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14063

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10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
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14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 84 / 282
CAN-106 DB18389
biotech

CAN-106 a novel, long-acting monoclonal antibody directed against human complement C5.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Canagliflozin Approved DB08907
small molecule | CAS: 842133-18-0

Canagliflozin, also known as _Invokana_, is a sodium-glucose cotransporter 2 (SGLT2) inhibitor used in the management of type 2 diabetes mellitus along with lifestyle changes including diet and exercise [FDA label]. It was initially approved by the FDA in …

Kategori:
Agents causing hyperkalemiaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +15
Target Protein:
Sodium/glucose cotransporter 2
Waktu ParuhIn a clinical study…
Vol. DistribusiThis drug is extens…
KlirensIn healthy subjects…
Genetik -
Canakinumab Approved DB06168
biotech | CAS: 914613-48-2

Canakinumab is a recombinant, human anti-human-IL-1? monoclonal antibody that belongs to the IgG1/? isotype subclass. It is expressed in a murine Sp2/0-Ag14 cell line and comprised of two 447- (or 448-) residue heavy chains and two 214-residue light chains, w…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +13
Target Protein:
Interleukin-1 beta
Waktu Paruh26 days
Vol. DistribusiThe steady-state vo…
KlirensThe clearance of ca…
Genetik -
Canaline DB02821
small molecule | CAS: 496-93-5

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +1
Target Protein:
Ornithine aminotransferase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Canavanine DB01833
small molecule | CAS: 543-38-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
Nitric oxide synthase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2259683-77-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Candesartan DB13919
small molecule | CAS: 139481-59-7

Candesartan is an angiotensin-receptor blocker (ARB) that may be used alone or with other agents to treat hypertension. It is available as a prodrug in the form of [candesartan cilexetil].

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAngiotensin 2 Receptor Blocker +22
Target Protein:
Type-1 angiotensin II receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Candicidin Approved DB01152
small molecule | CAS: 1403-17-4

Candicidin is an antibiotic obtained from a streptomyces (Streptomyces griseus) and active against some fungi of the genus Candida (C. albicans). Candicidin is administered intravaginally in the treatment of vulvovaginal candidiasis.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntifungal Agents +9
Target Protein:
Ergosterol
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Candida albicans Approved DB10429
biotech

Candida albicans is a fungus which can provoke allergic reactions. Candida albicans is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Candoxatril DB00616
small molecule | CAS: 123122-55-4

Candoxatril is the orally-active prodrug of candoxatrilat (UK-73967), a potent neutral endopeptidase (NEP) inhibitor.

Kategori:
Acids, AcyclicAntihypertensive AgentsCardiovascular Agents +8
Target Protein:
NeprilysinAngiotensin-converting enzyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Candoxatrilat DB11623
small molecule | CAS: 123122-54-3

A dicarboxylic acid monoamide obtained by formal condensation between the amino group of cis-4-aminocyclohexanecarboxylic acid and the cyclopentanecarboxylic acid group of 1-[(2S)-2-carboxy-3-(2-methoxyethoxy)propyl]cyclopentanecarboxylic acid. A potent inhib…

Kategori:
Acids, CarbocyclicCyclohexanesCycloparaffins +3
Target Protein:
Neprilysin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Canertinib DB05424
small molecule | CAS: 267243-28-7

Canertinib is a pan-erbB tyrosine kinase inhibitor which work against esophageal squamous cell carcinoma in vitro and in vivo. Canertinib treatment significantly affects tumour metabolism, proliferation and hypoxia as determined by PET.

Kategori:
Acids, AcyclicAnestheticsAntineoplastic Agents +10
Target Protein:
Receptor tyrosine-protein kinase erbB-2RAC-alpha serine/threonine-protein kinaseReceptor tyrosine-protein kinase erbB-4 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Canfosfamide DB04972
small molecule | CAS: 158382-37-7

Canfosfamide is an active agent in chemotherapy-resistant ovarian cancer.

Kategori:
Amino Acids, Peptides, and ProteinsCytotoxinsOligopeptides +1
Target Protein:
Glutathione S-transferase P
Waktu Paruh18 min
Vol. Distribusi-
Klirens-
Genetik -
Cangrelor Approved DB06441
small molecule | CAS: 163706-06-7

Cangrelor is an intravenous, direct-acting, reversible P2Y12 inhibitor for patients undergoing percutaneous coronary intervention (PCI) who have not been yet treated by oral P2Y12 inhibitors. An advantage Cangrelor provides over oral P2Y12 inhibitors (such as…

Kategori:
Adenine NucleotidesAnticoagulantsAntiplatelet agents +16
Target Protein:
P2Y purinoceptor 12
Waktu ParuhThe average elimina…
Vol. DistribusiIn a study in healt…
KlirensThe mean clearance …
Genetik -
Cannabichromene DB14735
small molecule | CAS: 20675-51-8

A natural product found in Cannabis sativa and Helichrysum species.

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cannabidiol Approved DB09061
small molecule | CAS: 13956-29-1

Cannabidiol, or CBD, is one of at least 85 active cannabinoids identified within the Cannabis plant. It is a major phytocannabinoid, accounting for up to 40% of the Cannabis plant's extract, that binds to a wide variety of physiological targets of the endocan…

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAnticonvulsants +56
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2G-protein coupled receptor 12 +36
Waktu ParuhThe CBD component o…
Vol. DistribusiCannabinoids are di…
Klirens-
Genetik -
small molecule | CAS: 1244-58-2

Cannabidiolic acid is under investigation in clinical trial NCT04103814 (Effect of Topical CBD Cream for Degenerative Hallux Disorders).

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cannabidivarin DB14050
small molecule | CAS: 24274-48-4

Cannabidivarin, also known as cannabidivarol or CBDV, is a non-psychoactive cannabinoid found within [DB14009]. It is one of over 100 cannabinoids identified from the Cannabis plant that can modulate the physiological activity of cannabis, or marijuana [A3258…

Kategori:
AnticonvulsantsCentral Nervous System DepressantsTerpenes
Target Protein:
Transient receptor potential cation channel subfamily V member 1Transient receptor potential cation channel subfamily V member 2Transient receptor potential cation channel subfamily A member 1 +1
Waktu ParuhOrally administered…
Vol. DistribusiDue to its lipophil…
Klirens-
Genetik -
Cannabigerol DB14734
small molecule | CAS: 25654-31-3

A natural product found in Cannabis sativa and Helichrysum species.

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cannabinol DB14737
small molecule | CAS: 521-35-7

Cannabinol (CBN) is a physiologically inactive constituent of Cannabis sativa.

Kategori:
BCRP/ABCG2 InhibitorsCannabinoids and similarsCytochrome P-450 CYP1A2 Inhibitors +30
Target Protein:
Cannabinoid receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cannabinor DB05048
small molecule | CAS: 573981-31-4

Cannabinor, a synthetic CB2-selective agonist, is in Phase 2 clinical testing as an analgesic.

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cannabivarin DB14736
small molecule | CAS: 33745-21-0

A natural product found in Cannabis sativa.

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Canrenone DB12221
small molecule | CAS: 976-71-6

Canrenone has been used in trials studying the diagnostic of Heart Failure.

Kategori:
Agents causing hyperkalemiaDiureticsFused-Ring Compounds +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cantharidin Approved DB12328
small molecule | CAS: 56-25-7

Cantharidin is a naturally occurring odorless, colorless fatty substance of the terpenoid class that is produced as an oral fluid in the alimentary canal of the male blister beetle.[A32891, A32892] For its natural purpose, the male blister beetle secretes and…

Kategori:
BenzofuransCompounds used in a research, industrial, or household settingEnzyme Inhibitors +4
Target Protein:
Serine/threonine-protein phosphatase PP1-alpha catalytic subunitAryl hydrocarbon receptor
Waktu ParuhLittle pharmacodyna…
Vol. DistribusiAfter oral or IP in…
KlirensLittle pharmacodyna…
Genetik -
biotech | CAS: 400010-39-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CAP-1 DB08027
small molecule | CAS: 564475-13-4

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capadenoson DB16118
small molecule | CAS: 544417-40-5

Capadenoson is under investigation in clinical trial NCT00518921 (Capadenoson in Angina Pectoris).

Kategori:
Adenosine A receptor agonistsAdenosine A1 Receptor AgonistsAmines +2
Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capecitabine Approved DB01101
small molecule | CAS: 154361-50-9

Capecitabine is an orally-administered chemotherapeutic agent used in the treatment of metastatic breast and colorectal cancers. Capecitabine is a prodrug, that is enzymatically converted to fluorouracil (antimetabolite) in the tumor, where it inhibits DNA sy…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +21
Target Protein:
Thymidylate synthaseDNARNA +1
Gen Terkait:
DPYD DPYD DPYD +4
Waktu ParuhThe elimination hal…
Vol. DistribusiIn colorectal cance…
KlirensIn colorectal cance…
Genetik 7 Varian
Capivasertib Approved DB12218
small molecule | CAS: 1143532-39-1

Hormone receptor (HR) positive, especially estrogen receptor-positive, HER2-negative breast cancer is the most common subtype of metastatic breast cancer, resulting in more than 400,000 deaths annually. Although endocrine-based therapy is the first line of tr…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +13
Target Protein:
RAC-alpha serine/threonine-protein kinaseRAC-beta serine/threonine-protein kinaseRAC-gamma serine/threonine-protein kinase
Waktu ParuhThe half-life of ca…
Vol. DistribusiThe steady-state or…
KlirensThe steady-state or…
Genetik -
Caplacizumab Approved DB06081
biotech | CAS: 915810-67-2

Caplacizumab, firstly called ALX-0081, is a humanized single-variable-domain immunoglobulin consisting of two identical humanized building blocks genetically linked by a three-alanine linker. Caplacizumab was developed by Ablynx, a Sanofi company and FDA appr…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
von Willebrand factor
Waktu ParuhThe reported half-l…
Vol. DistribusiThe reported volume…
KlirensAs the elimination …
Genetik -
Capmatinib Approved DB11791
small molecule | CAS: 1029712-80-8

Capmatinib is a small molecule kinase inhibitor targeted against c-Met (a.k.a. hepatocyte growth factor receptor [HGFR]), a receptor tyrosine kinase that, in healthy humans, activates signaling cascades involved in organ regeneration and tissue repair.[A19912…

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +20
Target Protein:
Hepatocyte growth factor receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -
Capravirine DB08502
small molecule | CAS: 178979-85-6

Deskripsi belum tersedia.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +11
Target Protein:
Gag-Pol polyproteinGag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2605-79-0

Deskripsi belum tersedia.

Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialPancreatic lipase-related protein 2Ferrichrome-iron receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capromab pendetide Approved DB00089
biotech | CAS: 145464-28-4

Capromab is a Murine IgG1 monoclonal 7E11-C5.3 antibody that recognizes prostate specific membrane antigen (PSMA – also known as glutamate carboxypeptidase 2) from prostate cancer cells and normal prostate tissue. When linked to pendetide, capromab is used as…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +13
Target Protein:
Glutamate carboxypeptidase 2
Waktu Paruh-
Vol. Distribusi* 4 ± 2.1 L
Klirens* 42 +/- 22 mL/hr
Genetik -
Capromorelin DB15205
small molecule | CAS: 193273-66-4

Capromorelin is under investigation in clinical trial NCT00527046 (Effects Of An Oral Growth Hormone Secretagogue In Older Functionally Limited Adults).

Target Protein:
Growth hormone secretagogue receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Caprospinol DB05263
small molecule | CAS: 4952-56-1

Caprospinol (SP-233) is the first drug ever to demonstrate the correlation of clearing beta-amyloid from the brain. It also improves the brain histopathology and recovers memory function.

Kategori:
Acids, AcyclicCholestanesFatty Acids +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Caprylic acid DB04519
small molecule | CAS: 124-07-2

Caprylic acid is an eight-carbon chain fatty acid, also known systematically as octanoic acid. It is found naturally in coconuts and breast milk. It is an oily liquid with a slightly unpleasant rancid-like smell that is minimally soluble in water.

Kategori:
Acids, AcyclicFatty AcidsLipids +2
Target Protein:
Peroxisome proliferator-activated receptor alpha3-oxoacyl-[acyl-carrier-protein] synthase 1Acyl-CoA thioesterase I
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 111-87-5

Caprylic alcohol has been used in trials studying the treatment of Essential Tremor.

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingFatty Alcohols +3
Target Protein:
Gap junction alpha-1 protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Caprylyl glycol DB14589
small molecule | CAS: 1117-86-8

Deskripsi belum tersedia.

Kategori:
AlcoholsFatty AlcoholsLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capsicum oleoresin Approved DB11131
biotech | CAS: 8023-77-6

Capsicum oleoresin is an oily organic resin derived from the fruit of plants in the Capsicum genus, such as chilli peppers. When the plants are finely ground, capsicum oleoresin is formed after the extraction process of capsaicin using oragnic solvents such a…

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +1
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu ParuhFor pharmacokinetic…
Vol. DistribusiFor pharmacokinetic…
KlirensFor pharmacokinetic…
Genetik -
Captodiame DB09014
small molecule | CAS: 486-17-9

Captodiame, also known as captodiamine, is an antihistamine which is used as a sedative and anxiolytic. It is a derivative of diphenhydramine. Captodiame has been suggested for use in preventing benzodiazepine withdrawal syndrome.

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsCentral Nervous System Depressants +7
Target Protein:
5-hydroxytryptamine receptor 2CSigma non-opioid intracellular receptor 1D(3) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Captopril Approved DB01197
small molecule | CAS: 62571-86-2

Captopril is a potent, competitive inhibitor of angiotensin-converting enzyme (ACE), the enzyme responsible for the conversion of angiotensin I (ATI) to angiotensin II (ATII). ATII regulates blood pressure and is a key component of the renin-angiotensin-aldos…

Kategori:
ACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin SystemAgents causing angioedema +19
Target Protein:
Angiotensin-converting enzyme72 kDa type IV collagenaseMatrix metalloproteinase-9 +2
Waktu Paruh2 hours
Vol. Distribusi-
Klirens-
Genetik -
Caramiphen DB11504
small molecule | CAS: 77-22-5

Caramiphen is a cholinergic antagonist used in Parkinson's disease. Additionally, it is used, in combination with [phenylpropanolamine], as a cough suppressant and nasal decongestant for the symptomatic treatment of seasonal respiratory conditions.

Kategori:
Cycloparaffins
Target Protein:
Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Poly [ADP-ribose] polymerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carbamazepine Approved DB00564
small molecule | CAS: 298-46-4

Carbamazepine, also known as Tegretol, is an anticonvulsant drug and analgesic drug used to control seizures and to treat pain resulting from trigeminal neuralgia. It was initially approved by the FDA in 1965.[A180301] Aside from the above uses, this drug is …

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnticonvulsants +65
Target Protein:
Voltage-gated sodium channel alpha subunitNeuronal acetylcholine receptor subunit alpha-4Nuclear receptor subfamily 1 group I member 2
Gen Terkait:
SCN1A HSPA1L HSPA1A +7
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe volume of distr…
KlirensIn a pharmacokineti…
Genetik 10 Varian
Carbamic Acid DB04261
small molecule | CAS: 463-77-4

Deskripsi belum tersedia.

Kategori:
Acids, Acyclic
Target Protein:
Beta-lactamaseBeta-lactamase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carbamide peroxide Approved DB11129
small molecule | CAS: 124-43-6

Carbamide peroxide, also known as urea-hydrogen peroxide, is a water-soluble, white crystalline solid compound consisting of hydrogen peroxide and urea. As it is a source of hydrogen peroxide, it can be found in disinfecting and dental bleaching products. Som…

Kategori:
AmidesAnionsAnti-Infective Agents +14
Waktu ParuhNo established phar…
Vol. DistribusiNo established phar…
KlirensNo established phar…
Genetik -
Carbamoylcholine Approved DB00411
small molecule | CAS: 462-58-8

Carbamoylcholine, also known as carbachol, is a muscarinic agonist discovered in 1932.[A226315] Carbamoylcholine was initially used as a treatment for migraines,[A226365] induction of diuresis,[A226370] and other parasympathetic effects. Carbamoylcholine w…

Kategori:
AlcoholsAminesAmino Alcohols +28
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Neuronal acetylcholine receptor subunit alpha-2 +2
Waktu ParuhData regarding the …
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Carbapenem DB18912
small molecule | CAS: 78854-41-8

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial Agentsbeta-Lactams +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4151–4200 dari 14063
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