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14063

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10481 (74.5%)
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8038 (57.2%)
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107 (0.8%)
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14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 71 / 282
Begelomab DB13241
biotech | CAS: 1403744-56-8

Begelomab is a murine monoclonal antibody against CD26.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic and Immunomodulating Agents +6
Waktu Paruh-
Vol. Distribusi-
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Beinaglutide DB15072
biotech | CAS: 123475-27-4

Beinaglutide is under investigation in clinical trial NCT03829891 (Study for Beinaglutide Versus Glargine Therapy in Glycemic Variability of Type 2 Diabetes Mellitus).

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +8
Waktu Paruh-
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Genetik -
biotech

Deskripsi belum tersedia.

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biotech

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biotech

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Belantamab mafodotin Approved DB15719
biotech | CAS: 2050232-20-5

Belantamab mafodotin, or GSK2857916, is an afucosylated monoclonal antibody that targets B cell maturation antigen conjugated to the microtubule disrupter monomethyl auristatin-F (MMAF).[A216756] Belantamab mafodotin was granted FDA accelerated approval on…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Tumor necrosis factor receptor superfamily member 17
Waktu ParuhThe terminal half l…
Vol. DistribusiThe mean steady sta…
KlirensThe clearance of be…
Genetik -
Belapectin DB15125
small molecule | CAS: 1980787-47-0

Belapectin is under investigation in clinical trial NCT02575404 (GR-MD-02 Plus Pembrolizumab in Melanoma, Non-small Cell Lung Cancer, and Squamous Cell Head and Neck Cancer Patients).

Kategori:
Biological ProductsBiopolymersCarbohydrates +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Belatacept Approved DB06681
biotech | CAS: 706808-37-9

Belatacept is a soluble fusion protein, which links the extracellular domain of human cytotoxic T-lymphocyte-associated antigen 4 (CTLA-4) to the modified Fc (hinge, CH2, and CH3 domains) portion of human immunoglobulin G1 (IgG1). Structurally, abatacept is a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents, Immunological +15
Target Protein:
T-lymphocyte activation antigen CD86T-lymphocyte activation antigen CD80
Waktu ParuhMean terminal elimi…
Vol. DistribusiVd, steady state, t…
KlirensIncreased body weig…
Genetik -
Belcesiran DB18226
biotech | CAS: 2375562-54-0

Deskripsi belum tersedia.

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Belimumab Approved DB08879
biotech | CAS: 356547-88-1

Belimumab is a fully human recombinant IgG1? monoclonal antibody that inhibits soluble human B lymphocyte stimulator protein (BLyS, also referred to as BAFF and TNFSF13B), a B cell survival factor.[L42630] BLyS levels are often elevated in immunodeficient and…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Tumor necrosis factor ligand superfamily member 13B
Waktu ParuhFollowing administr…
Vol. DistribusiFollowing administr…
KlirensFollowing administr…
Genetik -
Belinostat Approved DB05015
small molecule | CAS: 866323-14-0

Belinostat is a novel agent that inhibits the enzyme histone deacetylase (HDAC) with a sulfonamide-hydroxamide structure. It was developed as an orphan drug to target hematological malignancies and solid tumors by TopoTarget. The safety and efficacy of belino…

Kategori:
AmidesAminesAntineoplastic Agents +31
Target Protein:
Histone deacetylase
Gen Terkait:
UGT1A1 UGT1A1
Waktu ParuhDisplays a three-co…
Vol. DistribusiThe volume of distr…
Klirens1240 mL/min
Genetik 2 Varian
Belladonna Approved DB13913
biotech

Belladonna, also known as atropa belladonna or deadly nightshade, is a perennial herbaceous plant in the nightshade family _Solanaceae_. Its roots, leaves and fruits contain [DB00424], [DB00747], and mostly, [DB00572]. These alkaloids are naturally-occurring …

Kategori:
Anticholinergic AgentsAntimuscarinics AntispasmodicsMuscarinic Antagonists
Waktu ParuhFor pharmacokinetic…
Vol. DistribusiFor pharmacokinetic…
KlirensFor pharmacokinetic…
Genetik -
Beloranib DB12671
small molecule | CAS: 251111-30-5

Beloranib has been used in trials studying the treatment of Obesity, Over-weight, Type 2 Diabetes, Craniopharyngioma, and Hypothalamic Injury, among others.

Kategori:
Acids, CarbocyclicAngiogenesis InhibitorsAngiogenesis Modulating Agents +7
Target Protein:
Methionine aminopeptidase 2
Waktu Paruh-
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Belotecan DB12459
small molecule | CAS: 256411-32-2

Belotecan has been investigated for the treatment of Epithelial Ovarian Cancer.

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +4
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
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Belrestotug DB19066
biotech | CAS: 2574438-65-4

Belrestotug is under investigation in clinical trial NCT05565378 (A Platform Study of Novel Immunotherapy Combinations in Participants With Previously Untreated, Advanced/metastatic Non-small-cell Lung Cancer).

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Beludavimab DB18952
biotech | CAS: 2423016-74-2

Beludavimab is under investigation in clinical trial NCT04746183 (AGILE (Early Phase Platform Trial for COVID-19)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
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Belumosudil Approved DB16703
small molecule | CAS: 911417-87-3

Belumosudil is used in the treatment of chronic graft-versus-host disease (GVHD) and has been investigated for the treatment of pulmonary arterial hypertension.[A236634] It is an inhibitor of rho-associated coiled-coil-containing protein kinases (ROCK), with …

Kategori:
AcetatesAcids, AcyclicAmides +25
Target Protein:
Rho-associated protein kinase 2Rho-associated protein kinase 1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiFollowing a single …
KlirensThe mean clearance …
Genetik -
Belvarafenib DB17568
small molecule | CAS: 1446113-23-0

Deskripsi belum tersedia.

Target Protein:
RAF proto-oncogene serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2390462-37-8

Deskripsi belum tersedia.

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Belzutifan Approved DB15463
small molecule | CAS: 1672668-24-4

Belzutifan is an inhibitor of hypoxia-inducible factor 2? (HIF-2?) used in the treatment of von Hippel-Lindau (VHL) disease-associated cancers.[L35995] The HIF-2? protein was first identified in the 1990s by researchers at UT Southwestern Medical Center as a …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C19 Substrates +10
Target Protein:
Endothelial PAS domain-containing protein 1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
Bemarituzumab DB16105
biotech | CAS: 1952272-74-0

Bemarituzumab is under investigation in clinical trial NCT03694522 (A Study of Bemarituzumab (FPA144) Combined With Modified FOLFOX6 (Mfolfox6) in Gastric/gastroesophageal Junction Cancer (FIGHT)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bemcentinib DB12411
small molecule | CAS: 1037624-75-1

Bemcentinib has been investigated for the treatment of Non-Small Cell Lung Cancer.

Target Protein:
Spike glycoproteinTyrosine-protein kinase receptor UFO
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2766038-73-5

Deskripsi belum tersedia.

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Bemiparin Approved DB09258
small molecule | CAS: 91449-79-5

Bemiparin is an antithrombotic and belongs to the group of drugs known as the low molecular weight heparins (LMWH). Like semuloparin, bemiparin is classified as an ultra-LMH because of its low mean molecular mass of 3600 daltons, which is a unique property of…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +6
Target Protein:
Coagulation factor XAntithrombin-IIIHeparin cofactor 2
Waktu ParuhBemiparin, when adm…
Vol. Distribusi5.1 L [A32018].
KlirensElimination occurs …
Genetik -
Bemnifosbuvir DB19050
small molecule | CAS: 1998705-64-8

Bemnifosbuvir is under investigation in clinical trial NCT05629962 (SUNRISE-3: Efficacy and Safety of Bemnifosbuvir in High-risk Outpatients With COVID-19).

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Bemotrizinol Approved DB11206
small molecule | CAS: 187393-00-6

Bemotrizinol, or bis-ethylhexyloxyphenol methoxyphenyl triazine, is an organic UV filter found in over-the-counter sunscreen products. It primarily absorbs UV-A rays. Compared to older broad-spectrum chemical agents, bemotrizinol is more more fat soluble (oil…

Kategori:
Benzene DerivativesSunscreen Agents
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Bempedoic acid Approved DB11936
small molecule | CAS: 738606-46-7

High levels of LDL cholesterol (LDL-C) are a major risk factor for cardiovascular events. Caused by genetic mutations or lifestyle factors, hypercholesterolemia can significantly reduce quality of life and increase the risk of mortality from cardiovascular di…

Kategori:
Acids, AcyclicAdenosine Triphosphate-Citrate Lyase InhibitorAdenosine Triphosphate-Citrate Lyase Inhibitors +11
Target Protein:
ATP-citrate synthase
Waktu ParuhThe half-life of be…
Vol. DistribusiThe apparent volume…
KlirensThe clearance (CL/F…
Genetik -
biotech | CAS: 1939126-74-5

Bempegaldesleukin is under investigation in clinical trial NCT03729245 (A Study of NKTR-214 in Combination With Nivolumab Compared With the Investigator's Choice of a Tyrosine Kinase Inhibitor (TKI) Therapy (Either Sunitinib or Cabozantinib Monotherapy) for A…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Benactyzine DB09023
small molecule | CAS: 302-40-9

Benactyzine is an anticholinergic drug used as an antidepressant in the treatment of depression and associated anxiety. Benactyzine is no longer widely used in medicine, although it is still a useful drug for scientific research. It does not possess any an…

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAnticholinergic Agents +14
Target Protein:
Muscarinic acetylcholine receptor M5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benapenem DB18883
small molecule | CAS: 1312953-83-5

Benapenem is under investigation in clinical trial NCT04505683 (A Study to Assess Efficacy and Safety Intravenous Benapenem in Patients With Complicated Urinary Tract Infection (Cuti) or Acute Pyelonephritis (AP)).

Kategori:
Amidesbeta-LactamsHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benazepril Approved DB00542
small molecule | CAS: 86541-75-5

Benazepril, brand name Lotensin, is a medication used to treat high blood pressure (hypertension), congestive heart failure, and chronic renal failure[A838,A837]. Upon cleavage of its ester group by the liver, benazepril is converted into its active form bena…

Kategori:
ACE Inhibitors and Calcium Channel BlockersACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin System +13
Target Protein:
Angiotensin-converting enzyme
Waktu ParuhThe half life of th…
Vol. DistribusiThe final populatio…
KlirensThe final populatio…
Genetik -
Benazeprilat DB14125
small molecule | CAS: 86541-78-8

Deskripsi belum tersedia.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Bencyclane DB13488
small molecule | CAS: 2179-37-5

A vasodilator agent found to be effective in a variety of peripheral circulation disorders. It has various other potentially useful pharmacological effects. Its mechanism may involve block of calcium channels.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bendamustine Approved DB06769
small molecule | CAS: 16506-27-7

Bendamustine is a nitrogen mustard drug which has been used in the treatment of chronic lymphocytic leukemia (CLL) and indolent B-cell non-Hodgkin lymphoma (NHL). Bendamustine is a bifunctional mechlorethamine derivative capable of forming electrophilic alky…

Kategori:
Acids, AcyclicAlkylating ActivityAlkylating Drugs +19
Target Protein:
DNA
Waktu Paruh40 minutes
Vol. DistribusiThe mean steady-sta…
Klirens700 mL/min
Genetik -
Bendazac Approved DB13501
small molecule | CAS: 20187-55-7

Bendazac is an oxyacetic acid [A39863, A39869]. Despite possessing anti-inflammatory, anti-necrotic, choleretic, and anti-lipidemic characteristics, most research has revolved around studying and demonstrating the agent's principal action in inhibiting the de…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +18
Target Protein:
Free radicalsProstaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe volume of distr…
KlirensThe plasma clearanc…
Genetik -
Bendroflumethiazide Approved DB00436
small molecule | CAS: 73-48-3

A thiazide diuretic with actions and uses similar to those of hydrochlorothiazide. It has been used in the treatment of familial hyperkalemia, hypertension, edema, and urinary tract disorders. (From Martindale, The Extra Pharmacopoeia, 30th ed, p810)

Kategori:
Antihypertensive AgentsAntihypertensive Agents Indicated for HypertensionBenzothiadiazines +17
Target Protein:
Solute carrier family 12 member 3Solute carrier family 12 member 1Calcium-activated potassium channel subunit alpha-1 +3
Waktu Paruh8.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Benfluorex DB09022
small molecule | CAS: 23602-78-0

Benfluorex is an anorectic and hypolipidemic agent that is structurally related to fenfluramine. It was patented and manufactured by a French pharmaceutical company Servier. The European Medicines Agency (EMA) recommended withdrawing all benfluorex containing…

Kategori:
Alimentary Tract and MetabolismAminesAnti-Obesity Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Benfotiamine Approved DB11748
small molecule | CAS: 22457-89-2

Benfotiamine has been investigated for the treatment and prevention of Diabetic Nephropathy and Diabetes Mellitus, Type 2.

Kategori:
Adjuvants, ImmunologicAlimentary Tract and MetabolismCompounds used in a research, industrial, or household setting +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Benidipine DB09231
small molecule | CAS: 105979-17-7

Benidipine has the formula 1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3,5-pyridine-dicarboxylic acid methyl 1-(phenylmethyl)-3-piperidinyl ester hydrochloride. It is a synthetic dihydropyridine derivative that has anti-hypertensive and anti-anginal actions.[A…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +19
Target Protein:
Voltage-dependent L-type calcium channelVoltage-dependent N-type calcium channel subunit alpha-1BVoltage-dependent T-type calcium channel
Waktu ParuhThe elimination hal…
Vol. DistribusiBenidipine is highl…
Klirens-
Genetik -
Benmoxin DB09246
small molecule | CAS: 7654-03-7

Benmoxin is an irreversible and nonselective monoamine oxidase inhibitor (MAOI) of the hydrazine class. It was first synthesized in 1967 and rapidly used in Europe as an antidepressant. However, this agent is no longer marketed.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benoxaprofen Approved DB04812
small molecule | CAS: 51234-28-7

The use of benoxaprofen, formerly marketed as Oraflex tablets, was associated with fatal cholestatic jaundice among other serious adverse reactions. The holder of the approved application voluntarily withdrew Oraflex tablets from the market on August 5, 1982.

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +18
Target Protein:
Acetyl-CoA acetyltransferase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benperidol Approved DB12867
small molecule | CAS: 2062-84-2

Benperidol has been used in trials studying the treatment of Dementia, Depression, Schizophrenia, Anxiety Disorders, and Psychosomatic Disorders, among others.

Kategori:
Antipsychotic AgentsButyrophenone DerivativesButyrophenones +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benproperine DB13309
small molecule | CAS: 2156-27-6

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesCough and Cold Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benralizumab Approved DB12023
biotech | CAS: 1044511-01-4

Benralizumab is a humanized recombinant monoclonal antibody of the isotype IgG1k immunoglobulin that specifically binds to the alpha chain of the interleukin 5 receptor (IL-5R) expressed on eosinophils and basophils.[A31294] It inhibits the binding of IL-5 as…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAntibodies +13
Target Protein:
Interleukin-5 receptor subunit alphaLow affinity immunoglobulin gamma Fc region receptor III-A
Waktu ParuhThe half-life of Be…
Vol. DistribusiPharmacokinetic rep…
KlirensFor a subject weigh…
Genetik -
Benserazide Approved DB12783
small molecule | CAS: 322-35-0

When levodopa is used by itself as a therapy for treating Parkinson's disease, its ubiquitous metabolism into dopamine is responsible for a resultant increase in the levels of circulating dopamine in the blood and to various extracerebral tissues. This can re…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsAromatic L-amino Acid Decarboxylase Inhibitors +6
Target Protein:
Aromatic-L-amino-acid decarboxylase
Waktu ParuhThe half-life of be…
Vol. DistribusiReadily accessible …
KlirensReadily accessible …
Genetik -
Bentazepam DB14719
small molecule | CAS: 29462-18-8

Deskripsi belum tersedia.

Kategori:
Anti-Anxiety AgentsBenzodiazepines and benzodiazepine derivativesCentral Nervous System Agents +4
Target Protein:
GABA(A) ReceptorGamma-aminobutyric acid receptor subunit gamma-3GABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bentiromide DB00522
small molecule | CAS: 37106-97-1

Bentiromide is a dipeptide that is used in the bentiromide test, which is a screening test for evaluating pancreatic exocrine function and monitoring the adequacy of supplemental pancreatic therapy. It is typically administered orally. Cases of headache and g…

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +7
Target Protein:
Serine protease hepsin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bentracimab DB16659
biotech | CAS: 2260568-31-6

Bentracimab is under investigation in clinical trial NCT04286438 (Bentracimab (PB2452) in Ticagrelor-treated Patients With Uncontrolled Major or Life-threatening Bleeding or Requiring Urgent Surgery or Invasive Procedure).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Neutralizing +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzamidine DB03127
small molecule | CAS: 618-39-3

Deskripsi belum tersedia.

Kategori:
AmidinesEnzyme InhibitorsProtease Inhibitors +1
Target Protein:
Serine protease 1Urokinase-type plasminogen activatorSuppressor of tumorigenicity 14 protein +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benzatropine Approved DB00245
small molecule | CAS: 86-13-5

Benztropine, with the chemical formula 3alpha-diphenylmethoxytropane, is a tropane-based dopamine inhibitor used for the symptomatic treatment of Parkinson's disease. It is a combination molecule between a tropane ring, similar to cocaine, and a diphenyl ethe…

Kategori:
Agents producing tachycardiaAlkaloidsAnti-Dyskinesia Agents +23
Target Protein:
Muscarinic acetylcholine receptor M1Sodium-dependent dopamine transporterHistamine H1 receptor +2
Waktu ParuhThe elimination hal…
Vol. DistribusiBenztropine is expe…
KlirensExtensive pharmacod…
Genetik -
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