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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 77 / 321
Avutometinib DB15254
small molecule | CAS: 946128-88-7

Avutometinib (RO-5126766 free base) is under investigation in clinical trial NCT03875820 (Phase I Trial of VS-6063 and RO5126766.).

Kategori:
BenzopyransHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors +1
Target Protein:
Serine/threonine-protein kinase A-RafSerine/threonine-protein kinase B-rafRAF proto-oncogene serine/threonine-protein kinase
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AVX-001 DB19194
small molecule | CAS: 300553-18-8

AVX-001 is under investigation in clinical trial NCT05164393 (Phase I/iia Trial to Evaluate AVX001 Gel in Doses of 1% or 3% Compared With Vehicle Over Four Weeks of Field-directed Treatment Period in Adult Subjects With AK).

Kategori:
Dietary FatsDietary Fats, UnsaturatedFats +5
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AVX-470 DB18455
biotech

AVX-470 is an anti-tumor necrosis factor (TNF) polyclonal antibody (bovine).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +4
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AVXS-201 DB16997
biotech

Deskripsi belum tersedia.

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AVXS-301 DB17943
biotech

AVXS-301 consists of an adeno-associated virus serotype 9 (AAV9) designed to express the superoxide dismutase 1 (SOD1) gene. It is being investigated for the treatment of Amyotrophic Lateral Sclerosis (ALS).[L47077]

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AX200 DB05093
small molecule

AX200, which has been developed for the treatment of stroke, is the most advanced drug candidate and is halfway through the process of gaining clinical approval. The expression of the endogenous AX200 protein in the brain is increased after brain damage. Thus…

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biotech

Axalimogene filolisbac is under investigation in clinical trial NCT02853604 (Study of ADXS11-001 in Subjects With High Risk Locally Advanced Cervical Cancer).

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Axatilimab Approved DB16388
biotech | CAS: 2155851-88-8

Axatilimab is a humanized IgG4 monoclonal antibody produced in Chinese hamster ovary cells.[L51194] It is targeted against macrophage colony-stimulating factor 1 receptor (CSF-1R), causing a reduction in circulating levels of monocytes and macrophages respons…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Macrophage colony-stimulating factor 1 receptor
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe volume of distr…
KlirensThe total clearance…
Genetik -
Axelopran DB12013
small molecule | CAS: 949904-48-7

Axelopran has been used in trials studying the treatment of OIC and Opioid-induced Constipation.

Kategori:
Acids, CarbocyclicAlkaloidsAmides +5
Target Protein:
Mu-type opioid receptor
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Axicabtagene ciloleucel Approved DB13915
biotech

Axicabtagene ciloleucel is an anti-CD19 chimeric antigen receptor (CAR) T-cell therapy. The drug has a unique mechanism of action, as it utilizes the patient's own T cells, which play a central role in immune response to cancer.[A216163] Once T-cells are coll…

Kategori:
AntigensAntigens, CDAntigens, Differentiation +16
Target Protein:
B-lymphocyte antigen CD19
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Axitinib Approved DB06626
small molecule | CAS: 319460-85-0

Axitinib is a second generation tyrosine kinase inhibitor that works by selectively inhibiting vascular endothelial growth factor receptors (VEGFR-1, VEGFR-2, VEGFR-3).[L6676] Through this mechanism of action, axitinib blocks angiogenesis, tumour growth and m…

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +31
Target Protein:
Tyrosine-protein kinase ABL1Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2 +1
Waktu ParuhAxitinib has a half…
Vol. DistribusiThe volume of distr…
KlirensThe average clearan…
Genetik -
Axomadol DB16100
small molecule | CAS: 187219-99-4

Axomadol is under investigation in clinical trial NCT01043263 (Efficacy and Safety of EN3324 (Axomadol) in Subjects With Chronic Low Back Pain).

Kategori:
AlcoholsCyclohexanesCycloparaffins +3
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AZ-3102 DB18502
small molecule

AZ-3102 is a Biphenyl-substituted L-ido configured deoxynojirimycin derivative

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Azacitidine Approved DB00928
small molecule | CAS: 320-67-2

Azacitidine is a pyrimidine nucleoside analogue with anti-neoplastic activity. It differs from cytosine by the presence of nitrogen in the C5-position, key in its hypomethylating activity.[A1406,A1413,A1415] Two main mechanisms of action have been proposed fo…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
DNA (cytosine-5)-methyltransferase 1RNADNA
Waktu ParuhThe mean half-life …
Vol. DistribusiIn patients given a…
KlirensAzacitidine has an …
Genetik -
AZACYCLONOL DB19381
small molecule | CAS: 115-46-8

Deskripsi belum tersedia.

Target Protein:
Histamine H1 receptor
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Azadirachta indica leaf Approved DB14352
biotech

Azadirachta indica leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Azadirachtin DB19419
small molecule | CAS: 11141-17-6

Azadirachtin is under investigation in clinical trial NCT06617026 (Short-term Outcome of Medical vs. Surgical Management of Chronic Anal Fissure).

Kategori:
AgrochemicalsAzadirachtaCompounds used in a research, industrial, or household setting +5
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Azafenidin DB19031
small molecule | CAS: 68049-83-2

Azafenidin is under investigation in clinical trial NCT01726582 (Pancreas Cancer: Molecular Profiling as a Guide to Therapy Before and After Surgery ("Personalized Medicine")).

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Azanidazole DB13350
small molecule | CAS: 62973-76-6

Deskripsi belum tersedia.

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsGenito Urinary System and Sex Hormones +5
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Azapentacene DB15951
small molecule | CAS: 3863-80-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
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Azaperone DB11376
small molecule | CAS: 1649-18-9

Azaperone is a pyridinylpiperazine and butyrophenone agent that is capable of eliciting neuroleptic sedative and antiemetic effects. It is subsequently employed predominantly as a veterinary tranquilizer and mainly for pigs and elephants. At the same time, th…

Kategori:
Antipsychotic AgentsAntipsychotic Agents (First Generation [Typical])Butyrophenones +11
Target Protein:
D(3) dopamine receptorD(2) dopamine receptor
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Azapetine DB13727
small molecule | CAS: 146-36-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingPeripheral Vasodilators
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Azapropazone DB07402
small molecule | CAS: 13539-59-8

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +13
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Azaribine Approved DB19364
small molecule | CAS: 2169-64-4

Deskripsi belum tersedia.

Kategori:
Aza CompoundsDermatologicalsNucleic Acids, Nucleotides, and Nucleosides +4
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Azasetron DB16837
small molecule | CAS: 123040-69-7

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsAntiemeticsAutonomic Agents +7
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Azatadine Approved DB00719
small molecule | CAS: 3964-81-6

Antihistamines such as azatadine appear to compete with histamine for histamine H1- receptor sites on effector cells. The antihistamines antagonize those pharmacological effects of histamine which are mediated through activation of H1- receptor sites and ther…

Kategori:
Agents that reduce seizure thresholdAnticholinergic AgentsAntihistamines for Systemic Use +10
Target Protein:
Histamine H1 receptor
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Azathioprine Approved DB00993
small molecule | CAS: 446-86-6

Azathioprine is a prodrug of 6-mercaptopurine, first synthesized in 1956 by Gertrude Elion, William Lange, and George Hitchings in an attempt to produce a derivative of 6-mercaptopurine with a better therapeutic index.[A189678,A189687,A189690] Azathioprine is…

Kategori:
AntimetabolitesAntineoplastic and Immunomodulating AgentsAntirheumatic Agents +21
Target Protein:
AmidophosphoribosyltransferaseRas-related C3 botulinum toxin substrate 1
Gen Terkait:
TPMT TPMT TPMT
Waktu ParuhThe half life of az…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik 3 Varian
AZD-0328 DB12145
small molecule | CAS: 220099-91-2

AZD0328 has been used in trials studying the treatment and basic science of Schizophrenia and Alzheimer's Disease.

Kategori:
Receptors, Nicotinic
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
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AZD-0424 DB13088
small molecule | CAS: 692054-06-1

AZD0424 has been used in trials studying the treatment of Advanced Solid Tumours.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
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AZD-1236 DB11961
small molecule | CAS: 459814-89-2

AZD1236 has been used in trials studying the basic science and treatment of Cystic Fibrosis and Chronic Obstructive Pulmonary Disease.

Kategori:
AmidesImidazolesImidazolidines +2
Target Protein:
Macrophage metalloelastase
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AZD-1305 DB11766
small molecule | CAS: 872045-91-5

AZD1305 has been used in trials studying the treatment and basic science of Atrial Flutter, Atrial Fibrillation, and Left Ventricle Function.

Kategori:
Acids, AcyclicAza Compounds
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AZD-1386 DB15333
small molecule | CAS: 942937-80-6

AZD-1386 is under investigation in clinical trial NCT00945178 (Double-blind Placebo-controlled 2-part Study Assessing the Safety, Tolerability and PK of AZD1386 in Healthy Volunteers).

Kategori:
Heterocyclic Compounds, Fused-Ring
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AZD-1480 DB12588
small molecule | CAS: 935666-88-9

AZD1480 has been used in trials studying the treatment of Solid Malignancies, Post-Polycythaemia Vera, Primary Myelofibrosis (PMF), and Essential Thrombocythaemia Myelofibrosis.

Kategori:
Janus Kinase 2, antagonists & inhibitorsJanus Kinases, antagonists & inhibitors
Target Protein:
Tyrosine-protein kinase JAK2
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AZD-1656 DB14810
small molecule | CAS: 919783-22-5

AZD-1656 is under investigation in clinical trial NCT00747175 (A Study to Evaluate Safety, Tolerability and P-Glucose After Multiple Ascending Oral Doses of AZD1656 in Type 2 Diabetes).

Kategori:
AzetinesGlucokinase
Target Protein:
Hexokinase-4
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AZD-1940 DB17077
small molecule | CAS: 881413-29-2

Deskripsi belum tersedia.

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AZD-1981 DB11946
small molecule | CAS: 802904-66-1

AZD1981 has been used in trials studying the treatment and basic science of Asthma, Postmenopausal, Pharmakokinetic, Asthma Patients, and Drug Interaction, among others.

Target Protein:
Prostaglandin D2 receptor 2
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AZD-2066 DB12644
small molecule | CAS: 934282-55-0

AZD2066 has been used in trials studying the treatment and basic science of Pain, Chronic Pain, Reflux Episodes, Neuropathic Pain, and Diabetic Neuropathy, among others.

Target Protein:
Metabotropic glutamate receptor 5
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AZD-3043 DB12576
small molecule | CAS: 579494-66-9

AZD3043 has been used in trials studying the treatment and basic science of Safety, Sedation, Tolerability, and Pharmacokinetics.

Kategori:
Acids, CarbocyclicCentral Nervous System DepressantsHypnotics and Sedatives
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3
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AZD-3759 DB14795
small molecule | CAS: 1626387-80-1

AZD-3759 is under investigation in clinical trial NCT03360929 (Evaluate Safety, Tolerability, Pharmacokinetics and Anti-tumor Activity of AZD3759).

Kategori:
Heterocyclic Compounds, Fused-Ring
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AZD-3839 DB12368
small molecule | CAS: 1227163-84-9

AZD3839 has been used in trials studying the basic science of Safety, Tolerability, Alzheimer's Disease, and Blood Concentration.

Kategori:
Heterocyclic Compounds, Fused-Ring
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AZD-4017 DB14875
small molecule | CAS: 1024033-43-9

AZD-4017 is under investigation in clinical trial NCT01173471 (A Phase IIa Study to Assess the Tolerability, Safety, and Efficacy of AZD4017 for Raised Intra-ocular Pressure).

Kategori:
11-beta-Hydroxysteroid Dehydrogenase Type 1, antagonists & inhibitorsNicotinic AcidsPyridines
Target Protein:
11-beta-hydroxysteroid dehydrogenase 1
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AZD-4547 DB12247
small molecule | CAS: 1035270-39-3

AZD4547 has been used in trials studying the treatment of Cancer, LYMPHOMA, Gastric Cancer, Adenocarcinoma, and Solid Neoplasm, among others.

Target Protein:
Fibroblast growth factor receptor 1
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AZD-4818 DB12002
small molecule | CAS: 1003566-93-5

AZD4818 has been used in trials studying the treatment of Chronic Obstructive Pulmonary Disease (COPD).

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AZD-4877 DB11671
small molecule | CAS: 1176760-49-8

AZD4877 has been used in trials studying the treatment of NHL, Tumors, Cancer, Lymphoma, and Neoplasms, among others.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Kinesin-like protein KIF11
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AZD-5069 DB16822
small molecule | CAS: 878385-84-3

Deskripsi belum tersedia.

Kategori:
AmidesSulfonesSulfur Compounds
Target Protein:
C-X-C chemokine receptor type 2
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AZD-5153 DB17018
small molecule | CAS: 1869912-39-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Bromodomain-containing protein 4
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AZD-5423 DB12280
small molecule | CAS: 1034148-04-3

AZD5423 has been used in trials studying the basic science and treatment of Asthma, Bioavailability and AUC, and Chronic Obstructive Pulmonary Disease (COPD).

Kategori:
AcetatesAcids, AcyclicAmides +4
Target Protein:
Glucocorticoid receptor
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AZD-5672 DB11804
small molecule | CAS: 780750-65-4

Azd5672 has been used in trials studying the basic science and treatment of Pharmacokinetics, Renal Impairment, and Rheumatoid Arthritis.

Kategori:
AcetamidesAmidesAnti-HIV Agents +5
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AZD-5991 DB14792
small molecule | CAS: 2143010-83-5

AZD-5991 is under investigation in clinical trial NCT03218683 (Study of AZD5991 in Relapsed or Refractory Haematologic Malignancies.).

Kategori:
Antineoplastic Agents
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AZD-6280 DB12210
small molecule | CAS: 942436-93-3

AZD6280 has been used in trials studying the basic science of Anxiety.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Opioid, delta, agonists
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-3
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Menampilkan 3801–3850 dari 16004
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