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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 83 / 272
CBP-501 DB17277
small molecule | CAS: 565434-85-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCell Cycle ProteinsDual-Specificity Phosphatases +11
Target Protein:
MAP/microtubule affinity-regulating kinase 3MAP kinase-activated protein kinase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CC-115 DB12740
small molecule | CAS: 1228013-15-7

CC-115 has been used in trials studying the treatment of Prostate Cancer, Neoplasm Metastasis, Ewing's Osteosarcoma, Glioblastoma Multiforme, and Chronic Lymphocytic Leukemia, among others.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CC-401 DB12432
small molecule | CAS: 395104-30-0

CC-401 has been used in trials studying the treatment of Myeloid Leukemia.

Kategori:
JNK Mitogen-Activated Protein Kinases, antagonists & inhibitorsPyrazoles
Target Protein:
Mitogen-activated protein kinase 8Mitogen-activated protein kinase 9Mitogen-activated protein kinase 10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CC-90001 DB18445
small molecule | CAS: 1403859-14-2

Deskripsi belum tersedia.

Kategori:
AminesCyclohexanesCycloparaffins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CCX-354 DB12963
small molecule | CAS: 1010073-75-2

CCX354-C has been used in trials studying the treatment of Rheumatoid Arthritis.

Target Protein:
C-C chemokine receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CDD-0102 DB16945
small molecule | CAS: 146422-58-4

Deskripsi belum tersedia.

Kategori:
Muscarinic AgonistsOxazolesReceptor, Muscarinic M1, agonists
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CDP323 DB05092
small molecule

CDP323 is an antagonist of the _vascular cell adhesion molecule 1_ (VCAM-1) binding to alpha4-integrins (other adhesion molecules), a process thought to be implicated in the pathophysiology of Multiple Sclerosis (MS). It is considered a small-molecule prodrug…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +3
Target Protein:
Integrin alpha-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CDX-1135 DB17607
biotech

CDX-1135, formerly TP-10, is a soluble, recombinant human Complement Receptor Type 1 (sCR1) developed by Avant Immunotherapeutics (now Celldex). It was investigated in clinical trials for post-cardiopulmonary bypass syndrome and kidney damage.

Kategori:
Amino Acids, Peptides, and ProteinsMembrane ProteinsProteins +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CDX-301 DB19293
biotech

CDX-301 is under investigation in clinical trial NCT02129075 (A Vaccine (CDX-1401) With or Without a Biologic Drug (CDX-301) for the Treatment of Patients With Stage IIB-IV Melanoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CE-224535 DB12113
small molecule | CAS: 724424-43-5

CE-224535 has been used in trials studying the treatment of Osteoarthritis.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +4
Target Protein:
P2X purinoceptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CE-326597 DB12694
small molecule | CAS: 870615-40-0

CE-326,597 has been used in trials studying the treatment of Obesity.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Cholecystokinin receptor type A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cebranopadol DB12830
small molecule | CAS: 863513-91-1

Cebranopadol has been used in trials studying the treatment of Pain, Neoplasms, and Chronic Pain.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Mu-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceclazepide DB17270
small molecule | CAS: 1801749-44-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cedar leaf oil DB15836
biotech | CAS: 8007-20-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Cedazuridine Approved DB15694
small molecule | CAS: 1141397-80-9

Myelodysplastic syndromes (MDS) are a group of hematopoietic neoplasms that give rise to variable cytopenias progressing to secondary acute myeloid leukemia (sAML), which is invariably fatal if untreated.[A215082, A215092, A215097] Hypomethylating agents such…

Kategori:
Cytidine Deaminase, antagonists & inhibitorsNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Cytidine deaminase
Waktu ParuhCedazuridine has a …
Vol. DistribusiThe apparent volume…
KlirensCedazuridine has an…
Genetik -
Cediranib DB04849
small molecule | CAS: 288383-20-0

The novel indole-ether quinazoline Cediranib is a highly potent (IC<sub>50</sub> &lt; 1 nmol/L) ATP-competitive inhibitor of recombinant KDR tyrosine kinase in vitro. It is being developed clinically as a once-daily oral therapy for the treatment of cancer.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsEnzyme Inhibitors +4
Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh12 to 35 hours
Vol. Distribusi-
Klirens-
Genetik -
Cedirogant DB18951
small molecule | CAS: 2055496-11-0

Cedirogant is under investigation in clinical trial NCT05044234 (A Study to Assess Adverse Events and Disease Activity With Cedirogant (ABBV-157) in Adult Participants With Moderate to Severe Psoriasis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefaclor Approved DB00833
small molecule | CAS: 53994-73-3

Semisynthetic, broad-spectrum antibiotic derivative of cephalexin.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 1A
Waktu Paruh0.6-0.9 hour
Vol. Distribusi-
Klirens-
Genetik -
Cefadroxil Approved DB01140
small molecule | CAS: 50370-12-2

Long-acting, broad-spectrum, water-soluble, cephalexin derivative.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 1APenicillin-binding protein 1b +1
Waktu Paruh1.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Cefalonium DB11385
small molecule | CAS: 5575-21-3

Deskripsi belum tersedia.

Kategori:
Amidesbeta-LactamsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefaloridine DB09008
small molecule | CAS: 50-59-9

Cephaloridine or cefaloridine is a first generation semisynthetic cephalosporin. It is derived from cephalosporin C and is a zwitterion at physiological pH.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefalotin Approved DB00456
small molecule | CAS: 153-61-7

Cefalotin is a cephalosporin antibiotic.

Kategori:
Agents that reduce seizure thresholdAmidesAnti-Bacterial Agents +13
Target Protein:
D-alanyl-D-alanine carboxypeptidasePenicillin-binding protein 1APenicillin-binding protein 1b +5
Waktu Paruh30 minutes
Vol. Distribusi-
Klirens-
Genetik -
Cefamandole Approved DB01326
small molecule | CAS: 34444-01-4

Cefamandole is also known as cephamandole. It is a parenterally administered broad-spectrum cephalosporin antibiotic. It is generally formulated as a formate ester, [cefamandole nafate]. It is no longer marketed in the United States.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
Penicillin-binding protein 2
Waktu ParuhThe half-life after…
Vol. Distribusi-
Klirens-
Genetik -
Cefapirin Approved DB01139
small molecule | CAS: 21593-23-7

Cefapirin (INN, also spelled cephapirin), commonly marketed under the trade name Cefadyl, is a first-generation cephalosporin antibiotic that is available in injectable formulations. Production for use in humans has been discontinued in the United States. Cef…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefatrizine DB13266
small molecule | CAS: 51627-14-6

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefazedone DB13778
small molecule | CAS: 56187-47-4

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefazolin Approved DB01327
small molecule | CAS: 25953-19-9

A semisynthetic cephalosporin analog with broad-spectrum antibiotic action due to inhibition of bacterial cell wall synthesis. It attains high serum levels and is excreted quickly via the urine.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 1BPenicillin-binding protein 1C +5
Waktu ParuhThe serum half-life…
Vol. Distribusi-
Klirens-
Genetik -
Cefbuperazone DB13638
small molecule | CAS: 76610-84-9

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefcapene DB13461
small molecule | CAS: 135889-00-8

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefdinir Approved DB00535
small molecule | CAS: 91832-40-5

Cefdinir, also known as Omnicef, is a semi-synthetic, broad-spectrum antibiotic belonging to the third generation of the cephalosporin class. It has been proven to be effective for the treatment of common bacterial infections in the ear, sinus, throat, lungs,…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +14
Target Protein:
Penicillin-binding protein 2PBP3Myeloperoxidase +1
Waktu ParuhThe average plasma …
Vol. DistribusiThe average volume …
KlirensThe renal clearance…
Genetik -
Cefepime Approved DB01413
small molecule | CAS: 88040-23-7

Cefepime is a fourth-generation cephalosporin antibiotic developed in 1994. Cefepime is active against Gram-positive and Gram-negative bacteria, and has greater activity against both compared to third-generation antibiotics.[A2457,A249050] Cefepime is normall…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 1BPenicillin-binding protein 2 +4
Waktu ParuhHealthy adult male …
Vol. DistribusiThe average steady-…
KlirensCefepime has a tota…
Genetik -
Cefetamet DB13504
small molecule | CAS: 65052-63-3

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 65243-33-6

Cefetamet pivoxil is under investigation in clinical trial NCT04664803 (Safety and Efficacy of Cefecin Tab. in Patients With Acute Sinusitis).

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefiderocol Approved DB14879
small molecule | CAS: 1225208-94-5

Cefiderocol is a cephalosporin antibacterial drug and exerts a mechanism of action similar to other ?-lactam antibiotics.[FDA Label] Unlike other agents in this category, cefiderocol is a siderophore able to undergo active transport into the bacterial cell th…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Cell division proteinPenicillin-binding protein 1APenicillin-binding protein 1B +2
Waktu ParuhThe terminal elimin…
Vol. DistribusiCefiderocol has a m…
KlirensCefiderocol has a m…
Genetik -
Cefilavancin DB05735
small molecule | CAS: 722454-12-8

Cefilavancin is a covalently-linked glycopeptide-cephalosporin (beta-lactam) heterodimer antibiotic that exhibits substantially greater activity than its component parts against Gram-positive bacteria.

Kategori:
AmidesAmino Acids, Peptides, and Proteinsbeta-Lactams +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefixime Approved DB00671
small molecule | CAS: 79350-37-1

Bacteria possess a cell wall comprising a glycopeptide polymer commonly known as peptidoglycan, which is synthesized and remodelled through the action of a family of enzymes known as "penicillin-binding proteins" (PBPs).[A232920] ?-lactam antibiotics, includi…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
Penicillin-binding proteinPenicillin-binding protein 2
Waktu ParuhCefixime has a seru…
Vol. DistribusiCefixime has a volu…
KlirensCefixime administer…
Genetik -
Cefmenoxime Approved DB00267
small molecule | CAS: 65085-01-0

Cefmenoxime is a novel broad-spectrum and third-generation cephalosporin antibiotic that is typically used in the treatment of female gynecologic and obstetric infections. It is reported to exhibit high activity against a wide variety of gram-positive and gra…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1A
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
Cefmetazole Approved DB00274
small molecule | CAS: 56796-20-4

A semisynthetic cephamycin antibiotic with a broad spectrum of activity against both gram-positive and gram-negative microorganisms. It has a high rate of efficacy in many types of infection and to date no severe side effects have been noted.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
Penicillin binding protein 2aPenicillin-binding protein 1APenicillin-binding protein 1B +3
Waktu Paruh1.50 &plusmn;0.14 h…
Vol. Distribusi-
Klirens-
Genetik -
Cefminox DB09062
small molecule | CAS: 84305-41-9

Cefminox (INN) is a second generation cephalosporin antibiotic. It is approved for use in Japan.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefodizime DB13470
small molecule | CAS: 69739-16-8

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefonicid Approved DB01328
small molecule | CAS: 61270-58-4

A second-generation cephalosporin administered intravenously or intramuscularly. Its bactericidal action results from inhibition of cell wall synthesis. It is used for urinary tract infections, lower respiratory tract infections, and soft tissue and bone infe…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1APeptidoglycan synthase FtsIPenicillin-binding protein 1B +2
Waktu Paruh4.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Cefoperazone Approved DB01329
small molecule | CAS: 62893-19-0

Cefoperazone is a semisynthetic broad-spectrum cephalosporin proposed to be effective against <i>Pseudomonas</i> infections. It is a third-generation antiobiotic agent and it is used in the treatment of various bacterial infections caused by susceptible organ…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1BPenicillin-binding protein 2 +6
Waktu ParuhThe mean serum half…
Vol. Distribusi-
Klirens-
Genetik -
Ceforanide Approved DB00923
small molecule | CAS: 60925-61-3

Ceforanide is administered parenterally. It has a longer elimination half-life than any currently available cephalosporin. Its activity is very similar to that of cefamandole, another second-generation cephalosporin antibiotic, except that ceforanide is less …

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 2
Waktu Paruh2.6 to 2.98 hours
Vol. Distribusi-
Klirens-
Genetik -
Cefotaxime Approved DB00493
small molecule | CAS: 63527-52-6

Cefotaxime is a third-generation cephalosporin antibiotic. Like other third-generation cephalosporins, it has broad spectrum activity against Gram positive and Gram negative bacteria. In most cases, it is considered to be equivalent to ceftriaxone in terms of…

Kategori:
Agents that reduce seizure thresholdAmidesAnti-Bacterial Agents +13
Target Protein:
Penicillin-binding protein 1bPenicillin-binding protein 2aPenicillin-binding protein 3 +10
Waktu ParuhApproximately 1 hou…
Vol. Distribusi-
Klirens-
Genetik -
Cefotetan Approved DB01330
small molecule | CAS: 69712-56-7

A semisynthetic cephamycin antibiotic that is administered intravenously or intramuscularly. The drug is highly resistant to a broad spectrum of beta-lactamases and is active against a wide range of both aerobic and anaerobic gram-positive and gram-negative m…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
Penicillin-binding protein 3
Waktu ParuhIn volunteers with …
Vol. Distribusi* 10.4 L [elderly p…
Klirens* 1.8 +/- 0.1 L/h […
Genetik -
Cefotiam Approved DB00229
small molecule | CAS: 61622-34-2

One of the cephalosporins that has a broad spectrum of activity against both gram-positive and gram-negative microorganisms.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1A
Waktu ParuhApproximately 1 hou…
Vol. Distribusi-
Klirens-
Genetik -
Cefoxitin Approved DB01331
small molecule | CAS: 35607-66-0

Cefoxitin is a semi-synthetic, broad-spectrum cepha antibiotic for intravenous administration. It is derived from cephamycin C, which is produced by <i>Streptomyces lactamdurans</i>.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
D-alanyl-D-alanine carboxypeptidase DacCD-alanyl-D-alanine carboxypeptidase DacAD-alanyl-D-alanine endopeptidase +9
Waktu ParuhThe half-life after…
Vol. Distribusi-
Klirens-
Genetik -
Cefozopran DB13667
small molecule | CAS: 113359-04-9

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
Dihydropteroate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefpiramide Approved DB00430
small molecule | CAS: 70797-11-4

Cefpiramide is a third-generation cephalosporin antibiotic.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1BPenicillin-binding protein 1A +4
Waktu Paruh4.44 hours
Vol. Distribusi-
Klirens-
Genetik -
Cefpirome Approved DB13682
small molecule | CAS: 84957-29-9

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4101–4150 dari 13591
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