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6694

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3751 (56.0%)
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81 (1.2%)
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Halaman 87 / 134
Modakafusp alfa DB16399
biotech

Modakafusp alfa is under investigation in clinical trial NCT03215030 (A Study to Investigate the Safety, Tolerability, Efficacy, Pharmacokinetics, and Immunogenicity of TAK-573 in Participants With Refractory Multiple Myeloma (MM)).

Waktu Paruh-
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Moderna COVID-19 Vaccine Approved DB15654
biotech

The Moderna COVID-19 Vaccine (mRNA-1273) is a novel mRNA-based vaccine encapsulated in a lipid nanoparticle that encodes for a full-length pre-fusion stabilized spike (S) protein of severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2). Coronavirus dis…

Kategori:
Biological ProductsCOVID-19 VaccinesExperimental Unapproved Treatments for COVID-19 +5
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
Modified vaccinia ankara Approved DB15483
biotech

Modified Vaccinia Ankara (MVA) refers to an attenuated strain of the Vaccinia virus. Vaccines using MVA are live and non-replicating, and are produced using Modified Vaccinia Ankara-Bavarian Nordic (MVA-BN).[L42660,L42670]

Kategori:
Anti-Infective AgentsAntiviral AgentsBiological Products +5
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biotech | CAS: 2171576-44-4

Modified vaccinia virus Ankara-85A antigen is under investigation in clinical trial NCT00953927 (A Study of MVA85A in Healthy Infants).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBacterial Vaccines +8
Waktu Paruh-
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Modipafant DB16237
small molecule | CAS: 122957-06-6

Modipafant is under investigation in clinical trial NCT02569827 (Celgosivir or Modipafant as Treatment for Adult Participants With Uncomplicated Dengue Fever in Singapore).

Kategori:
Pyridines
Waktu Paruh-
Vol. Distribusi-
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Modithromycin DB16238
small molecule | CAS: 736992-12-4

Modithromycin is under investigation in clinical trial NCT00270517 (Comparative Study of EDP-420 Versus Another Antibiotic in the Treatment of Community Acquired Pneumonia).

Kategori:
LactonesPolyketides
Waktu Paruh-
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Modufolin DB12676
small molecule | CAS: 31690-11-6

Modufolin is under investigation for the treatment of Osteosarcoma.

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Mogamulizumab Approved DB12498
biotech | CAS: 1159266-37-1

Mogamulizumab is a humanized monoclonal antibody (mAb) directed against CC chemokine receptor 4 (CCR4) for the treatment of Mycosis Fungoides (MF) and Sézary Syndrome (SS), the most common subtypes of cutaneous T-cell lymphoma. Cutaneous T-cell lymphomas occu…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
C-C chemokine receptor type 4
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe central volume …
KlirensClearance is 12 mL/…
Genetik -
Molibresib DB16239
small molecule | CAS: 1260907-17-2

Molibresib is under investigation in clinical trial NCT01943851 (A Dose Escalation Study to Investigate the Safety, Pharmacokinetics (PK), Pharmacodynamics (PD) and Clinical Activity of GSK525762 in Subjects With Relapsed, Refractory Hematologic Malignancies).

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Bromodomain-containing protein 4
Waktu Paruh-
Vol. Distribusi-
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Molindone Approved DB01618
small molecule | CAS: 7416-34-4

An indole derivative effective in schizophrenia and other psychoses and possibly useful in the treatment of the aggressive type of undersocialized conduct disorder. Molindone has much lower affinity for D2 receptors than most antipsychotic agents and has a re…

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (First Generation [Typical]) +18
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2A +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Molnupiravir DB15661
small molecule | CAS: 2349386-89-4

Molnupiravir (EIDD-2801, MK-4482) is the isopropylester prodrug of [N4-hydroxycytidine].[A193014,A193026] With improved oral bioavailability in non-human primates, it is hydrolyzed _in vivo_, and distributes into tissues where it becomes the active 5’-triphos…

Kategori:
AminesAnti-Infective AgentsAntiinfectives for Systemic Use +13
Waktu ParuhThe half life of th…
Vol. Distribusi-
Klirens-
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Monalizumab DB12824
biotech | CAS: 1228763-95-8

Monalizumab has been used in trials studying the treatment of Gynecologic Cancer, Chronic Lymphocytic Leukemia, and Squamous Cell Carcinoma of the Oral Cavity.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Monensin DB11430
small molecule | CAS: 17090-79-8

Monensin is a polyether isolated from _Streptomyces cinnamonensis_ that presents antibiotic properties. It is widely used in ruminant animal feeds.

Kategori:
Acids, AcyclicAnti-Infective AgentsAntiparasitic Agents +21
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Monoctanoin DB06801
small molecule | CAS: 502-54-5

Monoctanoin is used to dissolve cholesterol gallstones.

Kategori:
Acids, AcyclicFatty AcidsLipids +1
Waktu Paruh-
Vol. Distribusi-
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Monomethyl fumarate Approved DB14219
small molecule | CAS: 2756-87-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDicarboxylic AcidsImmunosuppressive Agents
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAntigensAntigens, Bacterial +10
Waktu Paruh-
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Monopotassium phosphate Approved DB09413
small molecule | CAS: 7778-77-0

Monopotassium phosphate, MKP, (also potassium dihydrogenphosphate, KDP, or monobasic potassium phosphate), KH2PO4, is a soluble salt of potassium and the dihydrogen phosphate ion. It is a source of phosphorus and potassium as well as a buffering agent. It ca…

Kategori:
AcidsAcids, NoncarboxylicAnions +15
Waktu ParuhIn healthy children…
Vol. DistribusiPotassium first ent…
KlirensPhosphates are rapi…
Genetik -
Montelukast Approved DB00471
small molecule | CAS: 158966-92-8

Montelukast was first approved for clinical use by the US FDA in 1998 as Merck's brand name Singulair.[L6301] The medication is a member of the leukotriene receptor antagonist (LTRA) category of drugs.[L6301,L6304,L6307,L6310,L6325,L6328,L6331] Although capab…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityAgents to Treat Airway Disease +29
Target Protein:
Cysteinyl leukotriene receptor 1Polyunsaturated fatty acid 5-lipoxygenase
Waktu ParuhStudies have demons…
Vol. DistribusiThe steady-state vo…
KlirensThe plasma clearanc…
Genetik -
Moricizine Approved DB00680
small molecule | CAS: 31883-05-3

An antiarrhythmia agent used primarily for ventricular rhythm disturbances.

Kategori:
Antiarrhythmic agentsAntiarrhythmics, Class IAntiarrhythmics, Class Ic +15
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu Paruh2 hours (range 1.5-…
Vol. Distribusi* 300 L
Klirens-
Genetik -
Morinidazole DB15098
small molecule | CAS: 92478-27-8

Morinidazole is under investigation in clinical trial NCT03380793 (A Trial to Assess the Efficacy and Safety of Morinidazole in Patients With Appendicitis).

Kategori:
ImidazolesNitro Compounds
Waktu Paruh-
Vol. Distribusi-
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Morniflumate DB09285
small molecule | CAS: 65847-85-0

Morniflumate is a non-steroidal anti-inflammatory drug with antipyretic properties. It is the morpholinoethyl ester of niflumic acid [L1496]. In one study, post morniflumate ingestion, physical examination and clinical symptoms of those with bronchitis show…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +14
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Polyunsaturated fatty acid 5-lipoxygenase +2
Waktu Paruh2h [L1498]
Vol. Distribusi-
Klirens45 ml/min [L1498]
Genetik -
Moroctocog alfa Approved DB13999
biotech | CAS: 284036-24-4

Moroctocog alfa, also known as BDDrFVIII (B domain deleted recombinant factor VIII), is a recombinant DNA-based drug with functional characteristics comparable to those of endogenous coagulation Factor VIII, the essential human blood clotting protein that is …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +5
Target Protein:
Coagulation factor XCoagulation factor IXvon Willebrand factor +8
Waktu ParuhMean terminal elimi…
Vol. DistribusiMean steady-state v…
KlirensMean clearance = 4.…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin S
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin S
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin S
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Morrhuic acid DB14087
small molecule

Morrhuic acid is a mixture of unsaturated fatty acids obtained from cod liver oil.

Kategori:
Cardiovascular AgentsCompounds used in a research, industrial, or household settingFatty Acids +5
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Genetik -
biotech

Morus alba root bark is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Mosliciguat DB19425
small molecule | CAS: 2231749-54-3

Mosliciguat is under investigation in clinical trial NCT06635850 (A Phase 2 Study of Mosliciguat in PH-ILD).

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Mosunetuzumab Approved DB15434
biotech | CAS: 1905409-39-3

Mosunetuzumab is a humanized anti-CD20/CD3 bispecific antibody.[L42230] It can recognize and bind two different targets simultaneously, CD20 on cancer B-cells and CD3 on T-cells, allowing it to redirect T-cell cytotoxic activity to cancer cells.[A249320] The …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +13
Target Protein:
B-lymphocyte antigen CD20T-cell surface glycoprotein CD3 epsilon chain
Waktu ParuhMosunetuzumab has a…
Vol. DistribusiThe estimated centr…
KlirensThe mean steady-sta…
Genetik -
Moxetumomab pasudotox Approved DB12688
biotech | CAS: 1020748-57-5

CD22 is a lineage-restricted B-cell antigen that is expressed solely in on B-chronic lymphocytic leukemia, hairy cell leukemia, acute lymphocytic leukemiathe and Burkitt's lymphoma. The predecessor of Moxetumab pasudotox (MxP), named BL22, was first created b…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
B-cell receptor CD22Elongation factor 2
Waktu ParuhMxP presents a shor…
Vol. DistribusiThe mean volume of …
KlirensThe mean systemic c…
Genetik -
Moxidectin Approved DB11431
small molecule | CAS: 113507-06-5

Moxidectin is a potent, broad-spectrum endectocide (antiparasitic that is active against endo- and ecto-parasites) with activity against nematodes, insects, and acari. It was first used in cattle followed by an approved use in general animals. It is a semi-sy…

Kategori:
AgrochemicalsAnthelminticsAnti-Infective Agents +9
Target Protein:
Glutamate-gated chloride channelGABA-A gated chloride channelABC transporters
Waktu ParuhMoxidectin reporter…
Vol. DistribusiMoxidectin presents…
KlirensThe apparent cleara…
Genetik -
Moxifloxacin Approved DB00218
small molecule | CAS: 151096-09-2

Moxifloxacin is a synthetic fluoroquinolone antibiotic agent. Bayer AG developed the drug (initially called BAY 12-8039) and it is marketed worldwide (as the hydrochloride) under the brand name Avelox (in some countries also Avalox) for oral treatment.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +18
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +3
Waktu Paruh11.5-15.6 hours (si…
Vol. Distribusi* 1.7 to 2.7 L/kg
Klirens* 12 +/- 2 L/hr
Genetik -
Moxisylyte Approved DB09205
small molecule | CAS: 54-32-0

Moxisylyte, denominated as thymoxamine in the UK, is a specific and orally active ?1-adrenergic antagonist.[T45] According to the WHO, moxisylyte is approved since 1987[T91] and in the same year, it acquired the denomination of orphan product by the FDA.[L117…

Kategori:
Adrenergic AgentsAdrenergic alpha-AntagonistsAdrenergic Antagonists +17
Target Protein:
Alpha-1D adrenergic receptorAlpha adrenergic receptor
Waktu ParuhThe half-life of mo…
Vol. DistribusiIn preclinical tria…
KlirensIn preclinical tria…
Genetik -
Moxonidine Approved DB09242
small molecule | CAS: 75438-57-2

Moxonidine is a new-generation centrally acting antihypertensive drug approved for the treatment of mild to moderate essential hypertension. It is suggested to be effective in cases where other agents such as thiazides, beta-blockers, ACE inhibitors, and calc…

Kategori:
Adrenergic AgonistsAdrenergic alpha-2 Receptor AgonistsAdrenergic alpha-Agonists +8
Target Protein:
Alpha-2C adrenergic receptorAlpha-2B adrenergic receptorAlpha-2A adrenergic receptor +1
Waktu ParuhPlasma elimination …
Vol. Distribusi1.8±0.4L/kg. [FDA l…
KlirensAdministered twice …
Genetik -
MPI-674 DB05749
small molecule

MPI-674 is an aromatase inhibitor (AI) with a well-established, multi-year chronic safety and tolerability profile. AIs are a class of drugs that reduce the amount of estrogen circulating in the body by binding to and inhibiting the enzyme aromatase, which i…

Target Protein:
Aromatase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MPT0B640 DB16512
small molecule

MPT0B640 was under investigation in clinical trials NCT04526717 for COVID-19 infection and NCT04294875 for locally advanced or metastatic solid malignancies.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
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mRNA-1345 DB18739
biotech

mRNA-1345 is an investigational RSV vaccine.

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
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mRNA-3927 DB17669
biotech

mRNA-3927 is an investigational mRNA therapy that consists of two mRNAs that encode for the alpha and beta subunits of the mitochondrial enzyme propionyl-CoA carboxylase (PCC) encapsulated within a lipid nanoparticle (LNP). Developed by Moderna Inc., it is be…

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MT-401 DB18639
biotech

MT-401 is an allogeneic multi-tumor-associated antigen-specific T-cell therapy.

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Genetik -
biotech

Dendritic Cell (DC) Therapy is a newly emerging and potent form of immune therapy that amplifies the actions of the body's own immune system to help fight cancer, AIDS and other serious conditions. The Dendritic Cell is an immune cell whose role is the recogn…

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Vol. Distribusi-
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biotech

Mucor circinelloides f. circinelloides allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Mucor circinelloides f. lusitanicus allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MultiStem DB15742
biotech

MultiStem is an intravenously-administered, off-the-shelf proprietary product developed which comprises Multipotent Adult Progenitor Cells (MAPCs). Like mesenchymal stem cells, MAPCs are derived from bone-marrow stroma and are non-hematopoietically adherent. …

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Vol. Distribusi-
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Genetik -
biotech

Mumps virus strain B level jeryl lynn live antigen is a live attenuated virus vaccine for subcutenous injection. It is an active immunization against mumps, which is a common childhood disease.

Kategori:
Actively Acquired ImmunityLive Mumps Virus VaccineVaccines
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mupirocin Approved DB00410
small molecule | CAS: 12650-69-0

Mupirocin, formerly termed pseudomonic acid A,[A178531] is a novel antibacterial agent with a unique chemical structure and mode of action apart from other antibiotic agents. Produced by fermentation using the organism _Pseudomonas fluorescens_, mupirocin is …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics for Topical Use +12
Target Protein:
Isoleucine--tRNA ligase
Waktu ParuhIn healthy male vol…
Vol. DistribusiNo information avai…
KlirensNo information avai…
Genetik -
Muraglitazar DB06510
small molecule | CAS: 331741-94-7

Muraglitazar (Bristol-Myers Squibb/Merck) is a new agent under investigation for the treatment of patients with type 2 diabetes. It belongs to a novel class of drugs that target the peroxisome proliferator-activated receptors, both alpha and gamma subtypes. I…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsCytochrome P-450 CYP1A2 Substrates +6
Target Protein:
Peroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Muromonab Approved DB00075
biotech | CAS: 140608-64-6

Murine monoclonal antibody specific to CD3 T-cell lymphocyte antigens. More specifically it is a purified murine (mouse) monoclonal antibody, directed against the CD3 (T3) receptor on the surface of human T-cells (T-lymphocytes) cultured using the murine asci…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
T-cell surface glycoprotein CD3 delta chainT-cell surface glycoprotein CD3 epsilon chainT-cell surface glycoprotein CD3 gamma chain +2
Waktu Paruh0.8 hours (mammalia…
Vol. Distribusi-
Klirens-
Genetik -
Muscimol DB12458
small molecule | CAS: 2763-96-4

Muscimol has been used in trials studying the treatment of Epilepsy and Parkinson's Disease.

Kategori:
Biological FactorsGABA AgentsGABA Agonists +5
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit beta-3Gamma-aminobutyric acid receptor subunit gamma-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MV-NB-02 DB17305
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

MVA-BN-brachyury-TRICOM vaccine is an investigational cancer vaccine. It is composed of recombinant vaccinia viral vector, modified vaccinia Ankara-Bavarian Nordic (MVA-BN), encoding the human transcription factor and tumour-associated antigen (TAA) brachyury…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Menampilkan 4301–4350 dari 6694
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