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14361

Total database: 17430
Struktur (SMILES)
9916 (69.0%)
Target
7893 (55.0%)
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112 (0.8%)
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14361 (100.0%)

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Hasil Pencarian (14361)

Halaman 73 / 288
Bezitramide DB01459
small molecule | CAS: 15301-48-1

Bezitramide is a narcotic analgesic which was discovered in 1961, clinically tested around the 1970's [A14383], and marketed under the name Burgodin. After cases of fatal overdose in the Netherlands in 2004 the drug was withdrawn from the market. Bezitram…

Kategori:
AnalgesicsCentral Nervous System AgentsDiphenylpropylamine Derivatives +6
Waktu Paruh11-24h. [A14383]
Vol. Distribusi-
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Bezlotoxumab Approved DB13140
biotech | CAS: 1246264-45-8

Bezlotoxumab is a fully humanized ImmunoglobulinG1 (IgG1) kappa monoclonal antibody that binds to _Clostridium difficile_ toxin B and neutralizes its effects.[L46976] First approved by the FDA on October 21, 2016,[A260106] bezlotoxumab is used to reduce the r…

Kategori:
Amino Acids, Peptides, and ProteinsAntibacterial monoclonal antibodiesAntibodies +11
Target Protein:
Toxin B
Waktu ParuhBased on a populati…
Vol. DistribusiBased on a populati…
KlirensBased on a populati…
Genetik -
Bezuclastinib DB18041
small molecule | CAS: 1616385-51-3

Deskripsi belum tersedia.

Target Protein:
Mast/stem cell growth factor receptor Kit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BF-1 DB06029
small molecule | CAS: 518980-66-0

BF-1 is an investigational 5-HT2B receptor antagonist developed for the prophylaxis of Migraines.

Target Protein:
5-hydroxytryptamine receptor 2B
Waktu Paruh-
Vol. Distribusi-
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BF-37 DB05755
small molecule

BF-37 for the treatment of atopic dermatitis and/or psoriasis. The active ingredient in BF-37 is Riluzole, applied in a topical formulation, which is believed to correct the imbalances of the immune system that cause atopic dermatitis or psoriasis.

Waktu Paruh-
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BF-844 DB17801
small molecule | CAS: 1404506-35-9

Deskripsi belum tersedia.

Waktu Paruh-
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BFH772 DB16035
small molecule | CAS: 890128-81-1

BFH772 is under investigation in clinical trial NCT01449591 (Safety, Tolerability and Efficacy of BFH772 in Rosacea Patients).

Waktu Paruh-
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Bfpet F-18 DB15424
small molecule | CAS: 863644-14-8

Bfpet F-18 is under investigation in clinical trial NCT03265431 (Evaluation of PET/MR in Patients Selected for Ablation Therapy).

Waktu Paruh-
Vol. Distribusi-
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BG-777 DB05839
small molecule

BG-777 is an immunomodulator with proven efficacy against viral and bacterial infections in preclinical studies.

Waktu Paruh-
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BG-P-TAT DB18105
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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BG-P400-TAT DB17104
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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BG1805 DB18667
biotech

BG1805 is an investigational anti-CLL1 chimeric antigen receptor (CAR) T-cell therapy.

Waktu Paruh-
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BGA002 DB17125
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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BGB-DXP593 DB16357
biotech

BGB-DXP593 is a SARS-CoV-2 neutralizing antibody.[L27401] It is currently being investigated against COVID-19 in the clinical trial NCT04551898 (Severe Acute Respiratory Syndrome Coronavirus 2 (SARS-CoV-2) Neutralizing Antibody BGB-DXP593 in Participants With…

Waktu Paruh-
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BGT-DTDS DB18664
biotech

BGT-DTDS is an investigational gene therapy comprising an adeno-associated viral vector type 2 (AAV2) encoding the human _SLC6A3_ gene. It is under investigation for the treatment of dopamine transporter deficiency syndrome (DTDS).

Waktu Paruh-
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BHT-3034 DB18045
biotech

BHT-3034 is a DNA plasmid vaccine immunotherapy under investigation for the treatment of myasthenia gravis.[L48086]

Waktu Paruh-
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BHV-5000 DB17817
small molecule

BHV-5000 is an orally bioavailable, low-trapping, potent N-methyl-D-aspartate (NMDA) receptor antagonist. The active metabolite of BHV-5000 is [lanicemine].[L46446]

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BI-187004 DB18897
small molecule | CAS: 1303515-32-3

Deskripsi belum tersedia.

Waktu Paruh-
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BI-671800 DB12524
small molecule | CAS: 1093108-50-9

Bi 671800 has been used in trials studying the treatment of Asthma and Rhinitis, Allergic, Perennial.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Prostaglandin D2 receptor 2
Waktu Paruh-
Vol. Distribusi-
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BI-765063 DB17482
biotech

BI-765063 is a humanized IgG4 monoclonal antibody antagonist of signal regulatory protein ? (SIRP?).

Waktu Paruh-
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BI-836858 DB17267
biotech | CAS: 2206770-25-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
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BI-836880 DB17484
biotech

BI-836880 is a humanized bispecific nanobody that targets VEGF and Ang2.

Waktu Paruh-
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BI-K0376 DB05858
biotech

BI-K0376 is investigated for use/treatment in acne. BI-K0376 is a solid. It is under investigation by Pfizer and has gone through phase I of the clinical trails.

Waktu Paruh-
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Biapenem DB13028
small molecule | CAS: 120410-24-4

Biapenem has been used in trials studying the treatment of Bacterial Infections.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +6
Waktu Paruh-
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Bicalutamide Approved DB01128
small molecule | CAS: 90357-06-5

Bicalutamide is an oral non-steroidal anti-androgen for prostate cancer. It is comprised of a racemic mixture that is a 50:50 composition of the (R)-bicalutamide and (S)-bicalutamide enantionmers. Bicalutamide binds to the androgen receptor.

Kategori:
AmidesAminesAndrogen Receptor Antagonists +31
Target Protein:
Androgen receptor
Waktu Paruh5.9 days
Vol. Distribusi-
Klirens* Apparent oral cl=…
Genetik -
Bicifadine DB04889
small molecule | CAS: 71195-57-8

Bicifadine (DOV-220075) is a nonopioid analgesic. It is an inhibitor of both the norepinephrine and serotonin transporters and an NMDA antagonist with a non-narcotic profile. Bicifadine was shown to have potent analgesic activity in vivo and was chosen for fu…

Kategori:
AnalgesicsCytochrome P-450 CYP1A2 SubstratesCytochrome P-450 CYP2D6 Substrates +2
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Bicisate Approved DB11164
small molecule | CAS: 121251-02-3

Bicisate, also known as ethyl cysteinate dimer (ECD), is a N,N'-1,2-ethylene-di-yl-bis-L-cysteinate diethyl ester. It is used in conjunction with technetium Tc99m as a tracer to measure cerebral blood flow with single-photon emission computed tomography (SPEC…

Kategori:
Diagnostic AgentsDrugs that are Mainly Renally ExcretedRadioactive Diagnostic Agent
Waktu ParuhThe stability of bi…
Vol. DistribusiAfter intravenous a…
KlirensThe clearance of bi…
Genetik -
Bictegravir Approved DB11799
small molecule | CAS: 1611493-60-7

Bictegravir is a recently approved investigational drug that has been used in trials studying the treatment of HIV-1 and HIV-2 infection. It has been approved for HIV-1 monotherapy combined with 2 other antiretrovirals in a single tablet.[L43677]

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +11
Target Protein:
Reverse transcriptase/RNaseHIntegrase
Waktu ParuhHalf-life is 17.3 h…
Vol. Distribusi0.2 L/Kg in humans …
KlirensBictegravir is main…
Genetik -
Bicuculline DB11562
small molecule | CAS: 485-49-4

Bicuculline is a light-sensitive competitive antagonist of GABAA receptors. It was originally identified in 1932 in plant alkaloid extracts and has been isolated from Dicentra cucullaria, Adlumia fungosa, Fumariaceae, and several Corydalis species.

Kategori:
AlkaloidsBenzylisoquinolinesCentral Nervous System Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Bicyclol DB16014
small molecule | CAS: 118159-48-1

Bicyclol is under investigation in clinical trial NCT02944552 (The Multi Center, Randomized, Double-blind, Positive Controlled Study of Bicyclol in the Treatment of Acute DILI).

Kategori:
Benzene Derivatives
Waktu Paruh-
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Genetik -
biotech

Deskripsi belum tersedia.

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Bietaserpine DB13575
small molecule | CAS: 53-18-9

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntiadrenergic Agents, Centrally ActingAntihypertensive Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Bifenthrin DB15056
small molecule | CAS: 82657-04-3

Bifenthrin is under investigation in clinical trial NCT01560247 (Percutaneous Recanalization in Ischemic Stroke Management in Europe Observational Registry).

Kategori:
Cyclopentane MonoterpenesMonoterpenesSarcoma, Experimental, chemically induced +1
Waktu Paruh-
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Klirens-
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Bifeprunox DB04888
small molecule | CAS: 350992-10-8

Bifeprunox is a novel atypical antipsychotic agent which, along with SLV313, [aripiprazole] and SSR-181507 combines minimal D2 receptor agonism with 5-HT receptor agonism.

Kategori:
Antipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical])Central Nervous System Depressants +2
Target Protein:
5-hydroxytryptamine receptor 1AD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Probiotics
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Bifidobacterium Longum Infantis 35624 is a probiotic being investigated for the treatment of gastrointestinal disorders, such as Crohn's disease and irritable bowel syndrome.[A259872, A259877]

Waktu Paruh-
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biotech

Deskripsi belum tersedia.

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Bifikafusp alfa DB19185
biotech | CAS: 1957239-90-5

Bifikafusp alfa is under investigation in clinical trial NCT05329792 (L19IL2/L19TNF in Skin Cancer Patients).

Waktu Paruh-
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Bifonazole Approved DB04794
small molecule | CAS: 60628-96-8

Bifonazole is an azole antifungal drug.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +10
Target Protein:
Lanosterol 14-alpha demethylaseCytochrome P450 2B6
Waktu Paruh1-2 hours
Vol. Distribusi-
Klirens-
Genetik -
biotech

Bifunctional epoxide hydrolase 2 is under investigation in clinical trial NCT00654966 (Evaluation of the Effects of Urotensin-II and Soluble Epoxide Hydrolase Inhibitors on Skin Microvessel Tone in Patients With Heart Failure, and in Healthy Volunteers).

Waktu Paruh-
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BIIB015 DB06304
biotech

BIIB015 is a humanized, IgG1 [immunoglobulin G 1], DM4-Conjugated, anti-cripto, monoclonal antibody. It has been investigated for the treatment of subjects with relapsed or refractory solid tumours.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
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BIIB021 DB12359
small molecule | CAS: 848695-25-0

BIIB021 has been investigated for the treatment of Tumors and Lymphoma.

Kategori:
Heterocyclic Compounds, Fused-RingHSP90 Heat-Shock Proteins, antagonists & inhibitorsPurines
Target Protein:
Heat shock protein HSP 90-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
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BIIB115 DB18418
biotech

BIIB115 is an investigational antisense oligonucleotide in development for spinal muscular atrophy.

Waktu Paruh-
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Bilastine Approved DB11591
small molecule | CAS: 202189-78-4

Bilastine is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of action.

Kategori:
Antihistamines for Systemic UseDecongestants and AntiallergicsHeterocyclic Compounds, Fused-Ring +8
Target Protein:
Histamine H1 receptor
Waktu ParuhThe mean half life …
Vol. Distribusi-
KlirensBilastine has a tot…
Genetik -
Bilberry Approved DB14235
biotech

Deskripsi belum tersedia.

Kategori:
AngiospermsBenzopyransBiological Factors +21
Waktu Paruh-
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Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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small molecule | CAS: 114-25-0

Deskripsi belum tersedia.

Target Protein:
Heme oxygenase 1MyoglobinFlavin reductase (NADPH)
Waktu Paruh-
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Bimagrumab DB12584
biotech | CAS: 1356922-05-8

Bimagrumab has been used in trials studying the treatment and supportive care of Sarcopenia, Skeletal Muscle, Mechanical Ventilation, Sporadic Inclusion Body Myositis, and Sporadic Inclusion Body Myositis (sIBM), among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
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Bimatoprost Approved DB00905
small molecule | CAS: 155206-00-1

Bimatoprost, also known as Latisse or Lumigan, belongs to a group of drugs called prostamides, which are synthetic structural analogs of prostaglandin. Bimatoprost, marketed by Allergan, is administered in both the ophthalmic solution and implant form. It has…

Kategori:
AmidesAntiglaucoma Preparations and MioticsAntihypertensive Agents +19
Target Protein:
Prostaglandin F2-alpha receptorProstaglandin E2 receptor EP1 subtypeProstaglandin E2 receptor EP3 subtype
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance was m…
Genetik -
Bimekizumab Approved DB12917
biotech | CAS: 1418205-77-2

Bimekizumab is a humanized monoclonal antibody directed towards IL-17, which was approved for use in the EU on August 20, 2021, for the treatment of plaque psoriasis.[L39665,L39680] It is the first IL-17 inhibitor to target both IL-17A and IL-17F.[A244455] It…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +11
Target Protein:
Interleukin-17AInterleukin-17F
Waktu ParuhThe mean terminal e…
Vol. DistribusiIn patients with pl…
KlirensThe median apparent…
Genetik -
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