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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Hasil Pencarian (15718)

Halaman 77 / 315
small molecule | CAS: 403717-06-6

Bisphosphocin Nu-3 is under investigation in clinical trial NCT02737722 (Topically Applied Bisphosphocin Nu-3 on Infected Diabetic Ulcers of Subjects With Type I or II Diabetes Mellitus).

Waktu Paruh-
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Bithionol Approved DB04813
small molecule | CAS: 97-18-7

Bithionol, formerly marketed as an active ingredient in various topical drug products, was shown to be a potent photosensitizer with the potential to cause serious skin disorders. Approvals of the NDA's for bithionol drug products were withdrawn on October 24…

Kategori:
AnthelminticsAnti-Acne PreparationsAnti-Acne Preparations for Topical Use +10
Target Protein:
Estrogen receptorCalpain-2 catalytic subunitEstrogen receptor beta +1
Waktu Paruh-
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Bitolterol DB00901
small molecule | CAS: 30392-40-6

Bitolterol mesylate was used to treat bronchospasms in asthma and COPD. It is a beta-2-adrenergic receptor agonist. Bitolterol was withdrawn from the market by Elan Pharmaceuticals in 2001.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +15
Target Protein:
Beta-3 adrenergic receptorBeta-2 adrenergic receptor
Waktu Paruh-
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Genetik -
Bitopertin DB12426
small molecule | CAS: 845614-11-1

Bitopertin has been used in trials studying the treatment of Schizophrenia and Obsessive-Compulsive Disorder.

Kategori:
Sulfur Compounds
Waktu Paruh-
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Genetik -
Bivalirudin Approved DB00006
small molecule | CAS: 128270-60-0

Bivalirudin is a synthetic 20 residue peptide (thrombin inhibitor) which reversibly inhibits thrombin. Once bound to the active site, thrombin cannot activate fibrinogen into fibrin, the crucial step in the formation of thrombus. It is administered intravenou…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsAntithrombins +7
Target Protein:
Prothrombin
Waktu Paruh* Normal renal func…
Vol. Distribusi0.2L/kg
Klirens* 3.4 mL/min/kg [No…
Genetik -
Bivatuzumab DB06550
biotech

Bivatuzumab (previously BIWA 4) is a humanized monoclonal antibody against CD44 v6. [A31688,A31689]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
CD44 antigen
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Bixalomer DB15200
small molecule | CAS: 851373-13-2

Bixalomer is under investigation in clinical trial NCT01115985 (A Study to Assess the Effect of ASP1585 on Pharmacokinetics of Atorvastatin in Healthy Volunteers).

Kategori:
Amines
Waktu Paruh-
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biotech | CAS: 1977488-08-6

Bizalimogene ralaplasmid is under investigation in clinical trial NCT03499795 (VGX-3100 Delivered Intramuscularly (IM) Followed by Electroporation (EP) for the Treatment of HPV-16 And/or HPV-18 Related Anal or Anal/peri-anal, High Grade Squamous Intraepitheli…

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Bizaxofusp DB17345
biotech | CAS: 1236019-35-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bizelesin DB12352
small molecule | CAS: 129655-21-6

Bizelesin has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Alkylating DrugsAmidesAntibiotics, Antineoplastic +7
Waktu Paruh-
Vol. Distribusi-
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BJ-001 DB18585
biotech

BJ-001 is a recombinant human interleukin-15/IL-15 receptor alpha complex with linked integrin-binding motif.

Waktu Paruh-
Vol. Distribusi-
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BK-MDA DB12809
small molecule | CAS: 80535-73-5

BK-MDA has been used in trials studying the treatment of Bladder Exstrophy and Urinary Incontinence.

Waktu Paruh-
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BL-1020 DB05687
small molecule

BL-1020 is a first in class novel compound for the treatment of schizophrenia. It is being developed by BioLineRx (BioLine).

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +8
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Black cohosh DB13975
biotech

Black cohosh (_Actaea racemosa_ or _Cimicifuga racemosa_), a member of the buttercup family, is a perennial plant which native to North America. Historical names for this plant include snakeroot, black bugbane, rattleweed, macrotys, and rheumatism weed. Black…

Kategori:
AngiospermsBiological ProductsComplex Mixtures +21
Waktu ParuhApproximately 2h.[A…
Vol. Distribusi-
Klirens-
Genetik -
Black olive Approved DB10547
biotech

Black olive allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Black pepper Approved DB10557
biotech

Black pepper allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Black sea bass Approved DB15547
biotech

Black sea bass allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Black walnut Approved DB10919
biotech

Black walnut allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Black widow spider (_Latrodectus mactans_) antivenin is a treatment for black widow spider bites derived from the serum of healthy horses immunized against black widow spider venom.[L12792]

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Waktu Paruh-
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Black-eyed pea Approved DB10663
biotech

Black-eyed pea allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Blackberry Approved DB10628
biotech

Blackberry allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Blarcamesine DB05592
small molecule | CAS: 195615-83-9

Deskripsi belum tersedia.

Target Protein:
Sigma non-opioid intracellular receptor 1Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Blatella germanica Approved DB10418
biotech

German cockroach allergenic extract is used in allergenic testing.

Kategori:
AllergensAntigensBiological Factors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bleomycin Approved DB00290
small molecule | CAS: 11056-06-7

A complex of related glycopeptide antibiotics from <i>Streptomyces verticillus</i> consisting of bleomycin A2 and B2 (B2 CAS # 9060-10-0). It inhibits DNA metabolism and is used as an antineoplastic, especially for solid tumors. Bleomycin A2 is used as the re…

Kategori:
Amino Acids, Peptides, and ProteinsAntibiotics, AntineoplasticAntineoplastic Agents +11
Target Protein:
DNADNA ligase 1DNA ligase 3
Gen Terkait:
BLMH
Waktu Paruh115 minutes
Vol. Distribusi-
Klirens-
Genetik 1 Varian
Bleomycin A2 DB19091
small molecule | CAS: 11116-31-7

Bleomycin A2 is under investigation in clinical trial NCT00026208 (Combination Chemotherapy Plus Low-dose Radiation Therapy in Treating Patients With Stage I or Stage IIA Hodgkin's Lymphoma).

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Bleomycin A6 DB12992
small molecule | CAS: 37293-17-7

Bleomycin A6 (also known as boanmycin) has been used in trials studying the treatment of Squamous Cell Lung Cancer. It was developed in China as an antineoplastic antibiotic. This drug participated in clinical trials for the treatment of Squamous Cell Lung Ca…

Kategori:
Amino Acids, Peptides, and ProteinsCarbohydratesGlycoconjugates +2
Waktu Paruh-
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Bleselumab DB15253
biotech | CAS: 1453067-91-8

Bleselumab is under investigation in clinical trial NCT02921789 (Study to Assess the Efficacy and Safety of Bleselumab in Preventing the Recurrence of Focal Segmental Glomerulosclerosis in de Novo Kidney Transplant Recipients).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Bleximenib DB19328
small molecule | CAS: 2654081-35-1

Bleximenib is under investigation in clinical trials NCT04811560 (A Phase 1/2 Study of Bleximenib in Participants With Acute Leukemia) and NCT05453903 (A Study of Bleximenib in Combination With Acute Myeloid Leukemia (AML) Directed Therapies)

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Blinatumomab Approved DB09052
biotech | CAS: 853426-35-4

Blinatumomab is a BiTE-class (bi-specific T-cell engager) constructed monoclonal antibody formed by the recombinant fusion of an anti-CD3 single-chain variable fragment (scFV) and an anti-CD19 scFV through a short peptide linker.[A254836,L44311] CD3 is an ant…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
B-lymphocyte antigen CD19T-cell surface glycoprotein CD3 delta chain
Waktu ParuhBlinatumomab has a …
Vol. DistribusiBlinatumomab has a …
KlirensBlinatumomab has an…
Genetik -
Blisibimod DB12330
biotech | CAS: 1236126-45-6

Blisibimod has been used in trials studying the treatment of IgA Nephropathy, Microscopic Polyangiitis, Systemic Lupus Erythematosus, and Granulomatosis With Polyangiitis.

Kategori:
Amino Acids, Peptides, and ProteinsB-Cell Activating FactorImmunologic Factors +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Blonanserin DB09223
small molecule | CAS: 132810-10-7

Blonanserin is an atypical antipsychotic approved in Japan in January, 2008. It offers improved tolerability as it lacks side effects such as extrapyramidal symptoms, excessive sedation, or hypotension. As a second-generation (atypical) antipsychotic, it is s…

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical]) +13
Target Protein:
D(2) dopamine receptorD(3) dopamine receptor5-hydroxytryptamine receptor 2A
Waktu ParuhBlonanserin has a h…
Vol. DistribusiBlonanserin has a V…
KlirensBlonanserin has a c…
Genetik -
Blosozumab DB12560
biotech | CAS: 1132758-87-2

Blosozumab has been used in trials studying the basic science and treatment of Osteoporosis and Osteoporosis, Postmenopausal.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BLS-M22 DB16992
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
BLU-9931 DB17985
small molecule | CAS: 1538604-68-0

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAcrylatesAmides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Blue crab Approved DB10979
biotech

Blue crab allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Blueberry Approved DB10629
biotech

Blueberry allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bluefish Approved DB10613
biotech

Bluefish allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BLXA4 DB12133
small molecule | CAS: 864516-86-9

BLXA4 has been used in trials studying the treatment of Gingival Inflammation.

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BLZ-945 DB16838
small molecule | CAS: 953769-46-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingPyridinesReceptor, Macrophage Colony-Stimulating Factor, antagonists & inhibitors +1
Target Protein:
Granulocyte colony-stimulating factor receptorMacrophage colony-stimulating factor 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BM-3103 DB18056
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BMN-044 DB17003
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BMN-045 DB17004
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BMN-046 DB17005
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BMN-052 DB17006
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
BMN-053 DB17008
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
BMN-055 DB17009
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
BMN-331 DB18324
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
BMN-351 DB18186
biotech

BMN-351 is a fully modified 18-mer oligonucleotide with a TEG modification at its 5' end that binds to exon 51 of dystrophin pre-mRNA. It is under investigation for the treatment of Duchenne Muscular Dystrophy (DMD).

Waktu Paruh-
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BMS-181156 DB02466
small molecule | CAS: 110368-35-9

Deskripsi belum tersedia.

Target Protein:
Retinoic acid receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BMS-184476 DB12633
small molecule | CAS: 160237-25-2

BMS-184476 has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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