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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 72 / 321
ARG098 DB06338
biotech

ARG098 (anti-Fas IgM monoclonal antibody) was studied in a Phase I clinical trial in 2007 involving patients with rheumatoid arthritis.

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ARG201 DB06621
biotech

ARG201, a bovine-derived Type I collagen, aims to induce immune tolerance in patients with Diffuse Systemic Scleroderma (dcSSc). This drug was investigated in the completed clinical trial NCT0000567 (Multicenter Phase II Trial of Oral Type I Bovine Collagen i…

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Argadin DB04350
small molecule | CAS: 289665-92-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Chitotriosidase-1Endochitinase B1
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Argan oil DB14310
biotech

Argan oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsComplex MixturesLipids +3
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Argatroban Approved DB00278
small molecule | CAS: 74863-84-6

Argatroban is a direct, selective thrombin inhibitor. The American College of Cardiologists (ACC) recommend using bivalirudin or argatroban in patients who have had, or at risk for, heparin induced thrombocytopenia (HIT) and are undergoing percutaneous corona…

Kategori:
AmidesAmino AcidsAmino Acids, Basic +22
Target Protein:
Prothrombin
Waktu Paruh39 and 51 minutes
Vol. Distribusi* 174 mL/kg * 12.1…
Klirens* 5.1 L/kg/hr [infu…
Genetik -
Argifin DB03632
small molecule | CAS: 243975-37-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsChitinases, antagonists & inhibitorsPeptides
Target Protein:
Chitotriosidase-1Endochitinase B1
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Arginine DB00125
small molecule | CAS: 74-79-3

An essential amino acid that is physiologically active in the L-form.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Basic +14
Target Protein:
Cationic amino acid transporter 3Antizyme inhibitor 2Argininosuccinate lyase +6
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Genetik -
small molecule | CAS: 7675-83-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Basic +4
Waktu Paruh-
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Genetik -
small molecule | CAS: 4320-30-3

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBile and Liver Therapy +4
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Arginine PCA DB16025
small molecule | CAS: 56265-06-6

Deskripsi belum tersedia.

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Arginineamide DB02299
small molecule

Deskripsi belum tersedia.

Target Protein:
Potassium voltage-gated channel subfamily A member 4
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ARGX-119 DB18133
biotech

ARGX-119 is a monoclonal antibody that targets and activates muscle-specific kinase (MuSK).

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Arhalofenate DB11811
small molecule | CAS: 24136-23-0

Arhalofenate has been investigated for the treatment of Gout and Hyperuricemia.

Kategori:
AcetatesAcids, AcyclicAcids, Carbocyclic +1
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
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Arimoclomol Approved DB05025
small molecule | CAS: 289893-25-0

Arimoclomol is a hydroxylamine derivative [A264414] and a heat-shock protein-70 (HSP70) co-inducer.[L51384] Arimoclomol was approved by the FDA on September 20, 2024, making it the first treatment for Niemann-Pick disease, type C (NPC).[L51389] It is also bei…

Kategori:
AminesMATE 1 SubstratesMATE 2 Substrates +3
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Aripiprazole Approved DB01238
small molecule | CAS: 129722-12-9

Aripiprazole is an atypical antipsychotic orally indicated for the treatment of schizophrenia, bipolar I, major depressive disorder, irritability associated with autism, and Tourette's.[L45859] It is also indicated as an injection for agitation associated wit…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +48
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 1A +35
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe steady-state vo…
KlirensThe clearance of ar…
Genetik -
Aripiprazole lauroxil Approved DB14185
small molecule | CAS: 1259305-29-7

Aripiprazole lauroxil is a long-acting injectable atypical antipsychotic drug used in the treatment of schizophrenia in adult patients. It is a prodrug of [aripiprazole], which acts as a partial agonist at the D2 and 5-HT1A receptors, and as an antagonist at …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +29
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2A +22
Waktu ParuhThe mean aripiprazo…
Vol. DistribusiBased on population…
KlirensIn rats, the cleara…
Genetik -
Arketamine DB19150
small molecule | CAS: 33643-49-1

Arketamine is under investigation in clinical trial NCT05414422 (A Randomized, Placebo-controlled, Double-blind Study to Assess Safety and Efficacy of PCN-101 in TRD).

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ARM-210 DB16944
small molecule | CAS: 1467605-57-7

Deskripsi belum tersedia.

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Armodafinil Approved DB06413
small molecule | CAS: 112111-43-0

Armodafinil is the enantiopure of the wakefulness-promoting agent modafinil (Provigil), and is indicated to improve wakefulness in adult patients with excessive sleepiness associated with obstructive sleep apnea (OSA), narcolepsy, or shift work disorder (SWD)…

Kategori:
Benzene DerivativesBenzhydryl CompoundsCentral Nervous System Agents +21
Target Protein:
Alpha-1D adrenergic receptorSodium-dependent dopamine transporter
Waktu ParuhTerminal half-life …
Vol. DistribusiApparent volume of …
KlirensThe oral clearance …
Genetik -
Arnica montana DB14297
biotech | CAS: 8057-65-6

Arnica montana is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAsteraceaeBiological Products +8
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Arnica montana flower Approved DB14343
biotech

Arnica montana flower is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAsteraceaeBiological Products +8
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ARO-ANG3 DB17626
biotech

ARO-ANG3 is a subcutaneously administered RNA interference (RNAi)-based investigational medicine targeting angiopoietin-like protein 3 (ANGPTL3). It was granted an orphan drug designation for the treatment of homozygous familial hypercholesterolemia (HoFH).[L…

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ARO-APOC3 DB17625
biotech

ARO-APOC3 is an investigational RNAi therapeutic targeting apolipoprotein C-III (APOC3). It received an Orphan Drug designation by the FDA for the treatment of familial chylomicronemia syndrome.[L45864]

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Aroplatin DB17319
small molecule | CAS: 114488-24-3

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsOrganometallic Compounds
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Arotinoid acid DB02877
small molecule | CAS: 71441-28-6

Arotinoid acid is a retinoic acid analog which acts as a selective RAR agonist.

Kategori:
Acids, CarbocyclicAlkenesBenzene Derivatives +9
Target Protein:
Retinoic acid receptor beta
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Arotinolol DB09204
small molecule | CAS: 68377-92-4

Arotinolol is an alpha- and beta-receptor blocker developed in Japan. It is a thiopropanolamine with a tertiary butyl moiety. It has been studied for its potential to be an antihypertensive therapy.[T87] Artinolol is being developed by Sumitomo Pharmaceutical…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +11
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorAlpha-1 adrenergic receptors
Waktu ParuhThe reported half-l…
Vol. DistribusiThe stereospecifici…
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ARRY-502 DB16053
small molecule | CAS: 1202891-16-4

ARRY-502 is under investigation in clinical trial NCT01561690 (A Study of ARRY-502 in Patients With Persistent Asthma).

Target Protein:
Prostaglandin D2 receptor 2
Waktu Paruh-
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Arsanilic acid DB03006
small molecule | CAS: 98-50-0

An arsenical which has been used as a feed additive for enteric conditions in pigs and poultry. It causes blindness and is ototoxic and nephrotoxic in animals. [PubChem]

Kategori:
Adjuvants, ImmunologicAlkenesAnti-Infective Agents +10
Target Protein:
Lysozyme C
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Arsenic trioxide Approved DB01169
small molecule | CAS: 1327-53-3

Arsenic trioxide is a chemotherapeutic agent of idiopathic function used to treat leukemia that is unresponsive to first line agents. It is suspected that arsenic trisulfide induces cancer cells to undergo apoptosis. In general, arsenic is known to be a natur…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsArsenicals +16
Target Protein:
Inhibitor of nuclear factor kappa-B kinase subunit betaThioredoxin reductase 1, cytoplasmicTranscription factor Jun +7
Waktu Paruh-
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Arsenite ion DB18509
small molecule | CAS: 15502-74-6

Deskripsi belum tersedia.

Kategori:
AnionsArsenicalsElectrolytes +5
Waktu Paruh-
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Arsenous acid DB04456
small molecule | CAS: 13464-58-9

Deskripsi belum tersedia.

Kategori:
AnionsArsenicalsElectrolytes +1
Target Protein:
Arsenate reductaseArsenical pump-driving ATPase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Arsthinol DB08928
small molecule | CAS: 119-96-0

Arsthinol (INN) is an antiprotozoal agent that was first synthesized by Ernst A.H. Friedheim in 1949 via the complexing of acetarsol with 2,3-dimercaptopropanol. It has since been demonstrated that the agent possesses activity against amoebas and yaws. Consid…

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsArsenicals
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ART5803 DB18379
biotech

ART5803 is a humanized one-armed monoclonal antibody with a high affinity for the NMDA receptor.

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Artefenomel DB11809
small molecule | CAS: 1029939-86-3

Artefenomel has been investigated for the treatment of Malaria.

Kategori:
AnionsAnti-Infective AgentsAntimalarials +10
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Artemether Approved DB06697
small molecule | CAS: 71963-77-4

Artemether is an antimalarial agent used to treat acute uncomplicated malaria. It is administered in combination with lumefantrine for improved efficacy. This combination therapy exerts its effects against the erythrocytic stages of <i>Plasmodium spp.</i> and…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +25
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu ParuhArtemether, 1.6 +/-…
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Artemin DB15438
biotech | CAS: 309758-71-2

Artemin is under investigation in clinical trial NCT01842126 (Phase 1 Subcutaneous Single and Multiple Ascending Dose Study of BG00010 (Neublastin)).

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Artemisia vulgaris root Approved DB14170
biotech

Artemisia vulgaris root allergenic extract is used in allergenic testing.

Kategori:
Non-Standardized Food Allergenic Extract
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Artemisinin DB13132
small molecule | CAS: 63968-64-9

Artemisinin has been used in trials studying the treatment of Schizophrenia, Malaria, Falciparum, and Plasmodium Falciparum.

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Products, Insecticides and Repellents +13
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
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Artemisone DB16097
small molecule | CAS: 255730-18-8

Artemisone is under investigation in clinical trial NCT00936767 (Artemisone for the Treatment of Uncomplicated Falciparum Malaria in Western Cambodia).

Kategori:
Free RadicalsPeroxidesReactive Oxygen Species +2
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Artemotil Approved DB13851
small molecule | CAS: 75887-54-6

Artemotil, also known as ?-arteether, is a semi-synthetic derivative of artemisinin and a fast acting blood schizonticide specifically indicated for the treatment of chloroquine-resistant _Plasmodium falciparum_ malaria and cerebral malaria cases.

Kategori:
AmebicidesAnti-Infective AgentsAntimalarials +11
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Artenimol Approved DB11638
small molecule | CAS: 71939-50-9

Artenimol is an artemisinin derivative and antimalarial agent used in the treatment of uncomplicated *Plasmodium falciparum* infections [FDA Label]. It was first authorized for market by the European Medicines Agency in October 2011 in combination with [DB139…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +16
Target Protein:
Actin, cytoplasmic 2Alpha-aminoadipic semialdehyde dehydrogenaseAnnexin A2 +188
Waktu ParuhArtenimol was repor…
Vol. DistribusiArtenimol was obser…
KlirensArtenimol was obser…
Genetik -
Arterolane DB19027
small molecule | CAS: 664338-39-0

Arterolane is under investigation in clinical trial NCT03452475 (Comparison of Arterolane-piperaquine Versus Arterolane-piperaquine+mefloquine Versus Artemether-lumefantrine in Kenyan Children).

Kategori:
AnionsAntimalarialsAntiparasitic Products, Insecticides and Repellents +7
Waktu Paruh-
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Artesunate Approved DB09274
small molecule | CAS: 88495-63-0

Artesunate is indicated for the initial treatment of severe malaria.[L14099] The World Health Organization recommends artesunate as first line treatment for severe malaria.[L890] Artesunate was developed out of a need for a more hydrophilic derivative of [art…

Kategori:
Acids, AcyclicAnionsAnthelmintics +28
Target Protein:
Malaria protein EXP-1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ar…
Genetik -
Articaine Approved DB09009
small molecule | CAS: 23964-58-1

Articaine is a dental local anesthetic. Articaine is widely used around the world and is the most popular local anesthetic in many European countries.

Kategori:
AmidesAnestheticsAnesthetics, Local +11
Target Protein:
Voltage-gated sodium channel alpha subunit
Waktu Paruh-
Vol. Distribusi-
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Arundic acid DB05343
small molecule | CAS: 185517-21-9

Arundic acid has been investigated for the treatment of Amyotrophic Lateral Sclerosis (ALS).

Kategori:
Acids, AcyclicFatty AcidsLipids
Target Protein:
Beta-3 adrenergic receptorProtein S100-B
Waktu Paruh-
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Arverapamil DB06669
small molecule | CAS: 123932-43-4

Deskripsi belum tersedia.

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ARX201 DB05082
small molecule

ARX201 (PEG-ahGH) is a recombinant form of human growth hormone that has been modified using Ambrx’s patented ReCODE™ technology to achieve precise spatial positioning of the site of polyethylene glycol (PEG) attachment to human growth hormone, by biosyntheti…

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Arylacenamide DB05792
small molecule | CAS: 132173-07-0

Arylacenamide (SR31747) is a peripheral [sigma] ligand that binds four proteins in human cells, i.e. SRBP-1, [sigma]-2, HSI and its relative SRBP-2. It is a dual agent with both immunomodulatory and antiproliferative activities.

Kategori:
CycloparaffinsEnzyme InhibitorsImmunologic Factors +1
Target Protein:
3-beta-hydroxysteroid-Delta(8),Delta(7)-isomeraseHCG20471, isoform CRA_c
Waktu Paruh-
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Arzoxifene Approved DB06249
small molecule | CAS: 182133-25-1

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
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Genetik -
AS-8112 DB09207
small molecule

AS-8112 is a synthetic compound that acts as a selective antagonist at the dopamine receptor subtypes D2 and D3, and the serotonin receptor 5-HT3. It has been shown to exert potent antiemetic effects in animal studies and has been investigated for potential m…

Kategori:
Dopamine AgentsDopamine AntagonistsDopamine D2 Receptor Antagonists +1
Target Protein:
D(2) dopamine receptorD(3) dopamine receptor5HT3 serotonin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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