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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Hasil Pencarian (15718)

Halaman 79 / 315
BO-653 DB19216
small molecule | CAS: 157360-23-1

BO-653 is under investigation in clinical trial NCT00055510 (A Blinded Study Conducted at Multiple Centers Evaluating Various Doses of an Investigational Agent (BO-653) Against Placebo, for Safety and Effectiveness in Preventing Post-angioplasty Blood Vessel …

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Boceprevir Approved DB08873
small molecule | CAS: 394730-60-0

Boceprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine…

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +21
Target Protein:
Genome polyproteinGenome polyprotein
Waktu ParuhBoceprevir has a me…
Vol. DistribusiThe mean apparent v…
KlirensBoceprevir has a me…
Genetik -
Bocidelpar DB16906
small molecule | CAS: 2095128-20-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2356354-82-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bococizumab DB12456
biotech | CAS: 1407495-02-6

Bococizumab has been used in trials studying the treatment and prevention of Dyslipidemia, Hyperlipidemia, Hypercholesterolemia, Cardiovascular Disease, and Heterozygous Familial Hypercholesterolemia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bolandiol DB01554
small molecule | CAS: 19793-20-5

Deskripsi belum tersedia.

Kategori:
EstranesEstrenesFused-Ring Compounds +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bolasterone DB01471
small molecule | CAS: 1605-89-6

Deskripsi belum tersedia.

Kategori:
Anabolic AgentsAndrostanesAndrostenes +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Boldenone DB01541
small molecule | CAS: 846-48-0

Boldenone is an anabolic steroid developed for veterinary use, mostly for treatment of horses. It is not indicated for use in humans in the US and is only available through veterinary clinics.

Kategori:
Anabolic AgentsAndrostanesAndrostenes +9
Target Protein:
Androgen receptor
Waktu Paruh14 days
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 13103-34-9

Deskripsi belum tersedia.

Kategori:
AndrostanesAndrostenesAndrostenols +6
Target Protein:
Androgen receptor
Waktu Paruh14 days
Vol. Distribusi-
Klirens-
Genetik -
Boldione DB07373
small molecule | CAS: 897-06-3

Deskripsi belum tersedia.

Kategori:
AndrostanesAndrostenesFused-Ring Compounds +1
Target Protein:
AromatasePentaerythritol tetranitrate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Boldo leaf extract Approved DB15815
biotech

Boldo leaf extract allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bombesin DB11724
small molecule | CAS: 31362-50-2

Bombesin is under investigation in clinical trial NCT01205321 (PET/CT Imaging for Radiation Dosimetry, Plasma Pharmacokinetics, Biodistribution, Safety and Tolerability and Diagnostic Performance of BAY86-7548 in Patients With Prostate Cancer and Healthy Volu…

Kategori:
Amino Acids, Peptides, and ProteinsAmphibian VenomsBiological Factors +12
Target Protein:
Gastrin-releasing peptide receptorBombesin receptor subtype-3Neuromedin-B receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bombyx mori fiber Approved DB10609
biotech

Bombyx mori fiber is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bomedemstat DB17234
small molecule | CAS: 1990504-34-1

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2364477-20-1

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Borage oil Approved DB11238
biotech

Borage oil, or borage seed oil, is a rich source of gamma-linolenic acid (GLA) that is obtained from the seeds of the Borago officinalis (borage). Borage oil is used as an herbal treatment of skin disorders including eczema, seborrheic dermatitis, and neurode…

Kategori:
Agents that reduce seizure thresholdAntirheumatic AgentsBiological Products +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Borate ion DB14553
small molecule | CAS: 12258-53-6

Deskripsi belum tersedia.

Kategori:
AnionsBoric AcidsBoron Compounds +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Bordetella pertussis filamentous hemagglutinin antigen (formaldehyde inactivated) is a vaccine that contains inactivated acellular pertussis antigen that is isolated from Bordetella pertussis culture.

Kategori:
Actively Acquired ImmunityInactivated Bordetella Pertussis Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Bordetella pertussis fimbriae 2/3 antigen is a vaccine for the prophylaxis of the disease caused by Bordetella pertussis which is a a Gram-negative coccobacillus that expresses two serologically distinct fimbriae (Fim2 and Fim3).

Kategori:
Actively Acquired ImmunityInactivated Bordetella Pertussis Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Bordetella pertussis pertactin antigen is a vaccine for the prophylaxis of whooping cough that contains pertactin, a membrane-associated antigen of Bordetella pertussis [A31248].

Kategori:
Amino Acids, Peptides, and ProteinsBacterial ProteinsBacterial Toxins +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Actively Acquired ImmunityInactivated Bordetella Pertussis Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Bordetella pertussis toxoid antigen (formaldehyde inactivated) is a vaccine.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Bordetella pertussis toxoid antigen (formaldehyde, glutaraldehyde inactivated) is a vaccine that is used in the prophylaxis of Pertussis (whooping cough), which is caused by a small Gram-negative coccobacillus that infects the mucosal layers of the human resp…

Kategori:
Actively Acquired ImmunityBiological ProductsComplex Mixtures +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Actively Acquired ImmunityInactivated Bordetella Pertussis Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Boric acid Approved DB11326
small molecule | CAS: 10043-35-3

Boric acid, also known as hydrogen borate, is a weak monobasic Lewis acid of boron with the chemical formula H3BO3. Boric acid is typically utilized in industrial processing and manufacturing, but is also used as an additive in pharmaceutical products, cosmet…

Kategori:
AcidsAcids, NoncarboxylicAgrochemicals +12
Waktu ParuhAccording to human …
Vol. DistribusiVolume of distribut…
KlirensA case report of ac…
Genetik -
Bornaprine DB13619
small molecule | CAS: 20448-86-6

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAnti-Parkinson DrugsAnticholinergic Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Borneol DB11288
small molecule | CAS: 507-70-0

Deskripsi belum tersedia.

Kategori:
Bicyclic MonoterpenesBridged-Ring CompoundsMonoterpenes +3
Target Protein:
Transient receptor potential cation channel subfamily V member 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bornyl acetate DB14665
small molecule | CAS: 76-49-3

Deskripsi belum tersedia.

Kategori:
Bicyclic MonoterpenesBridged-Ring CompoundsMonoterpenes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Borocaptate DB17408
small molecule

Deskripsi belum tersedia.

Kategori:
BoranesBoron CompoundsBoron Neutron Capture Therapy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Boron DB11203
small molecule | CAS: 7440-42-8

Boron (B) is a chemical element with an atomic number 5 that belongs in the Period 2 and Group 13 in the periodic table. It is a low-abundant metalloid that is a poor electrical conductor at room temperature. Natural boron exists in 2 stable isotopes however …

Kategori:
Diet, Food, and NutritionElementsFood +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bortezomib Approved DB00188
small molecule | CAS: 179324-69-7

Bortezomib is a dipeptide boronic acid derivative and proteasome inhibitor used to treat multiple myeloma and mantle cell lymphoma.[A204083] The 26S proteasome is a protein complex that degrades ubiquitinated proteins in the ubiquitin-proteasome pathway: reve…

Kategori:
AcidsAcids, NoncarboxylicAntineoplastic Agents +36
Target Protein:
Proteasome subunit beta type-5Serine protease 1Proteasome subunit beta type-1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean distributi…
KlirensFollowing the admin…
Genetik -
Bortezomib D-mannitol Approved DB16741
small molecule | CAS: 444576-08-3

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsProteasome Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bos taurus dander Approved DB11020
biotech

Bos taurus dander allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Bos taurus gallstone is an animal extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Complex MixturesGallstones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bos taurus hair Approved DB10856
biotech

Bos taurus hair is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bos taurus skin Approved DB10406
biotech

Bos taurus skin or pelt is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BOS172722 DB15498
small molecule | CAS: 1578245-44-9

BOS172722 is a novel and selective Monopolar spindle 1 (Mps1) kinase inhibitor identified as a potential anticancer agent.[A187123] Normally, Mps1 supports the proper division of cancer cells, ensuring survival and replication. The key role of Mps1 in the gro…

Target Protein:
Dual specificity protein kinase TTK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bosakitug DB19101
biotech | CAS: 2762183-23-1

Bosakitug (BSI-045B) is under investigation in clinical trial NCT05932654 (POC Study to Evaluate BSI-045B Monotherapy and BSI-045B Add-on Therapy With Dupilumab in Atopic Dermatitis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Boscalid Approved DB12792
small molecule | CAS: 188425-85-6

Boscalid has been investigated for the treatment of OSDI, Glaucoma, Staining, Schirmers, and Disease Severity, among others.

Kategori:
Benzene DerivativesNicotinic AcidsPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bosentan Approved DB00559
small molecule | CAS: 147536-97-8

Bosentan is a dual endothelin receptor antagonist marketed under the trade name Tracleer by Actelion Pharmaceuticals. Bosentan is used to treat pulmonary hypertension by blocking the action of endothelin molecules that would otherwise promote narrowing of the…

Kategori:
AmidesAntihypertensive AgentsAntihypertensives for Pulmonary Arterial Hypertension +24
Target Protein:
Endothelin receptor type BEndothelin-1 receptor
Waktu ParuhTerminal eliminatio…
Vol. Distribusi* 18 L
Klirens* 4 L/h [patients w…
Genetik -
Boserolimab DB17452
biotech | CAS: 2444297-08-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bosutinib Approved DB06616
small molecule | CAS: 380843-75-4

Bosutinib is a 7-alkoxy-3-quinolinecarbonitrile that functions as a potent, dual SRC and ABL tyrosine kinase inhibitor indicated for chronic myelogenous leukemia (CML), specifically Philadelphia chromosome-positive (Ph+) CML. Philadelphia chromosome is a hall…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +22
Target Protein:
Tyrosine-protein kinase ABL1Tyrosine-protein kinase LynProto-oncogene tyrosine-protein kinase Src +8
Waktu ParuhThe mean (SD) bosut…
Vol. DistribusiThe mean (SD) appar…
KlirensThe mean (SD) appar…
Genetik -
biotech | CAS: 2417551-39-2

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Botensilimab DB16651
biotech | CAS: 2408310-37-0

Botensilimab is under investigation in clinical trial NCT03860272 (Fc-engineered Anti-ctla-4 Monoclonal Antibody in Advanced Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Botrytis cinerea Approved DB10428
biotech

Botrytis cinerea is a fungus which can provoke allergic reactions. Botrytis cinerea extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Botulinum toxin type A Approved DB00083
biotech | CAS: 93384-43-1

In 2002, botulinum toxin A, also known as onabotulinumtoxinA or Botox, was the first type A botulism toxin to be introduced into the market for cosmetic use.[A231824] With a wide variety of applications and favourable safety profile, Botulinum toxin A injecti…

Kategori:
Acetylcholine Release InhibitorsAgents that produce neuromuscular block (indirect)Amino Acids, Peptides, and Proteins +29
Target Protein:
Synaptosomal-associated protein 25Rho-related GTP-binding protein RhoB
Waktu ParuhThere is no readily…
Vol. DistribusiThere are extremely…
KlirensClearance informati…
Genetik -
biotech

Botulinum toxin type e is under investigation in clinical trial NCT03193593 (Study to Evaluate EB-001 in Reducing Musculoskeletal Pain).

Kategori:
Amino Acids, Peptides, and ProteinsBacterial ProteinsBacterial Toxins +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBacterial ProteinsBacterial Toxins +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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