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6694

Total database: 17430
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4518 (67.5%)
Target
3751 (56.0%)
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81 (1.2%)
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6694 (100.0%)

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Halaman 79 / 134
Lifibrol DB12448
small molecule | CAS: 96609-16-4

Lifibrol has been used in trials studying the basic science of Hyperlipoproteinemia and Hypercholesterolemia.

Kategori:
Acids, CarbocyclicAlcoholsBenzene Derivatives +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lifitegrast Approved DB11611
small molecule | CAS: 1025967-78-5

Lifitegrast is a FDA approved drug for the treatment of keratoconjunctivitis sicca (dry eye syndrome). It is a tetrahydroisoquinoline derivative and lymphocyte function-associated antigen-1 ( LFA-1) antagonist that was discovered through the rational design p…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +18
Target Protein:
Intercellular adhesion molecule 1Integrin alpha-L
Waktu ParuhNot possible to cal…
Vol. Distribusi-
KlirensNot possible to cal…
Genetik -
Ligelizumab DB11856
biotech | CAS: 1322627-61-1

Ligelizumab is a humanized IgG1k monoclonal antibody targeted against immunoglobulin E (IgE). Similar in mechanism to [omalizumab], another IgE-directed monoclonal antibody, ligelizumab has a distinct binding epitope as compared to its peer (with a small degr…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Immunoglobulin heavy constant epsilon
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Light green SF yellowish Approved DB11183
small molecule | CAS: 5141-20-8

Light green SF yellowish is a green triarylmethane dye that is used in the preparation of the staining solution which is widely used as a counterstain. It is used in histological applications and other labratory settings, and usually exists as a disodium salt…

Kategori:
AminesArylsulfonatesArylsulfonic Acids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Limaprost DB09211
small molecule | CAS: 74397-12-9

Limaprost (as Limaprost alfadex; CAS number 88852-12-4) is an oral prostaglandin E1 analog. Prostaglandins act on a variety of cells such as vascular smooth muscle cells causing constriction or dilation, on platelets causing aggregation or disaggregation and …

Kategori:
AnticoagulantsAutacoidsBiological Factors +11
Target Protein:
Prostaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtypeProstaglandin E2 receptor EP3 subtype +1
Waktu ParuhThe mean half life …
Vol. Distribusi-
KlirensMean total clearanc…
Genetik -
Lime (citrus) Approved DB10635
biotech

Lime (citrus) allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 138-86-3

Limonene, (+/-)- is under investigation in clinical trial NCT05525260 (Limonene for Pulmonary Nodule Chemoprevention).

Kategori:
Cyclohexane MonoterpenesCyclohexanesCyclohexenes +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Linaclotide Approved DB08890
small molecule | CAS: 851199-59-2

Linaclotide is a synthetic 14-amino acid cyclic peptide [A260271] and first-in-class guanylate cyclase-C (G-CC) agonist.[A260271, L47211] Linaclotide is structurally related to human guanylin and uroguanylin, paracrine peptide hormones that are endogenous act…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsDrugs for Constipation +7
Target Protein:
Guanylyl cyclase C
Waktu ParuhThere is no availab…
Vol. DistribusiGiven that linaclot…
KlirensNo information is a…
Genetik -
Lincomycin Approved DB01627
small molecule | CAS: 154-21-2

Lincomycin is a lincosamide antibiotic first isolated from the soil bacterium _Streptomyces lincolnensis_ in Lincoln, Nebraska.[A190621] Clinical use of lincomycin has largely been superseded by its semisynthetic derivative [clindamycin] due to its higher eff…

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
23S ribosomal RNA
Waktu ParuhLincomycin has a bi…
Vol. DistribusiLincomycin administ…
KlirensLincomycin administ…
Genetik -
Lindane Approved DB00431
small molecule | CAS: 58-89-9

An organochlorine insecticide that has been used as a pediculicide and a scabicide. Lindane has been banned in California, United Kingdom, Australia, and many western countries due to concerns about neurotoxicity and adverse effects on the environment. In Can…

Kategori:
Agents that reduce seizure thresholdAgrochemicalsAntiparasitic Products, Insecticides and Repellents +9
Target Protein:
Gamma-aminobutyric acid receptor subunit beta-1Glycine receptor subunit alpha-1Glycine receptor subunit alpha-2 +7
Waktu Paruh18 hours
Vol. Distribusi-
Klirens-
Genetik -
Linerixibat DB11729
small molecule | CAS: 1345982-69-5

GSK2330672 has been investigated for the treatment of Diabetes Mellitus, Type 2.

Kategori:
AminesAzepinesSulfur Compounds +1
Target Protein:
Ileal sodium/bile acid cotransporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Linezolid Approved DB00601
small molecule | CAS: 165800-03-3

Linezolid is a synthetic antibiotic which is used for the treatment of infections caused by aerobic Gram-positive bacteria. Its effects are bacteriostatic against both enterococci and staphylococci and bactericidal against most isolates of streptococci.[L3296…

Kategori:
AcetamidesAcetatesAcids, Acyclic +22
Target Protein:
23S ribosomal RNA
Waktu ParuhThe elimination hal…
Vol. DistribusiAt steady-state, th…
KlirensTotal clearance of …
Genetik -
Linifanib DB06080
small molecule | CAS: 796967-16-3

Linifanib (ABT-869) is a small molecule vascular endothelial growth factor (VEGF) receptor-based kinase inhibitor that is designed to suppress tumor growth by preventing the formation of new blood vessels that supply the tumor with oxygen and nutrients and by…

Kategori:
AmidesBenzene DerivativesHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Vascular endothelial growth factor receptor 3Receptor-type tyrosine-protein kinase FLT3Vascular endothelial growth factor receptor 1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Linoleic acid Approved DB14104
small molecule | CAS: 60-33-3

Deskripsi belum tersedia.

Kategori:
Fatty AcidsFatty Acids, EssentialFatty Acids, Omega-6 +3
Target Protein:
Fatty acid-binding protein, adipocyte
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Linopristin DB19296
small molecule | CAS: 325965-23-9

Linopristin is an antibiotic of the streptogramin B class. It is one part of the combination product NXL 103, along with [Virginiamycin M1]. The combination product was under investigation in clinical trials NCT00653172 and NCT00949130 for treatment of variou…

Waktu Paruh-
Vol. Distribusi-
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Linrodostat DB14986
small molecule | CAS: 1923833-60-6

Linrodostat is under investigation in clinical trial NCT03247283 (Pharmacokinetics and Metabolism Study in Healthy Male Participants).

Kategori:
AcetatesAcids, AcyclicAmides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Linseed oil DB11357
biotech | CAS: 66071-03-2

Linseed oil is a rich source of ?-Linolenic acid extracted from the dried, ripened seeds of the flax plant *Linum usitatissimum*. Other fatty acids contained in linseed oil include palmitic acid, stearic acid, oleic acid and linolenic acid. Linseed oil is par…

Kategori:
Biological ProductsComplex MixturesFats +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lintitript DB04867
small molecule | CAS: 136381-85-6

Lintitript is a new, highly specific and potent CCK-A receptor antagonist.

Kategori:
Heterocyclic Compounds, Fused-RingHormone AntagonistsHormones, Hormone Substitutes, and Hormone Antagonists +2
Target Protein:
Cholecystokinin receptor type A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2209911-94-2

Lintuzumab actinium Ac-225 is under investigation in clinical trial NCT00672165 (Targeted Atomic Nano-Generators (Actinium-225-Labeled Humanized Anti-CD33 Monoclonal Antibody HuM195) in Patients With Advanced Myeloid Malignancies).

Waktu Paruh-
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Linvoseltamab DB17447
biotech

Linvoseltamab is an investigational bispecific antibody. It promotes the interaction of B-cell maturation antigen (BCMA) on multiple myeloma cells with CD3-expressing T cells.

Waktu Paruh-
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Linzagolix Approved DB17083
small molecule | CAS: 935283-04-8

Linzagolix is a non-peptide, selective antagonist of the gonadotropin-releasing hormone (GnRH) receptor. It has been studied for the treatment of estrogen-dependent conditions such as uterine fibroids and endometriosis.[A253642,A253647] It is similar to other…

Kategori:
Anti-Gonadotropin-Releasing HormonesBCRP/ABCG2 SubstratesCytochrome P-450 CYP2C8 Inhibitors +18
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe half-life of li…
Vol. DistribusiAfter seven days of…
KlirensThe geometric mean …
Genetik -
LioCyx-M004 DB17368
biotech

LioCyx-M004 are autologous T cells transduced with a retroviral vector encoding a hepatitis B virus antigen-specific T cell receptor.

Waktu Paruh-
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Liotrix Approved DB01583
small molecule | CAS: 8065-29-0

Liotrix is a synthetically derived thyroid hormone replacement preparation. It consists of levothyroxine sodium (thyroxine, T4) and liothyronine sodium (triiodothyronine, T3) in a 4 to 1 ratio by weight. Liotrix was developed when it was believed that serum l…

Kategori:
Agents used to treat hypothyroidismAmino AcidsAmino Acids, Aromatic +19
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lipegfilgrastim Approved DB13200
biotech | CAS: 1117844-87-7

Lipegfilgrastim, previously known as XM22, is a pegylated, recombinant granulocyte colony-stimulating factor (G-CSF) that was synthetized using a highly site-specific glycoPEGylation technology [A32665]. It is used as an alternate to [DB00019] for prophylacti…

Kategori:
Adjuvants, ImmunologicAlcoholsAmino Acids, Peptides, and Proteins +17
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe average termina…
Vol. DistribusiLipegfilgrastim has…
KlirensIn a phase 1, multi…
Genetik -
Lipoic acid Approved DB00166
small molecule | CAS: 1200-22-2

A vitamin-like antioxidant.

Kategori:
Alimentary Tract and MetabolismAntioxidantsBiological Factors +15
Target Protein:
Lipoyl amidotransferase LIPT1, mitochondrialSodium-dependent multivitamin transporterLipoyl synthase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lipotecan DB17385
small molecule | CAS: 1432468-79-5

Deskripsi belum tersedia.

Kategori:
Alkaloids
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Carboxylic Ester HydrolasesEnzymesEnzymes and Coenzymes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Liquidambar styraciflua pollen is the pollen of the Liquidambar styraciflua plant. Liquidambar styraciflua pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 8046-19-3

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Liraglutide Approved DB06655
biotech | CAS: 204656-20-2

Victoza contains liraglutide, a synthetic analog of human glucagon-like peptide-1(GLP-1) and acts as a GLP-1 receptor agonist.[Label,A6932] Liraglutide is 97% similar to native human GLP-1, differing primarily by substituting arginine for lysine at position 3…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +17
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhTerminal half life …
Vol. Distribusi13L[Label].
Klirens1.2L/h[Label].
Genetik -
Lirentelimab DB16728
biotech | CAS: 2283348-97-8

Lirentelimab is under investigation in clinical trial NCT04856891 (A Study of Lirentelimab (AK002) in Patients With Active Eosinophilic Duodenitis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lisdexamfetamine Approved DB01255
small molecule | CAS: 608137-32-2

Lisdexamfetamine is a prodrug of [dextroamphetamine], a central nervous system stimulant known as d-amphetamine,[A40246] covalently attached to the naturally occurring amino acid L-lysine.[A2230] Lisdexamfetamine is the first chemically formulated prodrug sti…

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +17
Target Protein:
Trace amine-associated receptor 1
Waktu ParuhPlasma concentratio…
Vol. DistribusiDextroamphetamine, …
Klirens-
Genetik -
Lisocabtagene maraleucel Approved DB16582
biotech

Lisocabtagene maraleucel is a chimeric antigen receptor (CAR) T-cell therapy, similar to [brexucabtagene autoleucel] and [axicabtagene ciloleucel].[A228493,L31588] Lisocabtagene maraleucel is a genetically modified autologous T-cell therapy that targets CD19,…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAntineoplastic cell and gene therapy +3
Target Protein:
B-lymphocyte antigen CD19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lithium carbonate Approved DB14509
small molecule | CAS: 554-13-2

Lithium has been used to treat manic episodes since the 19th century[A176642]. Though it is widely used, its mechanism of action is still unknown[FDA Label][A14585,A176642,A176651,L5843]. Lithium carbonate has a narrow therapeutic range and so careful monitor…

Kategori:
AcidsAcids, NoncarboxylicAlkalies +26
Target Protein:
Inositol monophosphatase 2Inositol monophosphatase 1Glycogen synthase kinase-3 beta +1
Waktu ParuhThe half life of li…
Vol. DistribusiApparent volume of …
KlirensClearance is genera…
Genetik -
Lithium cation DB01356
small molecule | CAS: 7439-93-2

Lithium was used during the 19th century to treat gout. Lithium salts such as lithium carbonate (Li2CO3), lithium citrate, and lithium orotate are mood stabilizers. They are used in the treatment of bipolar disorder, since unlike most other mood altering drug…

Kategori:
Antidepressive AgentsAntimanic AgentsAntipsychotic Agents +11
Target Protein:
Glycogen synthase kinase-3 betaInositol monophosphatase 1Inositol monophosphatase 2 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lithium citrate Approved DB14507
small molecule | CAS: 919-16-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntidepressive AgentsAntimanic Agents +12
Target Protein:
Inositol monophosphatase 2Inositol monophosphatase 1Glycogen synthase kinase-3 beta +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 29126-50-9

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDermatologicalsDicarboxylic Acids +2
Target Protein:
Inositol monophosphatase 2Inositol monophosphatase 1Glycogen synthase kinase-3 beta +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Litifilimab DB18864
biotech | CAS: 2407378-48-5

Litifilimab is under investigation in clinical trial NCT05531565 (A Study to Assess the Efficacy and Safety of BIIB059 (Litifilimab) in Participants With Active Subacute Cutaneous Lupus Erythematosus (SCLE) And/or Chronic Cutaneous Lupus Erythematosus (CCLE) …

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lividomycin A DB04728
small molecule | CAS: 36441-41-5

Deskripsi belum tersedia.

Target Protein:
Telomerase reverse transcriptase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Livmoniplimab DB18939
biotech | CAS: 2412004-88-5

Livmoniplimab is under investigation in clinical trial NCT06109272 (A Study to Assess the Dose, Adverse Events, and Change in Disease Activity of Livmoniplimab as an Intravenous (IV) Solution in Combination With Budigalimab as an IV Solution in Adult Particip…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lixadesiran DB17295
biotech | CAS: 1152798-49-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lixisenatide Approved DB09265
biotech | CAS: 320367-13-3

Lixisenatide is a glucagon-like peptide-1 (GLP-1) receptor agonist used in the treatment of type II diabetes mellitus (T2DM). It is sold by Sanofi-Aventis under the brand name Adlyxin in the US[L763] and Lyxumia in the EU.[L764] Adlyxin recieved FDA approval …

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +11
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhFollowing the admin…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -
biotech | CAS: 2461531-19-9

Lixmabegagene relduparvovec, formerly known as LYS-GM101, is a recombinant adeno-associated virus vector serotype rh.10 (AAVrh.10) carrying the human ?-galactosidase gene (GBL1). It is under development for the treatment of GM1 gangliosidosis.[L45929]

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LJP 1082 DB05446
small molecule

LJP 1082 is a Toleragen that is designed to shut down the B cells that produce antibodies to ß2 GP1. LJP 1082 is undergoing trial for for the treatment of stroke, deep-vein thrombosis and other conditions associated with antibody-mediated thrombosis. Antibody…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsCarbohydrates +7
Target Protein:
Beta-2-glycoprotein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LL-37 DB16532
biotech

LL-37 is a human cathelicidin that inhibits viral replication and while also playing a role in host defense against infection.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LM-030 DB18283
small molecule | CAS: 1122484-55-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LM-609 DB05787
biotech

LM-609 (Vitaxin) is an artificial antibody that targets a protein on the surface of newly forming blood vessels, as well as on certain tumors. In addition to cancer, the protein has been implicated in bone destruction in rheumatoid arthritis and the inflammat…

Target Protein:
Integrin beta-3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
LMB-100 DB18591
biotech | CAS: 1841500-93-3

LMB-100 is a is an antibody-toxin conjugate with an antimesothelin Fab linked to a 24-kilodalton portion of Pseudomonas exotoxin A with mutations that decrease immunogenicity.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

LNP-nCoVsaRNA is a purified, synthetic mRNA vaccine candidate encoding the S glycoprotein of SARS-CoV-2, which is used primarily by the virus to attach to and invade human cells. The vaccine was developed in and tested by the Medical Research Council Clinical…

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Lobaplatin DB13049
small molecule | CAS: 135558-11-1

Lobaplatin has been used in trials studying the treatment of Breast Cancer, Hepatocellular Carcinoma, and Lobaplatin and Gemcitabine in Combination, Second-line Treatments on Advanced Osteosarcoma.

Kategori:
CycloparaffinsOrganometallic Compounds
Waktu Paruh-
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Genetik -
Menampilkan 3901–3950 dari 6694
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