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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Distribusi Wujud Zat

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Hasil Pencarian (12560)

Halaman 84 / 252
CRA_1802 DB02875
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CRA_23653 DB04246
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CRA_8696 DB03159
small molecule

Deskripsi belum tersedia.

Target Protein:
ProthrombinUrokinase-type plasminogen activatorSerine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CRA_9076 DB04215
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CRA_9678 DB04563
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CRA_9785 DB03595
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CRD5 DB05587
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Creatine Approved DB00148
small molecule | CAS: 57-00-1

An amino acid derivative that occurs in vertebrate tissues and in urine. In muscle tissue, creatine generally occurs as phosphocreatine. Creatine is excreted as creatinine in the urine.

Kategori:
AmidinesAmino AcidsAmino Acids, Peptides, and Proteins +3
Target Protein:
Creatine kinase M-typeCreatine kinase U-type, mitochondrialCreatine kinase B-type +3
Waktu Paruh3 hours
Vol. Distribusi-
Klirens-
Genetik -
Creatinine DB11846
small molecule | CAS: 60-27-5

Creatinine has been used in trials studying the treatment of Amyotrophic Lateral Sclerosis.

Kategori:
Imidazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Crefmirlimab DB17577
biotech | CAS: 2611099-93-3

Crefmirlimab is an anti-human CD8 probe targeting the CD8 antigen, for the diagnosis of various cancers.

Waktu Paruh-
Vol. Distribusi-
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Crenezumab DB11959
biotech | CAS: 1095207-05-8

Crenezumab has been used in trials studying the treatment of Alzheimer's Disease.

Kategori:
Alzheimer Disease, drug therapyAmino Acids, Peptides, and ProteinsAntibodies +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Crinecerfont DB18518
small molecule | CAS: 752253-39-7

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Target Protein:
Corticotropin-releasing factor receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Crisaborole Approved DB05219
small molecule | CAS: 906673-24-3

Crisaborole is a novel oxaborole approved by FDA on December 14, 2016 as Eucrisa, a topical treatment of for mild to moderate atopic dermatitis. This non-steroidal agent is efficacious in improving disease severity, reducing the risk of infection and reduci…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAnti-Inflammatory AgentsCytochrome P-450 CYP2B6 Inhibitors +9
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4B3',5'-cyclic-AMP phosphodiesterase 4C +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Crisdesalazine DB18405
small molecule | CAS: 927685-43-6

Deskripsi belum tersedia.

Kategori:
Anti-Inflammatory AgentsAnti-Inflammatory Agents, Non-SteroidalBenzene Derivatives +3
Target Protein:
Prostaglandin E synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Crisugabalin DB19300
small molecule | CAS: 2209104-84-5

Crisugabalin is under investigation in clinical trial NCT06490484 (Efficacy and Safety of HSK16149 Capsule in Chinese Patients With Diabetic Peripheral Neuropathic Pain Who Had an Inadequate Response to Pregabalin).

Waktu Paruh-
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Crizanlizumab Approved DB15271
biotech | CAS: 1690318-25-2

Crizanlizumab is a humanized IgG2 monoclonal antibody used to reduce the frequency of vaso-occlusive crises in patients with sickle cell disease.[L10097] Sickle cell disease is a genetically inherited condition prevalent in the Middle East, Africa, and certai…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
P-selectin
Waktu ParuhGiven a 5mg/kg dose…
Vol. DistribusiThe volume of distr…
KlirensGiven a 5mg/kg dose…
Genetik -
Crizotinib Approved DB08865
small molecule | CAS: 877399-52-5

Crizotinib is a tyrosine kinase receptor inhibitor used for the treatment of anaplastic lymphoma kinase (ALK) or ROS1-positive non-small cell lung cancer (NSCLC) tumors, as well as ALK-positive anaplastic large cell lymphoma (ALCL) and inflammatory myofibrobl…

Kategori:
AminopyridinesAnaplastic lymphoma kinase (ALK) inhibitorsAntineoplastic Agents +32
Target Protein:
ALK tyrosine kinase receptorHepatocyte growth factor receptorProto-oncogene tyrosine-protein kinase ROS +1
Waktu ParuhFollowing single do…
Vol. DistribusiFollowing a single …
KlirensAt steady-state (25…
Genetik -
Crocin DB11874
small molecule | CAS: 42553-65-1

Crocin has been investigated for the treatment of Hyperglycemia, Metabolic Syndrome, Hypertriglyceridemia, and Hypercholesterolemia.

Kategori:
AlkenesBiological FactorsCondiments +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Crofelemer Approved DB04941
small molecule | CAS: 148465-45-6

Crofelemer, previously known as the investigational drug SP-303, is a novel proanthocyanidin purified from the bark latex of the Amazonian Croton tree <i>Croton lechleri</i>. It is marketed under the brand name Fulyzaq and indicated for the symptomatic treatm…

Kategori:
Alimentary Tract and MetabolismAntidiarrhealsAntidiarrheals, Intestinal Antiinflammatory/antiinfective Agents +11
Target Protein:
Anoctamin-1Cystic fibrosis transmembrane conductance regulator
Waktu ParuhSince crofelemer is…
Vol. DistribusiSince crofelemer is…
KlirensSince crofelemer is…
Genetik -
Crolibulin DB12925
small molecule | CAS: 1000852-17-4

Crolibulin has been used in trials studying the treatment of Solid Tumor and Anaplastic Thyroid Cancer.

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Waktu Paruh-
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Cromoglicic acid Approved DB01003
small molecule | CAS: 16110-51-3

A chromone complex that acts by inhibiting the release of chemical mediators from sensitized mast cells. It is used in the prophylactic treatment of both allergic and exercise-induced asthma, but does not affect an established asthmatic attack.

Kategori:
Adrenergics, InhalantsAgents for Dermatitis, Excluding CorticosteroidsAlimentary Tract and Metabolism +24
Target Protein:
Heat shock protein HSP 90-alphaProtein S100-P
Waktu Paruh1.3 hours
Vol. Distribusi-
Klirens-
Genetik -
Cronidipine DB09233
small molecule | CAS: 113759-50-5

Cronidipine is a calcium channel blocker.

Waktu Paruh-
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Genetik -
biotech

Each year it is estimated there are 45,000 snakebites in the US and 300,000 to 400,000 bites worldwide. About 8000 of these snakebites involve venomous snake species. The majority of people bitten are males and about 50% occur in the age group of 18 to 28 [F1…

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Target Protein:
Group 10 secretory phospholipase A2
Waktu Paruh12 to 23 hours [FDA…
Vol. Distribusi-
KlirensThis product was sh…
Genetik -
Crotalus atrox antivenin Approved DB13892
biotech

Each year it is estimated there are 45,000 snakebites in the US and 300,000 to 400,000 bites worldwide. About 8000 of these snakebites involve venomous snake species. The majority of people bitten are males and about 50% occur in the age group of 18 to 28 [F1…

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Waktu Paruh12-23 hours [F113]
Vol. Distribusi-
Klirens-
Genetik -
biotech

Crotalus scutulatus antivenin is derived and purified immunoglobulin fragments obtained from other domestic animals such as sheep previously immunized with Crotalus scutulatus (also known as the _Mojave rattlesnake_ [L2856]). The final purified antivenin …

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Waktu ParuhApproximately 15 ho…
Vol. Distribusi0.3 L/kg [FDA label]
Klirens32 mL/min (approxim…
Genetik -
Crotamiton Approved DB00265
small molecule | CAS: 483-63-6

Crotamiton is a scabicidal and antipruritic agent available as a cream or lotion for topical use only. It is a colorless to slightly yellowish oil, having a faint amine-like odor. It is miscible with alcohol and with methanol.

Kategori:
AgrochemicalsAminesAniline Compounds +6
Target Protein:
Transient receptor potential cation channel subfamily V member 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Crotedumab DB12815
biotech | CAS: 1452387-69-7

Crotedumab has been used in trials studying the treatment of Diabetes Mellitus, Type 2.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Crovalimab Approved DB16128
biotech | CAS: 1917321-26-6

Crovalimab is a humanized monoclonal antibody and complement C5 inhibitor.[L50908] It consists of two heavy chains (451 amino acid residues each) and two light chains (217 amino acid residues each).[L50908] First developed by Chugai Pharmaceutical, in collabo…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic and Immunomodulating Agents +7
Target Protein:
Complement C5
Waktu ParuhThe mean estimated …
Vol. DistribusiThe mean central an…
KlirensIn PNH treatment-na…
Genetik -
Crozbaciclib DB18081
small molecule | CAS: 2099128-41-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CRS-3123 DB12262
small molecule | CAS: 1013915-71-3

CRS3123 has been used in trials studying the treatment of Clostridial Infection and Clostridium Difficile Colitis.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CRx-119 DB05688
small molecule

CRx-119 is a novel synergistic combination drug candidate discovered using the CombinatoRx combination High Throughput Screening (cHTS(TM)) technology with potential therapeutic use in a broad range of immuno-inflammatory conditions. CRx-119 is a combination …

Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CRx-139 DB05744
small molecule

CRx-139 is an oral synergistic combination drug candidates with novel mechanisms of action targeting multiple biological pathways simultaneously. It is a dissociated steroid designed to enhance the immuno-modulatory activity of a low-dose glucocorticoid stero…

Target Protein:
Tumor necrosis factorInterleukin-6C-reactive protein +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CRx-401 DB05775
small molecule

CRx-401 is a novel insulin sensitizer designed to provide anti-diabetic activity without promoting weight gain. It consists of a low dose of the analgesic diflunisal in conjunction with a modified-release therapeutic dose of bezafibrate, an anti-cholesterol a…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Cry5B DB17783
biotech

Cry5B is a pore-forming crystal protein produced by and derived from the soil bacterium _Bacillus thuringiensis_. With demonstrated anthelmintic properties, it has been investigated in the treatment of parasitic intestinal infections.[A259372, A259377]

Waktu Paruh-
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Genetik -
biotech

Vesta Therapeutics is a privately held company developing cell therapeutics for liver repair and regeneration. The Company's technology is centered on the isolation, expansion, and cryopreservation of liver cells (human hepatocytes) obtained from organ donor …

Waktu Paruh-
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Genetik -
Cryptenamine Approved DB00785
small molecule | CAS: 1356-18-9

Cryptenamine is a mixture of closely related hypotensive alkaloids from Veratrum album (Liliaceae). It has been used in the treatment of hypertension but has largely been replaced by drugs with fewer adverse effects. Cryptenamine has a marked and re-producibl…

Kategori:
AlkaloidsAntihypertensive AgentsCardiovascular Agents +3
Target Protein:
Muscarinic acetylcholine receptor M2Beta adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
small molecule | CAS: 35825-57-1

Deskripsi belum tersedia.

Kategori:
Drugs, Chinese HerbalPlant Extracts
Waktu Paruh-
Vol. Distribusi-
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Cryptoxanthin DB15914
small molecule | CAS: 472-70-8

Deskripsi belum tersedia.

Kategori:
AlkenesBiological FactorsCarotenoids +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CSIC002 DB18584
small molecule

CSIC002 is a small-molecule Sema-3A inhibitor. It is being investigated for the treatment of anterior ischemic optic neuropathy.

Waktu Paruh-
Vol. Distribusi-
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CSL324 DB16359
biotech

CSL324 is a fully human anti-G-CSFR antibody shown to have the ability to control G-CSF-mediated neutrophilia in cynomolgus macaques.[A225626] It has potential applications in various inflammatory conditions such as cystic fibrosis, inflammatory bowel disease…

Waktu Paruh-
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CT-001 DB18284
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CT-011 DB05916
biotech

CT-011 is a humanized monoclonal antibody directed against a B7 family-associated protein, in patients with advanced haematological malignancies. It is directed against human PD-1 (programmed cell death 1; PDCD1), with immunomodulating and antitumor activitie…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents +7
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CT-2584 DB13098
small molecule | CAS: 166981-13-1

CT-2584 has been used in trials studying the treatment of Prostate Cancer.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingPhospholipase D, antagonists & inhibitors +2
Target Protein:
Choline-phosphate cytidylyltransferase B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CTA018 DB05024
small molecule

CTA018 is a member of a new class of vitamin D analogues with a dual mechanism of action, called Vitamin D Signal Amplifiers. This proprietary new drug is both a potent inhibitor of CYP24 (the enzyme responsible for the breakdown of vitamin D) and a potent ac…

Target Protein:
1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrialVitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CTCE-0214 DB05934
small molecule | CAS: 577782-52-6

CTCE-0214 is a stable peptide agonist of stromal cell-derived factor-1 (SDF-1), a key signaling molecule in the proliferation, homing, engraftment and expansion of hematopoietic stem cells and white blood cells.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Inflammatory AgentsBiological Factors +8
Target Protein:
Stromal cell-derived factor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CTCE-9908 DB05625
small molecule | CAS: 1030384-98-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and Proteins
Target Protein:
C-X-C chemokine receptor type 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CTR-107 DB18583
biotech

CTR-107 is a synthetic targeted growth factor. It is being investigated for the treatment of familial exudative vitreoretinopathy.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CTT-1057 DB14965
small molecule | CAS: 1628717-55-4

CTT-1057 is under investigation in clinical trial NCT03427476 (CTT1057, a Small Molecular Inhibitor of PSMA, as a Novel Imaging Agent of Neovascularization in Renal Cell Carcinoma).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
CTx-PDE6b DB17858
biotech

CTx-PDE6b is an adeno-associated virus (AAV) based gene therapy designed to deliver a full-length non-mutated copy of the functional human _PDE6b_ gene. Being commercialied by Coave Therapeutics, it is being investigated for the treatment of retinitis pigment…

Waktu Paruh-
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