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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
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13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 84 / 272
Cefradine Approved DB01333
small molecule | CAS: 38821-53-3

A semi-synthetic cephalosporin antibiotic.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +18
Target Protein:
Penicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefroxadine DB11367
small molecule | CAS: 51762-05-1

Cefroxadine is an orally available cephalosporin antibiotic. As part of its drug class, it shares structural properties to [cefalexin] as well as its activity spectrum. It was used in Italy but has since been withdrawn.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +10
Target Protein:
Penicillin-binding protein 1B
Waktu ParuhThe serum half life…
Vol. DistribusiVolume of distrubut…
KlirensThe total body clea…
Genetik -
Cefsulodin DB13499
small molecule | CAS: 62587-73-9

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceftaroline fosamil Approved DB06590
small molecule | CAS: 229016-73-3

Ceftaroline fosamil is a cephalosporin antibacterial indicated for the treatment of the following infections caused by designated susceptible bacteria: Acute bacterial skin and skin structure infections. Community-acquired bacterial pneumonia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein
Waktu Paruh1.60 hours (600 mg …
Vol. DistribusiMedian 20.3 L (18.3…
Klirens-
Genetik -
Ceftazidime Approved DB00438
small molecule | CAS: 72558-82-8

Bacteria possess a cell wall comprising a glycopeptide polymer commonly known as peptidoglycan, which is synthesized and remodelled through the action of a family of enzymes known as "penicillin-binding proteins" (PBPs).[A232920] ?-lactam antibiotics, includi…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1APenicillin-binding protein 1B +2
Waktu ParuhCeftazidime has an …
Vol. DistribusiCeftazidime has a v…
KlirensThe mean renal clea…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-lactamaseBeta-lactamase TEMBeta-lactamase CTX-M
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceftezole DB13821
small molecule | CAS: 26973-24-0

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceftibuten Approved DB01415
small molecule | CAS: 97519-39-6

Ceftibuten is a third-generation cephalosporin antibiotic that is orally-administered. It is typically used to treat acute bacterial exacerbations of chronic bronchitis (ABECB), acute bacterial otitis media, pharyngitis, and tonsilitis.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1APenicillin-binding protein 1B +1
Waktu Paruh-
Vol. Distribusi* 0.21 L/kg [adult …
Klirens-
Genetik -
Ceftiofur DB11485
small molecule | CAS: 80370-57-6

Ceftiofur is a third generation cephalosporin antibiotic, first described in 1987, and now used in veterinary medicine. It is marketed by pharmaceutical company Zoetis as Excenel, and is the active ingredient in that company's Specramast LC (lactating cow for…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceftizoxime Approved DB01332
small molecule | CAS: 68401-81-0

A semisynthetic cephalosporin antibiotic which can be administered intravenously or by suppository. The drug is highly resistant to a broad spectrum of beta-lactamases and is active against a wide range of both aerobic and anaerobic gram-positive and gram-neg…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 1BPeptidoglycan transpeptidase +1
Waktu Paruh-
Vol. DistribusiThe mean apparent v…
Klirens-
Genetik -
Ceftobiprole medocaril Approved DB14733
small molecule | CAS: 376653-43-9

Ceftobiprole medocaril is a prodrug of [ceftobiprole], a fifth-generation semisynthetic cephalosporin antibacterial. Ceftobiprole is a broad-spectrum agent with demonstrated activity against both Gram-positive and Gram-negative bacteria, including antibiotic-…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
MecAPenicillin-binding protein 2BPenicillin-binding protein 2X
Waktu ParuhThe half-life of ac…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
Ceftolozane Approved DB09050
small molecule | CAS: 689293-68-3

Ceftolozane is a semi-synthetic broad-spectrum fifth generation cephalosporin.[L6685] It was approved by the FDA in 2014 for use in combination with [Tazobactam] for the treatment of serious infections, such as intra-abdominal infections and complicated urina…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +8
Target Protein:
Penicillin-binding protein 1BCell division proteinPenicillin-binding protein 1C +2
Waktu Paruh2.77 hours on day 1…
Vol. Distribusi13.5 L.[L41618] Tis…
KlirensThe renal clearance…
Genetik -
Ceftriaxone Approved DB01212
small molecule | CAS: 73384-59-5

Ceftriaxone is a broad-spectrum third-generation cephalosporin antibiotic.[A215582] It has a very long half-life compared to other cephalosporins and is high penetrable into the meninges[A215582], eyes[A215647], and inner ear[A215627]. Ceftriaxone has broader…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
Penicillin-binding protein 2BSolute carrier family 22 member 11Solute carrier family 22 member 6 +2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe plasma clearanc…
Genetik -
Cefuroxime Approved DB01112
small molecule | CAS: 55268-75-2

Broad-spectrum cephalosporin antibiotic resistant to beta-lactamase. It has been proposed for infections with gram-negative and gram-positive organisms, gonorrhea, and haemophilus.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
Penicillin-binding protein 1A
Waktu ParuhApproximately 80 mi…
Vol. Distribusi-
Klirens-
Genetik -
Celastrol DB18736
small molecule | CAS: 34157-83-0

Celastrol is a pentacyclic triterpenoid isolated from the root extracts of _Tripterygium wilfordii_.[L50567]

Kategori:
TerpenesTripterygiumTriterpenes
Target Protein:
Interleukin-1 betaTumor necrosis factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Celecoxib Approved DB00482
small molecule | CAS: 169590-42-5

Celecoxib, a selective cyclooxygenase-2 (COX-2) inhibitor, is a nonsteroidal anti-inflammatory drug (NSAID) which is known for its decreased risk of causing gastrointestinal bleeding compared to other NSAIDS.[A181544] It is used to manage symptoms of various …

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +41
Target Protein:
Prostaglandin G/H synthase 2Signal transducer and activator of transcription 3Sialidase-1 +4
Gen Terkait:
CYP2C9
Waktu ParuhThe effective half-…
Vol. DistribusiThe apparent volume…
KlirensApparent clearance …
Genetik 1 Varian
Celiprolol Approved DB04846
small molecule | CAS: 56980-93-9

Celiprolol is indicated for the management of mild to moderate hypertension and effort-induced angina pectoris. It is simultaneously a selective ?1 receptor antagonist, a ?2 receptor partial agonist and a weak ?2 receptor antagonist. In 2010 a clinical trial …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic Antagonists +30
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor +3
Waktu Paruh5 hours
Vol. DistribusiThe distribution vo…
KlirensCleared by both ren…
Genetik -
Celivarone DB16012
small molecule | CAS: 401925-43-7

Celivarone is under investigation in clinical trial NCT00233441 (Placebo Controlled Double-blind Dose Ranging Study of the Efficacy and Safety of SSR149744C 50, 100, 200 or 300 Mg OD With Amiodarone as Calibrator for the Maintenance of Sinus Rhythm in Patient…

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cellobiose DB02061
small molecule | CAS: 528-50-7

A disaccharide consisting of two glucose units in beta (1-4) glycosidic linkage. Obtained from the partial hydrolysis of cellulose. [PubChem]

Kategori:
CarbohydratesCelluloseCompounds used in a research, industrial, or household setting +4
Target Protein:
Endoglucanase GEndoglucanase 5AEndoglucanase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cellotetraose DB02717
small molecule | CAS: 38819-01-1

Deskripsi belum tersedia.

Kategori:
BiopolymersCarbohydratesCompounds used in a research, industrial, or household setting +5
Target Protein:
Glucanase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cemdisiran DB16121
biotech | CAS: 1639264-46-2

Cemdisiran is under investigation in clinical trial NCT03841448 (A Study of Cemdisiran in Adults With Immunoglobulin a Nephropathy (Igan)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cemdomespib DB18953
small molecule | CAS: 1450642-92-8

Cemdomespib is under investigation in clinical trial NCT05895552 (A Phase 2 Study of RTA 901 in Patients With Diabetic Peripheral Neuropathic Pain (CYPRESS)).

Kategori:
AminesCarbohydratesEthylamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cemiplimab Approved DB14707
biotech | CAS: 1801342-60-8

Cemiplimab is a fully human monoclonal antibody that works against programmed death receptor-1 (PD-1), which is a negative regulator of T cell function. By blocking PD-1, cemiplimab works to enhance T cell-mediated antitumour responses.[L39804] Cemiplimab …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Programmed cell death protein 1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensCemiplimab clearanc…
Genetik -
Cemsidomide DB18400
small molecule | CAS: 2504235-67-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cendakimab DB18427
biotech

Cendakimab is a recombinant humanized anti-interleukin 13 (IL-13) monoclonal antibody.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenegermin Approved DB13926
biotech | CAS: 1772578-74-1

Cenegermin is a human beta-nerve growth factor (beta-ngf)-(1-118)- peptide (non-covalent dimer) produced in escherichia coli. It received European Union Approval in July 2017 for the treatment of moderate to severe neurotrophic keratitis. Cenegermin received …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +7
Target Protein:
High affinity nerve growth factor receptorTumor necrosis factor receptor superfamily member 16
Waktu ParuhHalf-life data spec…
Vol. DistribusiAfter eye drop admi…
KlirensAlthough the system…
Genetik -
Cenersen DB15455
biotech | CAS: 415168-49-9

Cenersen is under investigation in clinical trial NCT02243124 (A Study of Aezea® (Cenersen) in Transfusion Dependent Anemia Associated With Myelodysplastic Syndrome (MDS)).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenicriviroc DB11758
small molecule | CAS: 497223-25-3

Cenicriviroc has been used in trials studying the treatment of HIV-infection/AIDS, AIDS Dementia Complex, Nonalcoholic Steatohepatitis, Human Immunodeficiency Virus, and HIV-1-Associated Cognitive Motor Complex.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +4
Target Protein:
C-C chemokine receptor type 5C-C chemokine receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenisertib DB06347
small molecule | CAS: 871357-89-0

Cenisertib is an aurora kinase inhibitor.

Kategori:
Bridged-Ring Compounds
Target Protein:
Aurora kinase BAurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenobamate Approved DB06119
small molecule | CAS: 913088-80-9

Cenobamate, or YKP-3089, is an antiepileptic drug developed by SK Pharmaceuticals and used to treat partial onset seizures.[A188442,L10653] The exact mechanism of action has not been described in the literature, though it positively modulates GABA<sub>A</sub>…

Kategori:
Acids, AcyclicAnticonvulsantsBenzene Derivatives +34
Target Protein:
Voltage-gated sodium channel alpha subunitGamma-aminobutyric acid receptor subunit alpha-1
Waktu ParuhThe terminal half l…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Cenplacel-L DB19188
biotech

Cenplacel-L is under investigation in clinical trial (Study of Human Placenta-derived Cells (PDA001) to Evaluate the Safety and Effectiveness for Patients With Ischemic Stroke) for the treatment of patients with Ischemic Stroke.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Censavudine DB12074
small molecule | CAS: 634907-30-5

Censavudine has been used in trials studying the treatment of HIV-1 Infection.

Kategori:
Anti-HIV AgentsDeoxyribonucleosidesNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Centanafadine DB14841
small molecule | CAS: 924012-43-1

Centanafadine is under investigation in clinical trial NCT02827513 (A Phase 1 Study to Investigate the Safety, Tolerance, Food Effect, Pharmacokinetics and Pharmacodynamics of Single and Multiple Doses of Extended Release Formulations of Centanafadine (CTN) i…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Centhaquine DB16122
small molecule | CAS: 57961-90-7

Centhaquine is under investigation in clinical trial NCT04045327 (Efficacy of PMZ-2010 (Centhaquine) a Resuscitative Agent for Hypovolemic Shock).

Kategori:
Adrenergic and Dopaminergic AgentsCardiac Stimulants Excl. Cardiac GlycosidesCardiac Therapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CEP-1347 DB05403
small molecule

CEP-1347 is a semi-synthetic compound shown to protect multiple nerve cell types from a variety of insults leading to programmed cell death (apoptosis) which could improve the survival of dopamine neurons prior to and after transplantation.

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
Target Protein:
Mitogen-activated protein kinase 12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CEP-37440 DB13060
small molecule | CAS: 1391712-60-9

CEP-37440 has been used in trials studying the treatment of Solid Tumors.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Focal adhesion kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CEP-9722 DB14882
small molecule | CAS: 916574-83-9

CEP-9722 is under investigation in clinical trial NCT01345357 (Study of CEP-9722 in Combination With Gemcitabine and Cisplatin in Patients With Advanced Solid Tumors or Mantle Cell Lymphoma).

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingImides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1192706-52-7

Cepeginterferon alfa-2B is under investigation in clinical trial NCT01889433 (An Open-label Comparative Efficacy and Safety Study of Algeron (Cepeginterferon Alfa-2b) in Treatment-naive Patients With Chronic Hepatitis C).

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP1A2 Inhibitors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cephalexin Approved DB00567
small molecule | CAS: 15686-71-2

Cephalexin is the first of the first generation cephalosporins.[A179071,A179074] This antibiotic contains a beta lactam and a dihydrothiazide.[A179071] Cephalexin is used to treat a number of susceptible bacterial infections through inhibition of cell wall s…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +23
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2aPenicillin-binding protein 1b +2
Waktu ParuhThe half life of ce…
Vol. Distribusi5.2-5.8L.[A179068]
KlirensClearance from one …
Genetik -
Cephaloglycin Approved DB00689
small molecule | CAS: 3577-01-3

A cephalorsporin antibiotic that is no longer commonly used.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +7
Target Protein:
Penicillin-binding protein 1B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Agents that reduce seizure threshold
Target Protein:
D-alanyl-D-alanine carboxypeptidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cephalosporin C DB03313
small molecule | CAS: 61-24-5

Deskripsi belum tersedia.

Kategori:
Agents that reduce seizure thresholdAmidesbeta-Lactams +4
Target Protein:
Penicillin-binding protein 1bPeptidoglycan synthase FtsIPenicillin-binding protein 1A +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cephalosporium roseum Approved DB10932
biotech

Cephalosporium roseum allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Cephalothin group is a solid. This compound belongs to the 1,3-thiazines. These are organic compounds containing 1,3-thiazine, a six-member ring with a nitrogen and a sulfur atom in ring positions 1 and 3 respectively, as well as two double bonds. This substa…

Kategori:
Nephrotoxic agents
Target Protein:
D-alanyl-D-alanine carboxypeptidaseBeta-lactamase Toho-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CER-001 DB18538
biotech

CER-001 is a negatively charged lipoprotein particle comprising human recombinant apolipoprotein A-I and two phospholipids: sphingomyelin and dipalmitoylphosphatidylglycerol.[L48290] It is under investigation for the treatment of lecithin-cholesterol acyltran…

Kategori:
Amino Acids, Peptides, and ProteinsApolipoproteinsApolipoproteins A +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceralasertib DB14917
small molecule | CAS: 1352226-88-0

Ceralasertib is under investigation in clinical trial NCT03682289 (Phase II Trial of AZD6738 Alone and in Combination With Olaparib).

Kategori:
AmidesHeterocyclic Compounds, Fused-RingOxazines +2
Target Protein:
Serine/threonine-protein kinase ATR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceralifimod DB16123
small molecule | CAS: 891859-12-4

Ceralifimod is under investigation in clinical trial NCT01226745 (Phase 2 Extension Trial in Patients With Relapsing-remitting Multiple Sclerosis (RRMS)).

Kategori:
AzetinesImmunologic FactorsImmunosuppressive Agents +1
Target Protein:
Sphingosine 1-phosphate receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceramide NG DB14706
small molecule | CAS: 2304-80-5

Deskripsi belum tersedia.

Kategori:
AmidesCarbohydratesGlycoconjugates +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceramide NP DB14111
small molecule | CAS: 100403-19-8

Ceramide NP is a lipid molecule included in a group of lipid molecules called ceramides. Ceramides are major lipid components in the stratum corneum of the human skin. Ceramide 3 consists of a phytosphingosine backbone N-acylated with a saturated fatty acid (…

Kategori:
AntigensAntigens, NeoplasmBiological Factors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CERC-301 DB12063
small molecule | CAS: 808732-98-1

Mk 0657 has been used in trials studying the treatment of Major Depressive Disorder.

Kategori:
Receptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Target Protein:
Glutamate receptor ionotropic, NMDA 2B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4151–4200 dari 13591
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