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14494

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9687 (66.8%)
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7525 (51.9%)
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14494 (100.0%)

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Halaman 71 / 290
Brefeldin A DB07348
small molecule | CAS: 20350-15-6

A metabolite from Penicillium brefeldianum that exhibits a wide range of antibiotic activity.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCytochrome P-450 CYP3A Inhibitors +9
Target Protein:
Cytohesin-2ADP-ribosylation factor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bremelanotide Approved DB11653
biotech | CAS: 189691-06-3

Bremelanotide is a 7 amino acid peptide used to treat hypoactive sexual desire disorder in premenopausal women.[L9635] Bremelanotide does not interact with alcohol.[A179686] The mechanism by which bremelanotide's action on receptors translates to a clinical e…

Kategori:
Amino Acids, Peptides, and ProteinsGenito Urinary System and Sex HormonesHormones +16
Target Protein:
Melanocyte-stimulating hormone receptorMelanocortin receptor 4Melanocortin receptor 3 +2
Waktu ParuhThe half life of br…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
Bremzalerbart DB19417
biotech | CAS: 2456307-07-4

Bremzalerbart is under investigation in clinical trial NCT06602739 (A Study to Demonstrate the Effect of REGN5713-5715 on Reducing Ocular Allergy Signs and Symptoms in Adult Participants With Birch Pollen Allergy).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
BREN-02 DB18264
biotech

BREN-02 is a recombinant human homeoprotein Engrailed 1 (rhEN1).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brenetafusp DB19441
biotech | CAS: 2736407-54-6

Brenetafusp is under investigation in clinical trial NCT04262466 (Safety and Efficacy of IMC-F106C as a Single Agent and in Combination With Checkpoint Inhibitors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brensocatib DB15638
small molecule | CAS: 1802148-05-5

Brensocatib is under investigation in clinical trial NCT03218917 (Assessment of INS1007 in Subjects With Non-cystic Fibrosis Bronchiectasis).

Kategori:
AzepinesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brentuximab vedotin Approved DB08870
biotech | CAS: 914088-09-8

Brentuximab vedotin, also known as Adcetris®, is an antibody-drug conjugate that combines an anti-CD30 antibody with the drug monomethyl auristatin E (MMAE). It is an anti-neoplastic agent used in the treatment of Hodgkin's lymphoma and systemic anaplastic la…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +35
Target Protein:
Tumor necrosis factor receptor superfamily member 8
Waktu ParuhThe terminal half-l…
Vol. DistribusiMMAE is unlikely to…
KlirensThe liver is the pr…
Genetik -
Bretylium Approved DB01158
small molecule | CAS: 59-41-6

Bretylium blocks the release of noradrenaline from the peripheral sympathetic nervous system, and is used in emergency medicine, cardiology, and other specialties for the acute management of ventricular tachycardia and ventricular fibrillation. The primary mo…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAmines +13
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1Beta-1 adrenergic receptor
Waktu ParuhThe terminal half-l…
Vol. Distribusi-
Klirens-
Genetik -
Brevenal DB17865
small molecule | CAS: 776331-34-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Brexanolone Approved DB11859
small molecule | CAS: 516-54-1

As of March 2019, brexanolone - developed and made available commercially by Sage Therapeutics Inc. as the brand name product Zulresso - is the first drug to have ever been approved by the US FDA specifically for the treatment of postpartum depression (PPD) i…

Kategori:
AnestheticsAnticonvulsantsAntidepressive Agents +28
Target Protein:
Gamma-aminobutyric acid receptor subunit deltaGamma-aminobutyric acid receptor subunit gamma-3GABA(A) Receptor +3
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe volume of distr…
KlirensThe total plasma cl…
Genetik -
Brexpiprazole Approved DB09128
small molecule | CAS: 913611-97-9

Brexpiprazole is an atypical antipsychotic and a novel D2 dopamine and serotonin 1A partial agonist called serotonin-dopamine activity modulator (SDAM). It has a high affinity for serotonin, dopamine and alpha (?)-adrenergic receptors.[L46417] Although it is …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +30
Target Protein:
5-hydroxytryptamine receptor 1AD(2) dopamine receptorD(3) dopamine receptor +9
Waktu ParuhAfter multiple once…
Vol. DistribusiThe volume of distr…
KlirensApparent oral clear…
Genetik -
Brexucabtagene autoleucel Approved DB15699
biotech

Mantle cell lymphoma is a heterogeneous sub-category of non-Hodgkin's lymphoma that can be classified as either an aggressive nodal or an indolent leukemic non-nodal variant. Despite the introduction of Bruton's tyrosine kinase (BTK) inhibitors such as [ibrut…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic Agents, Immunological +16
Target Protein:
B-lymphocyte antigen CD19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BRG01 DB18173
biotech

BRG01 is a genetically modified autologous CAR-T cell therapy under investigation for the treatment of nasopharyngeal carcinoma.[L48111]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Briakinumab DB05459
biotech | CAS: 339308-60-0

Briakinumab is a human anti-IL-12 monoclonal antibody being developed for the treatment of a number of T-cell driven autoimmune diseases. It targets and neutralize interleukin-12 and interleukin-23, two proteins associated with inflammation, such as pro-infla…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Interleukin-12 subunit betaInterleukin-23 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Briciclib DB12004
small molecule | CAS: 865783-99-9

Briciclib has been used in trials studying the treatment of Lymphoma, Neoplasms, Advanced Solid Tumor, and Acute Lymphocytic Leukemia.

Target Protein:
G1/S-specific cyclin-D1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brifentanil DB09172
small molecule | CAS: 101345-71-5

Brifentanil (also known as A-3331) is an analog of fentanyl, a potent opioid. This drug is classified as an opioid analgesic and was developed in the early 1990s. The effects of brifentanil are very similar to those of alfentanil, with strong but short lastin…

Kategori:
Piperidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brigatinib Approved DB12267
small molecule | CAS: 1197953-54-0

Brigatinib, originally named AP26113, is a reversible dual inhibitor of anaplastic lymphoma kinase (ALK) and epidermal growth factor receptor (EGFR). It presents selectivity against the mutant forms of EGFR compared to the wild-type.[A31311] It also exhibits …

Kategori:
Anaplastic lymphoma kinase (ALK) inhibitorsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
ALK tyrosine kinase receptorEpidermal growth factor receptorTyrosine-protein kinase ABL1 +6
Waktu ParuhThe half-life of br…
Vol. DistribusiThe apparent volume…
KlirensAfter oral administ…
Genetik -
Brilacidin DB12997
small molecule | CAS: 1224095-98-0

Brilacidin is under investigation for the supportive care of Mucositis, Stomatitis, Mouth Diseases, and Head and Neck Neoplasms.

Kategori:
AmidinesAnti-Infective Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brilaroxazine DB09226
small molecule | CAS: 1239729-06-6

Brilaroxazine (RP5063) is an investigational atypical antipsychotic which is under development by Reviva Pharmaceuticals for the treatment of schizophrenia and schizoaffective disorder. Reviva Pharmaceuticals also intends to investigate RP5063 for the treatme…

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical]) +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brilliant blue G Approved DB15594
small molecule | CAS: 6104-58-1

Brilliant Blue G is used in an ophthalmic solution for staining the internal limiting membrane (ILM) of the eye during ophthalmic procedures.[A188841,A188844] This membrane is thin and translucent, making it difficult to identify during eye surgeries that req…

Kategori:
AminesAniline CompoundsCompounds used in a research, industrial, or household setting +3
Target Protein:
Internal limiting membrane (ILM)
Waktu Paruh-
Vol. DistribusiThis drug is admini…
Klirens-
Genetik -
Brilliant green cation Approved DB11279
small molecule | CAS: 18198-35-1

Brilliant green, or ethanaminium, is a derivative of triarylmethane dye that has been used as a dye to color silk and wool. Due to its inhibitory actions against Gram positive microorganisms, brilliant green can be found in antiseptic products such as solutio…

Kategori:
AminesAmmonium CompoundsAnti-Infective Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brimapitide DB15231
small molecule | CAS: 1445179-97-4

Brimapitide is under investigation in clinical trial NCT01570205 (Safety, Tolerability and PK of a Single iv Infusion of 10, 40, and 80 µg/kg XG-102 Administered to Healthy Volunteers).

Kategori:
Amino Acids, Peptides, and ProteinsNeuroprotective Agents
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Brimonidine Approved DB00484
small molecule | CAS: 59803-98-4

Brimonidine is an alpha-adrenergic agonist and 2-imidazoline derivative that was first introduced in 1996.[A178951] It is considered to be a third generation alpha-2 aadrenergic receptor agonist, since it displays preferential binding at alpha-2 adrenoceptors…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +14
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptorAlpha-2C adrenergic receptor
Waktu ParuhFollowing ocular ad…
Vol. DistribusiThe volume of distr…
KlirensThe apparent cleara…
Genetik -
Brincidofovir Approved DB12151
small molecule | CAS: 444805-28-1

Brincidofovir is an oral antiviral drug used in the treatment of human smallpox infections. It is a lipid conjugate pro-drug of the acyclic nucleotide analogue [cidofovir][L34404,A235725] - this lipid conjugate improves drug delivery to the target cells and s…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +27
Target Protein:
DNA polymerase nuDNA polymerase delta subunit 4DNA polymerase delta catalytic subunit +7
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Brinzolamide Approved DB01194
small molecule | CAS: 138890-62-7

Brinzolamide is a highly specific, non-competitive, reversible carbonic anhydrase II (CA-II) inhibitor indicated to reduce ocular pressure in patients with ocular hypertension or open-angle glaucoma.[L35310] Although the exact pathophysiology of glaucoma is s…

Kategori:
AmidesAntiglaucoma Preparations and MioticsCarbonic Anhydrase Inhibitors +17
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 1Carbonic anhydrase 4 +2
Waktu ParuhDue to its affinity…
Vol. Distribusi-
Klirens-
Genetik -
Briquilimab DB18136
biotech | CAS: 2574591-89-0

Briquilimab is a humanized aglycosylated IgG1 kappa monoclonal antibody targeting CD117 (cKit).

Waktu Paruh-
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Genetik -
Brivanib DB11958
small molecule | CAS: 649735-46-6

Brivanib is under investigation for the treatment of HepatoCellular Carcinoma. Brivanib has been investigated for the treatment of Solid Tumors, Hepato Cellular Carcinoma (HCC), and Metastatic Colorectal Cancer (MCRC).

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 649735-63-7

Brivanib alaninate has been investigated for the treatment of Colorectal Cancer.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
Fibroblast growth factor receptor 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brivaracetam Approved DB05541
small molecule | CAS: 357336-20-0

Brivaracetam is a racetam derivative of levetiracetam used in the treatment of partial-onset seizures. Brivaracetam binds SV2A with 20 times higher affinity than levetiracetam [A19184]. It is available under the brand name Briviact made by UCB. Briviact recei…

Kategori:
AnticonvulsantsCentral Nervous System AgentsCentral Nervous System Depressants +11
Target Protein:
Synaptic vesicle glycoprotein 2ASodium channel protein
Waktu Paruh7-8h [A19180].
Vol. Distribusi0.5L/kg [FDA Label].
KlirensCL/F of 0.7-1.07 mL…
Genetik -
Brivoligide DB16116
biotech | CAS: 1803075-42-4

Brivoligide is under investigation in clinical trial NCT04104919 (Study to Evaluate a Preop Dose of Brivoligide Injection for Pain After Mastectomy in Patients With High PCS Scores).

Waktu Paruh-
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Brivudine Approved DB03312
small molecule | CAS: 69304-47-8

Brivudine is used in the treatment of herpes zoster. Although not approved in the U.S. or Canada, it is approved in several European countries.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +9
Target Protein:
Thymidine kinase 2, mitochondrialThymidine kinase, cytosolicDNA polymerase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BRM-421 DB18364
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Broccoli Approved DB10511
biotech

Broccoli allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brodalumab Approved DB11776
biotech | CAS: 1174395-19-7

Brodalumab has been used in trials studying the treatment of Asthma, Psoriasis, Crohn's Disease, Psoriatic Arthritis, and Rheumatoid Arthritis. Brodalumab was FDA approved in February, 2017 as Siliq for the treatment of moderate-to-severe plaque psoriasis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Interleukin-17 receptor A
Waktu Paruh-
Vol. Distribusi4.62 L.
Klirens0.223 L/day.
Genetik -
small molecule

Brodimoprim-4,6-dicarboxylate is a solid. This compound belongs to the anisoles. These are organic compounds contaiing a methoxybenzene or a derivative thereof. This medication is known to target the protein dihydrofolate reductase.

Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brofaromine DB13876
small molecule | CAS: 63638-91-5

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsEnzyme Inhibitors +3
Target Protein:
Amine oxidase [flavin-containing] A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Brogidirsen DB18884
biotech | CAS: 2409088-11-3

Brogidirsen is under investigation in clinical trial NCT05996003 (NS-089/NCNP-02-201 in Boys With Duchenne Muscular Dystrophy (DMD)).

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Genetik -
Brolucizumab Approved DB14864
biotech | CAS: 1531589-13-5

Brolucizumab, also known as RTH258 or ESBA1008,[A187211] is a monoclonal antibody indicated to treat neovascular age related macular degeneration.[L9089] Brolucizumab was granted FDA approval in October 2019.[L9089]

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAntibodies +14
Target Protein:
Vascular endothelial growth factor A, long form
Waktu ParuhThe systemic half l…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Bromamphenicol DB07492
small molecule | CAS: 16803-75-1

Deskripsi belum tersedia.

Kategori:
AlcoholsBenzene DerivativesGlycols +3
Target Protein:
Dr hemagglutinin structural subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromazepam Approved DB01558
small molecule | CAS: 1812-30-2

One of the benzodiazepines that is used in the treatment of anxiety disorders. It is a Schedule IV drug in the U.S. and Canada and under the Convention on Psychotropic Substances. It is a intermediate-acting benzodiazepine.

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepine hypnotics and sedatives +22
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh10-20 hours
Vol. Distribusi1.56 L/kg
Klirens0.82 mL/min/kg.
Genetik -
Bromelains DB13281
biotech | CAS: 9001-00-7

Bromelain is a protease enzyme derived from the stems of pineapples that is composed of a mixture of different thiol endopeptidases and other components like phosphatase, glucosidase, peroxidase, cellulase, escharase, and several protease inhibitors [A27198].…

Kategori:
Cysteine EndopeptidasesCysteine ProteasesDermatologicals +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromfenac Approved DB00963
small molecule | CAS: 91714-94-2

Bromfenac is a nonsteroidal anti-inflammatory drug (NSAID) for ophthalmic use. Ophthalmic NSAIDs are becoming a cornerstone for the management of ocular pain and inflammation. Their well-characterized anti-inflammatory activity, analgesic property, and establ…

Kategori:
Agents causing hyperkalemiaAnalgesicsAnalgesics, Non-Narcotic +16
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromhexine Approved DB09019
small molecule | CAS: 3572-43-8

Bromhexine is mucolytic agent used for a variety of respiratory conditions associated with increased mucus secretion. It is derived from the Adhatoda vasica plant and aids in the clearance of excess mucus, improving breathing and reducing cough. It was introd…

Kategori:
AminesAniline CompoundsCough and Cold Preparations +5
Target Protein:
Transmembrane protease serine 2Angiotensin-converting enzyme 2
Waktu ParuhFollowing single or…
Vol. DistribusiAfter intravenous a…
KlirensThe clearance of br…
Genetik -
small molecule | CAS: 3679-64-9

Deskripsi belum tersedia.

Kategori:
Antifungals for Dermatological UseAntifungals for Topical UseDermatologicals
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromocriptine Approved DB01200
small molecule | CAS: 25614-03-3

Bromocriptine mesylate is a semisynthetic ergot alkaloid derivative with potent dopaminergic activity. It inhibits prolactin secretion and may be used to treat dysfunctions associated with hyperprolactinemia. Bromocriptine is also indicated for the management…

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-1 Receptor Antagonists +41
Target Protein:
D(2) dopamine receptorD(3) dopamine receptor5-hydroxytryptamine receptor 1D +15
Waktu Paruh2-8 hours
Vol. Distribusi-
Klirens-
Genetik -
Bromodiphenhydramine Approved DB01237
small molecule | CAS: 118-23-0

Bromodiphenhydramine is an ethanolamine antihistamine with antimicrobial property. Bromodiphenhydramine is used in the control of cutaneous allergies. Ethanolamine antihistamines produce marked sedation in most patients.

Kategori:
AminesAminoalkyl EthersAntihistamines for Systemic Use +5
Target Protein:
Histamine H1 receptor
Waktu Paruh1 to 4 hours
Vol. Distribusi-
Klirens-
Genetik -
Bromopride DB09018
small molecule | CAS: 4093-35-0

Bromopride is a dopamine antagonist used as an antiemetic. Its prokinetic properties are similar to those of metoclopramide. It is unavailable in America or the United Kingdom.

Kategori:
Acids, CarbocyclicAlimentary Tract and MetabolismAmides +22
Target Protein:
D(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
KlirensRenal, 10-14% as or…
Genetik -
Bromopyruvate DB17135
small molecule | CAS: 1113-59-3

Deskripsi belum tersedia.

Kategori:
Affinity LabelsCompounds used in a research, industrial, or household settingEnzyme Inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromothalonil Approved DB14199
small molecule | CAS: 35691-65-7

Bromothalonil, also known as Methyldibromo glutaronitrile (MDBGN), is a widely used preservative that can be found in many personal hygiene and industrial products. It is also a known allergen and dermatological irritant that has been banned in many EU countr…

Kategori:
AllergensAntigensBiological Factors +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bromotheophylline Approved DB14018
small molecule | CAS: 10381-75-6

Bromotheophylline is the active moiety of pamabrom, a mixture of 2-amino-2-methyl-propanol and bromotheophylline. From this mixture, bromotheophylline acts as a weak diuretic that has been used along with some analgesics to relieve the symptoms of premenstrua…

Kategori:
AlcoholsAlkaloidsAmines +11
Target Protein:
Adenosine receptor
Waktu ParuhThe apparent elimin…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
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