Hasil Filter

12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (12560)

Halaman 74 / 252
Cefetamet DB13504
small molecule | CAS: 65052-63-3

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 65243-33-6

Cefetamet pivoxil is under investigation in clinical trial NCT04664803 (Safety and Efficacy of Cefecin Tab. in Patients With Acute Sinusitis).

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefiderocol Approved DB14879
small molecule | CAS: 1225208-94-5

Cefiderocol is a cephalosporin antibacterial drug and exerts a mechanism of action similar to other ?-lactam antibiotics.[FDA Label] Unlike other agents in this category, cefiderocol is a siderophore able to undergo active transport into the bacterial cell th…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Cell division proteinPenicillin-binding protein 1APenicillin-binding protein 1B +2
Waktu ParuhThe terminal elimin…
Vol. DistribusiCefiderocol has a m…
KlirensCefiderocol has a m…
Genetik -
Cefilavancin DB05735
small molecule | CAS: 722454-12-8

Cefilavancin is a covalently-linked glycopeptide-cephalosporin (beta-lactam) heterodimer antibiotic that exhibits substantially greater activity than its component parts against Gram-positive bacteria.

Kategori:
AmidesAmino Acids, Peptides, and Proteinsbeta-Lactams +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefixime Approved DB00671
small molecule | CAS: 79350-37-1

Bacteria possess a cell wall comprising a glycopeptide polymer commonly known as peptidoglycan, which is synthesized and remodelled through the action of a family of enzymes known as "penicillin-binding proteins" (PBPs).[A232920] ?-lactam antibiotics, includi…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
Penicillin-binding proteinPenicillin-binding protein 2
Waktu ParuhCefixime has a seru…
Vol. DistribusiCefixime has a volu…
KlirensCefixime administer…
Genetik -
Cefmenoxime Approved DB00267
small molecule | CAS: 65085-01-0

Cefmenoxime is a novel broad-spectrum and third-generation cephalosporin antibiotic that is typically used in the treatment of female gynecologic and obstetric infections. It is reported to exhibit high activity against a wide variety of gram-positive and gra…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1A
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
Cefmetazole Approved DB00274
small molecule | CAS: 56796-20-4

A semisynthetic cephamycin antibiotic with a broad spectrum of activity against both gram-positive and gram-negative microorganisms. It has a high rate of efficacy in many types of infection and to date no severe side effects have been noted.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
Penicillin binding protein 2aPenicillin-binding protein 1APenicillin-binding protein 1B +3
Waktu Paruh1.50 ±0.14 h…
Vol. Distribusi-
Klirens-
Genetik -
Cefminox DB09062
small molecule | CAS: 84305-41-9

Cefminox (INN) is a second generation cephalosporin antibiotic. It is approved for use in Japan.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefonicid Approved DB01328
small molecule | CAS: 61270-58-4

A second-generation cephalosporin administered intravenously or intramuscularly. Its bactericidal action results from inhibition of cell wall synthesis. It is used for urinary tract infections, lower respiratory tract infections, and soft tissue and bone infe…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1APeptidoglycan synthase FtsIPenicillin-binding protein 1B +2
Waktu Paruh4.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Cefoperazone Approved DB01329
small molecule | CAS: 62893-19-0

Cefoperazone is a semisynthetic broad-spectrum cephalosporin proposed to be effective against <i>Pseudomonas</i> infections. It is a third-generation antiobiotic agent and it is used in the treatment of various bacterial infections caused by susceptible organ…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1BPenicillin-binding protein 2 +6
Waktu ParuhThe mean serum half…
Vol. Distribusi-
Klirens-
Genetik -
Ceforanide Approved DB00923
small molecule | CAS: 60925-61-3

Ceforanide is administered parenterally. It has a longer elimination half-life than any currently available cephalosporin. Its activity is very similar to that of cefamandole, another second-generation cephalosporin antibiotic, except that ceforanide is less …

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 2
Waktu Paruh2.6 to 2.98 hours
Vol. Distribusi-
Klirens-
Genetik -
Cefotaxime Approved DB00493
small molecule | CAS: 63527-52-6

Cefotaxime is a third-generation cephalosporin antibiotic. Like other third-generation cephalosporins, it has broad spectrum activity against Gram positive and Gram negative bacteria. In most cases, it is considered to be equivalent to ceftriaxone in terms of…

Kategori:
Agents that reduce seizure thresholdAmidesAnti-Bacterial Agents +13
Target Protein:
Penicillin-binding protein 1bPenicillin-binding protein 2aPenicillin-binding protein 3 +10
Waktu ParuhApproximately 1 hou…
Vol. Distribusi-
Klirens-
Genetik -
Cefotetan Approved DB01330
small molecule | CAS: 69712-56-7

A semisynthetic cephamycin antibiotic that is administered intravenously or intramuscularly. The drug is highly resistant to a broad spectrum of beta-lactamases and is active against a wide range of both aerobic and anaerobic gram-positive and gram-negative m…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
Penicillin-binding protein 3
Waktu ParuhIn volunteers with …
Vol. Distribusi* 10.4 L [elderly p…
Klirens* 1.8 +/- 0.1 L/h […
Genetik -
Cefotiam Approved DB00229
small molecule | CAS: 61622-34-2

One of the cephalosporins that has a broad spectrum of activity against both gram-positive and gram-negative microorganisms.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1A
Waktu ParuhApproximately 1 hou…
Vol. Distribusi-
Klirens-
Genetik -
Cefovecin DB11505
small molecule

Cefovecin is a cephalosporin antibiotic used for the treatment of skin infections in cats and dogs. It is the first single-dose injectable antibiotic for dogs and cats that assures owner compliance with dosing for the animal. It is used for the treatment of s…

Kategori:
Amidesbeta-LactamsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefoxitin Approved DB01331
small molecule | CAS: 35607-66-0

Cefoxitin is a semi-synthetic, broad-spectrum cepha antibiotic for intravenous administration. It is derived from cephamycin C, which is produced by <i>Streptomyces lactamdurans</i>.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
D-alanyl-D-alanine carboxypeptidase DacCD-alanyl-D-alanine carboxypeptidase DacAD-alanyl-D-alanine endopeptidase +9
Waktu ParuhThe half-life after…
Vol. Distribusi-
Klirens-
Genetik -
Cefozopran DB13667
small molecule | CAS: 113359-04-9

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
Dihydropteroate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefpirome Approved DB13682
small molecule | CAS: 84957-29-9

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefprozil Approved DB01150
small molecule | CAS: 92665-29-7

Cefprozil is a cephalosporin antibiotic that is commonly employed to treat a variety of bacterial infections, including those of the ear and skin, bronchitis, and others.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 2xPenicillin-binding protein 2B
Waktu Paruh1.3 hours
Vol. Distribusi* 0.23 L/kg
Klirens* 3 mL/min/kg [fast…
Genetik -
Cefradine Approved DB01333
small molecule | CAS: 38821-53-3

A semi-synthetic cephalosporin antibiotic.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +18
Target Protein:
Penicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefroxadine DB11367
small molecule | CAS: 51762-05-1

Cefroxadine is an orally available cephalosporin antibiotic. As part of its drug class, it shares structural properties to [cefalexin] as well as its activity spectrum. It was used in Italy but has since been withdrawn.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +10
Target Protein:
Penicillin-binding protein 1B
Waktu ParuhThe serum half life…
Vol. DistribusiVolume of distrubut…
KlirensThe total body clea…
Genetik -
Cefsulodin DB13499
small molecule | CAS: 62587-73-9

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceftaroline fosamil Approved DB06590
small molecule | CAS: 229016-73-3

Ceftaroline fosamil is a cephalosporin antibacterial indicated for the treatment of the following infections caused by designated susceptible bacteria: Acute bacterial skin and skin structure infections. Community-acquired bacterial pneumonia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein
Waktu Paruh1.60 hours (600 mg …
Vol. DistribusiMedian 20.3 L (18.3…
Klirens-
Genetik -
Ceftazidime Approved DB00438
small molecule | CAS: 72558-82-8

Bacteria possess a cell wall comprising a glycopeptide polymer commonly known as peptidoglycan, which is synthesized and remodelled through the action of a family of enzymes known as "penicillin-binding proteins" (PBPs).[A232920] ?-lactam antibiotics, includi…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1APenicillin-binding protein 1B +2
Waktu ParuhCeftazidime has an …
Vol. DistribusiCeftazidime has a v…
KlirensThe mean renal clea…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-lactamaseBeta-lactamase TEMBeta-lactamase CTX-M
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceftibuten Approved DB01415
small molecule | CAS: 97519-39-6

Ceftibuten is a third-generation cephalosporin antibiotic that is orally-administered. It is typically used to treat acute bacterial exacerbations of chronic bronchitis (ABECB), acute bacterial otitis media, pharyngitis, and tonsilitis.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1APenicillin-binding protein 1B +1
Waktu Paruh-
Vol. Distribusi* 0.21 L/kg [adult …
Klirens-
Genetik -
Ceftiofur DB11485
small molecule | CAS: 80370-57-6

Ceftiofur is a third generation cephalosporin antibiotic, first described in 1987, and now used in veterinary medicine. It is marketed by pharmaceutical company Zoetis as Excenel, and is the active ingredient in that company's Specramast LC (lactating cow for…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceftizoxime Approved DB01332
small molecule | CAS: 68401-81-0

A semisynthetic cephalosporin antibiotic which can be administered intravenously or by suppository. The drug is highly resistant to a broad spectrum of beta-lactamases and is active against a wide range of both aerobic and anaerobic gram-positive and gram-neg…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 1BPeptidoglycan transpeptidase +1
Waktu Paruh-
Vol. DistribusiThe mean apparent v…
Klirens-
Genetik -
Ceftobiprole Approved DB04918
small molecule | CAS: 209467-52-7

Ceftobiprole is a fifth-generation semisynthetic cephalosporin antibacterial which is available commercially as the prodrug [ceftobiprole medocaril]. Ceftobiprole is a broad-spectrum agent with demonstrated activity against both Gram-positive and Gram-negativ…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
MecAPenicillin-binding protein 2xPenicillin-binding protein 2B +2
Waktu ParuhThe half-life of ac…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
Ceftobiprole medocaril Approved DB14733
small molecule | CAS: 376653-43-9

Ceftobiprole medocaril is a prodrug of [ceftobiprole], a fifth-generation semisynthetic cephalosporin antibacterial. Ceftobiprole is a broad-spectrum agent with demonstrated activity against both Gram-positive and Gram-negative bacteria, including antibiotic-…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
MecAPenicillin-binding protein 2BPenicillin-binding protein 2X
Waktu ParuhThe half-life of ac…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
Ceftolozane Approved DB09050
small molecule | CAS: 689293-68-3

Ceftolozane is a semi-synthetic broad-spectrum fifth generation cephalosporin.[L6685] It was approved by the FDA in 2014 for use in combination with [Tazobactam] for the treatment of serious infections, such as intra-abdominal infections and complicated urina…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +8
Target Protein:
Penicillin-binding protein 1BCell division proteinPenicillin-binding protein 1C +2
Waktu Paruh2.77 hours on day 1…
Vol. Distribusi13.5 L.[L41618] Tis…
KlirensThe renal clearance…
Genetik -
Ceftriaxone Approved DB01212
small molecule | CAS: 73384-59-5

Ceftriaxone is a broad-spectrum third-generation cephalosporin antibiotic.[A215582] It has a very long half-life compared to other cephalosporins and is high penetrable into the meninges[A215582], eyes[A215647], and inner ear[A215627]. Ceftriaxone has broader…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
Penicillin-binding protein 2BSolute carrier family 22 member 11Solute carrier family 22 member 6 +2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe plasma clearanc…
Genetik -
Cefuroxime Approved DB01112
small molecule | CAS: 55268-75-2

Broad-spectrum cephalosporin antibiotic resistant to beta-lactamase. It has been proposed for infections with gram-negative and gram-positive organisms, gonorrhea, and haemophilus.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
Penicillin-binding protein 1A
Waktu ParuhApproximately 80 mi…
Vol. Distribusi-
Klirens-
Genetik -
Celastrol DB18736
small molecule | CAS: 34157-83-0

Celastrol is a pentacyclic triterpenoid isolated from the root extracts of _Tripterygium wilfordii_.[L50567]

Kategori:
TerpenesTripterygiumTriterpenes
Target Protein:
Interleukin-1 betaTumor necrosis factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Celecoxib Approved DB00482
small molecule | CAS: 169590-42-5

Celecoxib, a selective cyclooxygenase-2 (COX-2) inhibitor, is a nonsteroidal anti-inflammatory drug (NSAID) which is known for its decreased risk of causing gastrointestinal bleeding compared to other NSAIDS.[A181544] It is used to manage symptoms of various …

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +41
Target Protein:
Prostaglandin G/H synthase 2Signal transducer and activator of transcription 3Sialidase-1 +4
Gen Terkait:
CYP2C9
Waktu ParuhThe effective half-…
Vol. DistribusiThe apparent volume…
KlirensApparent clearance …
Genetik 1 Varian
Celery Approved DB10517
biotech

Celery allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Celgosivir DB06580
small molecule | CAS: 121104-96-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingIndolizines
Target Protein:
Maltase-glucoamylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Celiprolol Approved DB04846
small molecule | CAS: 56980-93-9

Celiprolol is indicated for the management of mild to moderate hypertension and effort-induced angina pectoris. It is simultaneously a selective ?1 receptor antagonist, a ?2 receptor partial agonist and a weak ?2 receptor antagonist. In 2010 a clinical trial …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic Antagonists +30
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor +3
Waktu Paruh5 hours
Vol. DistribusiThe distribution vo…
KlirensCleared by both ren…
Genetik -
Celivarone DB16012
small molecule | CAS: 401925-43-7

Celivarone is under investigation in clinical trial NCT00233441 (Placebo Controlled Double-blind Dose Ranging Study of the Efficacy and Safety of SSR149744C 50, 100, 200 or 300 Mg OD With Amiodarone as Calibrator for the Maintenance of Sinus Rhythm in Patient…

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cellobiose DB02061
small molecule | CAS: 528-50-7

A disaccharide consisting of two glucose units in beta (1-4) glycosidic linkage. Obtained from the partial hydrolysis of cellulose. [PubChem]

Kategori:
CarbohydratesCelluloseCompounds used in a research, industrial, or household setting +4
Target Protein:
Endoglucanase GEndoglucanase 5AEndoglucanase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cemdomespib DB18953
small molecule | CAS: 1450642-92-8

Cemdomespib is under investigation in clinical trial NCT05895552 (A Phase 2 Study of RTA 901 in Patients With Diabetic Peripheral Neuropathic Pain (CYPRESS)).

Kategori:
AminesCarbohydratesEthylamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cemiplimab Approved DB14707
biotech | CAS: 1801342-60-8

Cemiplimab is a fully human monoclonal antibody that works against programmed death receptor-1 (PD-1), which is a negative regulator of T cell function. By blocking PD-1, cemiplimab works to enhance T cell-mediated antitumour responses.[L39804] Cemiplimab …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Programmed cell death protein 1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensCemiplimab clearanc…
Genetik -
Cemsidomide DB18400
small molecule | CAS: 2504235-67-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cendakimab DB18427
biotech

Cendakimab is a recombinant humanized anti-interleukin 13 (IL-13) monoclonal antibody.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenderitide DB11777
biotech | CAS: 507289-11-4

Cenderitide is under investigation for the treatment of ST Elevation (STEMI) Myocardial Infarction of Anterior Wall.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsComplex Mixtures +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenegermin Approved DB13926
biotech | CAS: 1772578-74-1

Cenegermin is a human beta-nerve growth factor (beta-ngf)-(1-118)- peptide (non-covalent dimer) produced in escherichia coli. It received European Union Approval in July 2017 for the treatment of moderate to severe neurotrophic keratitis. Cenegermin received …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +7
Target Protein:
High affinity nerve growth factor receptorTumor necrosis factor receptor superfamily member 16
Waktu ParuhHalf-life data spec…
Vol. DistribusiAfter eye drop admi…
KlirensAlthough the system…
Genetik -
Cenerimod DB12705
small molecule | CAS: 1262414-04-9

Cenerimod has been used in trials studying the treatment of Systemic Lupus Erythematosus.

Kategori:
AlcoholsGlycolsOxazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenersen DB15455
biotech | CAS: 415168-49-9

Cenersen is under investigation in clinical trial NCT02243124 (A Study of Aezea® (Cenersen) in Transfusion Dependent Anemia Associated With Myelodysplastic Syndrome (MDS)).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenicriviroc DB11758
small molecule | CAS: 497223-25-3

Cenicriviroc has been used in trials studying the treatment of HIV-infection/AIDS, AIDS Dementia Complex, Nonalcoholic Steatohepatitis, Human Immunodeficiency Virus, and HIV-1-Associated Cognitive Motor Complex.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +4
Target Protein:
C-C chemokine receptor type 5C-C chemokine receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenisertib DB06347
small molecule | CAS: 871357-89-0

Cenisertib is an aurora kinase inhibitor.

Kategori:
Bridged-Ring Compounds
Target Protein:
Aurora kinase BAurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 3651–3700 dari 12560
Sebelumnya Halaman 74 / 252 Berikutnya