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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 82 / 236
Danazol Approved DB01406
small molecule | CAS: 17230-88-5

A synthetic steroid with antigonadotropic and anti-estrogenic activities that acts as an anterior pituitary suppressant by inhibiting the pituitary output of gonadotropins. It possesses some androgenic properties. Danazol has been used in the treatment of end…

Kategori:
AndrogensAntigonadotropins and Similar AgentsCytochrome P-450 CYP3A Inhibitors +15
Target Protein:
Estrogen receptorAndrogen receptorProgesterone receptor +3
Waktu ParuhApproximately 24 ho…
Vol. Distribusi-
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Genetik -
Danburstotug DB19064
biotech | CAS: 2307144-65-4

Danburstotug is under investigation in clinical trial NCT04809012 (Study of STI-3031 in Patients With Selected Relapsed or Refractory Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
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Danicamtiv DB18962
small molecule | CAS: 1970972-74-7

Danicamtiv is under investigation in clinical trial NCT04572893 (Exploratory Study of Danicamtiv in Patients With Primary Dilated Cardiomyopathy (DCM) Due to Genetic Variants or Other Causalities).

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Danicopan Approved DB15401
small molecule | CAS: 1903768-17-1

Paroxysmal nocturnal hemoglobinuria (PNH) is a rare acquired hematologic disease characterized by hemolysis, thrombophilia, and bone marrow dysfunction.[A263501,L50417] Both hemolysis and thrombophilia are mediated primarily by the complement system.[A263501]…

Kategori:
AminesAmino AcidsAmino Acids, Cyclic +10
Target Protein:
Complement factor D
Waktu ParuhThe mean half-life …
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -
Daniquidone DB12804
small molecule | CAS: 67199-66-0

Daniquidone has been used in trials studying the treatment of Neoplasms.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
DNA topoisomerase 1DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
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Danoprevir DB11779
small molecule | CAS: 850876-88-9

Danoprevir has been used in trials studying the treatment of Hepatitis C, Chronic.

Kategori:
AmidesAmino AcidsAmino Acids, Cyclic +11
Target Protein:
Gag-Pol polyproteinGenome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dansyllysine DB04676
small molecule | CAS: 1101-84-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +1
Target Protein:
Immunoglobulin heavy constant alpha 2
Waktu Paruh-
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Klirens-
Genetik -
Dantrolene Approved DB01219
small molecule | CAS: 7261-97-4

Chemically, dantrolene is a hydantoin derivative, but does not exhibit antiepileptic activity like other hydantoin derivates such as phenytoin.

Kategori:
Agents causing hyperkalemiaAgents that produce neuromuscular block (indirect)Central Nervous System Agents +15
Target Protein:
Ryanodine receptor 1
Waktu ParuhThe mean biologic h…
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Dantron Approved DB04816
small molecule | CAS: 117-10-2

Withdrawn from the Canadian, US, and UK markets in 1998 due to genotoxicity.

Kategori:
Alimentary Tract and MetabolismAnthracenesContact Laxatives +8
Waktu Paruh-
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Danusertib DB11778
small molecule | CAS: 827318-97-8

Danusertib has been used in trials studying the treatment of Leukemia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Aurora kinase CAurora kinase AAurora kinase B
Waktu Paruh-
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Danvatirsen DB14825
biotech | CAS: 1402357-06-5

Danvatirsen is under investigation in clinical trial NCT03334617 (Phase II Umbrella Study of Novel Anti-cancer Agents in Patients With NSCLC Who Progressed on an Anti-PD-1/PD-L1 Containing Therapy.).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
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Dapaconazole DB11985
small molecule | CAS: 1269726-67-1

Dapaconazole has been used in trials studying the treatment of Tinea Pedis.

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Dapagliflozin Approved DB06292
small molecule | CAS: 461432-26-8

Dapagliflozin is a sodium-glucose cotransporter 2 (SGLT2) inhibitor, and it was the first SLGT2 inhibitor to be approved. indicated for managing diabetes mellitus type 2.[A261596] When combined with diet and exercise in adults, dapagliflozin helps to improve …

Kategori:
Alimentary Tract and MetabolismBenzene DerivativesBlood Glucose Lowering Agents +19
Target Protein:
Sodium/glucose cotransporter 2
Waktu ParuhThe mean plasma ter…
Vol. DistribusiThe volume of distr…
KlirensOral plasma clearan…
Genetik -
Dapansutrile DB16130
small molecule | CAS: 54863-37-5

Dapansutrile is under investigation in clinical trial NCT01768975 (Phase 2 Efficacy Trial of OLT1177 Gel in Subjects With Moderate to Severe Pain Associated With OA of the Knee).

Kategori:
Anti-Inflammatory AgentsSulfur Compounds
Target Protein:
NACHT, LRR and PYD domains-containing protein 3
Waktu Paruh-
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Daphnetin DB18965
small molecule | CAS: 486-35-1

Daphnetin is under investigation in clinical trial NCT06329167 (Daphnetin Capsules for Lower Limb Lymphoedema Following Gynaecological Surgery).

Kategori:
BenzopyransCoumarinsHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
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Dapiclermin DB17979
biotech | CAS: 444069-80-1

Dapiclermin is a recombinant ciliary neurotrophic factor.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +4
Waktu Paruh-
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Dapiglutide DB19182
biotech | CAS: 2296814-85-0

Dapiglutide is under investigation in clinical trial NCT05788601 (Dapiglutide for the Treatment of Obesity).

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Dapiprazole Approved DB00298
small molecule | CAS: 72822-12-9

Dapiprazole (U.S. trade name Rev-Eyes) is an alpha blocker. It is found in ophthalmic solutions used to reverse mydriasis after an eye examination.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +12
Target Protein:
D(2) dopamine receptorAlpha-1A adrenergic receptorAlpha-1D adrenergic receptor +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 1416147-64-2

Dapirolizumab pegol is under investigation in clinical trial NCT02804763 (A Phase 2 Efficacy and Safety Study of Dapirolizumab Pegol (DZP) in Systemic Lupus Erythematosus).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsAntibodies, Monoclonal +14
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Dapivirine DB08639
small molecule | CAS: 244767-67-7

Dapivirine has been investigated for the prevention of HIV-1 Infections and Topical Penile Exposures.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +4
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
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Daplusiran DB19331
biotech | CAS: 2202783-35-3

Daplusiran is under investigation in clinical trial NCT06537414 (A Study of Sequential Therapy With Daplusiran/tomligisiran (DAP/TOM) Followed by Bepirovirsen in Participants Living With Chronic Hepatitis B (CHB)).

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Daporinad DB12731
small molecule | CAS: 658084-64-1

Daporinad has been used in trials studying the treatment of Melanoma, Cutaneous T-cell Lymphoma, and B-cell Chronic Lymphocytic Leukemia.

Kategori:
Acids, AcyclicAcrylatesAmides
Target Protein:
Nicotinamide phosphoribosyltransferase
Waktu Paruh-
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Dapoxetine DB04884
small molecule | CAS: 119356-77-3

Dapoxetine is a selective serotonin reuptake inhibitor, for the treatment of premature ejaculation. In a phase II proof-of-concept study conducted by PPD, dapoxetine demonstrated a statistically significant increase in ejaculatory latency when compared to pla…

Kategori:
AminesAntidepressive AgentsBenzene Derivatives +17
Target Protein:
5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 2C
Waktu ParuhInitial half-life o…
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Daprodustat Approved DB11682
small molecule | CAS: 960539-70-2

Daprodustat is a small-molecule hypoxia-inducible factor (HIF) prolyl hydroxylase (PHD) inhibitor that was developed by GSK.[A254167,A254162] Patients with CKD cannot induce erythropoietin (EPO) production in response to hypoxia or anemia. As a potent inhibit…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntianemic Preparations +17
Target Protein:
Egl nine homolog 1Prolyl hydroxylase EGLN2Prolyl hydroxylase EGLN3
Waktu ParuhThe terminal elimin…
Vol. DistribusiDaprodustat has an …
KlirensMean clearance from…
Genetik -
Dapsone Approved DB00250
small molecule | CAS: 80-08-0

A sulfone active against a wide range of bacteria but mainly employed for its actions against mycobacterium leprae. Its mechanism of action is probably similar to that of the sulfonamides which involves inhibition of folic acid synthesis in susceptible organi…

Kategori:
Anti-Acne PreparationsAnti-Acne Preparations for Topical UseAnti-Bacterial Agents +32
Target Protein:
Inactive dihydropteroate synthase 2Dihydropteroate synthase
Waktu Paruh28 hours (range 10-…
Vol. Distribusi-
Klirens-
Genetik -
Daptomycin Approved DB00080
small molecule | CAS: 103060-53-3

Daptomycin is a cyclic lipopeptide antibacterial agent with a broad spectrum of activity against Gram-positive bacteria, including methicillin-susceptible and -resistant _Staphylococcus aureus_ (MSSA/MRSA) and vancomycin-resistant Enterococci (VRE).[A231379, …

Kategori:
Agents Causing Muscle ToxicityAmino Acids, Peptides, and ProteinsAnti-Bacterial Agents +11
Target Protein:
Dihydropteroate synthaseCytoplasmic membrane
Waktu ParuhDaptomycin has a re…
Vol. DistribusiDaptomycin has a ve…
KlirensDaptomycin administ…
Genetik -
DAR-0100A DB16139
small molecule | CAS: 174691-84-0

DAR-0100A is under investigation in clinical trial NCT01466205 (Clinical Testing of a D1 Agonist for Cognitive Enhancement in Schizotypal Personality Disorder).

Kategori:
Dopamine AgentsDopamine AgonistsDopamine D1 Receptor Agonists +2
Waktu Paruh-
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Darapladib DB06311
small molecule | CAS: 356057-34-6

Deskripsi belum tersedia.

Kategori:
AminesAnionsBenzene Derivatives +9
Target Protein:
Phospholipase A2Cytosolic phospholipase A2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Daratumumab Approved DB09331
biotech | CAS: 945721-28-8

Daratumumab is an immunoglobulin G1 kappa monoclonal antibody developed by Janssen and Genmab.[A7935] It was first described in the literature in 2010 as a monoclonal antibody that targets CD38+ multiple myeloma cells; the first of its kind.[A199002] Darat…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
Waktu ParuhIntravenous daratum…
Vol. DistribusiDaratumumab intrave…
KlirensIntravenous daratum…
Genetik -
Darbepoetin alfa Approved DB00012
biotech | CAS: 209810-58-2

Human erythropoietin with 2 aa substitutions to enhance glycosylation (5 N-linked chains), 165 residues (MW=37 kD). Produced in Chinese hamster ovary (CHO) cells by recombinant DNA technology.

Kategori:
Amino Acids, Peptides, and ProteinsAntianemic PreparationsBlood and Blood Forming Organs +10
Target Protein:
Erythropoietin receptor
Waktu Paruh-
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Daridorexant Approved DB15031
small molecule | CAS: 1505484-82-1

Daridorexant, formerly known as nemorexant, is a selective dual orexin receptor antagonist used to treat insomnia. Insomnia is characterized by difficulties with sleep onset and/or sleep maintenance and impairment of daytime functioning. It chronically affect…

Kategori:
Central Nervous System DepressantsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +6
Target Protein:
Orexin/Hypocretin receptor type 1Orexin receptor type 2
Waktu ParuhThe terminal half-l…
Vol. DistribusiDaridorexant has a …
KlirensThere is limited in…
Genetik -
Darigabat DB18966
small molecule | CAS: 1614245-70-3

Darigabat is under investigation in clinical trial NCT05941442 (A Study to Evaluate Efficacy, Safety, and Tolerability of Darigabat in Participants With Panic Disorder).

Kategori:
GABA AgentsGABA ModulatorsNeurotransmitter Agents
Waktu Paruh-
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Darinaparsin DB06179
small molecule | CAS: 69819-86-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Waktu Paruh-
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Klirens-
Genetik -
Darleukin DB17157
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Darodipine DB09234
small molecule | CAS: 72803-02-2

Darodipine is a calcium channel blocker.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +10
Waktu Paruh-
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Darolutamide Approved DB12941
small molecule | CAS: 1297538-32-9

Darolutamide is a nonsteroidal androgen receptor antagonist for the treatment of castrate-resistant, non-metastatic prostate cancer (nmCRPC). This condition occurs in the majority of patients with advanced prostate cancer who have been treated with androgen r…

Kategori:
Androgen Receptor InhibitorsAntiandrogensAntiandrogens, non-steroidal +14
Target Protein:
Androgen receptorProgesterone receptor
Waktu ParuhThe half-life of da…
Vol. DistribusiAfter intravenous a…
KlirensThe clearance of da…
Genetik -
Darovasertib DB16059
small molecule | CAS: 1874276-76-2

IDE-196 is under investigation in clinical trial NCT03947385 (Study of IDE196 in Patients With Solid Tumors Harboring GNAQ/11 Mutations or PRKC Fusions).

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Darunavir Approved DB01264
small molecule | CAS: 206361-99-1

Darunavir is a protease inhibitor used with other HIV protease inhibitor drugs as well as [ritonavir] for the effective management of HIV-1 infection.[L9227] As a second-generation protease inhibitor, darunavir is designed to combat resistance to standard HIV…

Kategori:
AmidesAnti-HIV AgentsAnti-Infective Agents +33
Target Protein:
Pol polyproteinGag-Pol polyprotein
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensDarunavir has a low…
Genetik -
Darusentan DB04883
small molecule | CAS: 171714-84-4

Darusentan is a selective endothelin ETA receptor antagonist. It is being evaluated as a treatment for congestive heart failure and hypertension.

Kategori:
Acids, CarbocyclicEndothelin Receptor Antagonists
Target Protein:
Endothelin-1 receptor
Waktu Paruh-
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Darvadstrocel Approved DB16581
biotech

Darvadstrocel is a suspension of expanded human allogeneic adipose-derived mesenchymal stem cells extracted from the subdermal adipose tissue of healthy donors via liposuction.[A244524] Darvadstrocel was first approved by the European Commission on March 23, …

Kategori:
Antineoplastic and Immunomodulating AgentsImmunomodulatory AgentsImmunosuppressive Agents +1
Waktu ParuhPharmacokinetic inf…
Vol. DistribusiIn preclinical tria…
KlirensPharmacokinetic inf…
Genetik -
DAS-181 DB15313
biotech | CAS: 946032-08-2

DAS-181 is under investigation in clinical trial NCT00527865 (Single Dose Escalating Study of DAS181 in Adults).

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
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Dasabuvir Approved DB09183
small molecule | CAS: 1132935-63-7

Dasabuvir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine …

Kategori:
AmidesAminesAntiinfectives for Systemic Use +20
Target Protein:
Genome polyproteinNonstructural protein 5b
Waktu ParuhThe half-life of el…
Vol. DistribusiDasabuvir has a vol…
KlirensClearance of Dasabu…
Genetik -
Dasatinib Approved DB01254
small molecule | CAS: 302962-49-8

Dasatinib is an orally available multikinase inhibitor indicated for the treatment of Philadelphia chromosome (Ph)-positive leukemias.[A2224,L45171] Ph is a chromosomal abnormality found in patients with chronic myelogenous leukemia (CML) and acute lymphocyti…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBcr-Abl Tyrosine Kinase Inhibitors +31
Target Protein:
Tyrosine-protein kinase ABL1Proto-oncogene tyrosine-protein kinase SrcEphrin type-A receptor 2 +20
Waktu ParuhThe terminal half-l…
Vol. DistribusiDasatinib has an ap…
KlirensThe clearance of da…
Genetik -
Dasiglucagon Approved DB15226
biotech | CAS: 1544300-84-6

Dasiglucagon is a glucagon analog that acts to increase blood sugar levels.[L39190] It consists of 29 amino acids similar to endogenous glucagon; however, it contains seven substituted amino acids for improved physical and chemical stability in its drug formu…

Kategori:
Amino Acids, Peptides, and ProteinsAntihypertensive AgentsAntihypoglycemic Agent +10
Target Protein:
Glucagon receptor
Waktu ParuhThe half-life was a…
Vol. DistribusiThe mean apparent v…
Klirens-
Genetik -
Dasiprotimut-T DB17287
biotech

Dasiprotimut-T is a personalized therapeutic vaccine against B-cell lymphomas.[A254701] It has been investigated in clinical trials.

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating Agents
Waktu Paruh-
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Dasotraline DB12305
small molecule | CAS: 675126-05-3

Dasotraline is a serotonin, norepinephrine and dopamine reuptake inhibitor (SNDRI) that is under investigation for the treatment of Binge Eating Disorder, Adult Attention Hyperactivity Disorder, Attention Deficit Hyperactivity Disorder, and Adult Attention De…

Kategori:
AminesCycloparaffinsNaphthalenes
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
Waktu Paruh-
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dATP DB03222
small molecule | CAS: 1927-31-7

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesDeoxyribonucleotidesHeterocyclic Compounds, Fused-Ring +4
Target Protein:
P2Y purinoceptor 11Anaerobic ribonucleoside-triphosphate reductaseProtein RecA +4
Waktu Paruh-
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Daunorubicin Approved DB00694
small molecule | CAS: 20830-81-3

A very toxic anthracycline aminoglycoside antineoplastic isolated from Streptomyces peucetius and others, used in treatment of leukemia and other neoplasms.

Kategori:
Anthracycline Topoisomerase InhibitorAnthracyclinesAnthracyclines and Related Substances +30
Target Protein:
DNADNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Gen Terkait:
CYP1B1 HNRNPD SEC14L3 +4
Waktu ParuhDaunorubicin has be…
Vol. DistribusiDaunorubicin has a …
KlirensDaunorubicin has a …
Genetik 7 Varian
Davalintide DB14956
biotech | CAS: 863919-85-1

Davalintide is under investigation in clinical trial NCT00785408 (Study to Examine Safety, Tolerability and Effect on Body Weight of Subcutaneous AC2307 in Obese or Overweight Subjects).

Kategori:
Amino Acids, Peptides, and Proteins
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Davanat DB15311
small molecule | CAS: 916851-14-4

Davanat is under investigation in clinical trial NCT00054977 (Safety of GM-CT-01 With and Without 5-Fluorouracil in Patients With Solid Tumors).

Kategori:
CarbohydratesHexosesMonosaccharides +1
Waktu Paruh-
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