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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 82 / 272
Cardarine DB05416
small molecule | CAS: 317318-70-0

Cardarine (GW-501516) is a peroxisome proliferator-activator receptor-delta agonist for the potential treatment of dyslipidemia. Cardarine has been investigated for the treatment of Obesity, Lipid Disorders, and Cardiovascular Disease.

Kategori:
Sulfur Compounds
Target Protein:
Peroxisome proliferator-activated receptor deltaPeroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cardiopet DB18913
small molecule | CAS: 855927-17-2

Cardiopet is under investigation in clinical trial NCT01826773 (Cardiopet as PET Imaging Agent to Assess Myocardial Perfusion and Fatty Acid Uptake in Known or Suspected CAD Subjects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cardiotrophin 1 DB18399
biotech | CAS: 1422101-11-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carfecillin DB13506
small molecule | CAS: 27025-49-6

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carfentanil DB01535
small molecule | CAS: 59708-52-0

Carfentanil or carfentanyl (Wildnil) is an analogue of the popular synthetic opioid analgesic fentanyl, and is one of the most potent opioids known (also the most potent opioid used commercially). Carfentanil was first synthesized in 1974 by a team of chemist…

Kategori:
AnalgesicsCarbon RadioisotopesCentral Nervous System Agents +9
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 98598-83-5

Carfentanil, C-11 is under investigation in clinical trial NCT01899170 (Towards Individualized Deep Brain Stimulation Treatment of Chronic Neuropathic Pain).

Kategori:
AnalgesicsCarbon RadioisotopesCentral Nervous System Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carfilzomib Approved DB08889
small molecule | CAS: 868540-17-4

Carfilzomib is an injectable antineoplastic agent (IV only). Chemically, it is a modified tetrapeptidyl epoxide and an analog of epoxomicin. It is also a selective proteasome inhibitor. FDA approved carfilzomib in July 2012 for the treatment of adults with re…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +8
Target Protein:
Proteasome subunit beta type-5Proteasome subunit beta type-8Proteasome subunit beta type-1 +3
Waktu ParuhFollowing intraveno…
Vol. DistribusiVd, steady state, 2…
KlirensSystemic clearance …
Genetik -
Carglumic acid Approved DB06775
small molecule | CAS: 1188-38-1

Carglumic acid is a drug used for the treatment of hyperammonemia in patients with a deficiency in N-acetyl glutamate synthase. This rare genetic disorder results in elevated blood levels of ammonia, which can eventually cross the blood–brain barrier and caus…

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids and Derivatives +6
Target Protein:
Carbamoyl-phosphate synthase [ammonia], mitochondrial
Waktu ParuhMedian values for t…
Vol. DistribusiThe apparent volume…
KlirensThe apparent total …
Genetik -
Caricotamide DB18950
small molecule | CAS: 64881-21-6

Caricotamide is under investigation in clinical trial NCT00746590 (Study of Anti-tumour Effects and Safety of Prolarix™ in Hepatocellular Carcinoma).

Target Protein:
Ribosyldihydronicotinamide dehydrogenase [quinone]
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carindacillin Approved DB09319
small molecule | CAS: 35531-88-5

Carindacillin or Carbenicillin isdanyl was an oral penicillin prodrug of [carbenicillin] marketed by Pfizer as Geocillin. It is no longer marketed in the United States.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cariporide DB06468
small molecule | CAS: 159138-80-4

Deskripsi belum tersedia.

Kategori:
AmidinesAntiarrhythmic agentsCardiovascular Agents +3
Target Protein:
Sodium/hydrogen exchanger 1Sodium/hydrogen exchanger 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cariprazine Approved DB06016
small molecule | CAS: 839712-12-8

Cariprazine is an atypical antipsychotic agent and a piperazine derivative that was first developed in Hungary.[A247100] It works as a partial agonist at central dopamine D2, dopamine D3, and serotonin 5-HT<sub>1A</sub> receptors and as an antagonist at serot…

Kategori:
Agents that produce hypertensionAntidepressive AgentsAntipsychotic Agents +48
Target Protein:
D(3) dopamine receptorD(2) dopamine receptor5-hydroxytryptamine receptor 1A +5
Waktu ParuhCariprazine and its…
Vol. Distribusi-
Klirens-
Genetik -
Carisbamate DB12338
small molecule | CAS: 194085-75-1

Carisbamate has been investigated in Alcohol Abuse, Substance Abuse, and Alcohol Dependence.

Kategori:
Acids, AcyclicAnticonvulsantsCentral Nervous System Depressants +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carisoprodol Approved DB00395
small molecule | CAS: 78-44-4

Originally approved by the FDA in 1959 [FDA label], carisoprodol is a centrally acting muscle relaxant used in painful musculoskeletal conditions in conjunction with physical therapy and other medications [A176047]. This drug is available by itself in an ora…

Kategori:
CarbamatesCarbamic Acid EstersCentral Nervous System Agents +7
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit gamma-2 +2
Waktu ParuhThe terminal half-l…
Vol. Distribusi0.93 to 1.3 L/kg, a…
KlirensFollowing an oral d…
Genetik -
Carlumab DB12718
biotech | CAS: 915404-94-3

Carlumab has been used in trials studying the treatment of Cancer and Prostate Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carmegliptin DB12268
small molecule | CAS: 813452-18-5

Carmegliptin has been used in trials studying the treatment of Diabetes Mellitus Type 2.

Kategori:
Agents causing angioedemaBlood Glucose Lowering AgentsDipeptidyl Peptidase 4 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carmustine Approved DB00262
small molecule | CAS: 154-93-8

A cell-cycle phase nonspecific alkylating antineoplastic agent. It is used in the treatment of brain tumors and various other malignant neoplasms. (From Martindale, The Extra Pharmacopoeia, 30th ed, p462) This substance may reasonably be anticipated to be a c…

Kategori:
Alkylating ActivityAlkylating DrugsAmides +15
Target Protein:
RNAGlutathione reductase, mitochondrialDNA
Waktu Paruh15-30 minutes
Vol. Distribusi-
Klirens-
Genetik -
Carnosine DB11695
small molecule | CAS: 305-84-0

Carnosine has been investigated for the treatment of Gulf War Illness.

Kategori:
Amino Acids, Peptides, and ProteinsDipeptidesNerve Tissue Proteins +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 401905-67-7

Carotegrast methyl is under investigation in clinical trial NCT03531892 (A Study to Evaluate the Safety and Efficacy of AJM300 in Participants With Active Ulcerative Colitis).

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carotuximab DB06322
biotech | CAS: 1268714-50-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Endoglin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Caroverine DB13835
small molecule | CAS: 23465-76-1

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAlimentary Tract and MetabolismAntiarrhythmic agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Caroxazone DB09254
small molecule | CAS: 18464-39-6

Caroxazone is an antidepressant that has been withdrawn from the market. It is a reversible monoamine oxidase inhibitor (MAOI) of both A and B monoamine oxidase subtypes. However, it presents a five-fold preference for the MAO-B subtype.

Kategori:
AcetamidesAgents that produce hypertensionAgents that reduce seizure threshold +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carphenazine DB01038
small molecule | CAS: 2622-30-2

Carphenazine is an antipsychotic drug, used in hospitalized patients in the management of chronic schizophrenic psychoses.

Kategori:
Dopamine AntagonistsDopamine D2 Receptor Antagonists
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptorD(1B) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carprofen Approved DB00821
small molecule | CAS: 53716-49-7

Carprofen is a non-steroidal anti-inflammatory drug (NSAID) that is used by veterinarians as a supportive treatment for the relief of arthritic symptoms in geriatric dogs. Carprofen was previously used in human medicine for over 10 years (1985-1995). It was g…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +15
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhApproximately 8 hou…
Vol. Distribusi-
Klirens-
Genetik -
Carpropamide DB02946
small molecule | CAS: 127640-90-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carumonam DB13553
small molecule | CAS: 87638-04-8

Deskripsi belum tersedia.

Kategori:
AmidesAntibacterials for Systemic UseAntiinfectives for Systemic Use +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carvedilol Approved DB01136
small molecule | CAS: 72956-09-3

Carvedilol is a racemic mixture where the S(-) enantiomer is both a beta and alpha-1 adrenoceptor blocker, and the R(+) enantiomer is an alpha-1 adrenoceptor blocker.[L7889,L7892] It is currently used to treat heart failure, left ventricular dysfunction, and …

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +40
Target Protein:
Beta-1 adrenergic receptorAlpha-1A adrenergic receptorAlpha-1 adrenergic receptors +16
Gen Terkait:
ADRB1
Waktu ParuhThe half life of ca…
Vol. DistribusiCarvedilol has a vo…
KlirensThe plasma clearanc…
Genetik 1 Varian
Carya glabra pollen Approved DB10883
biotech

Carya glabra pollen is the pollen of the Carya glabra plant. Carya glabra pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carya illinoinensis pollen Approved DB10380
biotech

Carya illinoinensis pollen allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carya ovata pollen Approved DB10364
biotech

Carya ovata pollen is the pollen of the Carya ovata plant. Carya ovata pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Caryophyllene DB16854
small molecule | CAS: 87-44-5

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +6
Target Protein:
Cannabinoid receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Casdozokitug DB17513
biotech | CAS: 2643331-37-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cashew Approved DB10653
biotech

Cashew allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Casimersen Approved DB14984
biotech | CAS: 1422958-19-7

Duchenne muscular dystrophy (DMD) is an X-linked recessive allelic disorder characterized by a lack of functional dystrophin protein, which leads to progressive impairment of ambulatory, pulmonary, and cardiac function and is invariably fatal. A related, albe…

Kategori:
Antisense OligonucleotidesCytochrome P-450 CYP2C19 InhibitorsCytochrome P-450 CYP2C19 inhibitors (strength unknown) +16
Target Protein:
DMD gene (exon 45 casimersen target site)
Waktu ParuhCasimersen has an e…
Vol. DistribusiCasimersen administ…
KlirensCasimersen administ…
Genetik -
Casimiroin DB08744
small molecule | CAS: 477-89-4

Casimiroin is a quinone reductase 2 inhibitor isolated from _Casimiroa edulis_.

Kategori:
AromataseDioxolesHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Ribosyldihydronicotinamide dehydrogenase [quinone]
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Casirivimab Approved DB15941
biotech | CAS: 2415933-42-3

Casirivimab is a monoclonal antibody combined with [Imdevimab] in Regeneron's antibody cocktail known as REGN-COV2 for the treatment of COVID-19.[L23539] This drug is a combination of antibodies derived from humanized VelocImmune® mice in addition to blood s…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Spike glycoprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Casopitant DB06634
small molecule | CAS: 414910-27-3

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAmidesAntiemetics +7
Target Protein:
Substance-P receptorCytochrome P450 3A4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Caspofungin Approved DB00520
small molecule | CAS: 162808-62-0

Caspofungin (brand name Cancidas worldwide) is an antifungal drug and the first member of a new drug class called the echinocandins, as coined by Merck & Co., Inc. It is typically administered intravenously. It shows activity against infections with Aspergill…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntifungal Agents +18
Target Protein:
1,3-beta-glucan synthase component FKS11,3-beta-glucan synthase component GSC2
Waktu Paruh9-11 hours
Vol. Distribusi-
Klirens* 12 mL/min [After …
Genetik -
Castanospermine DB01816
small molecule | CAS: 79831-76-8

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +10
Target Protein:
Glucan 1,3-beta-glucosidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Castor oil Approved DB11113
biotech | CAS: 8001-79-4

Castor oil is a vegetable oil obtained by pressing the seeds of the castor oil plant (_Ricinus communis_ L.) mainly cultivated in India, South America, Africa, and China. Castor oil is a rich source of [DB02955], which represents up to 90% of the total castor…

Kategori:
Alimentary Tract and MetabolismBiological ProductsComplex Mixtures +10
Target Protein:
Prostaglandin E2 receptor EP3 subtypeProstaglandin E2 receptor EP4 subtype
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Cat dander extract Approved DB13904
biotech

Cat dander extract is either subcutaneously or intracutaneously administered and contains dry cat dander or dry defatted cat pelt. It is used in the diagnosis and treatment (immunotherapy) of patients with a history of allergy to cats. An allergic reaction to…

Kategori:
Allergenic Extracts
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cathine DB01486
small molecule | CAS: 492-39-7

Cathine, also known as d-norpseudoephedrine and (+)-norpseudoephedrine, is a psychoactive drug with stimulant properties. It belongs to the phenethylamine and amphetamine chemical classes. In the United States, it is classified as a Schedule IV controlled sub…

Kategori:
AlcoholsAlimentary Tract and MetabolismAmines +7
Waktu Paruh5.2 +/- 3.4 hours
Vol. Distribusi-
Klirens-
Genetik -
Cathinone DB01560
small molecule | CAS: 71031-15-7

Cathinone is a monoamine alkaloid found in the shrub Catha edulis (Khat). Closely related to ephedrine, cathine and other amphetamines, it is probably the main contributor to the stimulant effect of Catha edulis. Cathinone differs from many other amphetamines…

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCentral Nervous System Stimulants +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Catridecacog Approved DB09310
biotech | CAS: 606138-08-3

Coagulation Factor XIII A-Subunit (Recombinant), also known as catridecacog, is a recombinant form of the Factor XIII-A2 homodimer composed of two factor XIII (FXIII) A-subunits [FDA Label]. For people with congenital deficiency or mutation of Factor XIII, a …

Kategori:
Blood and Blood Forming OrgansBlood Coagulation FactorsHemostatics
Target Protein:
Coagulation factor XIII B chain
Waktu Paruh7.1 days
Vol. Distribusi-
Klirens0.41 mL/h/kg
Genetik -
Cauliflower Approved DB10643
biotech

Cauliflower allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cavosonstat DB14775
small molecule | CAS: 1371587-51-7

Cavosonstat is under investigation in clinical trial NCT02589236 (Study of Cavosonstat (N91115) in Patients With CF Homozygous for the F508del-CFTR Mutation).

Kategori:
Benzene Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cavrotolimod DB18216
small molecule | CAS: 2378664-12-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CB-103 DB15279
small molecule | CAS: 218457-67-1

CB-103 is under investigation in clinical trial NCT03422679 (Study of CB-103 in Adult Patients With Advanced or Metastatic Solid Tumours and Haematological Malignancies).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CB-1158 DB15286
small molecule | CAS: 2095732-06-0

CB-1158 is under investigation in clinical trial NCT03910530 (A Study of INCMGA00012, INCB001158, and the Combination in Japanese Participants With Advanced Solid Tumors).

Kategori:
Enzyme Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CB-5083 DB16874
small molecule | CAS: 1542705-92-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Transitional endoplasmic reticulum ATPase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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