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11778

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8554 (72.6%)
Target
6383 (54.2%)
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96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 72 / 236
Chlortetracycline Approved DB09093
small molecule | CAS: 57-62-5

Chlortetracycline is a _tetracycline_ antibiotic, and historically the first member of this class to be identified. It was discovered in 1945 by the scientist, Benjamin Minge Duggar, working at Lederle Laboratories under the supervision of Yellapragada Subbar…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAnti-Bacterial Agents +15
Target Protein:
16S ribosomal RNA30S ribosomal protein S330S ribosomal protein S8 +8
Waktu ParuhThe half-life of Ch…
Vol. DistribusiChlortetracycline h…
Klirens-
Genetik -
Chlorthalidone Approved DB00310
small molecule | CAS: 77-36-1

Chlorthalidone is a thiazide-like diuretic used for the treatment of hypertension and for management of edema caused by conditions such as heart failure or renal impairment. Chlorthalidone improves blood pressure and swelling by preventing water absorption fr…

Kategori:
AmidesAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +25
Target Protein:
Carbonic anhydrase 1Solute carrier family 12 member 1
Waktu Paruh40-50 hours[FDA Lab…
Vol. DistribusiChlorthalidone has …
Klirens-
Genetik -
biotech

This vaccine candidate, developed in China, uses SARS-CoV-2 protein subunits that are entirely engineered, created, and secreted by Chinese Hamster Ovary (CHO) cells[A219758]. The vaccine candidate is sponsored by Anhui Zhifei Longcom Biologic Pharmacy Co., L…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cholecalciferol Approved DB00169
small molecule | CAS: 67-97-0

Vitamin D, in general, is a secosteroid generated in the skin when 7-dehydrocholesterol located there interacts with ultraviolet irradiation - like that commonly found in sunlight [L5689]. Both the endogenous form of vitamin D (that results from 7-dehydrochol…

Kategori:
Alimentary Tract and MetabolismBone Density Conservation AgentsCalcium-Regulating Hormones and Agents +28
Target Protein:
Vitamin D3 receptor
Waktu ParuhAt this time, there…
Vol. DistribusiStudies have determ…
KlirensStudies have determ…
Genetik -
Cholecystokinin Approved DB08862
small molecule | CAS: 9011-97-6

Cholecystokinin ( also known as _CCK or CCK-PZ_) is a peptide hormone of the gastrointestinal system which is responsible for stimulating the digestion of fat and protein. Cholecystokinin, previously called _pancreozymin_, is synthesized and secreted by enter…

Kategori:
Amino Acids, Peptides, and ProteinsCholagogues and CholereticsCholecystokinin, agonists +12
Target Protein:
Cholecystokinin receptor type ARAF proto-oncogene serine/threonine-protein kinaseMitogen-activated protein kinase 3 +3
Waktu Paruh2.5 min [L1642]
Vol. Distribusi-
Klirens-
Genetik -
Cholesterol Approved DB04540
small molecule | CAS: 57-88-5

The principal sterol of all higher animals, distributed in body tissues, especially the brain and spinal cord, and in animal fats and oils.

Kategori:
BCRP/ABCG2 InducersCholestanesCholestenes +6
Target Protein:
Choline-phosphate cytidylyltransferase BNuclear receptor subfamily 1 group I member 3Vitamin D3 receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Choline Approved DB00122
small molecule | CAS: 62-49-7

A basic constituent of lecithin that is found in many plants and animal organs. It is important as a precursor of acetylcholine, as a methyl donor in various metabolic processes, and in lipid metabolism.

Kategori:
AlcoholsAminesAmino Alcohols +23
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Neuronal acetylcholine receptor subunit alpha-7Choline-phosphate cytidylyltransferase B +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 28319-77-9

A component of phosphatidylcholines (lecithins), in which the two hydroxy groups of glycerol are esterified with fatty acids. (From Stedman, 26th ed) It counteracts the effects of urea on enzymes and other macromolecules. [PubChem]

Kategori:
AlcoholsBiological ProductsCarbohydrates +14
Target Protein:
Muscarinic acetylcholine receptor M5Ganglioside GM2 activator
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Choline C 11 Approved DB09277
small molecule | CAS: 87591-54-6

Choline C 11 is a marker for cellular proliferation as its main molecule is a precursor for the biosynthesis of phospholipids which are essential components of all cell membranes.[A32041] It was developed by MCPRF and FDA first approved in September 2012.

Kategori:
Drugs that are Mainly Renally Excreted
Waktu ParuhThe isotope half-li…
Vol. Distribusi-
KlirensAfter intravenous i…
Genetik -
Choline C-11 Approved DB09563
small molecule | CAS: 94793-58-5

Choline C 11 Injection is a radioactive diagnostic agent for positron emission tomography (PET) imaging of pat ients with suspected prostate cancer recurrence and non-informative bone scintigraphy, computerized tomography (CT) or magnetic resonance imaging.

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu Paruh-
Vol. Distribusi11C-choline distrib…
KlirensThe rate of 11C- ch…
Genetik -
small molecule | CAS: 64425-90-7

Choline magnesium trisalicylate is a non-acetylated salicylate used widely as a nonsteroidal anti-inflammatory drug. Trisalicylate significantly reduces methotrexate renal clearance, displacing methotrexate from protein, increasing the fraction unbound by 28%…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +23
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chondroitin sulfate Approved DB09301
small molecule | CAS: 24967-93-9

Chondroitin sulfate is a glycosaminoglycan considered as a symptomatic slow-acting drug for osteoarthritis (SYSADOA).[A7906] The SYSADOA status suggested a pain relief and increased joint mobility after a relative long regular administration, as well as a lon…

Kategori:
Antiinflammatory and Antirheumatic ProductsAntiinflammatory and Antirheumatic Products, Non-SteroidsCarbohydrates +5
Target Protein:
Neurotrophic factor BDNF precursor formGlial cell line-derived neurotrophic factorVascular endothelial growth factor A, long form +1
Waktu ParuhThe approximate hal…
Vol. DistribusiAfter intramuscular…
Klirens-
Genetik -
biotech

Chondrus crispus is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Choriogonadotropin alfa Approved DB00097
biotech | CAS: 177073-44-8

Recombinant human chorionic gonadotropin with 2 subunits, alpha = 92 residues, beta = 145 residues, each with N-and O-linked carbohydrate moieties linked to ASN-52 and ASN-78 (on alpha subunit) and ASN-13, ASN-30, SER-121, SER-127, SER-132 and SER-138 (on bet…

Kategori:
Genito Urinary System and Sex HormonesGonadotropinsGonadotropins and Antigonadotropins +1
Target Protein:
Follicle-stimulating hormone receptorLutropin-choriogonadotropic hormone receptor
Waktu ParuhThe mean terminal h…
Vol. Distribusi* 5.9 ± 1.0 L
Klirens* 0.29 +/- 0.04 L/h…
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chromic chloride Approved DB09129
small molecule | CAS: 10025-73-7

Chromic chloride, for injection, is a sterile, nonpyrogenic solution intended for use as an additive to solutions for Total Parenteral Nutrition (TPN).

Kategori:
AnionsAntioxidantsBiological Factors +8
Target Protein:
Insulin receptor
Waktu Paruh31- 41 hours
Vol. DistribusiChromium is stored …
Klirens-
Genetik -
Chromic citrate DB14526
small molecule | CAS: 57072-40-9

Deskripsi belum tersedia.

Kategori:
Drugs that are Mainly Renally Excreted
Target Protein:
Cytochrome b5
Waktu ParuhThe elimination hal…
Vol. DistribusiAbsorbed chromium i…
KlirensExcretion of chromi…
Genetik -
Chromic nitrate Approved DB14527
small molecule | CAS: 13548-38-4

Deskripsi belum tersedia.

Kategori:
AnionsDrugs that are Mainly Renally ExcretedElectrolytes +2
Target Protein:
Cytochrome b5
Waktu ParuhThe elimination hal…
Vol. DistribusiAbsorbed chromium i…
KlirensExcretion of chromi…
Genetik -
Chromium Approved DB11136
small molecule | CAS: 7440-47-3

Chromium is a transition element with the chemical symbol Cr and atomic number 24 that belongs to Group 6 of the periodic table. It is used in various chemical, industrial and manufacturing applications such as wood preservation and metallurgy. The uses of ch…

Kategori:
Cell-mediated ImmunityDiet, Food, and NutritionDrugs that are Mainly Renally Excreted +11
Target Protein:
Cytochrome b5
Waktu ParuhThe elimination hal…
Vol. DistribusiAbsorbed chromium i…
KlirensExcretion of chromi…
Genetik -
Chromium Cr-51 Approved DB11140
small molecule | CAS: 14392-02-0

Chromium Cr-51 is an isotope of chromium that has been used as a radioactive label for decades. It is used as a diagnostic radiopharmaceutical agent in nephrology to determine glomerular filtration rate,[A249765,A249770] and in hematology to determine red blo…

Kategori:
Chromium IsotopesElementsIsotopes +4
Waktu ParuhChromium Cr-51 has …
Vol. Distribusi-
Klirens-
Genetik -
Chromium picolinate Approved DB11255
small molecule | CAS: 14639-25-9

Chromium picolinate has a chemical formula CrPic3 and reddish-pink color. It is a coordination complex consisting of chromium(III) and picolinic acid. Chromium picolinate is used as a nutritional supplement for optimal insulin function in patients with Type 2…

Kategori:
Compounds used in a research, industrial, or household settingIron Chelating AgentsPyridines +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Chrysin DB15581
small molecule | CAS: 480-40-0

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Aldo-keto reductase family 1 member B1Cytochrome P450 1B1Aromatase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chrysoeriol DB17283
small molecule | CAS: 491-71-4

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +2
Target Protein:
Xanthine dehydrogenase/oxidaseCytochrome P450 1B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The ChulaCov19 vaccine is mRNA-based and was developed in Thailand’s Chulalongkorn University in collaboration with the University of Pennsylvania in the US[L30673, L30678]. Pre-clinical studies in mice and monkeys showed evidence that the vaccine facilitates…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Chymopapain Approved DB06752
biotech | CAS: 9001-09-6

Chymopapain was first isolated in 1941 from the crude latex derived from the fruit of Carica papaya by squeezing the green papaya while on the plant prior to harvest.[L2482]It is an extracellular plant cysteine proteinase similar to papain in specificity.[A32…

Kategori:
Cysteine EndopeptidasesCysteine ProteasesEndopeptidases +5
Target Protein:
Bone marrow proteoglycan
Waktu ParuhFollowing intra-dis…
Vol. Distribusi-
Klirens-
Genetik -
Chymostatin DB01683
small molecule | CAS: 9076-44-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsChymotrypsin, antagonists & inhibitorsEnzyme Inhibitors +3
Target Protein:
ChymasePeptide amidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chymotrypsin Approved DB09375
small molecule | CAS: 9004-07-3

Chymotrypsin (EC 3.4.21.1) is a digestive enzyme that promotes proteolysis, or the breakdown of proteins and polypeptides. It is a serine protease synthesized in the pancreas and is a vital component in the pancreatic juice. Like most proteolytic enzymes, chy…

Kategori:
Blood and Blood Forming OrgansEndopeptidasesEnzymes +8
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
CI-1040 DB12429
small molecule | CAS: 212631-79-3

CI-1040 has been used in trials studying the treatment of Lung Cancer, Breast Cancer, Breast Neoplasms, Pancreatic Cancer, and Colorectal Cancer, among others.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Target Protein:
Mitogen-activated protein kinase kinase kinase 1Mitogen-activated protein kinase kinase kinase 2Serine/threonine-protein kinase Sgk1 +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cibenzoline DB13358
small molecule | CAS: 53267-01-9

Deskripsi belum tersedia.

Kategori:
Antiarrhythmic agentsAntiarrhythmics, Class IAntiarrhythmics, Class Ia +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cibisatamab DB17349
biotech | CAS: 2101242-53-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ciclesonide Approved DB01410
small molecule | CAS: 126544-47-6

Ciclesonide is a glucocorticoid used to treat obstructive airway diseases. It is marketed under the brand name Alvesco.

Kategori:
Adrenal Cortex HormonesAdrenalsAgents to Treat Airway Disease +18
Target Protein:
Corticosteroid-binding globulinGlucocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens* 152 L/hr [Followi…
Genetik -
Cicletanine DB12766
small molecule | CAS: 89943-82-8

Cicletanine is under investigation for the treatment of Diabetes, Hypokalemia, Hyponatremia, and Arterial Hypertension.

Kategori:
Antiarrhythmic agentsAntihypertensive AgentsCardiovascular Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ciclonicate DB13709
small molecule | CAS: 53449-58-4

Deskripsi belum tersedia.

Kategori:
Nicotinic Acid and DerivativesPeripheral VasodilatorsPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 29546-59-6

Deskripsi belum tersedia.

Kategori:
Dioxoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cidofovir Approved DB00369
small molecule | CAS: 113852-37-2

Cidofovir is an injectable antiviral medication employed in the treatment of cytomegalovirus (CMV) retinitis in patients diagnosed with AIDS. It suppresses CMV replication through selective inhibition of viral DNA synthesis.[FDA label] It was manufactured by …

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +16
Target Protein:
DNA polymerase catalytic subunitDNA polymerase catalytic subunit
Waktu Paruh2.4 to 3.2 hours
Vol. Distribusi* 537 ± 126 mL/kg […
Klirens* 179 +/- 23.1 mL/m…
Genetik -
Cidoxepin DB14750
small molecule | CAS: 3607-18-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ciforadenant DB16125
small molecule | CAS: 1202402-40-1

Ciforadenant is under investigation in clinical trial NCT02253745 (Safety, Tolerability, PK & Efficacy of V81444 in Volunteers With Attention Deficit/ Hyperactivity Disorder (ADHD)).

Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CIGB 300 DB16464
biotech | CAS: 1072877-99-6

CIGB-300, is under investigation in clinical trials for its potential to treat various conditions, including NCT01639638 (recurrent and nonrecurrent condyloma) and NCT01639625 (squamous cell carcinoma and adenocarcinoma of the cervix)

Kategori:
Amino Acids, Peptides, and ProteinsExperimental Unapproved Treatments for COVID-19Peptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ciglitazone DB09201
small molecule | CAS: 74772-77-3

Developed by Takeda Pharmaceuticals in the early 1980s, it is considered the prototypical compound for the thiazolidinedione class. Ciglitazone was never used as a medication, but it sparked interest in the effects of thiazolidinediones. Several analogues …

Kategori:
Blood Glucose Lowering AgentsCytochrome P-450 CYP2C8 InhibitorsCytochrome P-450 CYP2C8 Inhibitors (strength unknown) +8
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cilansetron DB04885
small molecule | CAS: 120635-74-7

Cilansetron is a 5HT-3 antagonist made by Solvay Pharmaceuticals that is currently under trial phase in the EU and US.

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsCentral Nervous System Depressants +5
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Cilastatin Approved DB01597
small molecule | CAS: 82009-34-5

Cilastatin is an inhibitor of renal dehydropeptidase, an enzyme responsible for both the metabolism of thienamycin beta-lactam antibiotics as well as conversion of leukotriene D4 to leukotriene E4. Since the antibiotic, [imipenem], is one such antibiotic that…

Kategori:
CycloparaffinsCyclopropanesDipeptidase Inhibitors +5
Target Protein:
Dipeptidase 1
Waktu ParuhThe half-life of ci…
Vol. DistribusiCilastatin has a vo…
KlirensCilastatin has a to…
Genetik -
Cilazapril Approved DB01340
small molecule | CAS: 88768-40-5

Cilazapril is an ACE inhibtor class drug used in the treatment of hypertension and heart failure. It belongs to the angiotensin-converting enzyme inhibitors (ACE inhibitors) class of drugs. It is a prodrug that is hydrolyzed after absorption to its main meta…

Kategori:
ACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin SystemAgents causing angioedema +10
Target Protein:
Angiotensin-converting enzyme
Waktu ParuhHalf-lives for the …
Vol. Distribusi-
KlirensTotal clearance is …
Genetik -
Cilgavimab Approved DB16393
biotech | CAS: 2420563-99-9

SARS-CoV-2, the causative agent of COVID-19, enters cells via the interaction between the trimeric spike (S) glycoprotein and host cell angiotensin-converting enzyme 2 (ACE2). Blocking the interaction between the receptor-binding domain (RBD) of the S1 subuni…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Spike glycoprotein
Waktu ParuhCilgavimab has a ha…
Vol. DistribusiCilgavimab has an a…
KlirensCilgavimab has an a…
Genetik -
biotech | CAS: 133423-39-9

NT-501 is an intraocular implant that contains human cells that have been genetically modified to secrete ciliary neurotrophic factor (CNTF).[L46762] It is under investigation for the treatment of retinitis pigmentosa and age-related macular degeneration.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cilnidipine DB09232
small molecule | CAS: 132203-70-4

Cilnidipine is a dihydropyridine calcium antagonist. It was jointly developed by Fuji Viscera Pharmaceutical Company, Japan and Ajinomoto, Japan and approved in 1995. Compared with other calcium antagonists, cilnidipine can act on the N-type calcium channel t…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +12
Target Protein:
Voltage-dependent N-type calcium channel subunit alpha-1BVoltage-dependent L-type calcium channel
Waktu ParuhThe half-life of th…
Vol. DistribusiDrugs on the group …
Klirens-
Genetik -
Cilofexor DB15168
small molecule | CAS: 1418274-28-8

Cilofexor is under investigation in clinical trial NCT02943447 (Safety, Tolerability, and Efficacy of Cilofexor in Adults With Primary Biliary Cholangitis Without Cirrhosis).

Kategori:
AzetinesPyridines
Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cilomilast DB03849
small molecule | CAS: 153259-65-5

Cilomilast (Ariflo, SB-207,499) is a drug which was developed for the treatment of respiratory disorders such as asthma and Chronic Obstructive Pulmonary Disease (COPD). It is orally active and acts as a selective Phosphodiesterase-4 inhibitor. Following four…

Kategori:
Acids, CarbocyclicCyclohexanesCycloparaffins +3
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4D3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cilostazol Approved DB01166
small molecule | CAS: 73963-72-1

Cilostazol is a quinolinone derivative and antiplatelet agent with vasodilating properties that has been used in the symptomatic treatment of intermittent claudication in patients with peripheral ischaemia. It is marketed under the brand name Pletal by Otsuka…

Kategori:
Agents producing tachycardiaAnti-Asthmatic AgentsAntiplatelet agents +31
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A
Waktu Paruh11-13 hours.
Vol. Distribusi-
Klirens-
Genetik -
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