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11778

Total database: 17430
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8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
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11778 (100.0%)

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Halaman 75 / 236
Clove Approved DB10672
biotech | CAS: 84961-50-2

Clove allergenic extract is used in allergenic testing.

Kategori:
AngiospermsBiological ProductsCell-mediated Immunity +12
Waktu Paruh-
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Clove oil Approved DB11338
biotech | CAS: 8000-34-8

Clove oil is obtained by extraction from the dried flower buds of the clove plant. Traditionally, it has been used as a flavouring spice in foods, or as a fragrance. It is also found in topical analgesics. Clove oil has shown to exert some antimicrobial activ…

Kategori:
Biological ProductsComplex MixturesDrugs that are Mainly Renally Excreted +3
Target Protein:
Vascular cell adhesion protein 1C-X-C motif chemokine 10Collagen alpha-1(I) chain +1
Waktu ParuhIn a pharmacokineti…
Vol. Distribusi-
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Genetik -
Cloxacillin Approved DB01147
small molecule | CAS: 61-72-3

A semi-synthetic penicillin antibiotic which is a chlorinated derivative of [oxacillin].

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
D-alanyl-D-alanine carboxypeptidase DacAPenicillin-binding protein 2XPenicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clozapine Approved DB00363
small molecule | CAS: 5786-21-0

Clozapine is a tricyclic dibenzodiazepine, classified as an atypical antipsychotic agent.[A256708] Clozapine displays affinity to various neuroreceptors with a particularly low affinity to the dopamine receptors, thus breaking the mold of first-generation ant…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +65
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2AD(1A) dopamine receptor +30
Gen Terkait:
GNB3
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe median volume o…
KlirensThe median clearanc…
Genetik 1 Varian
CM-4307 DB15414
small molecule | CAS: 1130115-44-4

CM-4307 is under investigation in clinical trial NCT03602495 (Donafenib in 131I-Refractory Differentiated Thyroid Cancer).

Waktu Paruh-
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CM4620 DB16466
small molecule | CAS: 1713240-67-5

CM4620 (Zegocractin), is under investigation in multiple clinical trials, including NCT04195347 (pancreatitis due to asparaginase), NCT03709342 (PK/PD study in acute pancreatitis), NCT03401190 and NCT04681066 (pancreatitis and SIRS), and NCT04661540 (critical…

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CMX-2043 DB12795
small molecule | CAS: 910627-26-8

CMX-2043 has been used in trials studying the treatment and prevention of Non STEMI, Unstable Angina, Stable Coronary Artery Disease, and Percutaneous Coronary Intervention.

Kategori:
Amino Acids, Peptides, and ProteinsCoenzymesEnzymes and Coenzymes +6
Target Protein:
RAC-alpha serine/threonine-protein kinaseHepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
CN-105 DB18345
small molecule | CAS: 1632243-07-2

CN-105 is a neuroprotective pentapeptide with the sequence Acetyl-Valine-Serine-Arginine-Arginine-Arginine-NH2 (Ac-VSRRR- NH2).

Waktu Paruh-
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CN-201 DB18726
biotech

CN-201 is a humanized anti-CD3/CD19 bispecific antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CNDO-109 DB17290
biotech

CNDO-109 are CNDO-109-activated allogeneic natural killer cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CNM-Au8 DB17952
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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CNV-2197944 DB15229
small molecule | CAS: 1204535-44-3

CNV-2197944 is under investigation in clinical trial NCT01893125 (Efficacy and Safety of CNV2197944 Versus Placebo in Patients With Diabetic Peripheral Neuropathy).

Target Protein:
Voltage-dependent N-type calcium channel subunit alpha-1B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serotonin N-acetyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 102786-61-8

Recombinant human coagulation Factor VIIa (rFVIIa), intended for promoting hemostasis by activating the extrinsic pathway of the coagulation cascade. NovoSeven is a vitamin K-dependent glycoprotein consisting of 406 amino acid residues. Cloned and expressed i…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +15
Target Protein:
Coagulation factor XTissue factor
Waktu Paruh-
Vol. Distribusi* 121 ± 30 mL/kg [a…
Klirens* 33 - 37 mL/h x kg…
Genetik -
Coagulation factor X human Approved DB13148
biotech

Coagulation Factor X (Human), is a plasma-derived human blood coagulation factor is used by adults and children (aged 12 years and above) with hereditary Factor X deficiency. However its use is limited in the perioperative setting for the management of bleedi…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +11
Waktu ParuhFollowing a single …
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
biotech | CAS: 9013-55-2

Coagulation factor XIa is under investigation in clinical trial NCT01701947 (HEMOLEVEN® Expanded Access Program Prevention of Surgical/Postpartum Hemorrhage Severe Inherited Factor XI Deficiency).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coagulin-B DB17703
biotech

Coagulin-B is an adeno-associated viral vector expressing human blood-coagulation Factor IX.[A259038, A259043] It was previously investigated for the treatment of hemophilia; however, the manufacturing company discontinued the Phase I trial in 2004, halting i…

Waktu Paruh-
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Coal tar Approved DB11082
small molecule | CAS: 8007-45-2

Coal tar is a brown or black liquid of extremely high viscosity. Coal tar is among the by-products when coal is carbonized to make coke or gasified to make coal gas. Coal tars are complex and variable mixtures of phenols, polycyclic aromatic hydrocarbons (PAH…

Kategori:
Complex MixturesDermatologicalsKeratolytic Agents +2
Waktu ParuhIntended for local …
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
Cobalamin DB14098
small molecule | CAS: 13408-78-1

Deskripsi belum tersedia.

Kategori:
CorrinoidsHeterocyclic Compounds, Fused-RingMicronutrients +3
Waktu Paruh-
Vol. Distribusi-
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Cobalt Approved DB14574
small molecule | CAS: 7440-48-4

A trace element that is a component of vitamin B12. It has the atomic symbol Co, atomic number 27, and atomic weight 58.93. It is used in nuclear weapons, alloys, and pigments. Deficiency in animals leads to anemia; its excess in humans can lead to erythrocyt…

Kategori:
Cell-mediated ImmunityDiet, Food, and NutritionElements +9
Waktu Paruh-
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Cobalt chloride Approved DB14206
small molecule | CAS: 7646-79-9

Deskripsi belum tersedia.

Kategori:
Antimutagenic AgentsCompounds used in a research, industrial, or household settingElements +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobalt Co-60 DB15374
small molecule | CAS: 10198-40-0

Cobalt Co-60 is under investigation in clinical trial NCT02891083 (Adjuvant Therapies or Surgery Alone for High Risk pN0 Esophageal Cancer).

Kategori:
Cobalt IsotopesElementsIsotopes +4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 10124-43-3

Deskripsi belum tersedia.

Kategori:
ElementsMetalsMetals, Heavy +1
Waktu Paruh-
Vol. Distribusi-
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Cobamamide DB11191
small molecule | CAS: 13870-90-1

Cobamamide is one of the active forms of vitamin B12 that is also known as _adenosylcobalamin_ or _dibencozide_. This drug is available as a nutritional supplement to prevent vitamin B12 deficiency. Vitamin B12 is a collective term for these variously subs…

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansCoenzymes +6
Waktu Paruh-
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Cobitolimod DB14819
biotech | CAS: 1226822-98-5

Cobitolimod is under investigation in clinical trial NCT03178669 (The Efficacy of Cobitolimod in Patients With Moderate to Severe Active Ulcerative Colitis).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 2364477-18-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Cobolimab DB16372
biotech | CAS: 2022215-65-0

Cobolimab is under investigation in clinical trial NCT04655976 (Study of Cobolimab in Combination With Dostarlimab and Docetaxel in Advanced NSCLC Participants).

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Cobomarsen DB14931
biotech | CAS: 1848257-52-2

Cobomarsen is under investigation in clinical trial NCT02580552 (Safety, Tolerability and Pharmacokinetics of MRG-106 in Patients With Mycosis Fungoides (MF), CLL, DLBCL or ATLL).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
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Cocaine Approved DB00907
small molecule | CAS: 50-36-2

An alkaloid ester extracted from the leaves of plants including coca. It is a local anesthetic and vasoconstrictor and is clinically used for that purpose, particularly in the eye, ear, nose, and throat. It also has powerful central nervous system effects sim…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAlkaloids +36
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium channel protein +5
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
biotech

RBP-8000 is under investigation in clinical trials (A Randomized, 4-sequence, 2-period, Double-blind, Placebo Controlled Study With a DSM-IV-TR Diagnosis of Cocaine Abuse) for the treatment of Cocaine Abuse.

Kategori:
Amino Acids, Peptides, and ProteinsEnzymesEnzymes and Coenzymes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61789-40-0

Cocamidopropyl betaine is a mixture of closely related organic compounds derived from coconut oil and dimethylaminopropylamine that typically acts as an amphoteric surfactant in cosmetics and personal care products. It is a zwitterionic ammonium compound and …

Kategori:
AminesCompounds used in a research, industrial, or household settingOnium Compounds +3
Waktu Paruh-
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Genetik -
Cocarboxylase Approved DB01987
small molecule | CAS: 136-08-3

The coenzyme form of Vitamin B1 present in many animal tissues. It is a required intermediate in the pyruvate dehydrogenase complex and the ketoglutarate dehydrogenase complex.

Kategori:
CoenzymesEnzymes and CoenzymesMicronutrients +5
Target Protein:
RNAAcetolactate synthase, catabolicPyruvate dehydrogenase E1 component +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61791-31-9

Deskripsi belum tersedia.

Kategori:
AlcoholsAllergensAmines +3
Waktu Paruh-
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Genetik -
Cocoa Approved DB10977
biotech | CAS: 84649-99-0

Cocoa allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Cocoa butter Approved DB11086
biotech | CAS: 8002-31-1

Cocoa butter is an edible natural fat obtained from the _Theobroma cocoa_ seeds that is predominantly found in dark chocolate [A33033]. It is a rich source of monounsaturated and saturated fatty acids [A33040] that mainly contains approximately 33% [DB04224],…

Kategori:
Antipruritics and Local AnestheticsDiet, Food, and NutritionFats +3
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Codeine Approved DB00318
small molecule | CAS: 76-57-3

The relief of pain (analgesia) is a primary goal for enhancing the quality of life of patients and for increasing the ability of patients to engage in day to day activities. Codeine, an opioid analgesic, was originally approved in the US in 1950 and is a drug…

Kategori:
AlkaloidsAnalgesicsAntitussive Agents +26
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +6
Waktu ParuhPlasma half-lives o…
Vol. DistribusiApparent volume of …
KlirensRenal clearance of …
Genetik 9 Varian
small molecule | CAS: 125-27-9

Deskripsi belum tersedia.

Waktu Paruh-
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Codrituzumab DB14843
biotech | CAS: 1365267-33-9

Codrituzumab is under investigation in clinical trial NCT01507168 (A Study of RO5137382 (GC33) in Patients With Advanced or Metastatic Hepatocellular Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Coenzyme F420 DB03913
small molecule | CAS: 64885-97-8

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coenzyme M Approved DB09110
small molecule | CAS: 3375-50-6

Coenzyme M (commonly known by its salt form, Mesna) is a synthetic sulfhydryl (thiol) compound and is used for prophylaxis of Ifosfamide and cyclophosphamide induced hemorrhagic cystitis.[A18572]

Kategori:
AlkanesAlkanesulfonatesAlkanesulfonic Acids +12
Waktu ParuhThe elimination hal…
Vol. DistribusiVd = 0.652 ± 0.242 …
KlirensPlasma clearance of…
Genetik -
Cofirasersen DB19037
biotech | CAS: 2247669-96-9

Cofirasersen is under investigation in clinical trial NCT04441788 (A Study to Assess the Safety, Tolerability, and Efficacy of ION-827359 in Participants With Mild to Moderate Chronic Obstructive Pulmonary Disease (COPD) With Chronic Bronchitis (CB)).

Waktu Paruh-
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Col-118 DB05778
small molecule

COL-118, a topical compound based on the SansRosa technology, for the treatment of redness associated with rosacea and other skin disorders. It is a believed to reduce erythema by constricting enlarged blood vessels in facial tissue. Col-118 is a unique formu…

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Colchiceine Approved DB15534
small molecule | CAS: 477-27-0

Colchiceine is one of several metabolites of the anti-gout medication [colchicine].[A192714]

Kategori:
AlkaloidsColchicine DerivativesTubulin Inhibiting Agent
Target Protein:
Tubulin beta chainTubulin alpha-1A chain
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Colchicine Approved DB01394
small molecule | CAS: 64-86-8

Colchicine is an alkaloid drug derived from a plant belonging to the Lily family, known as _Colchicum autumnale_, or "autumn crocus."[A183611] Its use was first approved by the FDA in 1961.[L8192] Colchicine is used in the treatment of gout flares and Familia…

Kategori:
Agents Causing Muscle ToxicityAlkaloidsAntigout Preparations +23
Target Protein:
Tubulin beta chain
Waktu ParuhAfter several doses…
Vol. DistribusiThe mean apparent v…
KlirensIn one pharmacokine…
Genetik -
Coleneuramide DB14932
small molecule | CAS: 204200-47-5

Coleneuramide is under investigation in clinical trial NCT00307749 (Safety and Efficacy of MCC-257 in the Treatment of Diabetic Polyneuropathy).

Kategori:
Acids, AcyclicAmino SugarsCarbohydrates +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Colestipol Approved DB00375
small molecule | CAS: 26658-42-4

Bile acid sequestrants like colestipol have been in use since the 1970s.[FDA Label, F4555, F4567, L6262] And even though such an agent may very well be useful in reducing elevated cholesterol levels and decreasing the risk for atherosclerotic vascular disease…

Kategori:
AminesAnion Exchange ResinsBile Acid Sequestrants +12
Target Protein:
Bile acids
Waktu ParuhColestipol is not a…
Vol. DistribusiColestipol is not a…
KlirensColestipol is not a…
Genetik -
Colforsin DB02587
small molecule | CAS: 66575-29-9

Potent activator of the adenylate cyclase system and the biosynthesis of cyclic AMP. From the plant Coleus forskohlii. Has antihypertensive, positive inotropic, platelet aggregation inhibitory, and smooth muscle relaxant activities; also lowers intraocular pr…

Kategori:
Adjuvants, ImmunologicAnti-Asthmatic AgentsAutonomic Agents +12
Target Protein:
Adenylate cyclaseAdenylate cyclase type 2Guanine nucleotide-binding protein G(s) subunit alpha isoforms short +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Colfosceril palmitate Approved DB09114
small molecule | CAS: 63-89-8

Colfosceril palmitate is a synthetic pulmonary surfactant administered in infants with respiratory distress syndrome.[A31510] It was part of the first generation of commercially available artificial surfactants.[T70] It was developed by Burroughs Wellcome and…

Kategori:
GlycerophosphatesGlycerophospholipidsLipids +6
Waktu ParuhThe half-life of co…
Vol. DistribusiColfosceril palmita…
KlirensAfter 5 days of dru…
Genetik -
Colistimethate Approved DB01111
small molecule | CAS: 12705-41-8

Colistimethate is an antibiotic that has been shown to have bactericidal activity against aerobic gram-negative microorganisms. Colistimethate is particularly indicated when the infection is caused by sensitive strains of Pseudomonas aeruginosa.

Kategori:
Agents that produce neuromuscular block (indirect)Amino Acids, Peptides, and ProteinsAntimicrobial Cationic Peptides +11
Target Protein:
Dihydropteroate synthaseBacterial outer membrane
Waktu Paruh2-3 hours following…
Vol. Distribusi-
Klirens-
Genetik -
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