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12560

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9109 (72.5%)
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6912 (55.0%)
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12560 (100.0%)

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Halaman 75 / 252
Cenobamate Approved DB06119
small molecule | CAS: 913088-80-9

Cenobamate, or YKP-3089, is an antiepileptic drug developed by SK Pharmaceuticals and used to treat partial onset seizures.[A188442,L10653] The exact mechanism of action has not been described in the literature, though it positively modulates GABA<sub>A</sub>…

Kategori:
Acids, AcyclicAnticonvulsantsBenzene Derivatives +34
Target Protein:
Voltage-gated sodium channel alpha subunitGamma-aminobutyric acid receptor subunit alpha-1
Waktu ParuhThe terminal half l…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Cenplacel-L DB19188
biotech

Cenplacel-L is under investigation in clinical trial (Study of Human Placenta-derived Cells (PDA001) to Evaluate the Safety and Effectiveness for Patients With Ischemic Stroke) for the treatment of patients with Ischemic Stroke.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Censavudine DB12074
small molecule | CAS: 634907-30-5

Censavudine has been used in trials studying the treatment of HIV-1 Infection.

Kategori:
Anti-HIV AgentsDeoxyribonucleosidesNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Centanafadine DB14841
small molecule | CAS: 924012-43-1

Centanafadine is under investigation in clinical trial NCT02827513 (A Phase 1 Study to Investigate the Safety, Tolerance, Food Effect, Pharmacokinetics and Pharmacodynamics of Single and Multiple Doses of Extended Release Formulations of Centanafadine (CTN) i…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Centella asiatica Approved DB14256
biotech

Centella asiatica is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Agents that reduce seizure thresholdAngiospermsApiaceae +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Centhaquine DB16122
small molecule | CAS: 57961-90-7

Centhaquine is under investigation in clinical trial NCT04045327 (Efficacy of PMZ-2010 (Centhaquine) a Resuscitative Agent for Hypovolemic Shock).

Kategori:
Adrenergic and Dopaminergic AgentsCardiac Stimulants Excl. Cardiac GlycosidesCardiac Therapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CEP-1347 DB05403
small molecule

CEP-1347 is a semi-synthetic compound shown to protect multiple nerve cell types from a variety of insults leading to programmed cell death (apoptosis) which could improve the survival of dopamine neurons prior to and after transplantation.

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
Target Protein:
Mitogen-activated protein kinase 12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CEP-9722 DB14882
small molecule | CAS: 916574-83-9

CEP-9722 is under investigation in clinical trial NCT01345357 (Study of CEP-9722 in Combination With Gemcitabine and Cisplatin in Patients With Advanced Solid Tumors or Mantle Cell Lymphoma).

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingImides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1192706-52-7

Cepeginterferon alfa-2B is under investigation in clinical trial NCT01889433 (An Open-label Comparative Efficacy and Safety Study of Algeron (Cepeginterferon Alfa-2b) in Treatment-naive Patients With Chronic Hepatitis C).

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP1A2 Inhibitors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cephalexin Approved DB00567
small molecule | CAS: 15686-71-2

Cephalexin is the first of the first generation cephalosporins.[A179071,A179074] This antibiotic contains a beta lactam and a dihydrothiazide.[A179071] Cephalexin is used to treat a number of susceptible bacterial infections through inhibition of cell wall s…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +23
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2aPenicillin-binding protein 1b +2
Waktu ParuhThe half life of ce…
Vol. Distribusi5.2-5.8L.[A179068]
KlirensClearance from one …
Genetik -
Cephaloglycin Approved DB00689
small molecule | CAS: 3577-01-3

A cephalorsporin antibiotic that is no longer commonly used.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +7
Target Protein:
Penicillin-binding protein 1B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cephalosporin C DB03313
small molecule | CAS: 61-24-5

Deskripsi belum tersedia.

Kategori:
Agents that reduce seizure thresholdAmidesbeta-Lactams +4
Target Protein:
Penicillin-binding protein 1bPeptidoglycan synthase FtsIPenicillin-binding protein 1A +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Cephalothin group is a solid. This compound belongs to the 1,3-thiazines. These are organic compounds containing 1,3-thiazine, a six-member ring with a nitrogen and a sulfur atom in ring positions 1 and 3 respectively, as well as two double bonds. This substa…

Kategori:
Nephrotoxic agents
Target Protein:
D-alanyl-D-alanine carboxypeptidaseBeta-lactamase Toho-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CEQ508 DB17911
biotech

CEQ508 is a Live Attenuated E. Coli Expressing Beta Catenin ShRNA currently being investigated to treat Familial Adenomatous Polyposis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CER-001 DB18538
biotech

CER-001 is a negatively charged lipoprotein particle comprising human recombinant apolipoprotein A-I and two phospholipids: sphingomyelin and dipalmitoylphosphatidylglycerol.[L48290] It is under investigation for the treatment of lecithin-cholesterol acyltran…

Kategori:
Amino Acids, Peptides, and ProteinsApolipoproteinsApolipoproteins A +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceralasertib DB14917
small molecule | CAS: 1352226-88-0

Ceralasertib is under investigation in clinical trial NCT03682289 (Phase II Trial of AZD6738 Alone and in Combination With Olaparib).

Kategori:
AmidesHeterocyclic Compounds, Fused-RingOxazines +2
Target Protein:
Serine/threonine-protein kinase ATR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceralifimod DB16123
small molecule | CAS: 891859-12-4

Ceralifimod is under investigation in clinical trial NCT01226745 (Phase 2 Extension Trial in Patients With Relapsing-remitting Multiple Sclerosis (RRMS)).

Kategori:
AzetinesImmunologic FactorsImmunosuppressive Agents +1
Target Protein:
Sphingosine 1-phosphate receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceramide AP DB14705
small molecule | CAS: 212070-45-6

Deskripsi belum tersedia.

Kategori:
AmidesCarbohydratesGlycoconjugates +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceramide NG DB14706
small molecule | CAS: 2304-80-5

Deskripsi belum tersedia.

Kategori:
AmidesCarbohydratesGlycoconjugates +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CERC-301 DB12063
small molecule | CAS: 808732-98-1

Mk 0657 has been used in trials studying the treatment of Major Depressive Disorder.

Kategori:
Receptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Target Protein:
Glutamate receptor ionotropic, NMDA 2B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerdulatinib DB15499
small molecule | CAS: 1198300-79-6

Cerdulatinib is under investigation in clinical trial NCT04021082 (CELTIC-1: A Phase 2B Study of Cerdulatinib in Patients With Relapsed/refractory Peripheral T-cell Lymphoma (PTCL)).

Kategori:
Sulfur Compounds
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase JAK2Tyrosine-protein kinase SYK +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CERE-110 DB05898
biotech

CERE-110 is a gene-therapy product that involves in vivo delivery of nerve growth factor (NGF) genes through an adeno-associated viral vector (AAV) delivery system. This drug is developed by Ceregene and currently under phase I of clinical trial.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CERE-120 DB05637
biotech | CAS: 1148126-35-5

CERE-120 is an investigational drug consisting of an adeno-associated virus (AAV) that was engineered to carry the human gene for neurturin, a neurotrophic (growth) factor. It was under investigation in clinical trials for the treatment of Parkinson's Disease.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerebrolysin DB16599
biotech | CAS: 12656-61-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBrainCentral Nervous System Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1509916-03-3

Cergutuzumab amunaleukin is under investigation in clinical trial NCT02004106 (A Study to Evaluate Safety, Pharmacokinetics, and Efficacy of RO6895882 in Participants With Advanced and/or Metastatic Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceritinib Approved DB09063
small molecule | CAS: 1032900-25-6

Ceritinib is used for the treatment of adults with anaplastic lymphoma kinase (ALK)-positive metastatic non-small cell lung cancer (NSCLC) following failure (secondary to resistance or intolerance) of prior crizotinib therapy. About 4% of patients with NSCLC …

Kategori:
Anaplastic lymphoma kinase (ALK) inhibitorsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +25
Target Protein:
ALK tyrosine kinase receptor
Waktu ParuhThe terminal half l…
Vol. DistribusiThe apparent volume…
KlirensThe geometric mean …
Genetik -
Cerium oxalate DB13519
small molecule | CAS: 139-42-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAntiemetics and Antinauseants
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerivastatin Approved DB00439
small molecule | CAS: 145599-86-6

On August 8, 2001 the U.S. Food and Drug Administration (FDA) announced that Bayer Pharmaceutical Division voluntarily withdrew Baycol from the U.S. market, due to reports of fatal rhabdomyolysis, a severe adverse reaction from this cholesterol-lowering (lipi…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBCRP/ABCG2 Substrates +34
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh2-3 hours
Vol. Distribusi-
Klirens-
Genetik -
Cerlapirdine DB12229
small molecule | CAS: 925448-93-7

Cerlapirdine has been investigated for the treatment of Alzheimer Disease.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
5-hydroxytryptamine receptor 6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerliponase alfa Approved DB13173
biotech | CAS: 151662-36-1

Cerliponase alfa is a hydrolytic lysosomal N-terminal tripeptidyl peptidase-1 (TPP1).[L51319] On April 27, 2017, cerliponase alfa was first approved by the FDA as the first treatment for neuronal ceroid lipofuscinosis type 2 (CLN2), also known as TPP1 deficie…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsEnzymes +6
Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu ParuhFollowing intravent…
Vol. DistribusiFollowing intravent…
KlirensFollowing intravent…
Genetik -
Certepetide DB18721
biotech | CAS: 2580154-02-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Certolizumab pegol Approved DB08904
biotech | CAS: 428863-50-7

Certolizumab pegol is a pegylated monoclonal antibody against the tumor necrosis factor-alpha (TNF-alpha).[A176585] It is formed with a humanized Fab fragment of 50 kDa, from an IgG 1 isotype, fused to a 40 kDa polyethylene glycol moiety replacing the Fc anti…

Kategori:
Agents reducing cytokine levelsAlcoholsAmino Acids, Peptides, and Proteins +31
Target Protein:
Tumor necrosis factor
Waktu ParuhThe circulatory hal…
Vol. DistribusiCertolizumab pegol …
KlirensThe clearance rate …
Genetik -
Ceruletide Approved DB00403
small molecule | CAS: 17650-98-5

Caerulein is a specific decapeptide similar in action and composition to the natural gastrointestinal peptide hormone cholecystokinin. It exerts stimulatory effects on the gastric, biliary, and pancreatic secretion, as well as on certain smooth muscles.

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsOligopeptides +2
Target Protein:
Cholecystokinin receptor type AGastrin/cholecystokinin type B receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cesium DB15392
small molecule | CAS: 7440-46-2

Cesium is under investigation in clinical trial NCT02794675 (Intraoperative Placement of Cesium-131 Permanent Interstitial Brachytherapy in Head and Neck Cancer).

Kategori:
ElementsMetalsMetals, Alkali +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cesium Cs-131 DB19250
small molecule | CAS: 14914-76-2

Cesium Cs-131 is under investigation in clinical trial NCT04340258 (Trial Combining Pembrolizumab and Cesium 131 Brachytherapy With Salvage Surgery in HNSCC).

Kategori:
Cesium IsotopesElementsIsotopes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetalkonium Approved DB11583
small molecule | CAS: 10328-34-4

Cetalkonium is a C16 alkyl benzalkonium chloride derivative with an amphipathic property which allows it to be used in different types of formulations.[A27143] It is a quaternary ammonium salt that acts as an antiseptic against a variety of bacteria and fungi…

Kategori:
AlcoholsAminesAmmonium Compounds +7
Waktu ParuhAs cetalkonium is n…
Vol. DistribusiAs cetalkonium is n…
KlirensAs cetalkonium is n…
Genetik -
Cethromycin DB06419
small molecule | CAS: 205110-48-1

Cethromycin is a 3-keto (ketolide) derivative of erythromycin A with an 11,12-carbamate group and an O-6-linked aromatic ring system.[A203369] Cethromycin represents a joint development effort by Abbott Laboratories, Taisho Pharmaceuticals, and Advanced Life …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCytochrome P-450 CYP3A Inhibitors +15
Target Protein:
23S ribosomal RNA
Waktu ParuhCethromycin given i…
Vol. DistribusiCethromycin given i…
KlirensCethromycin clearan…
Genetik -
Cetiedil DB13753
small molecule | CAS: 14176-10-4

Deskripsi belum tersedia.

Kategori:
Antisickling AgentsCardiovascular AgentsHematologic Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetilistat DB06586
small molecule | CAS: 282526-98-1

Cetilistat is a novel inhibitor of pancreatic lipase being developed by Alizyme for the treatment of obesity and associated co-morbidities, including type 2 diabetes.

Kategori:
Anti-Obesity AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Endothelial lipaseGastric triacylglycerol lipasePancreatic triacylglycerol lipase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetirizine Approved DB00341
small molecule | CAS: 83881-51-0

Cetirizine, also commonly known as _Zyrtec_, is an orally active second-generation histamine H1 antagonist proven effective in the treatment of various allergic symptoms, such as sneezing, coughing, nasal congestion, hives, and other symptoms [A175051], [A175…

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseCentral Nervous System Depressants +14
Target Protein:
Histamine H1 receptor
Waktu ParuhPlasma elimination …
Vol. DistribusiApparent volume of …
KlirensApparent total body…
Genetik -
Cetrelimab DB15421
biotech | CAS: 2050478-92-5

Cetrelimab is under investigation in clinical trial NCT03547037 (A Study to Evaluate the Safety, Pharmacokinetics, Pharmacodynamics, and Immunogenicity of JNJ-63723283, an Anti-Programmed Cell Death (PD)-1 Monoclonal Antibody, as Monotherapy or in Combination…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetrorelix Approved DB00050
small molecule | CAS: 120287-85-6

Cetrorelix is a man-made hormone that blocks the effects of Gonadotropin Releasing Hormone (GnRH). GnRH controls another hormone that is called luteinizing hormone (LH), which is the hormone that starts ovulation during the menstrual cycle. When undergoing ho…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Gonadotropin-Releasing HormonesDecreased GnRH Secretion +18
Target Protein:
Gonadotropin-releasing hormone receptorLutropin-choriogonadotropic hormone receptor
Waktu Paruh~62.8 hours
Vol. Distribusi* 1.16 L/kg
Klirens* 1.28 ml/min·kg [a…
Genetik -
Cetuximab Approved DB00002
biotech | CAS: 205923-56-4

Cetuximab is a recombinant chimeric human/mouse IgG1 monoclonal antibody that competitively binds to epidermal growth factor receptor (EGFR) and competitively inhibits the binding of epidermal growth factor (EGF).[A227973] EGFR is a member of the ErbB family …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Epidermal growth factor receptorLow affinity immunoglobulin gamma Fc region receptor III-BComplement C1q subcomponent subunit A +5
Gen Terkait:
FCGR2A FCGR3A
Waktu ParuhAfter administratio…
Vol. DistribusiThe volume of the d…
KlirensIn patients with re…
Genetik 2 Varian
biotech | CAS: 2166339-33-7

Cetuximab sarotalocan is under investigation in clinical trial NCT03769506 (ASP-1929 Photoimmunotherapy (PIT) Study in Recurrent Head/Neck Cancer for Patients Who Have Failed at Least Two Lines of Therapy) for the treatment of Recurrent Head/Neck Cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetyl alcohol Approved DB09494
small molecule | CAS: 36653-82-4

Cetyl alcohol, also known as 1-hexadecanol or n-hexadecyl alcohol, is a 16-C fatty alcohol with the chemical formula CH3(CH2)15OH. It can be produced from the reduction of palmitic acid. Cetyl alcohol is present in a waxy white powder or flake form at room te…

Kategori:
AlcoholsDrugs that are Mainly Renally ExcretedLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 59130-69-7

Cetyl ethylhexanoate is an ester of cetyl alcohol and 2-ethylhexanoic acid. It is present in cosmetic products as a skin conditioning agent and emollient.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 64660-84-0

Deskripsi belum tersedia.

Kategori:
Lipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetyl oleate DB19454
small molecule | CAS: 22393-86-8

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cetyl palmitate DB15782
small molecule | CAS: 540-10-3

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipidsPalmitic Acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 22393-83-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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