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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Halaman 81 / 252
Clotiazepam Approved DB01559
small molecule | CAS: 33671-46-4

Clotiazepam is a thienodiazepine, not approved for sale in the U.S. or Canada, but has been approved in the U.K. It is a schedule IV drug in Canada.

Kategori:
Anti-Anxiety AgentsBenzodiazepines and benzodiazepine derivativesCentral Nervous System Depressants +8
Target Protein:
GABA(A) ReceptorTranslocator proteinGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh4 hours
Vol. Distribusi-
Klirens-
Genetik -
Clotrimazole Approved DB00257
small molecule | CAS: 23593-75-1

This drug is a broad spectrum antimycotic or antifungal agent. Clotrimazole's antimycotic properties were discovered in the late 1960s [A174094]. Clotrimazole falls under the _imidazole_ category of _azole_ antifungals, possessing broad-spectrum antimycotic a…

Kategori:
Anti-Infective AgentsAnti-Infective Agents, LocalAntifungal Agents +54
Target Protein:
C-X-C chemokine receptor type 2Lanosterol 14-alpha demethylaseIntermediate conductance calcium-activated potassium channel protein 4 +3
Waktu Paruh-
Vol. DistribusiThe topical form is…
Klirens-
Genetik -
Clove Approved DB10672
biotech | CAS: 84961-50-2

Clove allergenic extract is used in allergenic testing.

Kategori:
AngiospermsBiological ProductsCell-mediated Immunity +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cloxacillin Approved DB01147
small molecule | CAS: 61-72-3

A semi-synthetic penicillin antibiotic which is a chlorinated derivative of [oxacillin].

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
D-alanyl-D-alanine carboxypeptidase DacAPenicillin-binding protein 2XPenicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cloxazolam DB01553
small molecule | CAS: 24166-13-0

Cloxazolam is a benzodiazepine with anxiolytic, sedative/hypnotic, muscle relaxant, and antiepileptic effects. It is marketed in the Argentina, Australia, Portugal, Belgium, Switzerland, Luxembourg, Germany, Taiwan and Japan -- mainly for anti-anxiety. The us…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +4
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh65 hours
Vol. Distribusi-
Klirens-
Genetik -
Cloxyquin DB15933
small molecule | CAS: 130-16-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingHydroxyquinolinesQuinolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clozapine Approved DB00363
small molecule | CAS: 5786-21-0

Clozapine is a tricyclic dibenzodiazepine, classified as an atypical antipsychotic agent.[A256708] Clozapine displays affinity to various neuroreceptors with a particularly low affinity to the dopamine receptors, thus breaking the mold of first-generation ant…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +65
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2AD(1A) dopamine receptor +30
Gen Terkait:
GNB3
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe median volume o…
KlirensThe median clearanc…
Genetik 1 Varian
CLX-0921 DB05854
small molecule

CLX-0921 is investigated for use/treatment in diabetes mellitus type 2. CLX-0921 is a solid. CLX-0921 has a spectrum of activity that differs from commercially available thiazolidinediones. This substance targets the protein peroxisome proliferator-activated …

Kategori:
Sulfur Compounds
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CM-4307 DB15414
small molecule | CAS: 1130115-44-4

CM-4307 is under investigation in clinical trial NCT03602495 (Donafenib in 131I-Refractory Differentiated Thyroid Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CM4620 DB16466
small molecule | CAS: 1713240-67-5

CM4620 (Zegocractin), is under investigation in multiple clinical trials, including NCT04195347 (pancreatitis due to asparaginase), NCT03709342 (PK/PD study in acute pancreatitis), NCT03401190 and NCT04681066 (pancreatitis and SIRS), and NCT04661540 (critical…

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CMC 001 DB05353
small molecule

CMC 001 is an orally administered MRI contrast agent in development for enhancement of the liver, bile ducts and gastrointestinal tract.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CMLVAX100 DB05164
biotech

CMLVAX100 is a vaccine targeting the BCR-ABL-derived p210 fusion protein which reduces residual disease in some patients with chronic myeloid leukemia. It is developed by Breakthrough Therapeutics and has completed phase I of its clinical trial.

Target Protein:
BCR/ABL p210 fusion protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CMX-2043 DB12795
small molecule | CAS: 910627-26-8

CMX-2043 has been used in trials studying the treatment and prevention of Non STEMI, Unstable Angina, Stable Coronary Artery Disease, and Percutaneous Coronary Intervention.

Kategori:
Amino Acids, Peptides, and ProteinsCoenzymesEnzymes and Coenzymes +6
Target Protein:
RAC-alpha serine/threonine-protein kinaseHepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CN-105 DB18345
small molecule | CAS: 1632243-07-2

CN-105 is a neuroprotective pentapeptide with the sequence Acetyl-Valine-Serine-Arginine-Arginine-Arginine-NH2 (Ac-VSRRR- NH2).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CNM-Au8 DB17952
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CNS-5161 DB05824
small molecule

CNS 5161 is a blocker of the NMDA ion channel and has completed Phase IIa proof of concept clinical trials as a novel compound for the treatment of neuropathic pain.

Target Protein:
Glutamate receptor ionotropic, NMDA 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CNV-2197944 DB15229
small molecule | CAS: 1204535-44-3

CNV-2197944 is under investigation in clinical trial NCT01893125 (Efficacy and Safety of CNV2197944 Versus Placebo in Patients With Diabetic Peripheral Neuropathy).

Target Protein:
Voltage-dependent N-type calcium channel subunit alpha-1B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serotonin N-acetyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 181054-95-5

Recombinant Coagulation Factor IX is a purified Factor IX glycoprotein produced by recombinant DNA technology. It has a primary amino acid sequence that is identical to the Ala148 allelic form of human factor IX, and has structural and functional characterist…

Kategori:
Blood Coagulation FactorsHemostaticsIncreased Coagulation Activity
Target Protein:
Coagulation factor XCoagulation factor XICoagulation factor VII +4
Waktu Paruh18.8 ± 5.4 hours
Vol. Distribusi-
Klirens8.62 ± 1.7
Genetik -
Coagulation Factor IX Human Approved DB13152
biotech | CAS: 181054-95-5

Factor IX (or Christmas factor) is one of the serine proteases of the coagulation system; it belongs to peptidase family S1. Deficiency of this protein causes hemophilia B.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +9
Target Protein:
Coagulation factor XCoagulation factor XICoagulation factor VII +4
Waktu Paruh18.8 ± 5.4 hours.
Vol. Distribusi-
Klirens8.62 ± 1.7.
Genetik -
Coagulation factor VII human Approved DB13150
biotech

Coagulation factor VII is human serine protease type enzyme that is involved in the extrinsic coagulation cascade which results in blood clotting.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +8
Target Protein:
Tissue factorCoagulation factor XCoagulation factor IX
Waktu Paruh5 h
Vol. Distribusi45 ml/kg
Klirens7.4 ml/kgh
Genetik -
Coagulation factor X human Approved DB13148
biotech

Coagulation Factor X (Human), is a plasma-derived human blood coagulation factor is used by adults and children (aged 12 years and above) with hereditary Factor X deficiency. However its use is limited in the perioperative setting for the management of bleedi…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +11
Waktu ParuhFollowing a single …
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
biotech | CAS: 9013-55-2

Coagulation factor XIa is under investigation in clinical trial NCT01701947 (HEMOLEVEN® Expanded Access Program Prevention of Surgical/Postpartum Hemorrhage Severe Inherited Factor XI Deficiency).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coagulin-B DB17703
biotech

Coagulin-B is an adeno-associated viral vector expressing human blood-coagulation Factor IX.[A259038, A259043] It was previously investigated for the treatment of hemophilia; however, the manufacturing company discontinued the Phase I trial in 2004, halting i…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coal tar Approved DB11082
small molecule | CAS: 8007-45-2

Coal tar is a brown or black liquid of extremely high viscosity. Coal tar is among the by-products when coal is carbonized to make coke or gasified to make coal gas. Coal tars are complex and variable mixtures of phenols, polycyclic aromatic hydrocarbons (PAH…

Kategori:
Complex MixturesDermatologicalsKeratolytic Agents +2
Waktu ParuhIntended for local …
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
Cobalt Approved DB14574
small molecule | CAS: 7440-48-4

A trace element that is a component of vitamin B12. It has the atomic symbol Co, atomic number 27, and atomic weight 58.93. It is used in nuclear weapons, alloys, and pigments. Deficiency in animals leads to anemia; its excess in humans can lead to erythrocyt…

Kategori:
Cell-mediated ImmunityDiet, Food, and NutritionElements +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobalt Co-60 DB15374
small molecule | CAS: 10198-40-0

Cobalt Co-60 is under investigation in clinical trial NCT02891083 (Adjuvant Therapies or Surgery Alone for High Risk pN0 Esophageal Cancer).

Kategori:
Cobalt IsotopesElementsIsotopes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Outer membrane protein TolCChorismate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 22541-53-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 10124-43-3

Deskripsi belum tersedia.

Kategori:
ElementsMetalsMetals, Heavy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobamamide DB11191
small molecule | CAS: 13870-90-1

Cobamamide is one of the active forms of vitamin B12 that is also known as _adenosylcobalamin_ or _dibencozide_. This drug is available as a nutritional supplement to prevent vitamin B12 deficiency. Vitamin B12 is a collective term for these variously subs…

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansCoenzymes +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobicistat Approved DB09065
small molecule | CAS: 1004316-88-4

Cobicistat, marketed under the name Tybost (formerly GS-9350), indicated for treating infection with human immunodeficiency virus (HIV). Although it does not have any anti-HIV activity, cobicistat acts as a pharmacokinetic enhancer by inhibiting cytochrome P4…

Kategori:
Acids, AcyclicAnti-HIV AgentsAnti-Infective Agents +29
Target Protein:
Cytochrome P450 3A4Cytochrome P450 3A5Cytochrome P450 3A7
Waktu ParuhThe terminal plasma…
Vol. Distribusi-
Klirens-
Genetik -
Cobimetinib Approved DB05239
small molecule | CAS: 934660-93-2

Cobimetinib is an orally active, potent and highly selective small molecule inhibiting mitogen-activated protein kinase kinase 1 (MAP2K1 or MEK1), and central components of the RAS/RAF/MEK/ERK signal transduction pathway. It has been approved in Switzerland a…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2D6 Inhibitors +22
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 1
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe estimated appar…
KlirensFollowing oral admi…
Genetik -
Cobiprostone DB05514
small molecule | CAS: 333963-42-1

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +4
Target Protein:
Chloride channel protein 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobitolimod DB14819
biotech | CAS: 1226822-98-5

Cobitolimod is under investigation in clinical trial NCT03178669 (The Efficacy of Cobitolimod in Patients With Moderate to Severe Active Ulcerative Colitis).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coblopasvir DB15315
small molecule | CAS: 1312608-46-0

Coblopasvir is under investigation in clinical trial NCT03416491 (Safety and Efficacy of KW-136 and Sofosbuvir for Treatment of Chronic Hepatitis C).

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobolimab DB16372
biotech | CAS: 2022215-65-0

Cobolimab is under investigation in clinical trial NCT04655976 (Study of Cobolimab in Combination With Dostarlimab and Docetaxel in Advanced NSCLC Participants).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobomarsen DB14931
biotech | CAS: 1848257-52-2

Cobomarsen is under investigation in clinical trial NCT02580552 (Safety, Tolerability and Pharmacokinetics of MRG-106 in Patients With Mycosis Fungoides (MF), CLL, DLBCL or ATLL).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cocaine Approved DB00907
small molecule | CAS: 50-36-2

An alkaloid ester extracted from the leaves of plants including coca. It is a local anesthetic and vasoconstrictor and is clinically used for that purpose, particularly in the eye, ear, nose, and throat. It also has powerful central nervous system effects sim…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAlkaloids +36
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium channel protein +5
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
biotech

RBP-8000 is under investigation in clinical trials (A Randomized, 4-sequence, 2-period, Double-blind, Placebo Controlled Study With a DSM-IV-TR Diagnosis of Cocaine Abuse) for the treatment of Cocaine Abuse.

Kategori:
Amino Acids, Peptides, and ProteinsEnzymesEnzymes and Coenzymes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61789-40-0

Cocamidopropyl betaine is a mixture of closely related organic compounds derived from coconut oil and dimethylaminopropylamine that typically acts as an amphoteric surfactant in cosmetics and personal care products. It is a zwitterionic ammonium compound and …

Kategori:
AminesCompounds used in a research, industrial, or household settingOnium Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cocoa butter Approved DB11086
biotech | CAS: 8002-31-1

Cocoa butter is an edible natural fat obtained from the _Theobroma cocoa_ seeds that is predominantly found in dark chocolate [A33033]. It is a rich source of monounsaturated and saturated fatty acids [A33040] that mainly contains approximately 33% [DB04224],…

Kategori:
Antipruritics and Local AnestheticsDiet, Food, and NutritionFats +3
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Coconut Approved DB10523
biotech

Coconut allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CODA-001 DB14915
biotech | CAS: 1605326-11-1

CODA-001 is under investigation in clinical trial NCT01165450 (Efficacy and Safety Study of Nexagon for Persistent Corneal Epithelial Defects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Codeine Approved DB00318
small molecule | CAS: 76-57-3

The relief of pain (analgesia) is a primary goal for enhancing the quality of life of patients and for increasing the ability of patients to engage in day to day activities. Codeine, an opioid analgesic, was originally approved in the US in 1950 and is a drug…

Kategori:
AlkaloidsAnalgesicsAntitussive Agents +26
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +6
Waktu ParuhPlasma half-lives o…
Vol. DistribusiApparent volume of …
KlirensRenal clearance of …
Genetik 9 Varian
small molecule | CAS: 125-27-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Codeine-N-oxide DB01568
small molecule | CAS: 3688-65-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Codrituzumab DB14843
biotech | CAS: 1365267-33-9

Codrituzumab is under investigation in clinical trial NCT01507168 (A Study of RO5137382 (GC33) in Patients With Advanced or Metastatic Hepatocellular Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coenzyme A DB01992
small molecule | CAS: 85-61-0

Coenzyme A (CoA, CoASH, or HSCoA) is a coenzyme, well known for it's role in the synthesis and oxidation of fatty acids, and the oxidation of pyruvate in the citric acid cycle. All genomes sequenced to date encode enzymes that use coenzyme A as a substrate, a…

Kategori:
Adenine NucleotidesCoenzyme A, biosynthesisCoenzymes +7
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseCarnitine O-acetyltransferaseGalactoside O-acetyltransferase +42
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coenzyme F420 DB03913
small molecule | CAS: 64885-97-8

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 4001–4050 dari 12560
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