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13591

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10177 (74.9%)
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7625 (56.1%)
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104 (0.8%)
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13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 71 / 272
biotech | CAS: 2374772-30-0

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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Bexagliflozin Approved DB12236
small molecule | CAS: 1118567-05-7

Bexagliflozin is a highly specific and potent sodium-glucose co-transporter 2 (SGLT2) inhibitor.[A256408,A256413,L44758] Similar to other SGLT2 inhibitors, bexagliflozin contains three basic moieties: glucose, two benzene rings and a methylene bridge.[A256413…

Kategori:
Alimentary Tract and MetabolismBenzene DerivativesBlood Glucose Lowering Agents +16
Target Protein:
Sodium/glucose cotransporter 2
Waktu ParuhBexagliflozin has a…
Vol. DistribusiBexagliflozin has a…
KlirensPopulation pharmaco…
Genetik -
Bexarotene Approved DB00307
small molecule | CAS: 153559-49-0

Bexarotene (Targretin) is an antineoplastic agent indicated by the FDA for Cutaneous T cell lymphoma. It has been used off-label for lung cancer, breast cancer, and Kaposi's sarcoma.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCompounds used in a research, industrial, or household setting +18
Target Protein:
Retinoic acid receptor RXR-alphaRetinoic acid receptor RXR-betaRetinoic acid receptor RXR-gamma
Waktu Paruh7 hours
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Bexicaserin DB18885
small molecule | CAS: 2035818-24-5

Bexicaserin is under investigation in clinical trial NCT05626634 (Open-label, Long-term Safety Study of LP352 in Subjects With Developmental and Epileptic Encephalopathy).

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Bexmarilimab DB16383
biotech | CAS: 2259301-27-2

Bexmarilimab is under investigation in clinical trial NCT03733990 (A Study to Evaluate Safety, Tolerability and Preliminary Efficacy of FP-1305 in Cancer Patients).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Bexotegrast DB18444
small molecule | CAS: 2376257-44-0

Deskripsi belum tersedia.

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Bezafibrate Approved DB01393
small molecule | CAS: 41859-67-0

Antilipemic agent that lowers cholesterol and triglycerides. It decreases low density lipoproteins and increases high density lipoproteins.

Kategori:
Acids, AcyclicAcids, CarbocyclicAgents Causing Muscle Toxicity +26
Target Protein:
Peroxisome proliferator-activated receptor deltaPeroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha +4
Waktu Paruh1-2 hours
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Bezitramide DB01459
small molecule | CAS: 15301-48-1

Bezitramide is a narcotic analgesic which was discovered in 1961, clinically tested around the 1970's [A14383], and marketed under the name Burgodin. After cases of fatal overdose in the Netherlands in 2004 the drug was withdrawn from the market. Bezitram…

Kategori:
AnalgesicsCentral Nervous System AgentsDiphenylpropylamine Derivatives +6
Waktu Paruh11-24h. [A14383]
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Bezlotoxumab Approved DB13140
biotech | CAS: 1246264-45-8

Bezlotoxumab is a fully humanized ImmunoglobulinG1 (IgG1) kappa monoclonal antibody that binds to _Clostridium difficile_ toxin B and neutralizes its effects.[L46976] First approved by the FDA on October 21, 2016,[A260106] bezlotoxumab is used to reduce the r…

Kategori:
Amino Acids, Peptides, and ProteinsAntibacterial monoclonal antibodiesAntibodies +11
Target Protein:
Toxin B
Waktu ParuhBased on a populati…
Vol. DistribusiBased on a populati…
KlirensBased on a populati…
Genetik -
Bezuclastinib DB18041
small molecule | CAS: 1616385-51-3

Deskripsi belum tersedia.

Target Protein:
Mast/stem cell growth factor receptor Kit
Waktu Paruh-
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BF-37 DB05755
small molecule

BF-37 for the treatment of atopic dermatitis and/or psoriasis. The active ingredient in BF-37 is Riluzole, applied in a topical formulation, which is believed to correct the imbalances of the immune system that cause atopic dermatitis or psoriasis.

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BF-844 DB17801
small molecule | CAS: 1404506-35-9

Deskripsi belum tersedia.

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BFH772 DB16035
small molecule | CAS: 890128-81-1

BFH772 is under investigation in clinical trial NCT01449591 (Safety, Tolerability and Efficacy of BFH772 in Rosacea Patients).

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Bfpet F-18 DB15424
small molecule | CAS: 863644-14-8

Bfpet F-18 is under investigation in clinical trial NCT03265431 (Evaluation of PET/MR in Patients Selected for Ablation Therapy).

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BG-777 DB05839
small molecule

BG-777 is an immunomodulator with proven efficacy against viral and bacterial infections in preclinical studies.

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BG-P-TAT DB18105
small molecule

Deskripsi belum tersedia.

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BG-P400-TAT DB17104
small molecule

Deskripsi belum tersedia.

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BGB-DXP593 DB16357
biotech

BGB-DXP593 is a SARS-CoV-2 neutralizing antibody.[L27401] It is currently being investigated against COVID-19 in the clinical trial NCT04551898 (Severe Acute Respiratory Syndrome Coronavirus 2 (SARS-CoV-2) Neutralizing Antibody BGB-DXP593 in Participants With…

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BGT-DTDS DB18664
biotech

BGT-DTDS is an investigational gene therapy comprising an adeno-associated viral vector type 2 (AAV2) encoding the human _SLC6A3_ gene. It is under investigation for the treatment of dopamine transporter deficiency syndrome (DTDS).

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BHT-3034 DB18045
biotech

BHT-3034 is a DNA plasmid vaccine immunotherapy under investigation for the treatment of myasthenia gravis.[L48086]

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BI 2536 DB16107
small molecule | CAS: 755038-02-9

BI 2536 is under investigation in clinical trial NCT00376623 (Efficacy and Safety of BI 2536 in Advanced or Metastatic Non Small Cell Lung Cancer).

Kategori:
Antimitotic AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase PLK1
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BI 44370 TA DB16037
small molecule | CAS: 866086-05-7

BI 44370 TA is under investigation in clinical trial NCT00751803 (BI 44370 TA in Acute Migraine Attack).

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BI-1206 DB17429
biotech

BI-1206 is a fully human immunoglobulin G1 monoclonal antibody that targets CD32b.

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BI-187004 DB18897
small molecule | CAS: 1303515-32-3

Deskripsi belum tersedia.

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BI-671800 DB12524
small molecule | CAS: 1093108-50-9

Bi 671800 has been used in trials studying the treatment of Asthma and Rhinitis, Allergic, Perennial.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Prostaglandin D2 receptor 2
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BI-765063 DB17482
biotech

BI-765063 is a humanized IgG4 monoclonal antibody antagonist of signal regulatory protein ? (SIRP?).

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BI-836826 DB17322
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
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BI-836858 DB17267
biotech | CAS: 2206770-25-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
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BI-836880 DB17484
biotech

BI-836880 is a humanized bispecific nanobody that targets VEGF and Ang2.

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BI-K0376 DB05858
biotech

BI-K0376 is investigated for use/treatment in acne. BI-K0376 is a solid. It is under investigation by Pfizer and has gone through phase I of the clinical trails.

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Bi104 DB18743
biotech

Bi104 is being investigated for the treatment of Angelman syndrome.

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BIA DB03336
small molecule

Deskripsi belum tersedia.

Kategori:
COMT Inhibitors
Target Protein:
Catechol O-methyltransferase
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Biapenem DB13028
small molecule | CAS: 120410-24-4

Biapenem has been used in trials studying the treatment of Bacterial Infections.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +6
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Bibenzonium DB13630
small molecule | CAS: 59866-76-1

Deskripsi belum tersedia.

Kategori:
Cough and Cold Preparations
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Bibrocathol DB13818
small molecule | CAS: 6915-57-7

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsBenzene DerivativesOphthalmologicals +2
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Bicalutamide Approved DB01128
small molecule | CAS: 90357-06-5

Bicalutamide is an oral non-steroidal anti-androgen for prostate cancer. It is comprised of a racemic mixture that is a 50:50 composition of the (R)-bicalutamide and (S)-bicalutamide enantionmers. Bicalutamide binds to the androgen receptor.

Kategori:
AmidesAminesAndrogen Receptor Antagonists +31
Target Protein:
Androgen receptor
Waktu Paruh5.9 days
Vol. Distribusi-
Klirens* Apparent oral cl=…
Genetik -
Bicine DB03709
small molecule | CAS: 150-25-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
PlasminogenMembrane-bound lytic murein transglycosylase BUDP-galactopyranose mutase
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Bicisate Approved DB11164
small molecule | CAS: 121251-02-3

Bicisate, also known as ethyl cysteinate dimer (ECD), is a N,N'-1,2-ethylene-di-yl-bis-L-cysteinate diethyl ester. It is used in conjunction with technetium Tc99m as a tracer to measure cerebral blood flow with single-photon emission computed tomography (SPEC…

Kategori:
Diagnostic AgentsDrugs that are Mainly Renally ExcretedRadioactive Diagnostic Agent
Waktu ParuhThe stability of bi…
Vol. DistribusiAfter intravenous a…
KlirensThe clearance of bi…
Genetik -
Bictegravir Approved DB11799
small molecule | CAS: 1611493-60-7

Bictegravir is a recently approved investigational drug that has been used in trials studying the treatment of HIV-1 and HIV-2 infection. It has been approved for HIV-1 monotherapy combined with 2 other antiretrovirals in a single tablet.[L43677]

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +11
Target Protein:
Reverse transcriptase/RNaseHIntegrase
Waktu ParuhHalf-life is 17.3 h…
Vol. Distribusi0.2 L/Kg in humans …
KlirensBictegravir is main…
Genetik -
Bicuculline DB11562
small molecule | CAS: 485-49-4

Bicuculline is a light-sensitive competitive antagonist of GABAA receptors. It was originally identified in 1932 in plant alkaloid extracts and has been isolated from Dicentra cucullaria, Adlumia fungosa, Fumariaceae, and several Corydalis species.

Kategori:
AlkaloidsBenzylisoquinolinesCentral Nervous System Agents +8
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Bicyclol DB16014
small molecule | CAS: 118159-48-1

Bicyclol is under investigation in clinical trial NCT02944552 (The Multi Center, Randomized, Double-blind, Positive Controlled Study of Bicyclol in the Treatment of Acute DILI).

Kategori:
Benzene Derivatives
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Bietaserpine DB13575
small molecule | CAS: 53-18-9

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntiadrenergic Agents, Centrally ActingAntihypertensive Agents +7
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Bifemelane DB13550
small molecule | CAS: 90293-01-9

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsBenzene DerivativesCentral Nervous System Agents +5
Target Protein:
Amine oxidase [flavin-containing] A
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Bifenthrin DB15056
small molecule | CAS: 82657-04-3

Bifenthrin is under investigation in clinical trial NCT01560247 (Percutaneous Recanalization in Ischemic Stroke Management in Europe Observational Registry).

Kategori:
Cyclopentane MonoterpenesMonoterpenesSarcoma, Experimental, chemically induced +1
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Bifeprunox DB04888
small molecule | CAS: 350992-10-8

Bifeprunox is a novel atypical antipsychotic agent which, along with SLV313, [aripiprazole] and SSR-181507 combines minimal D2 receptor agonism with 5-HT receptor agonism.

Kategori:
Antipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical])Central Nervous System Depressants +2
Target Protein:
5-hydroxytryptamine receptor 1AD(2) dopamine receptor
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Bifidobacterium bifidum Approved DB16538
biotech

Deskripsi belum tersedia.

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Bifidobacterium longum Approved DB19248
biotech

Deskripsi belum tersedia.

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biotech

Bifidobacterium Longum Infantis 35624 is a probiotic being investigated for the treatment of gastrointestinal disorders, such as Crohn's disease and irritable bowel syndrome.[A259872, A259877]

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biotech

Deskripsi belum tersedia.

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Bifikafusp alfa DB19185
biotech | CAS: 1957239-90-5

Bifikafusp alfa is under investigation in clinical trial NCT05329792 (L19IL2/L19TNF in Skin Cancer Patients).

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