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11793

Total database: 17430
Struktur (SMILES)
8607 (73.0%)
Target
6418 (54.4%)
Genomik
102 (0.9%)
Referensi
11793 (100.0%)

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Hasil Pencarian (11793)

Halaman 73 / 236
Clorazepic acid Approved DB00628
small molecule | CAS: 23887-31-2

Clorazepic acid (clorazepate) is a water-soluble benzodiazepine with muscle-relaxant and anticonvulsant actions effective in the treatment of anxiety.[A957,L44788] Following administration, clorazepate is rapidly converted to nordiazepam (N-desmethyldiazepam)…

Kategori:
Anti-Anxiety AgentsAnticonvulsantsBenzazepines +15
Target Protein:
GABA(A) ReceptorTranslocator proteinGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhThe serum half-life…
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Clorexolone DB13617
small molecule | CAS: 2127-01-7

Deskripsi belum tersedia.

Kategori:
AmidesDiureticsHeterocyclic Compounds, Fused-Ring +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cloricromen DB13367
small molecule | CAS: 68206-94-0

Deskripsi belum tersedia.

Kategori:
Antiplatelet agentsBenzopyransBlood and Blood Forming Organs +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cloridarol DB13291
small molecule | CAS: 3611-72-1

Cloridarol is an experimental medication in the treatment of heart disease, which acts through vasodilation. It was studied for the treatment of coronary insufficiency in Italy in the 1970s [A176222].

Kategori:
Cardiac TherapyHeterocyclic Compounds, Fused-RingVasodilators Used in Cardiac Diseases
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clorindione DB13275
small molecule | CAS: 1146-99-2

Clorindione is a vitamin K antagonist, which may be useful to decrease prothrombin levels in humans.

Kategori:
AnticoagulantsBlood and Blood Forming OrgansIndenes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clorobiocin DB03966
small molecule | CAS: 39868-96-7

Clorobiocin is an aminocoumarin antibiotic, similar to [novobiocin] and coumermycin A1.

Kategori:
AminocoumarinsBenzopyransCarbohydrates +4
Target Protein:
DNA topoisomerase 2-betaDNA topoisomerase 2-alphaDNA gyrase subunit B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clorsulon DB11389
small molecule | CAS: 60200-06-8

Deskripsi belum tersedia.

Kategori:
AmidesAminesAniline Compounds +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 855-19-6

Deskripsi belum tersedia.

Kategori:
AndrostanesAndrostenesAndrostenols +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clostridium tetani Approved DB09876
biotech

Deskripsi belum tersedia.

Kategori:
Inactivated Clostridium Tetani Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clothiapine Approved DB13256
small molecule | CAS: 2058-52-8

Clothiapine has been approved in European countries and is an atypical antipsychotic, shown to be useful in some treatment-resistant patients.

Kategori:
Antipsychotic AgentsCentral Nervous System AgentsCentral Nervous System Depressants +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clotiazepam Approved DB01559
small molecule | CAS: 33671-46-4

Clotiazepam is a thienodiazepine, not approved for sale in the U.S. or Canada, but has been approved in the U.K. It is a schedule IV drug in Canada.

Kategori:
Anti-Anxiety AgentsBenzodiazepines and benzodiazepine derivativesCentral Nervous System Depressants +8
Target Protein:
GABA(A) ReceptorTranslocator proteinGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh4 hours
Vol. Distribusi-
Klirens-
Genetik -
Clotrimazole Approved DB00257
small molecule | CAS: 23593-75-1

This drug is a broad spectrum antimycotic or antifungal agent. Clotrimazole's antimycotic properties were discovered in the late 1960s [A174094]. Clotrimazole falls under the _imidazole_ category of _azole_ antifungals, possessing broad-spectrum antimycotic a…

Kategori:
Anti-Infective AgentsAnti-Infective Agents, LocalAntifungal Agents +54
Target Protein:
C-X-C chemokine receptor type 2Lanosterol 14-alpha demethylaseIntermediate conductance calcium-activated potassium channel protein 4 +3
Waktu Paruh-
Vol. DistribusiThe topical form is…
Klirens-
Genetik -
Clove Approved DB10672
biotech | CAS: 84961-50-2

Clove allergenic extract is used in allergenic testing.

Kategori:
AngiospermsBiological ProductsCell-mediated Immunity +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cloxacillin Approved DB01147
small molecule | CAS: 61-72-3

A semi-synthetic penicillin antibiotic which is a chlorinated derivative of [oxacillin].

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
D-alanyl-D-alanine carboxypeptidase DacAPenicillin-binding protein 2XPenicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cloxazolam DB01553
small molecule | CAS: 24166-13-0

Cloxazolam is a benzodiazepine with anxiolytic, sedative/hypnotic, muscle relaxant, and antiepileptic effects. It is marketed in the Argentina, Australia, Portugal, Belgium, Switzerland, Luxembourg, Germany, Taiwan and Japan -- mainly for anti-anxiety. The us…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +4
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh65 hours
Vol. Distribusi-
Klirens-
Genetik -
Cloxyquin DB15933
small molecule | CAS: 130-16-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingHydroxyquinolinesQuinolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Clozapine Approved DB00363
small molecule | CAS: 5786-21-0

Clozapine is a tricyclic dibenzodiazepine, classified as an atypical antipsychotic agent.[A256708] Clozapine displays affinity to various neuroreceptors with a particularly low affinity to the dopamine receptors, thus breaking the mold of first-generation ant…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +65
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2AD(1A) dopamine receptor +30
Gen Terkait:
GNB3
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe median volume o…
KlirensThe median clearanc…
Genetik 1 Varian
CLZ-2002 DB18638
biotech

CLZ-2002 consists of allogeneic mesenchymal stem cells derived neuronal regeneration-promoting cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CM-4307 DB15414
small molecule | CAS: 1130115-44-4

CM-4307 is under investigation in clinical trial NCT03602495 (Donafenib in 131I-Refractory Differentiated Thyroid Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CM4620 DB16466
small molecule | CAS: 1713240-67-5

CM4620 (Zegocractin), is under investigation in multiple clinical trials, including NCT04195347 (pancreatitis due to asparaginase), NCT03709342 (PK/PD study in acute pancreatitis), NCT03401190 and NCT04681066 (pancreatitis and SIRS), and NCT04661540 (critical…

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CMG901 DB18619
biotech

CMG901 is an anti-Claudin 18.2 monoclonal antibody conjugated with MMAE payload.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CMLVAX100 DB05164
biotech

CMLVAX100 is a vaccine targeting the BCR-ABL-derived p210 fusion protein which reduces residual disease in some patients with chronic myeloid leukemia. It is developed by Breakthrough Therapeutics and has completed phase I of its clinical trial.

Target Protein:
BCR/ABL p210 fusion protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CMX-2043 DB12795
small molecule | CAS: 910627-26-8

CMX-2043 has been used in trials studying the treatment and prevention of Non STEMI, Unstable Angina, Stable Coronary Artery Disease, and Percutaneous Coronary Intervention.

Kategori:
Amino Acids, Peptides, and ProteinsCoenzymesEnzymes and Coenzymes +6
Target Protein:
RAC-alpha serine/threonine-protein kinaseHepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CN-105 DB18345
small molecule | CAS: 1632243-07-2

CN-105 is a neuroprotective pentapeptide with the sequence Acetyl-Valine-Serine-Arginine-Arginine-Arginine-NH2 (Ac-VSRRR- NH2).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CN-201 DB18726
biotech

CN-201 is a humanized anti-CD3/CD19 bispecific antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CNS-5161 DB05824
small molecule

CNS 5161 is a blocker of the NMDA ion channel and has completed Phase IIa proof of concept clinical trials as a novel compound for the treatment of neuropathic pain.

Target Protein:
Glutamate receptor ionotropic, NMDA 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 102786-61-8

Recombinant human coagulation Factor VIIa (rFVIIa), intended for promoting hemostasis by activating the extrinsic pathway of the coagulation cascade. NovoSeven is a vitamin K-dependent glycoprotein consisting of 406 amino acid residues. Cloned and expressed i…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +15
Target Protein:
Coagulation factor XTissue factor
Waktu Paruh-
Vol. Distribusi* 121 ± 30 mL/kg [a…
Klirens* 33 - 37 mL/h x kg…
Genetik -
Coagulin-B DB17703
biotech

Coagulin-B is an adeno-associated viral vector expressing human blood-coagulation Factor IX.[A259038, A259043] It was previously investigated for the treatment of hemophilia; however, the manufacturing company discontinued the Phase I trial in 2004, halting i…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobalt chloride Approved DB14206
small molecule | CAS: 7646-79-9

Deskripsi belum tersedia.

Kategori:
Antimutagenic AgentsCompounds used in a research, industrial, or household settingElements +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobalt Co-60 DB15374
small molecule | CAS: 10198-40-0

Cobalt Co-60 is under investigation in clinical trial NCT02891083 (Adjuvant Therapies or Surgery Alone for High Risk pN0 Esophageal Cancer).

Kategori:
Cobalt IsotopesElementsIsotopes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 10124-43-3

Deskripsi belum tersedia.

Kategori:
ElementsMetalsMetals, Heavy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobamamide DB11191
small molecule | CAS: 13870-90-1

Cobamamide is one of the active forms of vitamin B12 that is also known as _adenosylcobalamin_ or _dibencozide_. This drug is available as a nutritional supplement to prevent vitamin B12 deficiency. Vitamin B12 is a collective term for these variously subs…

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansCoenzymes +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobicistat Approved DB09065
small molecule | CAS: 1004316-88-4

Cobicistat, marketed under the name Tybost (formerly GS-9350), indicated for treating infection with human immunodeficiency virus (HIV). Although it does not have any anti-HIV activity, cobicistat acts as a pharmacokinetic enhancer by inhibiting cytochrome P4…

Kategori:
Acids, AcyclicAnti-HIV AgentsAnti-Infective Agents +29
Target Protein:
Cytochrome P450 3A4Cytochrome P450 3A5Cytochrome P450 3A7
Waktu ParuhThe terminal plasma…
Vol. Distribusi-
Klirens-
Genetik -
Cobimetinib Approved DB05239
small molecule | CAS: 934660-93-2

Cobimetinib is an orally active, potent and highly selective small molecule inhibiting mitogen-activated protein kinase kinase 1 (MAP2K1 or MEK1), and central components of the RAS/RAF/MEK/ERK signal transduction pathway. It has been approved in Switzerland a…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2D6 Inhibitors +22
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 1
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe estimated appar…
KlirensFollowing oral admi…
Genetik -
Cobiprostone DB05514
small molecule | CAS: 333963-42-1

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +4
Target Protein:
Chloride channel protein 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobitolimod DB14819
biotech | CAS: 1226822-98-5

Cobitolimod is under investigation in clinical trial NCT03178669 (The Efficacy of Cobitolimod in Patients With Moderate to Severe Active Ulcerative Colitis).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Coblopasvir DB15315
small molecule | CAS: 1312608-46-0

Coblopasvir is under investigation in clinical trial NCT03416491 (Safety and Efficacy of KW-136 and Sofosbuvir for Treatment of Chronic Hepatitis C).

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2364477-18-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobolimab DB16372
biotech | CAS: 2022215-65-0

Cobolimab is under investigation in clinical trial NCT04655976 (Study of Cobolimab in Combination With Dostarlimab and Docetaxel in Advanced NSCLC Participants).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cobomarsen DB14931
biotech | CAS: 1848257-52-2

Cobomarsen is under investigation in clinical trial NCT02580552 (Safety, Tolerability and Pharmacokinetics of MRG-106 in Patients With Mycosis Fungoides (MF), CLL, DLBCL or ATLL).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cocaine Approved DB00907
small molecule | CAS: 50-36-2

An alkaloid ester extracted from the leaves of plants including coca. It is a local anesthetic and vasoconstrictor and is clinically used for that purpose, particularly in the eye, ear, nose, and throat. It also has powerful central nervous system effects sim…

Kategori:
Agents producing tachycardiaAgents that reduce seizure thresholdAlkaloids +36
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium channel protein +5
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61789-40-0

Cocamidopropyl betaine is a mixture of closely related organic compounds derived from coconut oil and dimethylaminopropylamine that typically acts as an amphoteric surfactant in cosmetics and personal care products. It is a zwitterionic ammonium compound and …

Kategori:
AminesCompounds used in a research, industrial, or household settingOnium Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cocarboxylase Approved DB01987
small molecule | CAS: 136-08-3

The coenzyme form of Vitamin B1 present in many animal tissues. It is a required intermediate in the pyruvate dehydrogenase complex and the ketoglutarate dehydrogenase complex.

Kategori:
CoenzymesEnzymes and CoenzymesMicronutrients +5
Target Protein:
RNAAcetolactate synthase, catabolicPyruvate dehydrogenase E1 component +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61791-31-9

Deskripsi belum tersedia.

Kategori:
AlcoholsAllergensAmines +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cocoa Approved DB10977
biotech | CAS: 84649-99-0

Cocoa allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cocoa butter Approved DB11086
biotech | CAS: 8002-31-1

Cocoa butter is an edible natural fat obtained from the _Theobroma cocoa_ seeds that is predominantly found in dark chocolate [A33033]. It is a rich source of monounsaturated and saturated fatty acids [A33040] that mainly contains approximately 33% [DB04224],…

Kategori:
Antipruritics and Local AnestheticsDiet, Food, and NutritionFats +3
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Cod liver oil DB11321
small molecule | CAS: 8001-69-2

Cod liver oil is extracted from the liver of cod fish and mainly consists of omega-3 fatty acids, eicosapentaenoic acid (EPA) and docosahexaenoic acid (DHA). Also being a rich source of vitamin A and D, cod liver oil can be taken orally as daily supplements. …

Kategori:
Diet, Food, and NutritionDietary FatsDietary Fats, Unsaturated +8
Waktu ParuhAs cod liver oil co…
Vol. DistribusiAs cod liver oil co…
KlirensAs cod liver oil co…
Genetik -
CODA-001 DB14915
biotech | CAS: 1605326-11-1

CODA-001 is under investigation in clinical trial NCT01165450 (Efficacy and Safety Study of Nexagon for Persistent Corneal Epithelial Defects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Codeine Approved DB00318
small molecule | CAS: 76-57-3

The relief of pain (analgesia) is a primary goal for enhancing the quality of life of patients and for increasing the ability of patients to engage in day to day activities. Codeine, an opioid analgesic, was originally approved in the US in 1950 and is a drug…

Kategori:
AlkaloidsAnalgesicsAntitussive Agents +26
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +6
Waktu ParuhPlasma half-lives o…
Vol. DistribusiApparent volume of …
KlirensRenal clearance of …
Genetik 9 Varian
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