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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 73 / 252
Catfish Approved DB14758
biotech

Catfish (unspecified) allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cathinone DB01560
small molecule | CAS: 71031-15-7

Cathinone is a monoamine alkaloid found in the shrub Catha edulis (Khat). Closely related to ephedrine, cathine and other amphetamines, it is probably the main contributor to the stimulant effect of Catha edulis. Cathinone differs from many other amphetamines…

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCentral Nervous System Stimulants +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Catridecacog Approved DB09310
biotech | CAS: 606138-08-3

Coagulation Factor XIII A-Subunit (Recombinant), also known as catridecacog, is a recombinant form of the Factor XIII-A2 homodimer composed of two factor XIII (FXIII) A-subunits [FDA Label]. For people with congenital deficiency or mutation of Factor XIII, a …

Kategori:
Blood and Blood Forming OrgansBlood Coagulation FactorsHemostatics
Target Protein:
Coagulation factor XIII B chain
Waktu Paruh7.1 days
Vol. Distribusi-
Klirens0.41 mL/h/kg
Genetik -
Catumaxomab Approved DB06607
biotech | CAS: 509077-98-9

Catumaxumab is a trifunctional monoclonal antibody developed for use in cancer treatment. It has affinity for T-cells, accessory immune cells, and cancer cells. Catumaxumab was initially authorized for market by the European Medicines Agency in April 2009 for…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Low affinity immunoglobulin gamma Fc region receptor II-aLow affinity immunoglobulin gamma Fc region receptor III-ALow affinity immunoglobulin gamma Fc region receptor III-B +3
Waktu ParuhCatumaxomab has an …
Vol. Distribusi-
Klirens-
Genetik -
Cavosonstat DB14775
small molecule | CAS: 1371587-51-7

Cavosonstat is under investigation in clinical trial NCT02589236 (Study of Cavosonstat (N91115) in Patients With CF Homozygous for the F508del-CFTR Mutation).

Kategori:
Benzene Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cavrotolimod DB18216
small molecule | CAS: 2378664-12-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CB-010 DB17711
biotech

CB-010 is a CRISPR-edited allogeneic CAR-T cell therapy targeting CD19. It is being investigated for the treatment of follicular lymphoma.[L46158]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CB-103 DB15279
small molecule | CAS: 218457-67-1

CB-103 is under investigation in clinical trial NCT03422679 (Study of CB-103 in Adult Patients With Advanced or Metastatic Solid Tumours and Haematological Malignancies).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CB-1158 DB15286
small molecule | CAS: 2095732-06-0

CB-1158 is under investigation in clinical trial NCT03910530 (A Study of INCMGA00012, INCB001158, and the Combination in Japanese Participants With Advanced Solid Tumors).

Kategori:
Enzyme Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CB-5083 DB16874
small molecule | CAS: 1542705-92-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Transitional endoplasmic reticulum ATPase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CBP-501 DB17277
small molecule | CAS: 565434-85-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCell Cycle ProteinsDual-Specificity Phosphatases +11
Target Protein:
MAP/microtubule affinity-regulating kinase 3MAP kinase-activated protein kinase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CC-115 DB12740
small molecule | CAS: 1228013-15-7

CC-115 has been used in trials studying the treatment of Prostate Cancer, Neoplasm Metastasis, Ewing's Osteosarcoma, Glioblastoma Multiforme, and Chronic Lymphocytic Leukemia, among others.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CC-401 DB12432
small molecule | CAS: 395104-30-0

CC-401 has been used in trials studying the treatment of Myeloid Leukemia.

Kategori:
JNK Mitogen-Activated Protein Kinases, antagonists & inhibitorsPyrazoles
Target Protein:
Mitogen-activated protein kinase 8Mitogen-activated protein kinase 9Mitogen-activated protein kinase 10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CC-90001 DB18445
small molecule | CAS: 1403859-14-2

Deskripsi belum tersedia.

Kategori:
AminesCyclohexanesCycloparaffins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CCR5 mAb DB05906
biotech

CCR5 mAb is a fully human monoclonal antibody that specifically recognizes and binds the chemokine receptor CCR5, which is known to be a key facilitator of infection with human immunodeficiency virus (HIV-1). It was generated by HGS using the Abgenix XenoMous…

Target Protein:
C-C chemokine receptor type 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CCT-018159 DB07594
small molecule | CAS: 171009-07-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Heat shock protein HSP 90-alphaHeat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CCX-354 DB12963
small molecule | CAS: 1010073-75-2

CCX354-C has been used in trials studying the treatment of Rheumatoid Arthritis.

Target Protein:
C-C chemokine receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CCX915 DB05159
small molecule

CCX915 is developed by ChemoCentryx which targets the chemokine receptor CCR2 and is in phase 1 of clinical trial for the treatment of Multiple Sclerosis and Neurologic Disorders. The CCR2 receptor is thought to be of central importance to inflammatory diseas…

Target Protein:
C-C chemokine receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CD564 DB02741
small molecule

Deskripsi belum tersedia.

Target Protein:
Retinoic acid receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CDC-801 DB15640
small molecule | CAS: 192819-27-5

CDC-801 is under investigation in clinical trial NCT00006097 (Chemotherapy in Treating Patients With Chronic Lymphocytic Leukemia).

Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4B3',5'-cyclic-AMP phosphodiesterase 4D3',5'-cyclic-AMP phosphodiesterase 4A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CDD-0102 DB16945
small molecule | CAS: 146422-58-4

Deskripsi belum tersedia.

Kategori:
Muscarinic AgonistsOxazolesReceptor, Muscarinic M1, agonists
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CDP323 DB05092
small molecule

CDP323 is an antagonist of the _vascular cell adhesion molecule 1_ (VCAM-1) binding to alpha4-integrins (other adhesion molecules), a process thought to be implicated in the pathophysiology of Multiple Sclerosis (MS). It is considered a small-molecule prodrug…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +3
Target Protein:
Integrin alpha-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CDX-1135 DB17607
biotech

CDX-1135, formerly TP-10, is a soluble, recombinant human Complement Receptor Type 1 (sCR1) developed by Avant Immunotherapeutics (now Celldex). It was investigated in clinical trials for post-cardiopulmonary bypass syndrome and kidney damage.

Kategori:
Amino Acids, Peptides, and ProteinsMembrane ProteinsProteins +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CDX-301 DB19293
biotech

CDX-301 is under investigation in clinical trial NCT02129075 (A Vaccine (CDX-1401) With or Without a Biologic Drug (CDX-301) for the Treatment of Patients With Stage IIB-IV Melanoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CDX-6512 DB17841
biotech

CDX-6512 is a modified, gastrointestinal-stable bacterial leucine decarboxylase. Developed by Codexis, it is being investigated for the treatment of homocystinuria And Maple Syrup Urine Disease.[L46651, L46656]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CE-224535 DB12113
small molecule | CAS: 724424-43-5

CE-224535 has been used in trials studying the treatment of Osteoarthritis.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +4
Target Protein:
P2X purinoceptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CE-326597 DB12694
small molecule | CAS: 870615-40-0

CE-326,597 has been used in trials studying the treatment of Obesity.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Cholecystokinin receptor type A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CEB-01 DB18505
small molecule

CEB-01 is a biocompatible polymeric PLGA nanofiber membrane containing the active substance 7-ethyl-10-hydroxycamptothecin

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cebranopadol DB12830
small molecule | CAS: 863513-91-1

Cebranopadol has been used in trials studying the treatment of Pain, Neoplasms, and Chronic Pain.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Mu-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceclazepide DB17270
small molecule | CAS: 1801749-44-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cedar leaf oil DB15836
biotech | CAS: 8007-20-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cedazuridine Approved DB15694
small molecule | CAS: 1141397-80-9

Myelodysplastic syndromes (MDS) are a group of hematopoietic neoplasms that give rise to variable cytopenias progressing to secondary acute myeloid leukemia (sAML), which is invariably fatal if untreated.[A215082, A215092, A215097] Hypomethylating agents such…

Kategori:
Cytidine Deaminase, antagonists & inhibitorsNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Cytidine deaminase
Waktu ParuhCedazuridine has a …
Vol. DistribusiThe apparent volume…
KlirensCedazuridine has an…
Genetik -
Cediranib DB04849
small molecule | CAS: 288383-20-0

The novel indole-ether quinazoline Cediranib is a highly potent (IC<sub>50</sub> &lt; 1 nmol/L) ATP-competitive inhibitor of recombinant KDR tyrosine kinase in vitro. It is being developed clinically as a once-daily oral therapy for the treatment of cancer.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsEnzyme Inhibitors +4
Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh12 to 35 hours
Vol. Distribusi-
Klirens-
Genetik -
Cedirogant DB18951
small molecule | CAS: 2055496-11-0

Cedirogant is under investigation in clinical trial NCT05044234 (A Study to Assess Adverse Events and Disease Activity With Cedirogant (ABBV-157) in Adult Participants With Moderate to Severe Psoriasis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefaclor Approved DB00833
small molecule | CAS: 53994-73-3

Semisynthetic, broad-spectrum antibiotic derivative of cephalexin.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 1A
Waktu Paruh0.6-0.9 hour
Vol. Distribusi-
Klirens-
Genetik -
Cefadroxil Approved DB01140
small molecule | CAS: 50370-12-2

Long-acting, broad-spectrum, water-soluble, cephalexin derivative.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 1APenicillin-binding protein 1b +1
Waktu Paruh1.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Cefalonium DB11385
small molecule | CAS: 5575-21-3

Deskripsi belum tersedia.

Kategori:
Amidesbeta-LactamsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefaloridine DB09008
small molecule | CAS: 50-59-9

Cephaloridine or cefaloridine is a first generation semisynthetic cephalosporin. It is derived from cephalosporin C and is a zwitterion at physiological pH.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefalotin Approved DB00456
small molecule | CAS: 153-61-7

Cefalotin is a cephalosporin antibiotic.

Kategori:
Agents that reduce seizure thresholdAmidesAnti-Bacterial Agents +13
Target Protein:
D-alanyl-D-alanine carboxypeptidasePenicillin-binding protein 1APenicillin-binding protein 1b +5
Waktu Paruh30 minutes
Vol. Distribusi-
Klirens-
Genetik -
Cefamandole Approved DB01326
small molecule | CAS: 34444-01-4

Cefamandole is also known as cephamandole. It is a parenterally administered broad-spectrum cephalosporin antibiotic. It is generally formulated as a formate ester, [cefamandole nafate]. It is no longer marketed in the United States.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
Penicillin-binding protein 2
Waktu ParuhThe half-life after…
Vol. Distribusi-
Klirens-
Genetik -
Cefamandole nafate Approved DB14725
small molecule | CAS: 57268-80-1

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefapirin Approved DB01139
small molecule | CAS: 21593-23-7

Cefapirin (INN, also spelled cephapirin), commonly marketed under the trade name Cefadyl, is a first-generation cephalosporin antibiotic that is available in injectable formulations. Production for use in humans has been discontinued in the United States. Cef…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefatrizine DB13266
small molecule | CAS: 51627-14-6

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefazedone DB13778
small molecule | CAS: 56187-47-4

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefazolin Approved DB01327
small molecule | CAS: 25953-19-9

A semisynthetic cephalosporin analog with broad-spectrum antibiotic action due to inhibition of bacterial cell wall synthesis. It attains high serum levels and is excreted quickly via the urine.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 1BPenicillin-binding protein 1C +5
Waktu ParuhThe serum half-life…
Vol. Distribusi-
Klirens-
Genetik -
Cefcapene DB13461
small molecule | CAS: 135889-00-8

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefdinir Approved DB00535
small molecule | CAS: 91832-40-5

Cefdinir, also known as Omnicef, is a semi-synthetic, broad-spectrum antibiotic belonging to the third generation of the cephalosporin class. It has been proven to be effective for the treatment of common bacterial infections in the ear, sinus, throat, lungs,…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +14
Target Protein:
Penicillin-binding protein 2PBP3Myeloperoxidase +1
Waktu ParuhThe average plasma …
Vol. DistribusiThe average volume …
KlirensThe renal clearance…
Genetik -
Cefditoren Approved DB01066
small molecule | CAS: 104145-95-1

Cefditoren is an oral third-generation cephalosporin. It is commonly marketed under the trade name Spectracef by Cornerstone BioPharma.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 2BPenicillin-binding protein 1A
Waktu ParuhMean terminal elimi…
Vol. Distribusi* 9.3 ± 1.6 L
Klirens* renal cl=4-5 L/h …
Genetik -
Cefepime Approved DB01413
small molecule | CAS: 88040-23-7

Cefepime is a fourth-generation cephalosporin antibiotic developed in 1994. Cefepime is active against Gram-positive and Gram-negative bacteria, and has greater activity against both compared to third-generation antibiotics.[A2457,A249050] Cefepime is normall…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 1BPenicillin-binding protein 2 +4
Waktu ParuhHealthy adult male …
Vol. DistribusiThe average steady-…
KlirensCefepime has a tota…
Genetik -
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