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11778

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11778 (100.0%)

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Halaman 76 / 236
Colistin Approved DB00803
biotech | CAS: 1066-17-7

Cyclic polypeptide antibiotic from Bacillus colistinus. It is composed of Polymyxins E1 and E2 (or Colistins A, B, and C) which act as detergents on cell membranes. Colistin is less toxic than Polymyxin B, but otherwise similar; the methanesulfonate is used o…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAmino Acids, Peptides, and Proteins +21
Target Protein:
Dihydropteroate synthaseBacterial outer membrane
Waktu Paruh5 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Collagen-polyvinylpyrrolidone is a copolymer generated from a mixture of type I collagen and low-molecular-weight PVP that has undergone ? irradiation[A227733]. It is characterized by antifibrotic, fibrolytic, and immunomodulatory properties[A227733].

Kategori:
AlkenesAmino Acids, Peptides, and ProteinsBiopolymers +11
Waktu Paruh-
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Genetik -
biotech | CAS: 9001-12-1

Collagenase clostridium histolyticum is an enzyme produced by the bacterium Clostridium histolyticum. It is beneficial in the breakdown of collagen plaques for the treatment of Dupuytren's contracture and Peyronie's disease.[L14882] The topical formulation is…

Kategori:
Collagen-specific EnzymeCollagenasesDermatologicals +11
Target Protein:
Collagen alpha-1(I) chainCollagen alpha-1(II) chainCollagen alpha-1(III) chain
Waktu Paruh-
Vol. DistribusiThere is no current…
KlirensClearance informati…
Genetik -
biotech | CAS: 1269764-99-9

Coltuximab ravtansine (SAR3419) targets CD19 and is being investigated for the treatment of acute lymphoblastic leukemia (ALL).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +16
Target Protein:
B-lymphocyte antigen CD19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 117048-59-6

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAntineoplastic Agents, PhytogenicBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Compound 18 DB02715
small molecule | CAS: 31112-66-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +1
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Compound 4-D DB03742
small molecule

Deskripsi belum tersedia.

Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Conatumumab DB11646
biotech | CAS: 896731-82-1

Conatumumab has been used in trials studying the treatment of Sarcoma, Lymphoma, Oncology, Colon Cancer, and Rectal Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Conbercept DB12460
biotech | CAS: 1227158-72-6

Conbercept has been investigated for the basic science of Age-related Macular Degeneration.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Concanamycin A DB14062
small molecule | CAS: 80890-47-7

Concanamycin A is an H+-ATPase (vacuolar) inhibitor.

Kategori:
Anti-Infective AgentsEnzyme InhibitorsLactones +3
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Concord grape Approved DB10875
biotech

Concord grape allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Condoliase DB12793
biotech | CAS: 9024-13-9

Condoliase has been used in trials studying the treatment of Lumbar Disc Disease, Lumbar Vertebra Hernia, and Intervertebral Disc Disease.

Waktu Paruh-
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Conivaptan Approved DB00872
small molecule | CAS: 210101-16-9

Conivaptan is a non-peptide inhibitor of antidiuretic hormone (vasopressin). It was approved in 2004 for hyponatremia (low blood sodium levels) caused by syndrome of inappropriate antidiuretic hormone (SIADH). Conivaptan inhibits both isotypes of the vasopres…

Kategori:
Antidiuretic Hormone Receptor AntagonistsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A Substrates +12
Target Protein:
Vasopressin V1a receptorVasopressin V2 receptor
Waktu Paruh5 hours
Vol. Distribusi-
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Genetik -
Conjugated estrogens Approved DB00286
small molecule | CAS: 12126-59-9

The conjugated estrogens are noncrystalline mixtures of purified female sex hormones obtained either by its isolation from the urine of pregnant mares or by synthetic generation from vegetal material. Both of these products are later conjugated to natrium sul…

Kategori:
Agents causing angioedemaBCRP/ABCG2 SubstratesCOMT Substrates +26
Target Protein:
Estrogen receptor betaEstrogen receptor
Waktu ParuhThe median half-lif…
Vol. DistribusiThe physiological d…
KlirensThe reported normal…
Genetik -
Copanlisib Approved DB12483
small molecule | CAS: 1032568-63-0

Copanlisib is a selective pan-Class I phosphoinositide 3-kinase (PI3K) inhibitor with preferential activity against the alpha and delta isoforms. PI3K, a lipid kinase that activates downstream signalling pathways involved in cell survival and growth, that exi…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +17
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform +1
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Copper Approved DB09130
small molecule | CAS: 7440-50-8

Copper is a transition metal and a trace element in the body. It is important to the function of many enzymes including cytochrome c oxidase, monoamine oxidase and superoxide dismutase [FDA Label]. Copper is commonly used in contraceptive intrauterine devices…

Kategori:
Copper-containing Intrauterine DeviceDecreased Embryonic ImplantationDecreased Sperm Motility +12
Target Protein:
Amyloid-beta precursor proteinAdenosylhomocysteinaseHistone H2B type 1-C/E/F/G/I +143
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Copper gluconate Approved DB11246
small molecule | CAS: 527-09-3

Copper gluconate is a copper salt of D-gluconic acid that displays a light blue to bluish-green color. It is prepared by the reaction of gluconic acid solutions with cupric oxide or basic cupric carbonate. According to the good manufacturing or feeding practi…

Kategori:
Acids, AcyclicCarbohydratesHydroxy Acids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Copper oxodotreotide Cu-64 Approved DB15873
small molecule | CAS: 1426155-87-4

Copper Cu 64 dotatate is a newly approved Cu labeled somatostatin analog and has several advantages over <sup>68</sup>Ga-labeled somatostatin analogs for positron emission tomography (PET).[A220348] Copper Cu 64 dotatate has a longer half-life and can be prod…

Kategori:
Amino Acids, Peptides, and ProteinsCopper RadioisotopesPeptides +4
Target Protein:
Somatostatin receptor type 2
Waktu ParuhThe half-life of Co…
Vol. Distribusi-
Klirens-
Genetik -
Coprelotamab DB16380
biotech | CAS: 2348469-84-9

Coprelotamab is under investigation in clinical trial NCT04170595 (Clinical Study of Recombinant Anti-her2 Humanized Monoclonal Antibody for Injection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coprogen DB01747
small molecule | CAS: 31418-71-0

Deskripsi belum tersedia.

Kategori:
AminesHydroxy AcidsHydroxylamines +1
Target Protein:
Iron(3+)-hydroxamate-binding protein FhuD
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Biological FactorsHeterocyclic Compounds, Fused-RingPigments, Biological +1
Target Protein:
Uroporphyrinogen decarboxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2624-63-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingPorphyrinogensPorphyrins
Target Protein:
Uroporphyrinogen decarboxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coptisine DB19308
small molecule | CAS: 3486-66-6

Deskripsi belum tersedia.

Kategori:
AlkaloidsBenzylisoquinolinesBerberine Alkaloids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Corcorus capsularis fiber Approved DB10711
biotech

Corcorus capsularis fiber is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Cordycepin DB12156
small molecule | CAS: 73-03-0

Cordycepin has been used in trials studying the treatment of Leukemia.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntineoplastic Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 73-04-1

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesDeoxyribonucleotidesHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Poly(A) polymerase alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Corifollitropin alfa Approved DB09066
biotech | CAS: 195962-23-3

Corifollitropin alfa, also known as _Elonva_ is used in women undergoing fertility treatment to stimulate the development of more than one mature egg (oocyte) at a time in the ovaries. This drug used together with _a gonadotropin-releasing hormone (GnRH) anta…

Kategori:
Drugs that are Mainly Renally ExcretedFollicle Stimulating HormoneGenito Urinary System and Sex Hormones +9
Target Protein:
Follicle-stimulating hormone receptor
Waktu ParuhCorifollitropin alf…
Vol. DistribusiDistribution, metab…
Klirens0.13 L/h (0.10-0.18…
Genetik -
Corn Approved DB10572
biotech

Corn allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CoronaVac DB15806
biotech

CoronaVac, previously known as PiCoVacc, is a SARS-CoV-2 purified, inactivated, and adsorbed vaccine candidate developed by SinoVac Biotech Corporation[A219758]. It was developed by propagating the SARS-CoV-2 CN2 strain inside Vero Cells and inactivating it w…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Corticorelin DB05394
small molecule | CAS: 86784-80-7

Corticotropin-releasing factor is studied in the treatment of brain cancer. It is made naturally by the hypothalamus (a part of the brain) and can also be made in the laboratory. Human corticotropin-releasing factor may help reduce symptoms caused by edema (s…

Kategori:
Amino Acids, Peptides, and ProteinsCorticotropin-Releasing HormoneDiagnostic Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 121249-14-7

Corticorelin, available commercially as corticorelin ovine triflutate (tradename Acthrel), is a synthetic form of the peptide human corticotropin-releasing hormone (hCRH), a potent stimulator of adrenocorticotropic hormone (ACTH) release from the anterior pit…

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsHormones +9
Target Protein:
Corticotropin-releasing factor receptor 1Corticotropin-releasing factor receptor 2
Waktu ParuhPlasma half-lives f…
Vol. DistribusiThe mean volume of …
Klirens95 ± 11 L/m2/day
Genetik -
Corticosterone DB04652
small molecule | CAS: 50-22-6

An adrenocortical steroid that has modest but significant activities as a mineralocorticoid and a glucocorticoid. (From Goodman and Gilman&#39;s The Pharmacological Basis of Therapeutics, 8th ed, p1437)

Kategori:
11-HydroxycorticosteroidsAdrenal Cortex HormonesAnti-Inflammatory Agents +11
Target Protein:
11-beta-hydroxysteroid dehydrogenase 1Glucocorticoid receptorNuclear receptor coactivator 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Corticotropin Approved DB01285
biotech | CAS: 12427-33-7

Corticotropin (ACTH or adrenocorticotropic hormone) is a polypeptide hormone produced and secreted by the pituitary gland. It is an important player in the hypothalamic-pituitary-adrenal axis.

Kategori:
Adrenal Cortex HormonesAdrenocorticotropic HormoneAmino Acids, Peptides, and Proteins +27
Target Protein:
Adrenocorticotropic hormone receptorCorticoliberin
Waktu ParuhAbout 15 minutes fo…
Vol. Distribusi-
Klirens-
Genetik -
Cortisone DB14681
small molecule | CAS: 53-06-5

A naturally occurring glucocorticoid. It has been used in replacement therapy for adrenal insufficiency and as an anti-inflammatory agent. Cortisone itself is inactive. It is converted in the liver to the active metabolite hydrocortisone. (From Martindale, Th…

Kategori:
17-HydroxycorticosteroidsAdrenal Cortex HormonesAnti-Inflammatory Agents +21
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cortisone acetate Approved DB01380
small molecule | CAS: 50-04-4

Cortisone acetate was first isolate in 1935 and became more widely researched in 1949.[A226295] Since then, glucocorticoids such as cortisone acetate have been used to treat a number of inflammatory conditions such as endocrine, rheumatic, collagen, dermatolo…

Kategori:
17-HydroxycorticosteroidsAdrenal Cortex HormonesAdrenals +25
Target Protein:
Steroid hormone receptor ERR2Estrogen-related receptor gammaGlucocorticoid receptor +2
Waktu Paruh-
Vol. Distribusi-
KlirensData regarding the …
Genetik -
Corydalis ambigua tuber Approved DB14279
biotech

Corydalis ambigua tuber is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
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Corynebacterium diphtheriae Approved DB09877
biotech

*Corynebacterium diphtheriae* toxin is extracted from the pathogenic actinobacterium *C. diphtheriae* that causes diphtheria. The bacteria culture is grown in a medium and through purification, diphtheria toxin is detoxified with formaldehyde and diafiltered.…

Kategori:
Inactivated Corynebacterium Diphtheriae Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1272033-67-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsDiphtheria ToxinInactivated Pneumococcal Vaccine +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 308079-75-6

Deskripsi belum tersedia.

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBacterial Vaccines +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cosfroviximab DB17774
biotech | CAS: 1792982-57-0

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Cosibelimab DB15770
biotech | CAS: 2216751-26-5

Deskripsi belum tersedia.

Kategori:
Immune Checkpoint Inhibitors
Target Protein:
Programmed cell death 1 ligand 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
COTI-2 DB17507
small molecule | CAS: 1039455-84-9

Deskripsi belum tersedia.

Target Protein:
Cellular tumor antigen p53
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2246424-95-1

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector TherapiesAmino Acids, Peptides, and ProteinsGenetic Phenomena +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cotsiranib DB18404
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Cotton Approved DB10707
biotech

Cotton allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coumaphos DB11390
small molecule | CAS: 56-72-4

This drug is a fat-soluble phosphorothioate agent that kills both insects and mites. It is non-volatile in nature and is well known by a variety of names as such a _dip_ or _wash_. Coumaphos is widely used for both farm and domestic animals to control ticks, …

Kategori:
AgrochemicalsAnthelminticsAnti-Infective Agents +22
Waktu Paruh-
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Klirens-
Genetik -
Coumarin 120 DB08168
small molecule | CAS: 26093-31-2

Deskripsi belum tersedia.

Kategori:
BenzopyransCompounds used in a research, industrial, or household settingHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Peptidyl-prolyl cis-trans isomerase APeptidyl-prolyl cis-trans isomerase APeptidyl-prolyl cis-trans isomerase F, mitochondrial +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Covax-19™ DB15846
biotech

Covax-19™, a protein-based vaccine, was developed through partnership between APC and Vaxine. It uses an insect-cell-produced recombinant SARS-CoV-2 spike protein and Vaxine’s adjuvant, Advax-SM. This adjuvant is designed to circumvent high fevers, fatigue, a…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

COVID-19 Spike-GM-CSF Protein Lactated Ringer's Injection is an intradermal injection currently being investigated in the clinical trial NCT03348670 (Discovery Stage (Proof-of-concept) COVID-19 Antigen Presentation Therapeutic Biologics (COVID-19--AP) (AP-TP-…

Waktu Paruh-
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Genetik -
CoviGlobulin DB15747
biotech

CoviGlobulin, a rabbit polyclonal antibody, was specifically designed as a potential therapy for COVID-19. Rabbit polyclonal antibodies are derived from the rabbit, a common animal host for polyclonal production. The antibodies themselves are produced in resp…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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