Hasil Filter

14494

Total database: 17430
Struktur (SMILES)
9687 (66.8%)
Target
7525 (51.9%)
Genomik
112 (0.8%)
Referensi
14494 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (14494)

Halaman 76 / 290
Candesartan cilexetil Approved DB00796
small molecule | CAS: 145040-37-5

Candesartan is an angiotensin-receptor blocker (ARB) that may be used alone or with other agents to treat hypertension. It is administered orally as the prodrug, candesartan cilexetil, which is rapidly converted to its active metabolite, candesartan, during a…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAngiotensin 2 Receptor Blocker +16
Target Protein:
Type-1 angiotensin II receptor
Waktu ParuhApproximately 9 hou…
Vol. Distribusi* 0.13 L/kg
Klirens* 0.37 mL/min/kg
Genetik -
Candicidin Approved DB01152
small molecule | CAS: 1403-17-4

Candicidin is an antibiotic obtained from a streptomyces (Streptomyces griseus) and active against some fungi of the genus Candida (C. albicans). Candicidin is administered intravaginally in the treatment of vulvovaginal candidiasis.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntifungal Agents +9
Target Protein:
Ergosterol
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Candida albicans Approved DB10429
biotech

Candida albicans is a fungus which can provoke allergic reactions. Candida albicans is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Candida tropicalis Approved DB10807
biotech

Candida tropicalis is a fungus which can provoke allergic reactions. Candida tropicalis is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Candoxatril DB00616
small molecule | CAS: 123122-55-4

Candoxatril is the orally-active prodrug of candoxatrilat (UK-73967), a potent neutral endopeptidase (NEP) inhibitor.

Kategori:
Acids, AcyclicAntihypertensive AgentsCardiovascular Agents +8
Target Protein:
NeprilysinAngiotensin-converting enzyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Candoxatrilat DB11623
small molecule | CAS: 123122-54-3

A dicarboxylic acid monoamide obtained by formal condensation between the amino group of cis-4-aminocyclohexanecarboxylic acid and the cyclopentanecarboxylic acid group of 1-[(2S)-2-carboxy-3-(2-methoxyethoxy)propyl]cyclopentanecarboxylic acid. A potent inhib…

Kategori:
Acids, CarbocyclicCyclohexanesCycloparaffins +3
Target Protein:
Neprilysin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Canertinib DB05424
small molecule | CAS: 267243-28-7

Canertinib is a pan-erbB tyrosine kinase inhibitor which work against esophageal squamous cell carcinoma in vitro and in vivo. Canertinib treatment significantly affects tumour metabolism, proliferation and hypoxia as determined by PET.

Kategori:
Acids, AcyclicAnestheticsAntineoplastic Agents +10
Target Protein:
Receptor tyrosine-protein kinase erbB-2RAC-alpha serine/threonine-protein kinaseReceptor tyrosine-protein kinase erbB-4 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Canfosfamide DB04972
small molecule | CAS: 158382-37-7

Canfosfamide is an active agent in chemotherapy-resistant ovarian cancer.

Kategori:
Amino Acids, Peptides, and ProteinsCytotoxinsOligopeptides +1
Target Protein:
Glutathione S-transferase P
Waktu Paruh18 min
Vol. Distribusi-
Klirens-
Genetik -
Cangrelor Approved DB06441
small molecule | CAS: 163706-06-7

Cangrelor is an intravenous, direct-acting, reversible P2Y12 inhibitor for patients undergoing percutaneous coronary intervention (PCI) who have not been yet treated by oral P2Y12 inhibitors. An advantage Cangrelor provides over oral P2Y12 inhibitors (such as…

Kategori:
Adenine NucleotidesAnticoagulantsAntiplatelet agents +16
Target Protein:
P2Y purinoceptor 12
Waktu ParuhThe average elimina…
Vol. DistribusiIn a study in healt…
KlirensThe mean clearance …
Genetik -
biotech

Canis lupus familiaris dander is the dander of Canis lupus familiaris. Canis lupus familiaris dander is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Canis lupus familiaris hair Approved DB10867
biotech

Domestic dog hair is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Canis lupus familiaris skin Approved DB10409
biotech

Canis lupus familiaris skin allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cannabichromene DB14735
small molecule | CAS: 20675-51-8

A natural product found in Cannabis sativa and Helichrysum species.

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cannabidiol Approved DB09061
small molecule | CAS: 13956-29-1

Cannabidiol, or CBD, is one of at least 85 active cannabinoids identified within the Cannabis plant. It is a major phytocannabinoid, accounting for up to 40% of the Cannabis plant's extract, that binds to a wide variety of physiological targets of the endocan…

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAnticonvulsants +56
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2G-protein coupled receptor 12 +36
Waktu ParuhThe CBD component o…
Vol. DistribusiCannabinoids are di…
Klirens-
Genetik -
small molecule | CAS: 1244-58-2

Cannabidiolic acid is under investigation in clinical trial NCT04103814 (Effect of Topical CBD Cream for Degenerative Hallux Disorders).

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cannabidivarin DB14050
small molecule | CAS: 24274-48-4

Cannabidivarin, also known as cannabidivarol or CBDV, is a non-psychoactive cannabinoid found within [DB14009]. It is one of over 100 cannabinoids identified from the Cannabis plant that can modulate the physiological activity of cannabis, or marijuana [A3258…

Kategori:
AnticonvulsantsCentral Nervous System DepressantsTerpenes
Target Protein:
Transient receptor potential cation channel subfamily V member 1Transient receptor potential cation channel subfamily V member 2Transient receptor potential cation channel subfamily A member 1 +1
Waktu ParuhOrally administered…
Vol. DistribusiDue to its lipophil…
Klirens-
Genetik -
Cannabigerol DB14734
small molecule | CAS: 25654-31-3

A natural product found in Cannabis sativa and Helichrysum species.

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cannabinol DB14737
small molecule | CAS: 521-35-7

Cannabinol (CBN) is a physiologically inactive constituent of Cannabis sativa.

Kategori:
BCRP/ABCG2 InhibitorsCannabinoids and similarsCytochrome P-450 CYP1A2 Inhibitors +30
Target Protein:
Cannabinoid receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cannabinor DB05048
small molecule | CAS: 573981-31-4

Cannabinor, a synthetic CB2-selective agonist, is in Phase 2 clinical testing as an analgesic.

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cannabivarin DB14736
small molecule | CAS: 33745-21-0

A natural product found in Cannabis sativa.

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Canoctakin DB18195
biotech | CAS: 1019859-03-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Canrenoic acid Approved DB09015
small molecule | CAS: 4138-96-9

Canrenoic acid (as the salt potassium canrenoate) is an aldosterone antagonist. Like spironolactone, it is a prodrug, which is metabolized to canrenone in the body.

Kategori:
Agents causing hyperkalemiaDiureticsFused-Ring Compounds +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Canrenone DB12221
small molecule | CAS: 976-71-6

Canrenone has been used in trials studying the diagnostic of Heart Failure.

Kategori:
Agents causing hyperkalemiaDiureticsFused-Ring Compounds +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cantaloupe Approved DB10514
biotech

Cantaloupe allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cantharidin Approved DB12328
small molecule | CAS: 56-25-7

Cantharidin is a naturally occurring odorless, colorless fatty substance of the terpenoid class that is produced as an oral fluid in the alimentary canal of the male blister beetle.[A32891, A32892] For its natural purpose, the male blister beetle secretes and…

Kategori:
BenzofuransCompounds used in a research, industrial, or household settingEnzyme Inhibitors +4
Target Protein:
Serine/threonine-protein phosphatase PP1-alpha catalytic subunitAryl hydrocarbon receptor
Waktu ParuhLittle pharmacodyna…
Vol. DistribusiAfter oral or IP in…
KlirensLittle pharmacodyna…
Genetik -
biotech | CAS: 400010-39-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 868747-45-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CAP-1 DB08027
small molecule | CAS: 564475-13-4

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capadenoson DB16118
small molecule | CAS: 544417-40-5

Capadenoson is under investigation in clinical trial NCT00518921 (Capadenoson in Angina Pectoris).

Kategori:
Adenosine A receptor agonistsAdenosine A1 Receptor AgonistsAmines +2
Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capecitabine Approved DB01101
small molecule | CAS: 154361-50-9

Capecitabine is an orally-administered chemotherapeutic agent used in the treatment of metastatic breast and colorectal cancers. Capecitabine is a prodrug, that is enzymatically converted to fluorouracil (antimetabolite) in the tumor, where it inhibits DNA sy…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +21
Target Protein:
Thymidylate synthaseDNARNA +1
Gen Terkait:
DPYD DPYD DPYD +4
Waktu ParuhThe elimination hal…
Vol. DistribusiIn colorectal cance…
KlirensIn colorectal cance…
Genetik 7 Varian
Capivasertib Approved DB12218
small molecule | CAS: 1143532-39-1

Hormone receptor (HR) positive, especially estrogen receptor-positive, HER2-negative breast cancer is the most common subtype of metastatic breast cancer, resulting in more than 400,000 deaths annually. Although endocrine-based therapy is the first line of tr…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +13
Target Protein:
RAC-alpha serine/threonine-protein kinaseRAC-beta serine/threonine-protein kinaseRAC-gamma serine/threonine-protein kinase
Waktu ParuhThe half-life of ca…
Vol. DistribusiThe steady-state or…
KlirensThe steady-state or…
Genetik -
Caplacizumab Approved DB06081
biotech | CAS: 915810-67-2

Caplacizumab, firstly called ALX-0081, is a humanized single-variable-domain immunoglobulin consisting of two identical humanized building blocks genetically linked by a three-alanine linker. Caplacizumab was developed by Ablynx, a Sanofi company and FDA appr…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
von Willebrand factor
Waktu ParuhThe reported half-l…
Vol. DistribusiThe reported volume…
KlirensAs the elimination …
Genetik -
Capmatinib Approved DB11791
small molecule | CAS: 1029712-80-8

Capmatinib is a small molecule kinase inhibitor targeted against c-Met (a.k.a. hepatocyte growth factor receptor [HGFR]), a receptor tyrosine kinase that, in healthy humans, activates signaling cascades involved in organ regeneration and tissue repair.[A19912…

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +20
Target Protein:
Hepatocyte growth factor receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -
Capra hircus hair Approved DB10876
biotech

Domestic goat hair is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capra hircus skin Approved DB10604
biotech

Capra hircus skin or pelt is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capravirine DB08502
small molecule | CAS: 178979-85-6

Deskripsi belum tersedia.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +11
Target Protein:
Gag-Pol polyproteinGag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capreomycin Approved DB00314
small molecule | CAS: 11003-38-6

Cyclic peptide antibiotic similar to viomycin. It is produced by Streptomyces capreolus.

Kategori:
Agents that produce neuromuscular block (indirect)Amino Acids, Peptides, and ProteinsAminoglycoside Antibacterials +14
Target Protein:
16S/23S rRNA (cytidine-2'-O)-methyltransferase TlyA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capric acid DB03600
small molecule | CAS: 334-48-5

Decanoic acid is a solid. This compound belongs to the straight chain fatty acids. These are fatty acids with a straight aliphatic chain. The proteins that decanoic acid targets include furin, octanoyltransferase, 3-oxoacyl-[acyl-carrier-protein] synthase 1, …

Kategori:
Anti-Infective AgentsAntifungal AgentsFatty Acids +1
Target Protein:
FurinPeptostreptococcal albumin-binding proteinGlycolipid transfer protein +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2605-79-0

Deskripsi belum tersedia.

Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialPancreatic lipase-related protein 2Ferrichrome-iron receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capromab pendetide Approved DB00089
biotech | CAS: 145464-28-4

Capromab is a Murine IgG1 monoclonal 7E11-C5.3 antibody that recognizes prostate specific membrane antigen (PSMA – also known as glutamate carboxypeptidase 2) from prostate cancer cells and normal prostate tissue. When linked to pendetide, capromab is used as…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +13
Target Protein:
Glutamate carboxypeptidase 2
Waktu Paruh-
Vol. Distribusi* 4 ± 2.1 L
Klirens* 42 +/- 22 mL/hr
Genetik -
Capromorelin DB15205
small molecule | CAS: 193273-66-4

Capromorelin is under investigation in clinical trial NCT00527046 (Effects Of An Oral Growth Hormone Secretagogue In Older Functionally Limited Adults).

Target Protein:
Growth hormone secretagogue receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Caprospinol DB05263
small molecule | CAS: 4952-56-1

Caprospinol (SP-233) is the first drug ever to demonstrate the correlation of clearing beta-amyloid from the brain. It also improves the brain histopathology and recovers memory function.

Kategori:
Acids, AcyclicCholestanesFatty Acids +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 7377-03-9

Deskripsi belum tersedia.

Kategori:
AminesHydroxy AcidsHydroxylamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Caprylic acid DB04519
small molecule | CAS: 124-07-2

Caprylic acid is an eight-carbon chain fatty acid, also known systematically as octanoic acid. It is found naturally in coconuts and breast milk. It is an oily liquid with a slightly unpleasant rancid-like smell that is minimally soluble in water.

Kategori:
Acids, AcyclicFatty AcidsLipids +2
Target Protein:
Peroxisome proliferator-activated receptor alpha3-oxoacyl-[acyl-carrier-protein] synthase 1Acyl-CoA thioesterase I
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 111-87-5

Caprylic alcohol has been used in trials studying the treatment of Essential Tremor.

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingFatty Alcohols +3
Target Protein:
Gap junction alpha-1 protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Caprylyl glycol DB14589
small molecule | CAS: 1117-86-8

Deskripsi belum tersedia.

Kategori:
AlcoholsFatty AlcoholsLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capsaicin Approved DB06774
small molecule | CAS: 404-86-4

Capsaicin is most often used as a topical analgesic and exists in many formulations of cream, liquid, and patch preparations of various strengths; however, it may also be found in some dietary supplements. Capsaicin is a naturally-occurring botanical irritant…

Kategori:
AlkaloidsAlkenesAmides +28
Target Protein:
Transient receptor potential cation channel subfamily V member 1Prohibitin-2
Waktu ParuhFollowing oral inge…
Vol. Distribusi-
Klirens-
Genetik -
Capsicum Approved DB10897
biotech

Capsicum (Chili pepper) allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Capsicum annuum whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 3751–3800 dari 14494
Sebelumnya Halaman 76 / 290 Berikutnya