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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 71 / 236
CHF 4227 DB05882
small molecule

CHF 4227 is a new selective estrogen receptor modulator (SERM). The compound has a high receptor affinity and has shown promising efficacy in the prevention of bone loss in animal models of osteoporosis. Additionally, the compound has shown no uterotrophic ac…

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CHF-6001 DB12800
small molecule | CAS: 1239278-59-1

CHF6001 has been used in trials studying the treatment of Asthma and Chronic Obstructive Pulmonary Disease.

Kategori:
Acids, CarbocyclicAmidesAminobenzoates +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CHF-6333 DB17815
small molecule | CAS: 1613621-54-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CHGN111 DB06376
small molecule

CHGN111 is an inhibitor of the mitochondrial enzyme CLK-1 which is a demethoxyubiquinone hydroxylase. Numerous parameters of mitochondrial function are altered when the activity of CLK-1 is reduced, which results in a decrease of ROS at critical cellular site…

Target Protein:
Dual specificity protein kinase CLK1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chiauranib DB16124
small molecule | CAS: 1256349-48-0

Chiauranib is under investigation in clinical trial NCT03974243 (Chiauranib in Combination With Chidamide in Patients With Relapsed/refractory Non-hodgkin's Lymphoma).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chicory leaf DB14376
biotech

Chicory leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chiglitazar DB19023
small molecule | CAS: 743438-45-1

Chiglitazar is under investigation in clinical trial NCT06125587 (Chiglitazar/metformin in Non-obese Women With PCOS).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +3
Target Protein:
Peroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Chikungunya virus (CHIKV) is a member of the Alphavirus genus that was first identified in Tanzania in 1952.[A262051] It is spread primarily by the bite of infected mosquitos of the _Aedes_ genus. Infection with CHIKV causes chikungunya fever, an illness char…

Kategori:
Live vaccinesVaccinesViral Vaccines
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
Chiniofon DB13379
small molecule | CAS: 8002-90-2

Deskripsi belum tersedia.

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 9012-76-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chloral hydrate Approved DB01563
small molecule | CAS: 302-17-0

A hypnotic and sedative used in the treatment of insomnia. The safety margin is too narrow for chloral hydrate to be used as a general anesthetic in humans, but it is commonly used for that purpose in animal experiments. It is no longer considered useful as a…

Kategori:
AlcoholsCentral Nervous System AgentsCentral Nervous System Depressants +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chloramphenicol Approved DB00446
small molecule | CAS: 56-75-7

An antibiotic first isolated from cultures of _Streptomyces venezuelae_ in 1947 but now produced synthetically. It has a relatively simple structure and was the first broad-spectrum antibiotic to be discovered. It acts by interfering with bacterial protein sy…

Kategori:
AlcoholsAmphenicolsAnti-Acne Preparations +34
Target Protein:
50S ribosomal protein L16Dr hemagglutinin structural subunitComplement decay-accelerating factor
Waktu ParuhHalf-life in adults…
Vol. Distribusi-
Klirens-
Genetik -
Chloramphenicol succinate Approved DB07565
small molecule | CAS: 3544-94-3

Chloramphenicol succinate is an ester prodrug of [chloramphenicol].[A192987] Chloramphenicol is a bacteriostatic antibiotic.[A204065] Use of chloramphenicol succinate and chloramphenicol has decreased due to the risk of potentially fatal blood dyscrasias.[L14…

Kategori:
AlcoholsAnti-Bacterial AgentsAnti-Infective Agents +8
Target Protein:
Dr hemagglutinin structural subunit
Waktu ParuhThe half life of ch…
Vol. DistribusiChloramphenicol suc…
KlirensChloramphenicol suc…
Genetik -
small molecule | CAS: 522-18-9

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Functional Gastrointestinal Disorders
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlordiazepoxide Approved DB00475
small molecule | CAS: 58-25-3

An anxiolytic benzodiazepine derivative with anticonvulsant, sedative, and amnesic properties. It has also been used in the symptomatic treatment of alcohol withdrawal.

Kategori:
Adjuvants, AnesthesiaAnti-Anxiety AgentsBenzazepines +22
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh24-48 hours
Vol. Distribusi-
Klirens-
Genetik -
Chlorfenson DB05377
small molecule | CAS: 80-33-1

Chlorfenson is developed by Moberg Derma for the treatment of onychomycosis (nail fungus) as the primary indication.

Kategori:
ArylsulfonatesArylsulfonic AcidsBenzene Derivatives +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlorhexidine Approved DB00878
small molecule | CAS: 55-56-1

Chlorhexidine is a broad-spectrum antimicrobial biguanide used as a topical antiseptic and in dental practice for the treatment of inflammatory dental conditions caused by microorganisms.[L11512] It is one of the most common skin and mucous membrane antisepti…

Kategori:
Alimentary Tract and MetabolismAmidinesAnti-Infective Agents +25
Target Protein:
Bacterial outer membrane
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chloric acid Approved DB14150
small molecule | CAS: 7790-93-4

Deskripsi belum tersedia.

Kategori:
AgrochemicalsAnionsChlorine Compounds +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chloride ion DB14547
small molecule | CAS: 16887-00-6

Deskripsi belum tersedia.

Kategori:
AnionsChloridesChlorine Compounds +2
Target Protein:
Lanosterol 14-alpha demethylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlorindanol DB19355
small molecule | CAS: 145-94-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlorine DB11109
small molecule | CAS: 7782-50-5

Chlorine is a stongly oxidizing agent and the third most electronegative element which belongs to the group of halogens with the atomic number 17 and symbol Cl. Being a yellow-green gas at room temperature, chlorine is the second most abundant halogen on Eart…

Kategori:
Compounds used in a research, industrial, or household settingElementsGases +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlorisondamine Approved DB19358
small molecule | CAS: 7701-62-4

Deskripsi belum tersedia.

Kategori:
AminesAnticholinergic AgentsAntihypertensive Agents +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlormadinone DB13528
small molecule | CAS: 1961-77-9

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAntiandrogensCombination Contraceptives (with Estrogen and derivatives) +23
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 302-22-7

Chlormadinone acetate is a progesterone derivative first synthesized in 1961. In the US, chlormadinone acetate was formerly marketed as a component of the combination drug products Estalor-21 and C-Quens. However, the use of these drugs was associated with th…

Kategori:
Adrenal Cortex HormonesAntiandrogensContraceptive Agents, Female +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlormerodrin Approved DB00534
small molecule | CAS: 62-37-3

Chlormerodrin is a mercurial compound with toxic side effects that was previously used as a diuretic. The radiolabeled form has been used as a diagnostic and research tool. It is no longer used and has been replaced with new classes of diuretic drugs.

Kategori:
Alkylmercury CompoundsOrganomercury CompoundsOrganometallic Compounds
Target Protein:
Solute carrier family 12 member 1Succinate-semialdehyde dehydrogenase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlormerodrin Hg-197 Approved DB09406
small molecule | CAS: 64461-80-9

Chlormerodrin Hg-197 is a radiolabelled form of chlormerodrin, an organomercury compound that was previously used as a diuretic. Its radiolabelled form was used as diagnostics in brain scans.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlormezanone Approved DB01178
small molecule | CAS: 80-77-3

A non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.

Kategori:
Anti-Anxiety AgentsCentral Nervous System AgentsCentral Nervous System Depressants +10
Target Protein:
Translocator protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlormidazole DB13611
small molecule | CAS: 3689-76-7

Deskripsi belum tersedia.

Kategori:
Antifungals for Dermatological UseAntifungals for Topical UseDermatologicals +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlorobutanol Approved DB11386
small molecule | CAS: 57-15-8

Chlorobutanol, or chlorbutol, is an alcohol-based preservative with no surfactant activity [A32746]. It also elicits sedative-hypnotic and weak local anesthetic actions in addition to antibacterial and antifungal properties. Similar in nature to chloral hydra…

Kategori:
AlcoholsAlimentary Tract and MetabolismAntiemetics and Antinauseants +8
Target Protein:
Voltage-gated inwardly rectifying potassium channel KCNH2
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe volume of distr…
KlirensIn healthy subjects…
Genetik -
Chlorocresol DB16864
small molecule | CAS: 59-50-7

Deskripsi belum tersedia.

Kategori:
AgrochemicalsBenzene DerivativesChlorobenzenes +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chloroform Approved DB11387
small molecule | CAS: 67-66-3

Chloroform is an organic small molecule, member of the family of the chloromethanes that presents a formula of CHCl3. It is a colorless, sweet-smelling, dense liquid that is produced on a large scale as a precursor to PTFE and refrigerants, but the latter app…

Kategori:
AnestheticsAnesthetics, GeneralCompounds used in a research, industrial, or household setting +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlorophyll A DB02133
small molecule | CAS: 479-61-8

Deskripsi belum tersedia.

Kategori:
ChlorophyllHeterocyclic Compounds, Fused-Ring
Target Protein:
Beta-lactamase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlorophyll B DB04506
small molecule | CAS: 519-62-0

A light, silvery, metallic element. It has the atomic symbol Mg, atomic number 12, and atomic weight 24.31. Its salts are essential in nutrition, being required for the activity of many enzymes, especially those concerned with oxidative phosphorylation. It is…

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 52080-57-6

Deskripsi belum tersedia.

Kategori:
OphthalmologicalsSensory Organs
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chloroprocaine Approved DB01161
small molecule | CAS: 133-16-4

Chloroprocaine is an ester local anesthetic commonly available in its salt form, chloroprocaine hydrochloride. Similar to other local anesthetics, it increases the threshold for electrical excitation in nerves by slowing the propagation of the nerve impulse a…

Kategori:
Acids, CarbocyclicAminobenzoatesAnesthetics +15
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1Voltage-gated sodium channel alpha subunitSodium-dependent dopamine transporter
Waktu ParuhIn adults, the aver…
Vol. Distribusi-
Klirens-
Genetik -
Chloroquine Approved DB00608
small molecule | CAS: 54-05-7

Chloroquine is an aminoquinolone derivative first developed in the 1940s for the treatment of malaria.[A191655] It was the drug of choice to treat malaria until the development of newer antimalarials such as [pyrimethamine], [artemisinin], and [mefloquine].[A…

Kategori:
Agents Causing Muscle ToxicityAgents that produce neuromuscular block (indirect)Agents that reduce seizure threshold +39
Target Protein:
Atypical chemokine receptor 1Glutathione S-transferase A2Tumor necrosis factor +5
Waktu ParuhThe half life of ch…
Vol. DistribusiThe volume of distr…
KlirensChloroquine has a t…
Genetik -
Chlorothiazide Approved DB00880
small molecule | CAS: 58-94-6

A thiazide diuretic with actions and uses similar to those of hydrochlorothiazide. (From Martindale, The Extra Pharmacopoeia, 30th ed, p812)

Kategori:
Antihypertensive AgentsBenzothiadiazinesCardiovascular Agents +17
Target Protein:
Solute carrier family 12 member 3Carbonic anhydrase 1Carbonic anhydrase 2
Waktu Paruh45-120 minutes
Vol. Distribusi-
Klirens-
Genetik -
Chlorothymol Approved DB19375
small molecule | CAS: 89-68-9

Chlorotymol is a [Thymol] derivative.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlorotoxin DB15210
biotech | CAS: 163515-35-3

Chlorotoxin is under investigation in clinical trial NCT00733798 (A Safety and Efficacy Study of Intravenous 131I-TM601 in Adult Patients With Malignant Melanoma).

Kategori:
Arthropod VenomsBiological FactorsComplex Mixtures +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 569-57-3

A powerful synthetic, non-steroidal estrogen. [PubChem]

Kategori:
Antineoplastic AgentsAntineoplastic Agents, HormonalBenzene Derivatives +9
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chloroxine Approved DB01243
small molecule | CAS: 773-76-2

Chloroxine is a synthetic antibacterial compound. Chloroxine is a compound used in some shampoos for the treatment of dandruff and seborrheic dermatitis of the scalp.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntifungal Agents +3
Target Protein:
Kappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlorphenesin carbamate Approved DB14656
small molecule | CAS: 886-74-8

Deskripsi belum tersedia.

Kategori:
AlcoholsGlycolsPropylene Glycols
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 77-38-3

Chlorphenoxamine is marketed under the name Phenoxene. It is an antihistamine and anticholinergic used to treat itching as well as for its antiparkinsonian effect.

Kategori:
Agents producing tachycardiaAminesAminoalkyl Ethers +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 461-78-9

A sympathomimetic agent that was formerly used as an anorectic. It has properties similar to those of dextroamphetamine. It has been implicated in lipid storage disorders and pulmonary hypertension. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1223)

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +7
Target Protein:
Sodium-dependent serotonin transporter
Waktu Paruh40 hours
Vol. Distribusi-
Klirens-
Genetik -
Chlorproguanil DB12314
small molecule | CAS: 537-21-3

Chlorproguanil has been used in trials studying the treatment of MALARIA. It is a dichloro-derivative of chloroguanide.

Kategori:
AmidinesAnti-Infective AgentsAntimalarials +4
Target Protein:
Peptide deformylase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Chlorpromazine Approved DB00477
small molecule | CAS: 50-53-3

The prototypical phenothiazine antipsychotic drug. Like the other drugs in this class, chlorpromazine's antipsychotic actions are thought to be due to long-term adaptation by the brain to blocking dopamine receptors. Chlorpromazine has several other actions a…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +63
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptor5-hydroxytryptamine receptor 1A +21
Waktu Paruh~ 30 hours
Vol. Distribusi* 20 L/kg
Klirens-
Genetik -
Chlorpropamide Approved DB00672
small molecule | CAS: 94-20-2

Chlorpropamide is an oral antihyperglycemic agent used for the treatment of non-insulin-dependent diabetes mellitus (NIDDM). It belongs to the sulfonylurea class of insulin secretagogues, which act by stimulating ? cells of the pancreas to release insulin. Su…

Kategori:
Alimentary Tract and MetabolismAmidesBenzene Derivatives +17
Target Protein:
ATP-binding cassette sub-family C member 8ATP-sensitive inward rectifier potassium channel 10
Waktu ParuhApproximately 36 ho…
Vol. Distribusi-
Klirens-
Genetik -
Chlorprothixene Approved DB01239
small molecule | CAS: 113-59-7

Chlorprothixene is a typical antipsychotic drug of the thioxanthene (tricyclic) class. Chlorprothixene exerts strong blocking effects by blocking the 5-HT2 D1, D2, D3, histamine H1, muscarinic and alpha1 adrenergic receptors.

Kategori:
Agents producing tachycardiaAnticholinergic AgentsAntidepressive Agents +28
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptorD(3) dopamine receptor +8
Waktu Paruh8 to 12 hours
Vol. Distribusi-
Klirens-
Genetik -
Chlorquinaldol Approved DB13306
small molecule | CAS: 72-80-0

Chlorquinaldol was used historically as a topical antiseptic under the trade name Sterosan.[F4549] It was marketed in the 1950s as an iodine-free alternative which was also unrelated to sulfa drugs or hormones. Chlorquinaldol is currently approved by the Euro…

Kategori:
Anti-Infective AgentsAnti-Infective Agents, LocalAntiparasitic Products, Insecticides and Repellents +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 97919-22-7

Chlorsulfaquinoxaline has been used in trials studying the treatment of Lung Cancer and Colorectal Cancer.

Kategori:
AmidesAminesAniline Compounds +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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