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11778

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8554 (72.6%)
Target
6383 (54.2%)
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96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 79 / 236
Cusatuzumab DB15100
biotech | CAS: 1864871-20-4

CD70 is a ligand expressed on the surface of activated lymphocytes and mature dendritic cells that, in its binding to CD27 receptors, plays an important role in cell proliferation and survival. An overexpression of CD70 can result in the proliferation of mali…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Target Protein:
CD70 antigen
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Custirsen DB05487
biotech | CAS: 890056-27-6

Custirsen is a benzopyran with potential antineoplastic activity. Custirsen acts as a selective estrogen receptor modulator (SERM), inhibiting the proliferation of estrogen-sensitive breast cancer cells. This agent also inhibits growth and induces apoptosis o…

Kategori:
Antisense OligonucleotidesHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +3
Target Protein:
ClusterinEstrogen receptorNuclear factor NF-kappa-B p100 subunit +1
Waktu Paruh-
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Cutamesine DB06618
small molecule | CAS: 165377-43-5

Deskripsi belum tersedia.

Kategori:
Central Nervous System AgentsNootropic AgentsReceptors, sigma, agonists
Target Protein:
Sigma non-opioid intracellular receptor 1
Waktu Paruh-
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CV-8102 DB19184
biotech

CV-8102 is under investigation in clinical trial NCT03203005 (IMA970A Plus CV8102 in Very Early, Early and Intermediate Stage Hepatocellular Carcinoma Patients).

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CVac Approved DB17351
small molecule

Deskripsi belum tersedia.

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CVN-424 DB18958
small molecule | CAS: 2254706-21-1

CVN-424 is under investigation in clinical trial NCT06006247 (Early Parkinson's Disease Monotherapy With CVN424).

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CVnCoV DB15844
biotech

The CVnCov Vaccine (or CV07050101) is in development by CureVac AG. The vaccine uses mRNA technology to create a protein associated with SARS-CoV2, and upon administration and replication, to initiate subsequent immune responses in the body. As of June 2020, …

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CVnCoV Vaccine DB15843
biotech

The CVnCov Vaccine (or CV07050101) is in development by CureVac AG. The vaccine uses mRNA technology to create a protein associated with SARS-CoV2, and upon administration and replication, to initiate subsequent immune responses in the body. As of June 2020, …

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +10
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CVT-6883 DB05936
small molecule | CAS: 752222-83-6

CVT-6883 is a selective, potent and orally available A2B-adenosine receptor antagonist which CV Therapeutics is investigating for the potential treatment of asthma and other conditions related to inflammation and fibrosis.

Kategori:
Adenosine A2 Receptor AntagonistsHeterocyclic Compounds, Fused-Ring
Target Protein:
Adenosine receptor A2b
Waktu Paruh-
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CX-046684 Approved DB19414
biotech

CX-046684 is a COVID-19 mRNA vaccine encoding the pre-fusion stabilized Spike glycoprotein (S) of the SARS-CoV-2 Omicron variant lineage KP.2. It is the active ingredient of the 2024-2025 formulation of Moderna's Spikevax vaccine.[L40074]

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CX-717 DB05047
small molecule | CAS: 867276-98-0

CX-717 is an ampakine compound previously investigated for the treatment of Attention-Deficit/Hyperactivity Disorder (ADHD) and Alzheimer's disease.

Target Protein:
Neurotrophic factor BDNF precursor formGlutamate receptor 1Glutamate receptor 2 +2
Waktu Paruh-
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CX157 DB05205
small molecule

CX157,3-fluoro-7-(2,2,2,-trifluoroethoxy)phenoxathiin-10,10-dioxide, is a reversible, selective inhibitor of MAO-A designed to have improved oral bioavailability and reduced clearance compared to previous MAO-A inhibitors of this class.

Target Protein:
Amine oxidase [flavin-containing] A
Waktu Paruh-
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CX501 DB05174
small molecule

Cx501 is used to treat epidermolysis bullosa (EB), a rare genetic condition which can lead to contraction of the joints, fusion of fingers and toes, contraction of the mouth membranes and narrowing of the oesophagus. It is developed by Cellerix and is in phas…

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CX516 DB06247
small molecule | CAS: 154235-83-3

Deskripsi belum tersedia.

Kategori:
Receptors, AMPA
Target Protein:
Glutamate receptor 1
Waktu Paruh-
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CXA-10 DB15026
small molecule | CAS: 875685-46-4

CXA-10 is under investigation in clinical trial NCT03422510 (FIRSTx - A Study of Oral CXA-10 in Primary Focal Segmental Glomerulosclerosis (FSGS)).

Kategori:
Anti-Inflammatory AgentsFatty AcidsFatty Acids, Monounsaturated +2
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CXD101 DB16182
small molecule | CAS: 934828-12-3

CXD101 is under investigation in clinical trial NCT03873025 (A Study of CXD101 in Combination With Pembrolizumab for Relapsed or Refractory Diffuse Large B-cell Lymphoma).

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CXL-1020 DB15326
small molecule | CAS: 950834-06-7

CXL-1020 is under investigation in clinical trial NCT01092325 (Safety and Hemodynamic Effects and Pharmacokinetics of CXL-1020 in Patients With Stable Heart Failure).

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CY 1899 DB17797
biotech

Deskripsi belum tersedia.

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CY-1503 DB17605
small molecule | CAS: 168678-84-0

CY-1503 is a pentasaccharide ethyl glycoside consisting of one alpha-D-sialylosyl residue as a sodium salt, two beta-D-galactopyranosyl residues, one 2-acetamido-beta-Dglucopyranosyl unit, and one alpha-L-fucopyranosyl unit. It was investigated in cardiopulmo…

Kategori:
CarbohydratesPolysaccharides
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Cyanamide DB02679
small molecule | CAS: 420-04-2

A cyanide compound which has been used as a fertilizer, defoliant and in many manufacturing processes. It often occurs as the calcium salt, sometimes also referred to as cyanamide. The citrated calcium salt is used in the treatment of alcoholism. [PubChem]

Kategori:
CarbodiimidesCyanidesImines +1
Target Protein:
Cathepsin KCarbonic anhydrase 2
Waktu Paruh-
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Cyanocobalamin Approved DB00115
small molecule | CAS: 68-19-9

Cyanocobalamin (commonly known as Vitamin B12) is a highly complex, essential vitamin, owing its name to the fact that it contains the mineral, cobalt. This vitamin is produced naturally by bacteria [A175276], and is necessary for DNA synthesis and cellular e…

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansCorrinoids +10
Target Protein:
Methionine synthaseMethylmalonyl-CoA mutase, mitochondrialMethionine synthase reductase +3
Waktu ParuhApproximately 6 day…
Vol. DistribusiCobalamin is distri…
KlirensDuring vitamin load…
Genetik -
Cyanocobalamin Co-57 Approved DB09385
small molecule | CAS: 13115-03-2

Deskripsi belum tersedia.

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
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Cyanocobalamin Co-60 Approved DB09387
small molecule | CAS: 13422-53-2

Cyanocobalamin Co-60 is an analog of Vitamin B12 labeled with Co60. Cyanocobalamin Co-60 was used for the diagnosis of pernicious anemia, but now it is withdrawn from the market in the US for unknown reasons.

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CYC-065 DB15425
small molecule | CAS: 1070790-89-4

CYC-065 is under investigation in clinical trial NCT03739554 (CYC065 CDK Inhibitor and Venetoclax Study in Relapsed/Refractory CLL).

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Cyclin-dependent kinase 9Cyclin-dependent kinase 2
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Cyclacillin Approved DB01000
small molecule | CAS: 3485-14-1

A cyclohexylamido analog of penicillanic acid.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +8
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 3Penicillin binding protein 2a +1
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Cyclandelate Approved DB04838
small molecule | CAS: 456-59-7

A direct-acting smooth muscle relaxant used to dilate blood vessels. It may cause gastrointestinal distress and tachycardia. Cyclandelate is not approved for use in the U.S. or Canada, but is approved in various European countries.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAntiarrhythmic agents +10
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1Liver carboxylesterase 1
Waktu Paruh-
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small molecule | CAS: 6453-60-7

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleotidesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
Target Protein:
5'(3')-deoxyribonucleotidase, mitochondrial
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small molecule | CAS: 60-92-4

Cyclic adenosine monophosphate (cAMP, cyclic AMP or 3'-5'-cyclic adenosine monophosphate) is a molecule that is important in many biological processes; it is derived from adenosine triphosphate (ATP).

Kategori:
Adenine NucleotidesCyclic AMPHeterocyclic Compounds, Fused-Ring +8
Target Protein:
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2cAMP-dependent protein kinase type I-alpha regulatory subunitcAMP-dependent protein kinase type II-beta regulatory subunit +3
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Cyclic GMP DB02315
small molecule | CAS: 7665-99-8

Cyclic guanosine monophosphate (Cyclic GMP) is a guanine nucleotide containing one phosphate group which is esterified to the sugar moiety in both the 3'- and 5'-positions. It is a cellular regulatory agent and has been described as a second messenger…

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +5
Target Protein:
cGMP-dependent 3',5'-cyclic phosphodiesterasePotassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2cAMP-dependent protein kinase type I-alpha regulatory subunit
Waktu Paruh-
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Cyclizine Approved DB01176
small molecule | CAS: 82-92-8

A histamine H1 antagonist given by mouth or parenterally for the control of postoperative and drug-induced vomiting and in motion sickness. (From Martindale, The Extra Pharmacopoeia, 30th ed, p935)

Kategori:
AntiemeticsAntihistamines for Systemic UseAutonomic Agents +15
Target Protein:
Histamine H1 receptorSulfotransferase 1E1
Waktu Paruh20 hours
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small molecule | CAS: 97011-16-0

NA-831 (Traneurocin), is under investigation in two clinical trials: NCT03538522 (completed, for mild cognitive impairment and Alzheimer’s disease) and NCT04452565 (unknown status, combination therapy with Atazanavir and Dexamethasone for COVID-19).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Chitinase B
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Vanadates
Target Protein:
Mono-ADP-ribosyltransferase C3
Waktu Paruh-
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Cyclobarbital DB13737
small molecule | CAS: 52-31-3

Deskripsi belum tersedia.

Kategori:
Barbiturates, PlainCentral Nervous System DepressantsHypnotics and Sedatives +4
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Cyclobenzaprine Approved DB00924
small molecule | CAS: 303-53-7

Cyclobenzaprine, a centrally-acting muscle relaxant, was first synthesized in 1961[A185039] and has been available for human use since 1977.[A184982] It was initially studied for use as antidepressant given its structural similarity to tricyclic antidepressan…

Kategori:
Agents that reduce seizure thresholdAntidepressive AgentsBenzocycloheptenes +23
Target Protein:
Alpha-2C adrenergic receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2B +7
Waktu ParuhThe effective half-…
Vol. DistribusiThe volume of distr…
KlirensThe approximate pla…
Genetik -
Cyclocreatine DB17624
small molecule | CAS: 35404-50-3

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntineoplastic Agents +2
Waktu Paruh-
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Cyclofenil DB13472
small molecule | CAS: 2624-43-3

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesCresolsFertility Agents +7
Target Protein:
Estrogen receptor
Waktu Paruh-
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Cycloguanil Approved DB14763
small molecule | CAS: 516-21-2

Cycloguanil is the active metabolite of [proguanil].

Kategori:
AmidinesAnti-Infective AgentsAntimalarials +7
Target Protein:
Peptide deformylase, mitochondrial
Waktu Paruh-
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small molecule | CAS: 701-97-3

Deskripsi belum tersedia.

Target Protein:
Aromatic-amino-acid aminotransferase
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Cyclohexanol DB03703
small molecule | CAS: 108-93-0

Monohydroxy derivatives of cyclohexanes that contain the general formula R-C6H11O. They have a camphorlike odor and are used in making soaps, insecticides, germicides, dry cleaning, and plasticizers. [PubChem]

Kategori:
AlcoholsCyclohexanesCycloparaffins +3
Target Protein:
Beta-lactamaseAll-trans-retinol dehydrogenase [NAD(+)] ADH1B
Waktu Paruh-
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small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-lactamase SHV-1Beta-lactamase SHV-2
Waktu Paruh-
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small molecule | CAS: 766-93-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAlcohol Dehydrogenase, antagonists & inhibitorsAmides +1
Target Protein:
Alcohol dehydrogenase 1CAll-trans-retinol dehydrogenase [NAD(+)] ADH4
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin D
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Cyclopenthiazide Approved DB13532
small molecule | CAS: 742-20-1

Cyclopenthiazide is a thiazide diuretic with antihypertensive properties. In a double blind, randomized crossover study, cyclopenthiazide was effective in reducing diastolic blood pressure in mildly hypertensive non-insulin dependent diabetic patients [A27180…

Kategori:
Antihypertensive AgentsBenzothiadiazinesCardiovascular Agents +13
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Cyclopentolate Approved DB00979
small molecule | CAS: 512-15-2

A parasympatholytic anticholinergic used solely to obtain mydriasis or cycloplegia.

Kategori:
Acids, CarbocyclicAnticholinergic AgentsAutonomic Agents +11
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M5
Waktu Paruh-
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Cyclopropane DB13984
small molecule | CAS: 75-19-4

Cyclopropane was initially investigated because it was thought to be the toxic element in ethylene. Instead, it turned out to be an excellent anesthetic with very rapid onset and recovery while maintaining stable hemodynamics. Its use was ultimately limited b…

Kategori:
AnestheticsCentral Nervous System AgentsCentral Nervous System Depressants +1
Waktu Paruh-
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Cycloserine Approved DB00260
small molecule | CAS: 68-41-7

Antibiotic substance produced by Streptomyces garyphalus.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +14
Target Protein:
Glutamate receptor ionotropic, NMDA 1D-alanine--D-alanine ligase AAlanine racemase
Waktu ParuhHalf-life in patien…
Vol. Distribusi-
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Cyclosporine Approved DB00091
small molecule | CAS: 59865-13-3

Cyclosporine is a calcineurin inhibitor known for its immunomodulatory properties that prevent organ transplant rejection and treat various inflammatory and autoimmune conditions. It is isolated from the fungus _Beauveria nivea_.[A174049] Initially manufactur…

Kategori:
Agents causing hyperkalemiaAgents Causing Muscle ToxicityAgents that produce hypertension +45
Target Protein:
Guided entry of tail-anchored proteins factor CAMLGProtein phosphatase 3 catalytic subunit alphaCalcineurin subunit B type 2 +2
Waktu ParuhThe half-life of cy…
Vol. DistribusiThe distribution of…
KlirensCyclosporin shows a…
Genetik -
Cyclothiazide Approved DB00606
small molecule | CAS: 2259-96-3

As a diuretic, cyclothiazide inhibits active chloride reabsorption at the early distal tubule via the Na-Cl cotransporter, resulting in an increase in the excretion of sodium, chloride, and water. Thiazides like cyclothiazide also inhibit sodium ion transport…

Kategori:
Antihypertensive AgentsCardiovascular AgentsDiuretics +11
Target Protein:
Sodium/potassium-transporting ATPase subunit gammaCarbonic anhydraseCarbonic anhydrase 2 +2
Waktu Paruh-
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Cyclouridine DB04627
small molecule | CAS: 3736-77-4

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosidesPyrimidine Nucleosides +2
Target Protein:
Uridine phosphorylase
Waktu Paruh-
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Cycrimine Approved DB00942
small molecule | CAS: 77-39-4

Cycrimine is a drug used to reduce levels of acetylcholine to return a balance with dopamine in the treatment and management of Parkinson's disease.

Kategori:
Agents producing tachycardiaAnticholinergic AgentsMuscarinic Antagonists
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
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Menampilkan 3901–3950 dari 11778
Sebelumnya Halaman 79 / 236 Berikutnya