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11793

Total database: 17430
Struktur (SMILES)
8607 (73.0%)
Target
6418 (54.4%)
Genomik
102 (0.9%)
Referensi
11793 (100.0%)

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Hasil Pencarian (11793)

Halaman 74 / 236
Codeine-N-oxide DB01568
small molecule | CAS: 3688-65-1

Deskripsi belum tersedia.

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Codrituzumab DB14843
biotech | CAS: 1365267-33-9

Codrituzumab is under investigation in clinical trial NCT01507168 (A Study of RO5137382 (GC33) in Patients With Advanced or Metastatic Hepatocellular Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
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Coenzyme A DB01992
small molecule | CAS: 85-61-0

Coenzyme A (CoA, CoASH, or HSCoA) is a coenzyme, well known for it's role in the synthesis and oxidation of fatty acids, and the oxidation of pyruvate in the citric acid cycle. All genomes sequenced to date encode enzymes that use coenzyme A as a substrate, a…

Kategori:
Adenine NucleotidesCoenzyme A, biosynthesisCoenzymes +7
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseCarnitine O-acetyltransferaseGalactoside O-acetyltransferase +42
Waktu Paruh-
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small molecule | CAS: 81918-99-2

Coenzyme A persulfide is a possible in vivo inhibitor of mammalian short chain acyl-CoA dehydrogenase.

Kategori:
Adenine NucleotidesCoenzymesEnzymes and Coenzymes +6
Target Protein:
Isovaleryl-CoA dehydrogenase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coenzyme F420 DB03913
small molecule | CAS: 64885-97-8

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +4
Waktu Paruh-
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Genetik -
Coenzyme M Approved DB09110
small molecule | CAS: 3375-50-6

Coenzyme M (commonly known by its salt form, Mesna) is a synthetic sulfhydryl (thiol) compound and is used for prophylaxis of Ifosfamide and cyclophosphamide induced hemorrhagic cystitis.[A18572]

Kategori:
AlkanesAlkanesulfonatesAlkanesulfonic Acids +12
Waktu ParuhThe elimination hal…
Vol. DistribusiVd = 0.652 ± 0.242 …
KlirensPlasma clearance of…
Genetik -
Coffea arabica seed, roasted Approved DB15603
biotech

Coffea arabica seed, roasted allergenic extract is used in allergenic testing.

Waktu Paruh-
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Cofirasersen DB19037
biotech | CAS: 2247669-96-9

Cofirasersen is under investigation in clinical trial NCT04441788 (A Study to Assess the Safety, Tolerability, and Efficacy of ION-827359 in Participants With Mild to Moderate Chronic Obstructive Pulmonary Disease (COPD) With Chronic Bronchitis (CB)).

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Col-Treg DB18451
biotech

Col-Treg is an autologous T-cell therapy comprising type I regulatory T-cells specific for human type II collagen.[A261635]

Waktu Paruh-
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Colchicine Approved DB01394
small molecule | CAS: 64-86-8

Colchicine is an alkaloid drug derived from a plant belonging to the Lily family, known as _Colchicum autumnale_, or "autumn crocus."[A183611] Its use was first approved by the FDA in 1961.[L8192] Colchicine is used in the treatment of gout flares and Familia…

Kategori:
Agents Causing Muscle ToxicityAlkaloidsAntigout Preparations +23
Target Protein:
Tubulin beta chain
Waktu ParuhAfter several doses…
Vol. DistribusiThe mean apparent v…
KlirensIn one pharmacokine…
Genetik -
Colesevelam Approved DB00930
small molecule | CAS: 182815-43-6

Colesevelam is a bile acid sequestrant. Colesevelam is used with exercise and diet changes (restriction of cholesterol and fat intake) to reduce the amount of cholesterol and certain fatty substances in the blood. It works by binding bile acids in the intesti…

Kategori:
AlkenesAllyl CompoundsAllylamine +11
Target Protein:
Bile acids
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Colestilan chloride Approved DB11634
small molecule | CAS: 95522-45-5

Colestilan is an ingredient in the EMA-withdrawn product BindRen.

Kategori:
Drugs for Treatment of Hyperkalemia and HyperphosphatemiaFused-Ring CompoundsSteroids
Waktu Paruh-
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Colestipol Approved DB00375
small molecule | CAS: 26658-42-4

Bile acid sequestrants like colestipol have been in use since the 1970s.[FDA Label, F4555, F4567, L6262] And even though such an agent may very well be useful in reducing elevated cholesterol levels and decreasing the risk for atherosclerotic vascular disease…

Kategori:
AminesAnion Exchange ResinsBile Acid Sequestrants +12
Target Protein:
Bile acids
Waktu ParuhColestipol is not a…
Vol. DistribusiColestipol is not a…
KlirensColestipol is not a…
Genetik -
Colforsin DB02587
small molecule | CAS: 66575-29-9

Potent activator of the adenylate cyclase system and the biosynthesis of cyclic AMP. From the plant Coleus forskohlii. Has antihypertensive, positive inotropic, platelet aggregation inhibitory, and smooth muscle relaxant activities; also lowers intraocular pr…

Kategori:
Adjuvants, ImmunologicAnti-Asthmatic AgentsAutonomic Agents +12
Target Protein:
Adenylate cyclaseAdenylate cyclase type 2Guanine nucleotide-binding protein G(s) subunit alpha isoforms short +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Colfosceril palmitate Approved DB09114
small molecule | CAS: 63-89-8

Colfosceril palmitate is a synthetic pulmonary surfactant administered in infants with respiratory distress syndrome.[A31510] It was part of the first generation of commercially available artificial surfactants.[T70] It was developed by Burroughs Wellcome and…

Kategori:
GlycerophosphatesGlycerophospholipidsLipids +6
Waktu ParuhThe half-life of co…
Vol. DistribusiColfosceril palmita…
KlirensAfter 5 days of dru…
Genetik -
Colistin Approved DB00803
biotech | CAS: 1066-17-7

Cyclic polypeptide antibiotic from Bacillus colistinus. It is composed of Polymyxins E1 and E2 (or Colistins A, B, and C) which act as detergents on cell membranes. Colistin is less toxic than Polymyxin B, but otherwise similar; the methanesulfonate is used o…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAmino Acids, Peptides, and Proteins +21
Target Protein:
Dihydropteroate synthaseBacterial outer membrane
Waktu Paruh5 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Collagen-polyvinylpyrrolidone is a copolymer generated from a mixture of type I collagen and low-molecular-weight PVP that has undergone ? irradiation[A227733]. It is characterized by antifibrotic, fibrolytic, and immunomodulatory properties[A227733].

Kategori:
AlkenesAmino Acids, Peptides, and ProteinsBiopolymers +11
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biotech | CAS: 9001-12-1

Collagenase clostridium histolyticum is an enzyme produced by the bacterium Clostridium histolyticum. It is beneficial in the breakdown of collagen plaques for the treatment of Dupuytren's contracture and Peyronie's disease.[L14882] The topical formulation is…

Kategori:
Collagen-specific EnzymeCollagenasesDermatologicals +11
Target Protein:
Collagen alpha-1(I) chainCollagen alpha-1(II) chainCollagen alpha-1(III) chain
Waktu Paruh-
Vol. DistribusiThere is no current…
KlirensClearance informati…
Genetik -
Colloidal oatmeal Approved DB11286
biotech

Colloidal oatmeal is produced by grinding fine granules of oatmeal and boiling it to extract the colloidal material. It contains high concentrations of starches and beta-glucan that exhibits water-absorbing properties. Phenols are also contained in colloidal …

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
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biotech | CAS: 1269764-99-9

Coltuximab ravtansine (SAR3419) targets CD19 and is being investigated for the treatment of acute lymphoblastic leukemia (ALL).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +16
Target Protein:
B-lymphocyte antigen CD19
Waktu Paruh-
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Combretastatin DB12596
small molecule | CAS: 82855-09-2

Combretastatin has been investigated for the treatment of Anaplastic Thyroid Cancer.

Kategori:
Antimitotic AgentsAntineoplastic AgentsAntineoplastic Agents, Phytogenic +5
Waktu Paruh-
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small molecule | CAS: 117048-59-6

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAntineoplastic Agents, PhytogenicBenzene Derivatives +1
Waktu Paruh-
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Common carp Approved DB10614
biotech

Common carp allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Compound 18 DB02715
small molecule | CAS: 31112-66-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +1
Target Protein:
Estrogen receptor
Waktu Paruh-
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Compound 19 DB02615
small molecule

Deskripsi belum tersedia.

Target Protein:
Estrogen receptorTyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
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Conatumumab DB11646
biotech | CAS: 896731-82-1

Conatumumab has been used in trials studying the treatment of Sarcoma, Lymphoma, Oncology, Colon Cancer, and Rectal Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents +7
Waktu Paruh-
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Conbercept DB12460
biotech | CAS: 1227158-72-6

Conbercept has been investigated for the basic science of Age-related Macular Degeneration.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
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Concanamycin A DB14062
small molecule | CAS: 80890-47-7

Concanamycin A is an H+-ATPase (vacuolar) inhibitor.

Kategori:
Anti-Infective AgentsEnzyme InhibitorsLactones +3
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Conivaptan Approved DB00872
small molecule | CAS: 210101-16-9

Conivaptan is a non-peptide inhibitor of antidiuretic hormone (vasopressin). It was approved in 2004 for hyponatremia (low blood sodium levels) caused by syndrome of inappropriate antidiuretic hormone (SIADH). Conivaptan inhibits both isotypes of the vasopres…

Kategori:
Antidiuretic Hormone Receptor AntagonistsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A Substrates +12
Target Protein:
Vasopressin V1a receptorVasopressin V2 receptor
Waktu Paruh5 hours
Vol. Distribusi-
Klirens-
Genetik -
Conjugated estrogens Approved DB00286
small molecule | CAS: 12126-59-9

The conjugated estrogens are noncrystalline mixtures of purified female sex hormones obtained either by its isolation from the urine of pregnant mares or by synthetic generation from vegetal material. Both of these products are later conjugated to natrium sul…

Kategori:
Agents causing angioedemaBCRP/ABCG2 SubstratesCOMT Substrates +26
Target Protein:
Estrogen receptor betaEstrogen receptor
Waktu ParuhThe median half-lif…
Vol. DistribusiThe physiological d…
KlirensThe reported normal…
Genetik -
Copanlisib Approved DB12483
small molecule | CAS: 1032568-63-0

Copanlisib is a selective pan-Class I phosphoinositide 3-kinase (PI3K) inhibitor with preferential activity against the alpha and delta isoforms. PI3K, a lipid kinase that activates downstream signalling pathways involved in cell survival and growth, that exi…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +17
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform +1
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Copper Cu-64 Approved DB13980
small molecule | CAS: 13981-25-4

Copper-64 is a radiopharmaceutical usually found in the +2 oxidation state as the complexes including the +1 state tend to be more unstable.[T604] It is used in molecular radiotherapy and positron emission tomography.

Waktu Paruh-
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Copper gluconate Approved DB11246
small molecule | CAS: 527-09-3

Copper gluconate is a copper salt of D-gluconic acid that displays a light blue to bluish-green color. It is prepared by the reaction of gluconic acid solutions with cupric oxide or basic cupric carbonate. According to the good manufacturing or feeding practi…

Kategori:
Acids, AcyclicCarbohydratesHydroxy Acids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Copper oxodotreotide Cu-64 Approved DB15873
small molecule | CAS: 1426155-87-4

Copper Cu 64 dotatate is a newly approved Cu labeled somatostatin analog and has several advantages over <sup>68</sup>Ga-labeled somatostatin analogs for positron emission tomography (PET).[A220348] Copper Cu 64 dotatate has a longer half-life and can be prod…

Kategori:
Amino Acids, Peptides, and ProteinsCopper RadioisotopesPeptides +4
Target Protein:
Somatostatin receptor type 2
Waktu ParuhThe half-life of Co…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 68341-09-3

Deskripsi belum tersedia.

Kategori:
SemicarbazidesSemicarbazonesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coprelotamab DB16380
biotech | CAS: 2348469-84-9

Coprelotamab is under investigation in clinical trial NCT04170595 (Clinical Study of Recombinant Anti-her2 Humanized Monoclonal Antibody for Injection).

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small molecule | CAS: 2624-63-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingPorphyrinogensPorphyrins
Target Protein:
Uroporphyrinogen decarboxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coptisine DB19308
small molecule | CAS: 3486-66-6

Deskripsi belum tersedia.

Kategori:
AlkaloidsBenzylisoquinolinesBerberine Alkaloids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coramitug DB19411
biotech | CAS: 2626841-92-5

Deskripsi belum tersedia.

Waktu Paruh-
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Cordycepin DB12156
small molecule | CAS: 73-03-0

Cordycepin has been used in trials studying the treatment of Leukemia.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntineoplastic Agents +9
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 73-04-1

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesDeoxyribonucleotidesHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Poly(A) polymerase alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Corifollitropin alfa Approved DB09066
biotech | CAS: 195962-23-3

Corifollitropin alfa, also known as _Elonva_ is used in women undergoing fertility treatment to stimulate the development of more than one mature egg (oocyte) at a time in the ovaries. This drug used together with _a gonadotropin-releasing hormone (GnRH) anta…

Kategori:
Drugs that are Mainly Renally ExcretedFollicle Stimulating HormoneGenito Urinary System and Sex Hormones +9
Target Protein:
Follicle-stimulating hormone receptor
Waktu ParuhCorifollitropin alf…
Vol. DistribusiDistribution, metab…
Klirens0.13 L/h (0.10-0.18…
Genetik -
CoronaVac DB15806
biotech

CoronaVac, previously known as PiCoVacc, is a SARS-CoV-2 purified, inactivated, and adsorbed vaccine candidate developed by SinoVac Biotech Corporation[A219758]. It was developed by propagating the SARS-CoV-2 CN2 strain inside Vero Cells and inactivating it w…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Corticorelin DB05394
small molecule | CAS: 86784-80-7

Corticotropin-releasing factor is studied in the treatment of brain cancer. It is made naturally by the hypothalamus (a part of the brain) and can also be made in the laboratory. Human corticotropin-releasing factor may help reduce symptoms caused by edema (s…

Kategori:
Amino Acids, Peptides, and ProteinsCorticotropin-Releasing HormoneDiagnostic Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1312542-61-2

Corticorelin acetate has been investigated for the treatment of Brain Edema and Brain Tumor.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 121249-14-7

Corticorelin, available commercially as corticorelin ovine triflutate (tradename Acthrel), is a synthetic form of the peptide human corticotropin-releasing hormone (hCRH), a potent stimulator of adrenocorticotropic hormone (ACTH) release from the anterior pit…

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsHormones +9
Target Protein:
Corticotropin-releasing factor receptor 1Corticotropin-releasing factor receptor 2
Waktu ParuhPlasma half-lives f…
Vol. DistribusiThe mean volume of …
Klirens95 ± 11 L/m2/day
Genetik -
Corticosterone DB04652
small molecule | CAS: 50-22-6

An adrenocortical steroid that has modest but significant activities as a mineralocorticoid and a glucocorticoid. (From Goodman and Gilman&#39;s The Pharmacological Basis of Therapeutics, 8th ed, p1437)

Kategori:
11-HydroxycorticosteroidsAdrenal Cortex HormonesAnti-Inflammatory Agents +11
Target Protein:
11-beta-hydroxysteroid dehydrogenase 1Glucocorticoid receptorNuclear receptor coactivator 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cortisone DB14681
small molecule | CAS: 53-06-5

A naturally occurring glucocorticoid. It has been used in replacement therapy for adrenal insufficiency and as an anti-inflammatory agent. Cortisone itself is inactive. It is converted in the liver to the active metabolite hydrocortisone. (From Martindale, Th…

Kategori:
17-HydroxycorticosteroidsAdrenal Cortex HormonesAnti-Inflammatory Agents +21
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cortisone acetate Approved DB01380
small molecule | CAS: 50-04-4

Cortisone acetate was first isolate in 1935 and became more widely researched in 1949.[A226295] Since then, glucocorticoids such as cortisone acetate have been used to treat a number of inflammatory conditions such as endocrine, rheumatic, collagen, dermatolo…

Kategori:
17-HydroxycorticosteroidsAdrenal Cortex HormonesAdrenals +25
Target Protein:
Steroid hormone receptor ERR2Estrogen-related receptor gammaGlucocorticoid receptor +2
Waktu Paruh-
Vol. Distribusi-
KlirensData regarding the …
Genetik -
Corylus americana pollen Approved DB10363
biotech

Corylus americana pollen is the pollen of the Corylus americana plant. Corylus americana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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