
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Chlorobutanol Approved DB11386
small molecule | CAS: 57-15-8

Chlorobutanol, or chlorbutol, is an alcohol-based preservative with no surfactant activity [A32746]. It also elicits sedative-hypnotic and weak local anesthetic actions in addition to antibacterial and antifungal properties. Similar in nature to chloral hydra…

Kategori:
AlcoholsAlimentary Tract and MetabolismAntiemetics and Antinauseants +8
Target Protein:
Voltage-gated inwardly rectifying potassium channel KCNH2
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe volume of distr…
KlirensIn healthy subjects…
Genetik -
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