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14494

Total database: 17430
Struktur (SMILES)
9687 (66.8%)
Target
7525 (51.9%)
Genomik
112 (0.8%)
Referensi
14494 (100.0%)

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Hasil Pencarian (14494)

Halaman 87 / 290
Cinnamyl alcohol Approved DB14186
small molecule | CAS: 4407-36-7

Cinnamyl alcohol is a naturally occurring compound that is found within cinnamon. Due to the low levels found in cinnamon, cinnamyl alcohol is usually supplied as [DB14184] within commercial products. Cinnamyl alcohol has been shown to be a skin sensitizer…

Kategori:
AlcoholsCell-mediated ImmunityDrugs that are Mainly Renally Excreted +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cinnarizine Approved DB00568
small molecule | CAS: 298-57-7

First synthesized by Janssen Pharmaceuticals in 1955, cinnarizine is an anti-histaminic drug mainly used for the control of vestibular disorders and motion sickness. Cinnarizine is a specific calcium channel blocker that primarily works on the central vestibu…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntivertigo Preparations +22
Target Protein:
Histamine H1 receptorVoltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent L-type calcium channel subunit alpha-1D +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cinolazepam DB01594
small molecule | CAS: 75696-02-5

Cinolazepam is a benzodiazepine derivative with anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant activity. It is not approved in Canada or America.

Kategori:
BenzazepinesBenzodiazepine hypnotics and sedativesBenzodiazepines and benzodiazepine derivatives +5
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh9 hours
Vol. Distribusi-
Klirens-
Genetik -
Cinoxacin Approved DB00827
small molecule | CAS: 28657-80-9

Synthetic antimicrobial related to oxolinic acid and nalidixic acid and used in urinary tract infections.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +12
Target Protein:
DNA gyrase subunit ADNA topoisomerase 2-betaDNA topoisomerase 2-alpha +1
Waktu ParuhWhile the mean seru…
Vol. Distribusi-
Klirens-
Genetik -
Cinoxate Approved DB15467
small molecule | CAS: 104-28-9

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicSunscreen Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cinpanemab DB16127
biotech | CAS: 2094516-02-4

Cinpanemab is under investigation in clinical trial NCT03318523 (Evaluating the Efficacy, Safety, Pharmacokinetics, and Pharmacodynamics of BIIB054 in Participants With Parkinson's Disease).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 2218515-90-1

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
biotech | CAS: 372075-36-0

Cintredekin besudotox has been developed as a specific tumor-targeting agent, which is administered by positive-pressure convection-enhanced delivery (CED) directly to brain tissue at risk for residual infiltrating glioblastoma multiforme (GBM) after tumor re…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +6
Target Protein:
Interleukin-13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cipaglucosidase alfa Approved DB16708
biotech | CAS: 2359727-71-0

Cipaglucosidase alfa (ATB200) is a novel recombinant human acid alpha-glucosidase (GAA) investigated for the treatment of patients with Pompe disease, a rare inherited metabolic disorder characterized by a deficiency in GAA.[A232955] Other types of enzyme rep…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +1
Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu ParuhThe mean terminal e…
Vol. DistribusiThe mean volume of …
KlirensCoadministration of…
Genetik -
Cipargamin DB12306
small molecule | CAS: 1193314-23-6

Cipargamin has been used in trials studying the treatment of Malaria, Cure Rate, and Plasmodium Falciparum Malaria.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Adenosine receptor A3Voltage-gated inwardly rectifying potassium channel KCNH2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cipatinib DB16752
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ciprocinonide Approved DB18738
small molecule | CAS: 58524-83-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ciprofibrate Approved DB09064
small molecule | CAS: 52214-84-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityBenzene Derivatives +14
Target Protein:
Peroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ciprofloxacin Approved DB00537
small molecule | CAS: 85721-33-1

Ciprofloxacin is a second generation fluoroquinolone that has spawned many derivative antibiotics.[A178870] It is formulated for oral, intravenous, intratympanic, ophthalmic, and otic administration for a number of bacterial infections.[L6469,L6472,L6475,L647…

Kategori:
4-QuinolonesAgents Causing Muscle ToxicityAnti-Bacterial Agents +38
Target Protein:
DNA topoisomerase 4 subunit ADNA gyrase subunit BThymidylate synthase +10
Waktu ParuhThe average half li…
Vol. DistribusiCirpofloxacin follw…
KlirensThe average renal c…
Genetik -
Ciraparantag DB15199
small molecule | CAS: 1438492-26-2

Ciraparantag is under investigation in clinical trial NCT01826266 (Effects of a Double-Blind, Single Dose of PER977 Administered Alone, and Following a Single Dose of Edoxaban).

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cirazoline DB09202
small molecule | CAS: 59939-16-1

Cirazoline acts on a number of ? adrenergic receptors. It is an agonist of ?1A, partial agonist of ?1B and ?1D, and a nonselective antagonist of ?2. It is believed that this combination of properties could make cirazoline an effective vasoconstricting agent. …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +8
Target Protein:
Alpha-1A adrenergic receptorAlpha-2C adrenergic receptorAlpha-1B adrenergic receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cirtuvivint DB17269
small molecule | CAS: 2143917-62-6

Cirtuvivint is a first-in-class CDC-like kinase (CLK) inhibitor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Phenylethanolamine N-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Lanosterol 14-alpha demethylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 191595-91-2

Deskripsi belum tersedia.

Kategori:
Bile Acids and SaltsCholanesFused-Ring Compounds +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 151057-28-2

Deskripsi belum tersedia.

Target Protein:
Antigen-presenting glycoprotein CD1d
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 506-17-2

Deskripsi belum tersedia.

Kategori:
Fatty AcidsFatty Acids, MonounsaturatedFatty Acids, Unsaturated +1
Target Protein:
Peroxisome proliferator-activated receptor delta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
E3 ubiquitin-protein ligase Mdm2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
E3 ubiquitin-protein ligase Mdm2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cisapride Approved DB00604
small molecule | CAS: 81098-60-4

In many countries (including Canada) cisapride has been either withdrawn or has had its indications limited due to reports about long QT syndrome due to cisapride, which predisposes to arrhythmias. The FDA issued a warning letter regarding this risk to health…

Kategori:
Acids, CarbocyclicAlimentary Tract and MetabolismAmides +36
Target Protein:
5-hydroxytryptamine receptor 45-hydroxytryptamine receptor 3A5-hydroxytryptamine receptor 2A +1
Waktu Paruh6-12 hours
Vol. Distribusi-
Klirens-
Genetik -
Cisatracurium Approved DB00565
small molecule | CAS: 96946-41-7

Cisatracurium is a non-depolarising neuromuscular blocking agent of the benzylisoquinolinium class, available in its salt form, cisatracurium besylate.[A243416,A253592] Cisatracurium has an intermediate duration of action and is one of the most commonly used …

Kategori:
Anticholinergic AgentsBenzylisoquinolinesCentral Nervous System Depressants +11
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Neuronal Acetylcholine (nACh) Receptor SubunitsAcetylcholine receptor subunit alpha +1
Waktu ParuhCisatracurium has a…
Vol. DistribusiCisatracurium has a…
KlirensCisatracurium has a…
Genetik -
Cisplatin Approved DB00515
small molecule | CAS: 15663-27-1

Cisplatin, cisplatinum or cis-diamminedichloroplatinum(II) (CDDP) is a platinum-based chemotherapy drug used to treat various types of cancers, including sarcomas, some carcinomas (e.g. small cell lung cancer, and ovarian cancer), lymphomas and germ cell tumo…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +24
Target Protein:
DNADNA-3-methyladenine glycosylaseAlpha-2-macroglobulin +2
Gen Terkait:
GSTM1 LRP2 GSTP1 +1
Waktu ParuhCisplatin decays mo…
Vol. DistribusiVolume of distribut…
Klirens* 15-16 L/h/m^2 [to…
Genetik 4 Varian
Citalopram Approved DB00215
small molecule | CAS: 59729-33-8

Citalopram is an antidepressant belonging to the class of selective _serotonin-reuptake inhibitors_ (SSRIs) widely used to treat the symptoms of depression. It is a racemic bicyclic phthalate derivate and is the only compound with a tertiary amine and 2 nitro…

Kategori:
AminesAntidepressive AgentsAntidepressive Agents Indicated for Depression +41
Target Protein:
Sodium-dependent serotonin transporterHistamine H1 receptor
Gen Terkait:
ABCB1 HTR2A GRIK4 +3
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe volume of distr…
KlirensThe systemic cleara…
Genetik 6 Varian
Citarinostat DB15449
small molecule | CAS: 1316215-12-9

Citarinostat is under investigation in clinical trial NCT02886065 (A Study of PVX-410, a Cancer Vaccine, and Citarinostat +/- Lenalidomide for Smoldering MM).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHistone Deacetylase Inhibitors
Target Protein:
Histone deacetylase 6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 945228-49-9

VB6-845 is a humanized antibody fragment targeting EpCAM fused with the deimmunized form of the cytotoxin Bouganin and is designed for systemic use against metastatic cancer. VB6-845 has demonstrated effective cancer cell killing properties in pre-clinical te…

Target Protein:
Epithelial cell adhesion molecule
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Citicoline Approved DB12153
small molecule | CAS: 987-78-0

Citicoline is a donor of choline in biosynthesis of choline-containing phosphoglycerides. It has been investigated for the treatment, supportive care, and diagnosis of Mania, Stroke, Hypomania, Cocaine Abuse, and Bipolar Disorder, among others.

Kategori:
AminesCentral Nervous System AgentsCytidine Diphosphate +13
Target Protein:
LicC protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Citiolone DB13442
small molecule | CAS: 1195-16-0

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismBile and Liver TherapyExpectorants +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Citraconic acid DB04734
small molecule | CAS: 498-23-7

Citraconic acid is one of the isomeric dicarboxylic acids produced by the distillation of citric acid, or as metabolites by microorganisms, cis-CH3-C(CO2H)=CHCO2H; the trans-isomer is mesaconic acid.

Kategori:
Acids, AcyclicDermatologicalsDicarboxylic Acids
Target Protein:
Fumarate reductase flavoprotein subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Citric acid Approved DB04272
small molecule | CAS: 77-92-9

A key intermediate in metabolism. It is an acid compound found in citrus fruits. The salts of citric acid (citrates) can be used as anticoagulants due to their calcium-chelating ability. Citric acid is one of the active ingredients in Phexxi, a non-hormona…

Kategori:
Acid PreparationsAcidifying ActivityAcids, Acyclic +16
Target Protein:
Metallo-beta-lactamase type 2Lanosterol 14-alpha demethylaseTransient receptor potential cation channel subfamily V member 4 +49
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Citronella oil DB16601
biotech | CAS: 8000-29-1

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesLipids +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Citrulline DB00155
small molecule | CAS: 372-75-8

Citrulline is an amino acid. It is made from ornithine and carbamoyl phosphate in one of the central reactions in the urea cycle. It is also produced from arginine as a by-product of the reaction catalyzed by NOS family. Its name is derived from citrullus, th…

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Diamino +8
Target Protein:
Nitric oxide synthase 3Argininosuccinate synthasePutative hydrolase DDAH2 +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Citrus bioflavonoids Approved DB14586
small molecule | CAS: 12002-36-7

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Citrus junos fruit is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Citrus sinensis pollen Approved DB10743
biotech

Citrus sinensis pollen is the pollen of the Citrus sinensis plant. Citrus sinensis pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cixutumumab DB12250
biotech | CAS: 947687-12-9

Cixutumumab has been used in trials studying the treatment of Lung Cancer, Malignant Neoplasm, Leukemia, Mast-Cell, Non-Small-Cell Lung Carcinoma, and Adenocarcinoma of the Prostate. Cixutumumab is a highly specific recombinant human monoclonal antibody wi…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Insulin-like growth factor 1 receptor
Waktu Paruh148 h (3 mg/kg dose…
Vol. Distribusi-
Klirens-
Genetik -
CK0802 DB15866
biotech

CK0802 is an off-the-shelf product composed of allogeneic umbilical cord blood derived regulatory T-cells (T-Reg cells), which can be used intravenously and without HLA matching.[L16358] On the surface of these T-Reg cells, T-cell lung homing markers are expr…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
CKD-504 DB18235
small molecule

CKD-504 is a novel, selective histone deacetylase 6 inhibitor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CL-315555 DB18757
small molecule | CAS: 133513-12-9

CL-315555 is the C isomer of [Verteporfin].

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CL-315585 DB18758
small molecule | CAS: 142878-05-5

CL-315585 is the D isomer of [Verteporfin].

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cladosporium cladosporioides Approved DB10431
biotech

Cladosporium cladosporioides is a fungus which can provoke allergic reactions. Cladosporium cladosporioides extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cladosporium herbarum Approved DB10865
biotech

Cladosporium herbarum is a fungus which can provoke allergic reactions. Cladosporium herbarum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cladosporium sphaerospermum Approved DB10432
biotech

Cladosporium sphaerospermum is a fungus which can provoke allergic reactions. Cladosporium sphaerospermum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cladribine Approved DB00242
small molecule | CAS: 4291-63-8

Cladribine is a purine analogue or a chlorinated derivative of adenine [A263733] that causes apoptosis of B and T lymphocytes.[A350] Cladribine was first approved in the United States in 1993 [A263713] initially as a treatment for a number of hematological ma…

Kategori:
2-ChloroadenosineAgents Causing Muscle ToxicityAntimetabolites +19
Target Protein:
Ribonucleoside-diphosphate reductase large subunitAdenosine deaminaseRibonucleoside-diphosphate reductase subunit M2 +9
Waktu ParuhCladribine plasma c…
Vol. DistribusiIn general, the app…
KlirensIn patients with he…
Genetik -
Clarithromycin Approved DB01211
small molecule | CAS: 81103-11-9

Clarithromycin, a semisynthetic macrolide antibiotic derived from erythromycin, inhibits bacterial protein synthesis by binding to the bacterial 50S ribosomal subunit. Binding inhibits peptidyl transferase activity and interferes with amino acid translocation…

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +31
Target Protein:
50S ribosomal protein L10Voltage-gated inwardly rectifying potassium channel KCNH2Solute carrier organic anion transporter family member 1B1 +1
Waktu Paruh3-4 hours
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4301–4350 dari 14494
Sebelumnya Halaman 87 / 290 Berikutnya