Hasil Filter

13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (13591)

Halaman 85 / 272
Cerdulatinib DB15499
small molecule | CAS: 1198300-79-6

Cerdulatinib is under investigation in clinical trial NCT04021082 (CELTIC-1: A Phase 2B Study of Cerdulatinib in Patients With Relapsed/refractory Peripheral T-cell Lymphoma (PTCL)).

Kategori:
Sulfur Compounds
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase JAK2Tyrosine-protein kinase SYK +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CERE-120 DB05637
biotech | CAS: 1148126-35-5

CERE-120 is an investigational drug consisting of an adeno-associated virus (AAV) that was engineered to carry the human gene for neurturin, a neurotrophic (growth) factor. It was under investigation in clinical trials for the treatment of Parkinson's Disease.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1509916-03-3

Cergutuzumab amunaleukin is under investigation in clinical trial NCT02004106 (A Study to Evaluate Safety, Pharmacokinetics, and Efficacy of RO6895882 in Participants With Advanced and/or Metastatic Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceritinib Approved DB09063
small molecule | CAS: 1032900-25-6

Ceritinib is used for the treatment of adults with anaplastic lymphoma kinase (ALK)-positive metastatic non-small cell lung cancer (NSCLC) following failure (secondary to resistance or intolerance) of prior crizotinib therapy. About 4% of patients with NSCLC …

Kategori:
Anaplastic lymphoma kinase (ALK) inhibitorsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +25
Target Protein:
ALK tyrosine kinase receptor
Waktu ParuhThe terminal half l…
Vol. DistribusiThe apparent volume…
KlirensThe geometric mean …
Genetik -
Cerium dioxide DB18493
small molecule | CAS: 1306-38-3

Deskripsi belum tersedia.

Kategori:
ElementsLanthanoid Series ElementsMetals +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerium oxalate DB13519
small molecule | CAS: 139-42-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAntiemetics and Antinauseants
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerivastatin Approved DB00439
small molecule | CAS: 145599-86-6

On August 8, 2001 the U.S. Food and Drug Administration (FDA) announced that Bayer Pharmaceutical Division voluntarily withdrew Baycol from the U.S. market, due to reports of fatal rhabdomyolysis, a severe adverse reaction from this cholesterol-lowering (lipi…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBCRP/ABCG2 Substrates +34
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh2-3 hours
Vol. Distribusi-
Klirens-
Genetik -
Cerlapirdine DB12229
small molecule | CAS: 925448-93-7

Cerlapirdine has been investigated for the treatment of Alzheimer Disease.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
5-hydroxytryptamine receptor 6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerliponase alfa Approved DB13173
biotech | CAS: 151662-36-1

Cerliponase alfa is a hydrolytic lysosomal N-terminal tripeptidyl peptidase-1 (TPP1).[L51319] On April 27, 2017, cerliponase alfa was first approved by the FDA as the first treatment for neuronal ceroid lipofuscinosis type 2 (CLN2), also known as TPP1 deficie…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsEnzymes +6
Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu ParuhFollowing intravent…
Vol. DistribusiFollowing intravent…
KlirensFollowing intravent…
Genetik -
Certepetide DB18721
biotech | CAS: 2580154-02-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Certolizumab pegol Approved DB08904
biotech | CAS: 428863-50-7

Certolizumab pegol is a pegylated monoclonal antibody against the tumor necrosis factor-alpha (TNF-alpha).[A176585] It is formed with a humanized Fab fragment of 50 kDa, from an IgG 1 isotype, fused to a 40 kDa polyethylene glycol moiety replacing the Fc anti…

Kategori:
Agents reducing cytokine levelsAlcoholsAmino Acids, Peptides, and Proteins +31
Target Protein:
Tumor necrosis factor
Waktu ParuhThe circulatory hal…
Vol. DistribusiCertolizumab pegol …
KlirensThe clearance rate …
Genetik -
Cerulenin DB01034
small molecule | CAS: 17397-89-6

Cerulenin is an antifungal agent whose activity interferes with or otherwise acts to prevent the formation of fatty acids and sterols. In fatty acid synthesis, reported to bind in equimolar ratio to b-keto-acyl-ACP synthase. In sterol synthesis, inhibits HMG-…

Kategori:
AmidesAnti-Infective AgentsAntifungal Agents +3
Target Protein:
3-oxoacyl-[acyl-carrier-protein] synthase 13-oxoacyl-[acyl-carrier-protein] synthase 23-oxoacyl-[acyl-carrier-protein] synthase 3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceruletide Approved DB00403
small molecule | CAS: 17650-98-5

Caerulein is a specific decapeptide similar in action and composition to the natural gastrointestinal peptide hormone cholecystokinin. It exerts stimulatory effects on the gastric, biliary, and pancreatic secretion, as well as on certain smooth muscles.

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsOligopeptides +2
Target Protein:
Cholecystokinin receptor type AGastrin/cholecystokinin type B receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cesium DB15392
small molecule | CAS: 7440-46-2

Cesium is under investigation in clinical trial NCT02794675 (Intraoperative Placement of Cesium-131 Permanent Interstitial Brachytherapy in Head and Neck Cancer).

Kategori:
ElementsMetalsMetals, Alkali +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cesium Cs-131 DB19250
small molecule | CAS: 14914-76-2

Cesium Cs-131 is under investigation in clinical trial NCT04340258 (Trial Combining Pembrolizumab and Cesium 131 Brachytherapy With Salvage Surgery in HNSCC).

Kategori:
Cesium IsotopesElementsIsotopes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetalkonium Approved DB11583
small molecule | CAS: 10328-34-4

Cetalkonium is a C16 alkyl benzalkonium chloride derivative with an amphipathic property which allows it to be used in different types of formulations.[A27143] It is a quaternary ammonium salt that acts as an antiseptic against a variety of bacteria and fungi…

Kategori:
AlcoholsAminesAmmonium Compounds +7
Waktu ParuhAs cetalkonium is n…
Vol. DistribusiAs cetalkonium is n…
KlirensAs cetalkonium is n…
Genetik -
Cethromycin DB06419
small molecule | CAS: 205110-48-1

Cethromycin is a 3-keto (ketolide) derivative of erythromycin A with an 11,12-carbamate group and an O-6-linked aromatic ring system.[A203369] Cethromycin represents a joint development effort by Abbott Laboratories, Taisho Pharmaceuticals, and Advanced Life …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCytochrome P-450 CYP3A Inhibitors +15
Target Protein:
23S ribosomal RNA
Waktu ParuhCethromycin given i…
Vol. DistribusiCethromycin given i…
KlirensCethromycin clearan…
Genetik -
Cetiedil DB13753
small molecule | CAS: 14176-10-4

Deskripsi belum tersedia.

Kategori:
Antisickling AgentsCardiovascular AgentsHematologic Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetirizine Approved DB00341
small molecule | CAS: 83881-51-0

Cetirizine, also commonly known as _Zyrtec_, is an orally active second-generation histamine H1 antagonist proven effective in the treatment of various allergic symptoms, such as sneezing, coughing, nasal congestion, hives, and other symptoms [A175051], [A175…

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseCentral Nervous System Depressants +14
Target Protein:
Histamine H1 receptor
Waktu ParuhPlasma elimination …
Vol. DistribusiApparent volume of …
KlirensApparent total body…
Genetik -
Cetrelimab DB15421
biotech | CAS: 2050478-92-5

Cetrelimab is under investigation in clinical trial NCT03547037 (A Study to Evaluate the Safety, Pharmacokinetics, Pharmacodynamics, and Immunogenicity of JNJ-63723283, an Anti-Programmed Cell Death (PD)-1 Monoclonal Antibody, as Monotherapy or in Combination…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetuximab Approved DB00002
biotech | CAS: 205923-56-4

Cetuximab is a recombinant chimeric human/mouse IgG1 monoclonal antibody that competitively binds to epidermal growth factor receptor (EGFR) and competitively inhibits the binding of epidermal growth factor (EGF).[A227973] EGFR is a member of the ErbB family …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Epidermal growth factor receptorLow affinity immunoglobulin gamma Fc region receptor III-BComplement C1q subcomponent subunit A +5
Gen Terkait:
FCGR2A FCGR3A
Waktu ParuhAfter administratio…
Vol. DistribusiThe volume of the d…
KlirensIn patients with re…
Genetik 2 Varian
biotech | CAS: 2166339-33-7

Cetuximab sarotalocan is under investigation in clinical trial NCT03769506 (ASP-1929 Photoimmunotherapy (PIT) Study in Recurrent Head/Neck Cancer for Patients Who Have Failed at Least Two Lines of Therapy) for the treatment of Recurrent Head/Neck Cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetyl alcohol Approved DB09494
small molecule | CAS: 36653-82-4

Cetyl alcohol, also known as 1-hexadecanol or n-hexadecyl alcohol, is a 16-C fatty alcohol with the chemical formula CH3(CH2)15OH. It can be produced from the reduction of palmitic acid. Cetyl alcohol is present in a waxy white powder or flake form at room te…

Kategori:
AlcoholsDrugs that are Mainly Renally ExcretedLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 59130-69-7

Cetyl ethylhexanoate is an ester of cetyl alcohol and 2-ethylhexanoic acid. It is present in cosmetic products as a skin conditioning agent and emollient.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetyl oleate DB19454
small molecule | CAS: 22393-86-8

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetyl palmitate DB15782
small molecule | CAS: 540-10-3

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipidsPalmitic Acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 22393-83-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetylpyridinium Approved DB11073
small molecule | CAS: 7773-52-6

Cetylpyridinium is a quaternary ammonium with broad-spectrum antiseptic properties. Its salt form, cetylpyridinium chloride, is typically found as an active ingredient in mouthwashes, toothpastes, lozenges, throat sprays, breath sprays, and nasal sprays. In t…

Kategori:
Alimentary Tract and MetabolismAnti-Infective AgentsAnti-Infective Agents, Local +19
Waktu ParuhNo readily availabl…
Vol. DistribusiNo readily availabl…
KlirensNo readily availabl…
Genetik -
Cevidoplenib DB18725
small molecule | CAS: 1703788-21-9

Deskripsi belum tersedia.

Kategori:
Oxazoles
Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cevimeline Approved DB00185
small molecule | CAS: 107233-08-9

Cevimeline is a parasympathomimetic agent that act as an agonist at the muscarinic acetylcholine receptors M1 and M3. It is indicated by the Food and Drug Administration for the treatment of dry mouth associated with Sjögren's syndrome.

Kategori:
Autonomic AgentsCholinergic AgentsCholinergic Agonists +12
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1
Waktu Paruh5 ± 1 hours
Vol. Distribusi* 6 L/kg
Klirens-
Genetik -
Cevipabulin DB12533
small molecule | CAS: 849550-05-6

Cevipabulin has been used in trials studying the treatment and educational/counseling/training of Tumors and Neoplasms.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cevostamab DB18374
biotech | CAS: 2249888-53-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CFG-920 DB19193
small molecule | CAS: 1260006-20-9

CFG-920 is under investigation in clinical trial NCT04060394 (Dose-escalation and Efficacy Study of Lae001/prednisone Plus Afuresertib Patients With M-crpc).

Target Protein:
Steroid 17-alpha-hydroxylase/17,20 lyase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CFT-8634 DB18443
small molecule | CAS: 2704617-96-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CG-200745 DB12259
small molecule | CAS: 936221-33-9

Cg200745 has been used in trials studying the treatment of Solid Tumour.

Kategori:
AminesAntineoplastic AgentsHistone Deacetylase Inhibitors +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CG-400549 DB12347
small molecule | CAS: 934628-27-0

CG400549 has been used in trials studying the treatment of Skin Infection.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CGI-1842 DB12744
small molecule | CAS: 900573-88-8

JI-101 has been used in trials studying the treatment of Cancer, Colon Cancer, Neuroendocrine, Ovarian Cancer, and Advanced Solid Tumors.

Kategori:
AmidesBenzene DerivativesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Receptor tyrosine-protein kinase erbB-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CGP 4832 DB04220
small molecule | CAS: 113303-81-4

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingLactams, Macrocyclic
Target Protein:
Ferrichrome-iron receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CGS-27023 DB07556
small molecule | CAS: 161314-70-1

Deskripsi belum tersedia.

Kategori:
AmidesAminesEnzyme Inhibitors +8
Target Protein:
Neutrophil collagenaseA disintegrin and metalloproteinase with thrombospondin motifs 472 kDa type IV collagenase +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CGX-1321 DB17491
small molecule

CGX-1321 is a porcupine inhibitor that affects Wnt production and can block Wnt downstream signaling.[A257038]

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CH-5132799 DB13051
small molecule | CAS: 1007207-67-1

CH5132799 has been used in trials studying the treatment of Solid Tumors.

Kategori:
AmidesClass I Phosphatidylinositol 3-Kinases, antagonists & inhibitorsSulfones +1
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chaetomium globosum Approved DB10430
biotech

Chaetomium globosum is a fungus which can provoke allergic reactions. Chaetomium globosum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Chamaecyparis obtusa wood oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Chamaemelum nobile flower is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAsteraceaeBiological Products +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chamazulene DB15931
small molecule | CAS: 529-05-5

Deskripsi belum tersedia.

Kategori:
CycloheptanesCycloparaffins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chamomile Approved DB14357
biotech

Chamomile is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAsteraceaeBiological Products +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chelerythrine DB17024
small molecule | CAS: 34316-15-9

A benzophenanthridine alkaloid evaluated as a kinase-inhibitor.[A252982]

Kategori:
AlkaloidsAnti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
P2X purinoceptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chenodeoxycholic acid Approved DB06777
small molecule | CAS: 474-25-9

Chenodeoxycholic acid (or Chenodiol) is an epimer of ursodeoxycholic acid (DB01586). Chenodeoxycholic acid is a bile acid naturally found in the body. It works by dissolving the cholesterol that makes gallstones and inhibiting production of cholesterol in the…

Kategori:
Alimentary Tract and MetabolismBile Acid PreparationsBile acids and derivatives +12
Target Protein:
Bile acid receptorNuclear receptor subfamily 1 group I member 2G-protein coupled bile acid receptor 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chenopodium album pollen Approved DB10368
biotech

Chenopodium album pollen is the pollen of the Chenopodium album plant. Chenopodium album pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4201–4250 dari 13591
Sebelumnya Halaman 85 / 272 Berikutnya