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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
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17430 (100.0%)

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Halaman 76 / 349
biotech | CAS: 1349719-22-7

Asparaginase _Erwinia chrysanthemi_ is an asparaginase-specific enzyme derived from _Erwinia_ _chrysanthemi_ used as an anticancer agent. It works by depleting the stores of an important amino acid called asparagine, which is involved in DNA synthesis and cel…

Kategori:
AmidohydrolasesAntineoplastic AgentsAsparaginase +7
Waktu ParuhThe apparent half-l…
Vol. DistribusiThe volume of distr…
KlirensThe geometric mean …
Genetik -
biotech | CAS: 9015-68-3

Asparaginase derived from _Escherichia coli_ (L-asparagine amidohydrolase, EC 3.5.1.1) is an enzyme responsible for the metabolism of L-asparagine, by catalyzing L-asparagine into L-aspartic acid and ammonia. It also facilitates the production of oxaloacetate…

Kategori:
AmidohydrolasesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +7
Target Protein:
L-asparagine
Waktu ParuhPlasma half life of…
Vol. DistribusiApparent volume of …
Klirens-
Genetik -
Asparagine Approved DB00174
small molecule | CAS: 70-47-3

A non-essential amino acid that is involved in the metabolic control of cell functions in nerve and brain tissue. It is biosynthesized from aspartic acid and ammonia by asparagine synthetase. (From Concise Encyclopedia Biochemistry and Molecular Biology, 3rd …

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +5
Target Protein:
Sodium-coupled neutral amino acid transportersNeutral amino acid transporter B(0)Asparagine synthetase [glutamine-hydrolyzing] +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asparagus Approved DB10503
biotech

Asparagus allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspartame DB00168
small molecule | CAS: 22839-47-0

Flavoring agent sweeter than sugar, metabolized as phenylalanine and aspartic acid.

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingDiet, Food, and Nutrition +13
Target Protein:
Taste receptor type 1 member 3Taste receptor type 1 member 2Transient receptor potential cation channel subfamily V member 1
Waktu ParuhAt room temperature…
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1Sugar phosphatase YbiVChemotaxis protein CheY
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +2
Target Protein:
Aspartate-semialdehyde dehydrogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspartic acid Approved DB00128
small molecule | CAS: 56-84-8

One of the non-essential amino acids commonly occurring in the L-form. It is found in animals and plants, especially in sugar cane and sugar beets. It may be a neurotransmitter.

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +5
Target Protein:
Glutamate receptor ionotropic, NMDA 2AGlutamate receptor ionotropic, NMDA 2BGlutamate receptor ionotropic, NMDA 1 +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
(S)-2-haloacid dehalogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Aspartate--tRNA(Asp) ligase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 110954-19-3

Aspartyl-alanyl-diketopiperazine is under investigation in clinical trial NCT03349645 (An Open Label Extension Study to Assess the Safety of Long-Term Treatment With Ampion for Severe OA of the Knee).

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspergillus flavus Approved DB10694
biotech

Aspergillus flavus is a fungus which can provoke allergic reactions. Aspergillus flavus extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Fungal Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspergillus fumigatus Approved DB10425
biotech

Aspergillus fumigatus is a fungus which can provoke allergic reactions. Aspergillus fumigatus extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Fungal Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspergillus nidulans Approved DB11022
biotech

Aspergillus nidulans is a fungus which can provoke allergic reactions. Aspergillus nidulans extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspergillus niger var. niger Approved DB10426
biotech

Aspergillus niger var. niger is a fungus which can provoke allergic reactions. Aspergillus niger var. niger extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspergillus oryzae Approved DB10448
biotech

Aspergillus oryzae allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspergillus repens Approved DB10449
biotech

Aspergillus repens is a fungus which can provoke allergic reactions. Aspergillus repens extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspergillus terreus Approved DB10450
biotech

Aspergillus terreus is a fungus which can provoke allergic reactions. Aspergillus terreus extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aspoxicillin DB13816
small molecule | CAS: 63358-49-6

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Astaxanthin DB06543
small molecule | CAS: 472-61-7

Astaxanthin is a keto-carotenoid in the terpenes class of chemical compounds. It is classified as a xanthophyll but it is a carotenoid with no vitamin A activity. It is found in the majority of aquatic organisms with red pigment. Astaxanthin has shown to medi…

Kategori:
AlkenesAnticoagulantsBiological Factors +9
Target Protein:
NF-kappa-B inhibitor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Astegolimab DB16386
biotech | CAS: 2173054-79-8

Astegolimab is under investigation in clinical trial NCT04386616 (A Study to Evaluate the Safety and Efficacy of MSTT1041A (Astegolimab) or UTTR1147A in Patients With Severe COVID-19 Pneumonia).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Inflammatory Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Astemizole Approved DB00637
small molecule | CAS: 68844-77-9

Astemizole is a long-acting, non-sedating second generation antihistamine used in the treatment of allergy symptoms. It was withdrawn from market by the manufacturer in 1999 due to the potential to cause arrhythmias at high doses, especially when when taken …

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseBenzimidazoles +27
Target Protein:
Histamine H1 receptorVoltage-gated inwardly rectifying potassium channel KCNH2Voltage-gated delayed rectifier potassium channel KCNH1 +1
Waktu Paruh1 day
Vol. Distribusi-
Klirens-
Genetik -
Astodrimer DB11854
biotech | CAS: 1379746-42-5

Astodrimer has been used in trials studying the treatment and prevention of Bacterial Vaginosis. It is a lysine-based dendrimer with naphthalene disulfonic acid surface groups.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +10
Target Protein:
Envelope glycoprotein gp160
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AstraZeneca COVID-19 Vaccine Approved DB15656
biotech | CAS: 2420395-83-9

The AstraZeneca COVID-19 Vaccine (previously known as ChAdOx1 nCoV-19 or AZD1222) is one of several vaccines developed in 2020 for the prevention of COVID-19 caused by SARS-CoV-2.[L12669,L32649] The ChAdOx1 viral vector was developed at the University of Oxfo…

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ASTX-029 DB18900
small molecule | CAS: 2095719-92-7

ASTX-029 is under investigation in clinical trial NCT03520075 (Study of ASTX029 in Subjects With Advanced Solid Tumors).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asunaprevir Approved DB11586
small molecule | CAS: 630420-16-5

Asunaprevir, also named BMS-650032, is a potent hepatitis C virus (HCV) NS3 protease inhibitor. It has been shown to have a very high efficacy in dual-combination regimens with daclatasvir in patients chronically infected with HCV genotype 1b.[A32528] It was …

Kategori:
AmidesAntiinfectives for Systemic UseAntiviral Agents +35
Target Protein:
Gag-Pol polyproteinGenome polyprotein
Waktu ParuhClinical pharmacoki…
Vol. DistribusiThe registered volu…
KlirensClinical pharmacoki…
Genetik -
Asundexian DB19088
small molecule | CAS: 2064121-65-7

Asundexian is under investigation in clinical trial NCT05686070 (A Study to Test Asundexian for Preventing a Stroke Caused by a Clot in Participants After an Acute Ischemic Stroke or After a High-risk Transient Ischemic Attack, a So-called Mini Stroke).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Coagulation factor XI
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asunercept DB15160
biotech | CAS: 1450882-18-4

Asunercept is under investigation in clinical trial NCT02853565 (A Study of CAN008 for Newly Diagnosed Glioblastoma Multiforme).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Asvasiran DB05638
biotech | CAS: 870094-26-1

Asvasiran is an siRNA that targets the respiratory syncytial virus (RSV) N gene and inhibits viral replication. It has the potential to treat or prevent RSV infection.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT-001 DB15121
small molecule | CAS: 1355612-71-3

AT-001 is under investigation in clinical trial NCT03062384 (AT-001 for Long-term Preservation of Brain Health in Aging).

Kategori:
Heterocyclic Compounds, Fused-RingPyridinesThiazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT-301 DB16507
biotech

AT-301 was under investigation in clinical trial NCT01675284 to evaluate the safety, reactogenicity, and humoral immune responses to an inactivated H5N1 influenza vaccine

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT-527 DB16451
small molecule | CAS: 2241337-84-6

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicExperimental Unapproved Treatments for COVID-19 +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT-7519 DB08142
small molecule | CAS: 844442-38-2

AT7519 is a selective inhibitor of certain Cyclin Dependent Kinases (CDKs) leading to tumour regression. It is developed by Astex for the treatment of solid tumours and haematological malignancies.

Kategori:
Cyclin-Dependent Kinases, antagonists & inhibitors
Target Protein:
Cyclin-dependent kinase 2Cyclin-dependent kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT-GTX-502 DB17001
biotech

AT-GTX-502 is an experimental, one-time gene therapy that uses AAV9 to deliver a functional copy of CLN3.

Kategori:
Non-Replicating Recombinant, Self-Complementary Adeno-Associated Virus Serotype 9 Containing the Human CLN3 Gene
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT1022 DB04995
small molecule

AT1022 is a hydromorphone skin patch designed to provide rapid and sustained delivery of a potent opiate for the management of severe pain. AT1022 incorporates PassPort(TM) system, developed to deliver protein and peptide drugs, small-molecule drugs, genes a…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT1391 DB05120
small molecule

AT1391 is a daily insulin skin patch designed to provide continuous basal levels of insulin for patients with diabetes.

Target Protein:
Insulin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT2220 DB05200
small molecule

AT2220 is an experimental, oral therapy for the treatment of Pompe disease and belongs to a class of molecules known as pharmacological chaperones. It is a small molecule designed to act as a pharmacological chaperone that specifically binds, stabilizes, and …

Target Protein:
Lysosomal alpha-glucosidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT3022 DB05172
small molecule

AT3022, the Altea Therapeutics’s fentanyl citrate transdermal patch designed to provide safe and rapid management of moderate to severe chronic pain.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT845 DB17638
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AT9283 DB05169
small molecule | CAS: 896466-04-9

AT9283 is an aurora Kinase inhibitor developed by Astex Therapeutics for the treatment of cancer. It was discovered and developed internally using Astex’s fragment-based drug discovery platform, Pyramid.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Aurora kinase BAurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ATA-100 DB18329
biotech

ATA-100 is an adeno-associated virus serotype 9 carrying the human Fukutin-Related protein gene and target sequence of the miR-208a

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atabecestat DB15307
small molecule | CAS: 1200493-78-2

Atabecestat is under investigation in clinical trial NCT02211079 (A Study to Assess Effect of JNJ-54861911 on Pharmacokinetics of Cocktail Representatives for Cytochrome P450 (CYP) 3A4, CYP2B6, CYP2C9, and CYP1A2 Substrates).

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atacicept DB06399
biotech | CAS: 845264-92-8

Atacicept is a recombinant fusion protein combined with the extracellular ligand binding portion of TACI.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ataciguat DB12805
small molecule | CAS: 254877-67-3

Ataciguat has been investigated for the basic science of Aortic Valve Stenosis.

Kategori:
Acids, CarbocyclicAmidesAminobenzoates +5
Target Protein:
Atrial natriuretic peptide receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atagabalin DB12032
small molecule | CAS: 223445-75-8

Atagabalin has been used in trials studying the treatment of Insomnia, Primary Insomnia, and Nonrestorative Sleep.

Kategori:
Acids, AcyclicCycloparaffinsFatty Acids +2
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ataluren Approved DB05016
small molecule | CAS: 775304-57-9

Ataluren is a novel, orally administered drug that targets nonsense mutations. Ataluren is approved for use by the European Medicines Agency to treat Duchenne Muscular Dystrophy in patients aged 5 years and older who are able to walk. More specifically, atalu…

Kategori:
Musculo-Skeletal SystemOAT1/SLC22A6 inhibitorsOAT3/SLC22A8 Inhibitors +3
Target Protein:
Dystrophin
Waktu ParuhAtaluren plasma hal…
Vol. Distribusi-
Klirens-
Genetik -
Atamestane DB12194
small molecule | CAS: 96301-34-7

Atamestane has been used in trials studying the treatment of Breast Cancer, Breast Neoplasms, and Neoplasms, Hormone-Dependent.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesAndrostanes +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atamparib DB19028
small molecule | CAS: 2381037-82-5

Atamparib is under investigation in clinical trial NCT05127590 (RBN-2397 in Combination With Pembrolizumab in Patients With SCCL).

Target Protein:
Protein mono-ADP-ribosyltransferase TIPARP
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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