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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 78 / 321
AZD-6482 DB14980
small molecule | CAS: 1173900-33-8

AZD-6482 is under investigation in clinical trial NCT00688714 (Study to Investigate Safety and Tolerability of a Single Dose of AZD6482).

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +3
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AZD-7268 DB19203
small molecule | CAS: 1018988-00-5

AZD-7268 is under investigation in clinical trial NCT01020799 (AZD7268 Safety and Tolerability Study).

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Opioid, delta, agonists
Waktu Paruh-
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AZD-7295 DB12724
small molecule | CAS: 929890-64-2

AZD7295 has been investigated for the treatment of Hepatitis C.

Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
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AZD-7325 DB13994
small molecule | CAS: 942437-37-8

AZD7325 is a high affinity, selective modulator of the GABAA receptor system. [L2936]

Kategori:
GABA ModulatorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-3Gamma-aminobutyric acid receptor subunit alpha-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AZD-7648 DB16834
small molecule | CAS: 2230820-11-6

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
DNA-dependent protein kinase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AZD-7687 DB14949
small molecule | CAS: 1166827-44-6

AZD-7687 is under investigation in clinical trial NCT01119352 (AZD7687 Multiple Ascending Dose Study).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AZD-7762 DB12242
small molecule | CAS: 860352-01-8

AZD7762 has been investigated for the treatment of Cancer, Solid Tumors, and Advanced Solid Malignancies.

Kategori:
AmidesSulfur Compounds
Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
AZD-8055 DB12774
small molecule | CAS: 1009298-09-2

AZD8055 has been used in trials studying the treatment of Cancer, Lymphomas, Solid Tumors, MALIGNANT GLIOMA, and brainstem glioma, among others.

Kategori:
Oxazines
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
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Genetik -
AZD-8165 DB15132
small molecule | CAS: 1201686-72-7

AZD-8165 is under investigation in clinical trial NCT01150812 (Oral AZD8165 After Single Oral Ascending Doses in Healthy Male Subjects).

Target Protein:
Prothrombin
Waktu Paruh-
Vol. Distribusi-
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AZD-8186 DB15029
small molecule | CAS: 1627494-13-6

AZD-8186 is under investigation in clinical trial NCT03218826 (PI3Kbeta Inhibitor AZD8186 and Docetaxel in Treating Patients Advanced Solid Tumors With PTEN or PIK3CB Mutations That Are Metastatic or Cannot Be Removed by Surgery).

Kategori:
AminesBenzopyransHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AZD-8330 DB06061
small molecule | CAS: 869357-68-6

AZD-8330 is a potent, selective, orally active MEK inhibitor that blocks signal transduction pathways implicated in cancer cell proliferation and survival. AZD-8330 has shown tumor suppressive activity in multiple preclinical models of human cancer including …

Kategori:
Protein Kinase InhibitorsPyridines
Target Protein:
Mitogen-activated protein kinase kinase kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AZD-8418 DB13102
small molecule | CAS: 1198309-73-7

Azd8418 is under investigation in clinical trial NCT01027234 (This Study Will Assess the Safety and Tolerability of AZD8418 After Single Increasing Oral Doses).

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AZD-8848 DB14868
small molecule | CAS: 866269-28-5

AZD-8848 is under investigation in clinical trial NCT01818869 (To Assess the Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Multiple Doses AZD8848 in Healthy Subjects).

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Toll-like receptor 7
Waktu Paruh-
Vol. Distribusi-
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Genetik -
AZD-9056 DB12594
small molecule | CAS: 345304-65-6

AZD9056 has been used in trials studying the basic science and treatment of Rheumatoid Arthritis.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Target Protein:
P2X purinoceptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AZD-9164 DB12115
small molecule | CAS: 1034978-04-5

AZD9164 has been used in trials studying the basic science and treatment of Chronic Obstructive Pulmonary Disease.

Kategori:
Receptor, Muscarinic M3, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
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AZD-9496 DB15138
small molecule | CAS: 1639042-08-2

AZD-9496 is under investigation in clinical trial NCT02248090 (AZD9496 First Time in Patients Ascending Dose Study).

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-Ring
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
AZD-9684 DB05712
small molecule

AZD-9684 is the first member of a new anti-thrombotic class (CPU inhibitors). It is being developed by AstraZeneca.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Target Protein:
Carboxypeptidase B2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
AZD-9977 DB15418
small molecule | CAS: 1850385-64-6

AZD-9977 is under investigation in clinical trial NCT03843060 (A Phase 1 Study to Assess the Pharmacokinetics of AZD9977 Administered Alone and in Combination With Itraconazole in Healthy Volunteers).

Kategori:
Acids, CarbocyclicBenzene Derivatives
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AZD2066 DB17078
small molecule | CAS: 934282-55-0

Deskripsi belum tersedia.

Kategori:
Gastrointestinal AgentsReceptor, Metabotropic Glutamate 5, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
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Genetik -
AZD2315 DB06540
biotech | CAS: 457937-78-9

The drug AZD2315, an immunosuppressant developed by AstraZeneca, was in Phase 1 clinical trials for the treatment of rheumatoid arthritis but was discontinued during this phase

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AZD3409 DB04893
small molecule

AZD3409 is a farnesyl-transferase inhibitor (FAR) indicated for the treatment of solid tumors. Phase I trials were initiated January 2003, and were ongoing as of February 2004. As of February 2007 the development of AZD3409 had been discontinued.

Target Protein:
Protein farnesyltransferase subunit betaProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha
Waktu Paruh15–20 hours for the…
Vol. Distribusi-
Klirens-
Genetik -
AZD7442 DB15787
biotech

AZD7442 is a combination of SARS-CoV-2 antibodies (AZD8895 + AZD1061) currently undergoing phase I clinical trials for the prevention and treatment of COVID-19.[L15596] It was developed by AstraZeneca with the goal of conferring at least 6 months of protecti…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +9
Waktu Paruh-
Vol. Distribusi-
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Genetik -
AZD8529 DB16073
small molecule | CAS: 1092453-15-0

AZD8529 is under investigation in clinical trial NCT00921804 (Study to Assess the Efficacy, Safety, and Tolerability of AZD8529 in Adult Schizophrenia Patients).

Kategori:
Heterocyclic Compounds, Fused-RingOxazoles
Target Protein:
Metabotropic glutamate receptor 1
Waktu Paruh-
Vol. Distribusi-
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AZD8630 DB19397
biotech

AZD8630 is an experimental drug under investigation, as described in the Phase I clinical study titled "Randomised, Blinded, Placebo-controlled Study to Evaluate the Safety, Tolerability, Pharmacokinetics and Pharmacodynamics (NCT05110976)

Target Protein:
Thymic stromal lymphopoietin
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Azelaic acid Approved DB00548
small molecule | CAS: 123-99-9

Azelaic acid is a saturated dicarboxylic acid found naturally in wheat, rye, and barley. It is also produced by _Malassezia furfur_, also known as _Pityrosporum ovale_, which is a species of fungus that is normally found on human skin. Azelaic acid is effecti…

Kategori:
Acids, AcyclicAnti-Acne PreparationsAnti-Acne Preparations for Topical Use +5
Target Protein:
Thioredoxin reductasePolyprenal reductase3-oxo-5-alpha-steroid 4-dehydrogenase 1 +4
Waktu ParuhThe observed half-l…
Vol. Distribusi-
Klirens-
Genetik -
Azelaprag DB19329
small molecule | CAS: 2049980-18-7

Azelaprag is under investigation in clinical trial NCT06515418 (Efficacy and Safety of Oral Azelaprag Plus Once Weekly Tirzepatide Compared With Tirzepatide Alone in Participants With Obesity Aged 55 Years and Over).

Target Protein:
Apelin receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Azelastine Approved DB00972
small molecule | CAS: 58581-89-8

Azelastine, a phthalazine derivative, is an antihistamine available as an intranasal spray for the treatment of allergic and vasomotor rhinitis and as an ophthalmic solution for the treatment of allergic conjunctivitis.[L8240,L8270] It is a racemic mixture, t…

Kategori:
Anti-Allergic AgentsAntiallergic Agents, Excl. CorticosteroidsAntihistamines for Systemic Use +41
Target Protein:
Histamine H1 receptorHistamine H2 receptorPhospholipase A2 +1
Waktu ParuhBased on intravenou…
Vol. DistribusiAfter intravenous a…
KlirensBased on intravenou…
Genetik -
Azeliragon DB12689
small molecule | CAS: 603148-36-3

Azeliragon has been used in trials studying the treatment of Alzheimer's Disease.

Target Protein:
Advanced glycosylation end product-specific receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Azelnidipine DB09230
small molecule | CAS: 123524-52-7

Azelnidipine is a dihydropyridine calcium channel blocker. It is marketed by Daiichi-Sankyo pharmaceuticals, Inc. in Japan. It has a gradual onset of action and produces a long-lasting decrease in blood pressure, with only a small increase in heart rate, unl…

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAmino Acids +14
Target Protein:
Voltage-dependent L-type calcium channel subunit beta-1
Waktu Paruh16 –28 hours [L1383…
Vol. DistribusiIn a Chinese study …
Klirens-
Genetik -
Azemiglitazone DB16028
small molecule | CAS: 1133819-87-0

Azemiglitazone is under investigation in clinical trial NCT01280695 (A Randomized, Double-blind, Comparator- and Placebo-controlled, Multiple-dose Study to Evaluate the Safety, Tolerability and Efficacy of Three Dose Levels of MSDC-0602 in Type 2 Diabetic Pat…

Kategori:
KetonesSulfur CompoundsThiazoles
Target Protein:
Insulin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Azenosertib DB18028
small molecule | CAS: 2376146-48-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Azficel-T Approved DB11051
biotech

Azficel-T is an autologous cellular product composed of fibroblasts indicated for improvement of the appearance of moderate to severe nasolabial fold wrinkles in adults. Dermal fibroblasts are collected from the post-auricular biopsy tissue and aseptically ex…

Kategori:
Autologous Cultured Cell
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Azidamfenicol DB13294
small molecule | CAS: 13838-08-9

Deskripsi belum tersedia.

Kategori:
AlcoholsAnti-Bacterial AgentsAnti-Infective Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Azidocillin DB08795
small molecule | CAS: 17243-38-8

Azidocillin is a penicillin antibiotic similir to ampicillin.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +8
Target Protein:
Penicillin-binding protein 2aPenicillin-binding protein 1bPenicillin-binding protein 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Azilsartan medoxomil Approved DB08822
small molecule | CAS: 863031-21-4

Azilsartan medoxomil is a prodrug that is broken down to azilsartan, which belongs in the angiotensin-receptor blocking (ARB) drug class. It is a selective AT1 subtype angiotensin II receptor antagonist. Azilsartan medoxomil is a relatively recently-developed…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +18
Target Protein:
Type-1 angiotensin II receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensRenal clearance of …
Genetik -
Azimilide DB04957
small molecule | CAS: 149908-53-2

Azimilide is an investigational class III anti-arrhythmic drug that blocks fast and slow components of the delayed rectifier cardiac potassium channels. It is not approved for use in any country, but is currently in clinical trials in the United States.

Kategori:
Antiarrhythmic agentsAntiarrhythmics, Class IIICalcium-Regulating Hormones and Agents +11
Target Protein:
Potassium voltage-gated channel subfamily E member 1Potassium voltage-gated channel subfamily KQT member 1Voltage-gated inwardly rectifying potassium channel KCNH2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Azintamide DB13992
small molecule | CAS: 1830-32-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1826819-58-2

Azintuxizumab vedotin is under investigation in clinical trial NCT02951117 (A Study of Venetoclax and ABBV-838 Combination Therapy With Dexamethasone in Participants With Multiple Myeloma Whose Cancer Has Come Back or Had No Response to Recent Cancer Treatmen…

Waktu Paruh-
Vol. Distribusi-
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Azithromycin Approved DB00207
small molecule | CAS: 83905-01-5

Azithromycin is a broad-spectrum macrolide antibiotic with a long half-life and a high degree of tissue penetration [A174172]. It was initially approved by the FDA in 1991 [A174175]. It is primarily used for the treatment of respiratory, enteric and genito…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +22
Target Protein:
23S ribosomal RNAProtein-arginine deiminase type-4
Waktu ParuhTerminal eliminatio…
Vol. DistribusiAfter oral administ…
KlirensMean apparent plasm…
Genetik -
Azlocillin Approved DB01061
small molecule | CAS: 37091-66-0

Azlocillin is a semisynthetic ampicillin-derived acylureido penicillin.

Kategori:
Agents that reduce seizure thresholdAmidesAnti-Bacterial Agents +11
Target Protein:
Penicillin-binding protein 1A
Waktu ParuhMean elimination ha…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 123-77-3

Deskripsi belum tersedia.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Azosemide DB08961
small molecule | CAS: 27589-33-9

Azosemide is a loop diuretic used to treat hypertension, edema, and ascites.

Kategori:
AmidesAminesAniline Compounds +7
Waktu ParuhTerminal half life …
Vol. DistribusiPoor affinity for h…
Klirens-
Genetik -
small molecule | CAS: 892497-01-7

Azoximer bromide is under investigation in clinical trial NCT04381377 (Efficacy and Safety of Polyoxidonium® in Hospitalized Patients With Coronavirus Disease COVID-19).

Kategori:
Macromolecular Substances
Waktu Paruh-
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Azoxystrobin DB07401
small molecule | CAS: 131860-33-8

Azoxystrobin is a methoxyacrylate analog and a strobilurin fungicide.

Kategori:
Acids, AcyclicAcrylatesElectron Transport Complex III +2
Target Protein:
Cytochrome c1, heme protein, mitochondrialCytochrome bCytochrome b-c1 complex subunit 1, mitochondrial +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aztreonam Approved DB00355
small molecule | CAS: 78110-38-0

A monocyclic beta-lactam antibiotic originally isolated from Chromobacterium violaceum. It is resistant to beta-lactamases and is used in gram-negative infections, especially of the meninges, bladder, and kidneys. It may cause a superinfection with gram-posit…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
Penicillin-binding protein 3Peptidoglycan synthase FtsIBeta-lactamase +1
Waktu ParuhThe serum half-life…
Vol. Distribusi* 12.6 L
Klirens* 91 mL/min [health…
Genetik -
Azurin-p28 DB17241
biotech | CAS: 897026-25-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBacterial ProteinsMetalloproteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Azvudine DB16407
small molecule | CAS: 1011529-10-4

Azvudine is under investigation in clinical trial NCT04668235 (Study on Safety and Clinical Efficacy of AZVUDINE in COVID-19 Patients (Sars-cov-2 Infected)).

Kategori:
DeoxyribonucleosidesExperimental Unapproved Treatments for COVID-19Nitrogen Compounds +4
Target Protein:
Broad substrate specificity ATP-binding cassette transporter ABCG2ATP-binding cassette sub-family C member 2ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AZX-100 DB06323
biotech | CAS: 1217194-46-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsHeat-Shock ProteinsMolecular Chaperones +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
H subunit of photosynthetic reaction center complexAquaporin ZCytochrome b +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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