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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
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16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 76 / 321
Avadomide DB14857
small molecule | CAS: 1015474-32-4

Avadomide is under investigation in clinical trial NCT02031419 (Novel Combinations of CC-122, CC-223, CC-292, and Rituximab in Diffuse Large B-cell Lymphoma and Follicular Lymphoma).

Kategori:
Heterocyclic Compounds, Fused-RingPiperidinesQuinazolines
Target Protein:
Protein cereblon
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Avagacestat DB11893
small molecule | CAS: 1146699-66-2

Avagacestat has been investigated for the basic science and treatment of Alzheimer Disease.

Kategori:
AmidesAmyloid Precursor Protein Secretases, antagonists & inhibitorsEnzyme Inhibitors +4
Target Protein:
Gamma-secretase subunit APH-1ANicastrinGamma-secretase subunit APH-1B +2
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Avalglucosidase alfa Approved DB16099
biotech | CAS: 1802558-87-7

Avalglucosidase alfa, or NeoGAA, is a drug for enzyme replacement therapy specifically designed for Pompe disease, a rare inherited neuromuscular disorder caused by the deficiency of the alpha-glucosidase (GAA) enzyme. GAA is an essential enzyme that hydrolyz…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +2
Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu ParuhThe mean avalglucos…
Vol. DistribusiThe volume of distr…
KlirensThe mean avalglucos…
Genetik -
biotech | CAS: 2227000-30-6

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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Avanafil Approved DB06237
small molecule | CAS: 330784-47-9

Avanafil is a phosphodiesterase-5 (PDE5) inhibitor used in the treatment of erectile dysfunction. In comparison with other drugs of the same class, it shows greater selectivity for PDE5 over PDE6 than both [sildenafil] and [vardenafil] but less selectivity th…

Kategori:
BCRP/ABCG2 InhibitorsCytochrome P-450 CYP2C9 SubstratesCytochrome P-450 CYP3A Substrates +9
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesterase
Waktu ParuhStudies have demons…
Vol. DistribusiThe apparent volume…
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Avapritinib Approved DB15233
small molecule | CAS: 1703793-34-3

Avapritinib, or BLU-285,[A189327] is a selective tyrosine kinase inhibitor of KIT and platelet derived growth factor receptor alpha indicated for the treatment of unresectable, metastatic gastrointestinal stromal tumors and advanced systemic mastocytosis.[A18…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +17
Target Protein:
Platelet-derived growth factor receptor alphaMast/stem cell growth factor receptor Kit
Waktu ParuhThe half life of av…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent o…
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Avasimibe DB06442
small molecule | CAS: 166518-60-1

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicAmides +14
Target Protein:
Liver carboxylesterase 1
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Avasopasem DB18481
small molecule

Deskripsi belum tersedia.

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small molecule | CAS: 435327-40-5

Avasopasem manganese, also known as GC4419, is a highly-selective small molecule mimetic of superoxide dismutase (SOD) being investigated for the reduction of radiation-induced severe oral mucositis.[L27246, L27256] This drug has potential application for rad…

Kategori:
AntioxidantsFree Radical Scavengers
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Avatrombopag Approved DB11995
small molecule | CAS: 570406-98-3

Avatrombopag (_Doptelet_), is an orally administered, small molecule thrombopoietin receptor (c-Mpl) agonist that increases platelet number without increasing platelet activation,[A33097,L2824] thereby decreasing the need for blood transfusions.[L2824] Patien…

Kategori:
BCRP/ABCG2 InhibitorsBlood and Blood Forming OrgansCytochrome P-450 CYP2C8 Inducers +14
Target Protein:
Thrombopoietin receptor
Waktu ParuhThe mean plasma eli…
Vol. DistribusiAvatrombopag has an…
KlirensThe mean (%CV) of t…
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AVB-001 DB18452
biotech

AVB-001 is an encapsulated, engineered human ARPE-19 cell line that constitutively expresses the native human IL-2 cytokine

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AVB-101 DB18416
biotech

AVB-101 is a recombinant AAV9 vector encoding the human progranulin (PGRN) gene.

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Avdoralimab DB16392
biotech | CAS: 2226393-85-5

Avdoralimab is under investigation in clinical trial NCT04333914 (Prospective Study in Patients With Advanced or Metastatic Cancer and Sars-cov-2 Infection).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Inflammatory Agents +9
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AVE-2865 DB07396
small molecule | CAS: 648917-13-9

Deskripsi belum tersedia.

Target Protein:
Glycogen phosphorylase, liver form
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AVE9633 DB06318
biotech

AVE9633 is an anti-CD33 monoclonal antibody-DM4 conjugate.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +14
Target Protein:
Myeloid cell surface antigen CD33
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Avelumab Approved DB11945
biotech | CAS: 1537032-82-8

Avelumab is a human IgG1 lambda monoclonal antibody that binds programmed cell death ligand-1 (PD-L1) to block its interaction with its receptors found on T cells and antigen-presenting cells.[A261496] Avelumab was first approved by the FDA on March 23, 2017.…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Programmed cell death 1 ligand 1
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe geometric mean …
KlirensThe total systemic …
Genetik -
Avena sativa flowering top Approved DB14253
biotech

Avena sativa flowering top is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Avenciguat DB18882
small molecule | CAS: 1579514-06-9

Avenciguat is under investigation in clinical trial NCT05282121 (A Study to Test Whether BI 685509 Alone or in Combination With Empagliflozin Helps People With Liver Cirrhosis Caused by Viral Hepatitis or Non-alcoholic Steatohepatitis (NASH) Who Have High Blo…

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Avexitide DB14806
small molecule | CAS: 133514-43-9

Avexitide is under investigation in clinical trial NCT02996812 (Evaluation of Single Ascending Doses of Subcutaneous Exendin 9-39 in Patients With Post-Bariatric Hypoglycemia).

Kategori:
Amino Acids, Peptides, and ProteinsGlucagon-Like Peptide 1Peptides
Target Protein:
Glucagon-like peptide 1 receptor
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AVI-014 DB17086
biotech

AVI-014 is a glycosylated, recombinant human granulocyte colony-stimulating factor (G-CSF).

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AVI-4020 DB05873
small molecule

AVI-4020 is a neugene antisense drug candidate for the treatment of patients with acute West Nile virus disease who have serious neurological impairment (WNV neuroinvasive disease).

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AVI-4065 DB05620
small molecule

AVI-4065, a phosphorodiamidate Morpholino oligomer (PMO), is an investigational antisense HCV drug. It was developed by Sarepta Therapeutics, Inc. After phase II trials it was cancelled due to lack of potency. [L2917]

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AVI-4557 DB05447
small molecule

AVI-4557 is an oral antisense compound that selectively inhibits the metabolic enzyme cytochrome P450 3A4 (CYP), a liver enzyme responsible for the metabolism or breakdown of approximately half of currently marketed drugs. Studies indicate that AVI-4557 can s…

Target Protein:
Hepatocyte nuclear factor 4-alpha
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AVI-5126 DB05726
small molecule

AVI-526 is an improved formulation of [AVI-4557], developed for use on Vein Grafts before use in Heart by-Pass Graft Surgery. AVI-526 works by silencing a gene known as c-myc, a key regulatory gene involved in cardiovascular restenosis. The drug was under inv…

Kategori:
MorpholinesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
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AVI-7287 DB17799
biotech

Deskripsi belum tersedia.

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AVI-7288 DB17800
biotech

Deskripsi belum tersedia.

Kategori:
MorpholinesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
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AVI-7537 DB15433
biotech

AVI-7537 is an antisense molecule that binds to the Ebola virus mRNA to prevent the viral replication.[L46207] AVI-7537 is under investigation in clinical trial NCT01593072 (A Study to Assess the Safety, Tolerability and Pharmacokinetics of AVI-7537 in Health…

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Avibactam Approved DB09060
small molecule | CAS: 1192500-31-4

Avibactam is a non-?-lactam ?-lactamase inhibitor that is available in combination with ceftazidime (Avycaz). This combination was approved by the FDA on February 25, 2015 for the treatment of complicated intra-abdominal infections in combination with metroni…

Kategori:
Anti-Infective AgentsAza Compoundsbeta-Lactamase Inhibitors +2
Target Protein:
Beta-lactamase TEMBeta-lactamase CTX-MBeta-lactamase +7
Waktu ParuhCeftazidime-avibact…
Vol. DistribusiThe steady state vo…
KlirensAvibactam and cefta…
Genetik -
Avicin D DB17240
small molecule | CAS: 197787-20-5

Deskripsi belum tersedia.

Kategori:
CarbohydratesGlycosides
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AVID-200 DB18454
biotech | CAS: 2269485-28-9

AVID-200 is an Anti-transforming growth factor beta (TGF-?) trap fusion protein.

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Avidin DB15228
biotech | CAS: 110539-97-4

Avidin is under investigation in clinical trial NCT00345618 (Clinical Study Assessing Idrabiotaparinux Sodium Injections Once-weekly in Pulmonary Embolism Therapeutic Approach).

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsAnimal Proteins, Dietary +10
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Avilamycin DB11375
small molecule | CAS: 11051-71-1

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCarbohydrates +2
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Aviptadil DB06260
small molecule | CAS: 40077-57-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsErectile DysfunctionGastrointestinal Hormones +9
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Aviscumine DB12684
biotech | CAS: 223577-45-5

Cy 503 is under investigation in clinical trial NCT00658437 (Aviscumine for the Treatment of Malignant Melanoma Stage IV After Failure of Prior Therapy).

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsBiological Factors +12
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Avizakimab DB18842
biotech | CAS: 2229685-51-0

Avizakimab is under investigation in clinical trial NCT03371251 (Study of BOS161721 in Systemic Lupus Erythematosus (SLE) Patients on a Background of Limited Standard of Care).

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AVL-3288 DB18707
small molecule | CAS: 917837-54-8

Deskripsi belum tersedia.

Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
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AVN-944 DB05500
biotech

AVN944 is a biotech drug that demonstrated a statistically meaningful impact on IMPDH and other proteins that are critical to activities in cancer cells, including nucleotide biosynthesis, energy and metabolism, DNA replication, apoptosis and cell cycle contr…

Kategori:
Acids, AcyclicAmidesBenzene Derivatives +1
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Avobenzone Approved DB09495
small molecule | CAS: 70356-09-1

Avobenzone is dibenzoyl methane derivative. It is oil soluble ingredient. Avobenzone has the ability to absorb ultraviolet light over wider range of wavelengths. It is included in many commercially available sunscreens which are used as wide spectrum sunscree…

Kategori:
Compounds used in a research, industrial, or household settingCosmeticsDermatologicals +4
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Avoplacel DB18659
biotech

Avoplacel (PLX-R18) is an allogeneic cell therapy under investigation for the treatment of acute radiation syndrome.[L48370]

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Avoralstat DB12120
small molecule | CAS: 918407-35-9

Avoralstat has been used in trials studying the prevention of HAE and Hereditary Angioedema.

Kategori:
Acids, CarbocyclicAlkenesAmides +6
Target Protein:
Kallikrein-2Kininogen-1
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Avotaciclib DB16652
small molecule | CAS: 1983983-41-0

Avotaciclib is under investigation in clinical trial NCT03579836 (Evaluation of Safety and Efficacy in BEY1107 in Monotherapy Gemcitabine Combination in Patient With Pancreatic Cancer).

Target Protein:
Cyclin-dependent kinase 1
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Avotermin DB11955
biotech | CAS: 182212-66-4

Juvista has been investigated for the treatment, prevention, and basic science of Scars, Keloid, and Cicatrix.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
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AVP-21D9 DB17798
biotech

AVP-21D9 is a fully human anthrax monoclonal antibody that is being investigated as an anthrax antitoxin.[A259522]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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AVR-48 DB18294
small molecule | CAS: 3459-18-5

Deskripsi belum tersedia.

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AVR-RD-01 DB17651
biotech

AVR-RD-01 is an investigational _ex vivo_ lentiviral gene therapy developed by AVROBIO Inc. It consists of autologous CD34+ cells that transduced with Lentiviral Vector/alpha-galactosidase A (AGA) encoding for the human AGA complementary deoxyribonucleic acid…

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AVR-RD-02 DB17650
biotech

AVR-RD-02 is an investigational _ex vivo_ lentiviral gene therapy developed by AVROBIO Inc. It consists of autologous CD34+ enriched hematopoietic stem cells (HSCs) that have been genetically modified _ex vivo_ with a lentiviral vector (LV) to contain a ribon…

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AVR-RD-04 DB18644
biotech

AVR-RD-04 is an investigational gene therapy for cystinosis. It consists of autologous CD34+ enriched cells transduced with a lentiviral vector containing RNA resulting in codon-optimized cDNA encoding for functional human cystinosin.

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AVR-RD-05 DB18631
biotech

AVR-RD-05 is a gene therapy comprising genetically modified autologous stem cells transduced _ex vivo_ with a lentiviral vector encoding the human iduronate-2-sulfatase (IDS) enzyme. It is under investigation for the treatment of Hunter Syndrome (Mucopolysacc…

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AVR118 DB04979
biotech

AVR118 represents a new type of biopolymer chemistry that also possesses novel immunomodulator activity. This non-toxic peptide-nucleic acid, which to date has shown no indication of human toxicity, appears to stimulate the proinflammatory responses required …

Kategori:
HIVNucleic Acids, Nucleotides, and NucleosidesNucleotides +2
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AVS-100 DB18068
small molecule | CAS: 2245942-72-5

Deskripsi belum tersedia.

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