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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 88 / 282
Celecoxib Approved DB00482
small molecule | CAS: 169590-42-5

Celecoxib, a selective cyclooxygenase-2 (COX-2) inhibitor, is a nonsteroidal anti-inflammatory drug (NSAID) which is known for its decreased risk of causing gastrointestinal bleeding compared to other NSAIDS.[A181544] It is used to manage symptoms of various …

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +41
Target Protein:
Prostaglandin G/H synthase 2Signal transducer and activator of transcription 3Sialidase-1 +4
Gen Terkait:
CYP2C9
Waktu ParuhThe effective half-…
Vol. DistribusiThe apparent volume…
KlirensApparent clearance …
Genetik 1 Varian
Celgosivir DB06580
small molecule | CAS: 121104-96-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingIndolizines
Target Protein:
Maltase-glucoamylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Celiprolol Approved DB04846
small molecule | CAS: 56980-93-9

Celiprolol is indicated for the management of mild to moderate hypertension and effort-induced angina pectoris. It is simultaneously a selective ?1 receptor antagonist, a ?2 receptor partial agonist and a weak ?2 receptor antagonist. In 2010 a clinical trial …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic Antagonists +30
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor +3
Waktu Paruh5 hours
Vol. DistribusiThe distribution vo…
KlirensCleared by both ren…
Genetik -
Celivarone DB16012
small molecule | CAS: 401925-43-7

Celivarone is under investigation in clinical trial NCT00233441 (Placebo Controlled Double-blind Dose Ranging Study of the Efficacy and Safety of SSR149744C 50, 100, 200 or 300 Mg OD With Amiodarone as Calibrator for the Maintenance of Sinus Rhythm in Patient…

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cellobiose DB02061
small molecule | CAS: 528-50-7

A disaccharide consisting of two glucose units in beta (1-4) glycosidic linkage. Obtained from the partial hydrolysis of cellulose. [PubChem]

Kategori:
CarbohydratesCelluloseCompounds used in a research, industrial, or household setting +4
Target Protein:
Endoglucanase GEndoglucanase 5AEndoglucanase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cellotetraose DB02717
small molecule | CAS: 38819-01-1

Deskripsi belum tersedia.

Kategori:
BiopolymersCarbohydratesCompounds used in a research, industrial, or household setting +5
Target Protein:
Glucanase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Celtis occidentalis pollen Approved DB10472
biotech

Celtis occidentalis pollen is the pollen of the Celtis occidentalis plant. Celtis occidentalis pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cemdisiran DB16121
biotech | CAS: 1639264-46-2

Cemdisiran is under investigation in clinical trial NCT03841448 (A Study of Cemdisiran in Adults With Immunoglobulin a Nephropathy (Igan)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cemdomespib DB18953
small molecule | CAS: 1450642-92-8

Cemdomespib is under investigation in clinical trial NCT05895552 (A Phase 2 Study of RTA 901 in Patients With Diabetic Peripheral Neuropathic Pain (CYPRESS)).

Kategori:
AminesCarbohydratesEthylamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cemiplimab Approved DB14707
biotech | CAS: 1801342-60-8

Cemiplimab is a fully human monoclonal antibody that works against programmed death receptor-1 (PD-1), which is a negative regulator of T cell function. By blocking PD-1, cemiplimab works to enhance T cell-mediated antitumour responses.[L39804] Cemiplimab …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Programmed cell death protein 1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensCemiplimab clearanc…
Genetik -
Cemsidomide DB18400
small molecule | CAS: 2504235-67-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cendakimab DB18427
biotech

Cendakimab is a recombinant humanized anti-interleukin 13 (IL-13) monoclonal antibody.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenderitide DB11777
biotech | CAS: 507289-11-4

Cenderitide is under investigation for the treatment of ST Elevation (STEMI) Myocardial Infarction of Anterior Wall.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsComplex Mixtures +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenegermin Approved DB13926
biotech | CAS: 1772578-74-1

Cenegermin is a human beta-nerve growth factor (beta-ngf)-(1-118)- peptide (non-covalent dimer) produced in escherichia coli. It received European Union Approval in July 2017 for the treatment of moderate to severe neurotrophic keratitis. Cenegermin received …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +7
Target Protein:
High affinity nerve growth factor receptorTumor necrosis factor receptor superfamily member 16
Waktu ParuhHalf-life data spec…
Vol. DistribusiAfter eye drop admi…
KlirensAlthough the system…
Genetik -
Cenerimod DB12705
small molecule | CAS: 1262414-04-9

Cenerimod has been used in trials studying the treatment of Systemic Lupus Erythematosus.

Kategori:
AlcoholsGlycolsOxazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenersen DB15455
biotech | CAS: 415168-49-9

Cenersen is under investigation in clinical trial NCT02243124 (A Study of Aezea® (Cenersen) in Transfusion Dependent Anemia Associated With Myelodysplastic Syndrome (MDS)).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenicriviroc DB11758
small molecule | CAS: 497223-25-3

Cenicriviroc has been used in trials studying the treatment of HIV-infection/AIDS, AIDS Dementia Complex, Nonalcoholic Steatohepatitis, Human Immunodeficiency Virus, and HIV-1-Associated Cognitive Motor Complex.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +4
Target Protein:
C-C chemokine receptor type 5C-C chemokine receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenobamate Approved DB06119
small molecule | CAS: 913088-80-9

Cenobamate, or YKP-3089, is an antiepileptic drug developed by SK Pharmaceuticals and used to treat partial onset seizures.[A188442,L10653] The exact mechanism of action has not been described in the literature, though it positively modulates GABA<sub>A</sub>…

Kategori:
Acids, AcyclicAnticonvulsantsBenzene Derivatives +34
Target Protein:
Voltage-gated sodium channel alpha subunitGamma-aminobutyric acid receptor subunit alpha-1
Waktu ParuhThe terminal half l…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Cenplacel-L DB19188
biotech

Cenplacel-L is under investigation in clinical trial (Study of Human Placenta-derived Cells (PDA001) to Evaluate the Safety and Effectiveness for Patients With Ischemic Stroke) for the treatment of patients with Ischemic Stroke.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Censavudine DB12074
small molecule | CAS: 634907-30-5

Censavudine has been used in trials studying the treatment of HIV-1 Infection.

Kategori:
Anti-HIV AgentsDeoxyribonucleosidesNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Centanafadine DB14841
small molecule | CAS: 924012-43-1

Centanafadine is under investigation in clinical trial NCT02827513 (A Phase 1 Study to Investigate the Safety, Tolerance, Food Effect, Pharmacokinetics and Pharmacodynamics of Single and Multiple Doses of Extended Release Formulations of Centanafadine (CTN) i…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Centella asiatica Approved DB14256
biotech

Centella asiatica is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Agents that reduce seizure thresholdAngiospermsApiaceae +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Centhaquine DB16122
small molecule | CAS: 57961-90-7

Centhaquine is under investigation in clinical trial NCT04045327 (Efficacy of PMZ-2010 (Centhaquine) a Resuscitative Agent for Hypovolemic Shock).

Kategori:
Adrenergic and Dopaminergic AgentsCardiac Stimulants Excl. Cardiac GlycosidesCardiac Therapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CEP-37440 DB13060
small molecule | CAS: 1391712-60-9

CEP-37440 has been used in trials studying the treatment of Solid Tumors.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Focal adhesion kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CEP-9722 DB14882
small molecule | CAS: 916574-83-9

CEP-9722 is under investigation in clinical trial NCT01345357 (Study of CEP-9722 in Combination With Gemcitabine and Cisplatin in Patients With Advanced Solid Tumors or Mantle Cell Lymphoma).

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingImides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1192706-52-7

Cepeginterferon alfa-2B is under investigation in clinical trial NCT01889433 (An Open-label Comparative Efficacy and Safety Study of Algeron (Cepeginterferon Alfa-2b) in Treatment-naive Patients With Chronic Hepatitis C).

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP1A2 Inhibitors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cephalexin Approved DB00567
small molecule | CAS: 15686-71-2

Cephalexin is the first of the first generation cephalosporins.[A179071,A179074] This antibiotic contains a beta lactam and a dihydrothiazide.[A179071] Cephalexin is used to treat a number of susceptible bacterial infections through inhibition of cell wall s…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +23
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2aPenicillin-binding protein 1b +2
Waktu ParuhThe half life of ce…
Vol. Distribusi5.2-5.8L.[A179068]
KlirensClearance from one …
Genetik -
Cephaloglycin Approved DB00689
small molecule | CAS: 3577-01-3

A cephalorsporin antibiotic that is no longer commonly used.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +7
Target Protein:
Penicillin-binding protein 1B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Agents that reduce seizure threshold
Target Protein:
D-alanyl-D-alanine carboxypeptidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cephalosporin C DB03313
small molecule | CAS: 61-24-5

Deskripsi belum tersedia.

Kategori:
Agents that reduce seizure thresholdAmidesbeta-Lactams +4
Target Protein:
Penicillin-binding protein 1bPeptidoglycan synthase FtsIPenicillin-binding protein 1A +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cephalosporium roseum Approved DB10932
biotech

Cephalosporium roseum allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cepharanthine DB16824
small molecule | CAS: 481-49-2

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnalgesicsAnalgesics, Non-Narcotic +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CER-001 DB18538
biotech

CER-001 is a negatively charged lipoprotein particle comprising human recombinant apolipoprotein A-I and two phospholipids: sphingomyelin and dipalmitoylphosphatidylglycerol.[L48290] It is under investigation for the treatment of lecithin-cholesterol acyltran…

Kategori:
Amino Acids, Peptides, and ProteinsApolipoproteinsApolipoproteins A +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceralasertib DB14917
small molecule | CAS: 1352226-88-0

Ceralasertib is under investigation in clinical trial NCT03682289 (Phase II Trial of AZD6738 Alone and in Combination With Olaparib).

Kategori:
AmidesHeterocyclic Compounds, Fused-RingOxazines +2
Target Protein:
Serine/threonine-protein kinase ATR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceralifimod DB16123
small molecule | CAS: 891859-12-4

Ceralifimod is under investigation in clinical trial NCT01226745 (Phase 2 Extension Trial in Patients With Relapsing-remitting Multiple Sclerosis (RRMS)).

Kategori:
AzetinesImmunologic FactorsImmunosuppressive Agents +1
Target Protein:
Sphingosine 1-phosphate receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceramide AP DB14705
small molecule | CAS: 212070-45-6

Deskripsi belum tersedia.

Kategori:
AmidesCarbohydratesGlycoconjugates +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceramide NG DB14706
small molecule | CAS: 2304-80-5

Deskripsi belum tersedia.

Kategori:
AmidesCarbohydratesGlycoconjugates +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceramide NP DB14111
small molecule | CAS: 100403-19-8

Ceramide NP is a lipid molecule included in a group of lipid molecules called ceramides. Ceramides are major lipid components in the stratum corneum of the human skin. Ceramide 3 consists of a phytosphingosine backbone N-acylated with a saturated fatty acid (…

Kategori:
AntigensAntigens, NeoplasmBiological Factors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CERC-301 DB12063
small molecule | CAS: 808732-98-1

Mk 0657 has been used in trials studying the treatment of Major Depressive Disorder.

Kategori:
Receptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Target Protein:
Glutamate receptor ionotropic, NMDA 2B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerdulatinib DB15499
small molecule | CAS: 1198300-79-6

Cerdulatinib is under investigation in clinical trial NCT04021082 (CELTIC-1: A Phase 2B Study of Cerdulatinib in Patients With Relapsed/refractory Peripheral T-cell Lymphoma (PTCL)).

Kategori:
Sulfur Compounds
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase JAK2Tyrosine-protein kinase SYK +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CERE-120 DB05637
biotech | CAS: 1148126-35-5

CERE-120 is an investigational drug consisting of an adeno-associated virus (AAV) that was engineered to carry the human gene for neurturin, a neurotrophic (growth) factor. It was under investigation in clinical trials for the treatment of Parkinson's Disease.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerebrolysin DB16599
biotech | CAS: 12656-61-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBrainCentral Nervous System Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1509916-03-3

Cergutuzumab amunaleukin is under investigation in clinical trial NCT02004106 (A Study to Evaluate Safety, Pharmacokinetics, and Efficacy of RO6895882 in Participants With Advanced and/or Metastatic Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceritinib Approved DB09063
small molecule | CAS: 1032900-25-6

Ceritinib is used for the treatment of adults with anaplastic lymphoma kinase (ALK)-positive metastatic non-small cell lung cancer (NSCLC) following failure (secondary to resistance or intolerance) of prior crizotinib therapy. About 4% of patients with NSCLC …

Kategori:
Anaplastic lymphoma kinase (ALK) inhibitorsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +25
Target Protein:
ALK tyrosine kinase receptor
Waktu ParuhThe terminal half l…
Vol. DistribusiThe apparent volume…
KlirensThe geometric mean …
Genetik -
Cerium oxalate DB13519
small molecule | CAS: 139-42-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAntiemetics and Antinauseants
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerivastatin Approved DB00439
small molecule | CAS: 145599-86-6

On August 8, 2001 the U.S. Food and Drug Administration (FDA) announced that Bayer Pharmaceutical Division voluntarily withdrew Baycol from the U.S. market, due to reports of fatal rhabdomyolysis, a severe adverse reaction from this cholesterol-lowering (lipi…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBCRP/ABCG2 Substrates +34
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh2-3 hours
Vol. Distribusi-
Klirens-
Genetik -
Cerlapirdine DB12229
small molecule | CAS: 925448-93-7

Cerlapirdine has been investigated for the treatment of Alzheimer Disease.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
5-hydroxytryptamine receptor 6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerliponase alfa Approved DB13173
biotech | CAS: 151662-36-1

Cerliponase alfa is a hydrolytic lysosomal N-terminal tripeptidyl peptidase-1 (TPP1).[L51319] On April 27, 2017, cerliponase alfa was first approved by the FDA as the first treatment for neuronal ceroid lipofuscinosis type 2 (CLN2), also known as TPP1 deficie…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsEnzymes +6
Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu ParuhFollowing intravent…
Vol. DistribusiFollowing intravent…
KlirensFollowing intravent…
Genetik -
Certepetide DB18721
biotech | CAS: 2580154-02-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Certolizumab pegol Approved DB08904
biotech | CAS: 428863-50-7

Certolizumab pegol is a pegylated monoclonal antibody against the tumor necrosis factor-alpha (TNF-alpha).[A176585] It is formed with a humanized Fab fragment of 50 kDa, from an IgG 1 isotype, fused to a 40 kDa polyethylene glycol moiety replacing the Fc anti…

Kategori:
Agents reducing cytokine levelsAlcoholsAmino Acids, Peptides, and Proteins +31
Target Protein:
Tumor necrosis factor
Waktu ParuhThe circulatory hal…
Vol. DistribusiCertolizumab pegol …
KlirensThe clearance rate …
Genetik -
Menampilkan 4351–4400 dari 14063
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