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16749

Total database: 17430
Struktur (SMILES)
11810 (70.5%)
Target
9015 (53.8%)
Genomik
112 (0.7%)
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16749 (100.0%)

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Hasil Pencarian (16749)

Halaman 70 / 335
AP-001 DB18511
small molecule | CAS: 660430-03-5

Deskripsi belum tersedia.

Kategori:
Dietary FatsDietary Fats, UnsaturatedFats +6
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AP-101 DB17947
biotech

AP-101 is a recombinant human antibody directed against human misfolded superoxide dismutase 1.

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AP-102 DB18206
small molecule | CAS: 846569-60-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
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AP103 DB18234
biotech

AP103 is a non-viral gene therapy that uses a delivery vector, HPAE (Highly Branched Poly ?-Amino Ester), to deliver the correct collagen VII gene into skin cells.

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AP1081 DB05233
small molecule

A transdermal gel containing ethinyl estradiol and norelgestromin being investigated by Antares Pharma for use as a female contraceptive.

Target Protein:
Estrogen receptor
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AP5280 DB05112
small molecule

AP5280 is a novel N-(2-hydroxypropyl)methacrylamide (HPMA) copolymer-bound platinum (Pt) therapeutic designed to increase the therapeutic index relative to conventional, small-molecule platinum agents.

Kategori:
Acids, AcyclicAcrylatesAmides +2
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AP5346 DB04992
small molecule

AP5346 is designed to target a diaminocyclohexane platinum (Pt) moiety to tumors through pH-sensitive linkage to a 25 kDa hydroxypropylmethacrylamide polymer. It is being pursued by Access Pharmaceuticals, Inc.

Kategori:
Organometallic Compounds
Target Protein:
DNA
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Apabetalone DB12000
small molecule | CAS: 1044870-39-4

Apabetalone has been investigated for the treatment of Diabetes, Atherosclerosis, and Coronary Artery Disease.

Kategori:
Heterocyclic Compounds, Fused-RingQuinazolines
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Apadamtase alfa Approved DB15164
biotech | CAS: 2086325-24-6

Thrombotic thrombocytopenic purpura (TTP) is a rare blood clotting disorder characterized by thrombocytopenia, microangiopathic hemolytic anemia, and various degrees of organ damage.[A262076] It may be inherited (congenital TTP; cTTP) or acquired due to autoa…

Kategori:
ADAM ProteinsADAMTS ProteinsAmino Acids, Peptides, and Proteins +12
Target Protein:
von Willebrand factor
Waktu ParuhFollowing the intra…
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Apadenoson DB05009
small molecule | CAS: 250386-15-3

Apadenoson is a selective A2a adenosine receptor agonist designed for use as a pharmacologic stress agent in cardiac perfusion imaging studies. It is developed by Bristol-Myers Squibb and is in phase II of clinical trials.

Kategori:
Acids, CarbocyclicAdenosine A receptor agonistsAdenosine A2 Receptor Agonists +7
Target Protein:
Adenosine receptor A2a
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Apalutamide Approved DB11901
small molecule | CAS: 956104-40-8

Apalutamide is a potent androgen receptor (AR) antagonist that selectively binds to the ligand-binding domain of AR and blocks AR nuclear translocation or binding to androgen response elements [A31846]. It has been used in trials studying the treatment of Pro…

Kategori:
Androgen Receptor InhibitorsAntiandrogensAntineoplastic Agents +28
Target Protein:
Androgen receptorGABA(A) Receptor
Waktu ParuhThe mean effective …
Vol. DistribusiThe mean apparent v…
KlirensThe CL/F of apaluta…
Genetik -
biotech | CAS: 2097132-02-8

Deskripsi belum tersedia.

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Apararenone DB15024
small molecule | CAS: 945966-46-1

Apararenone is under investigation in clinical trial NCT02531568 (Drug Interaction Study of Warfarin and MT-3995).

Kategori:
AmidesSulfonesSulfur Compounds
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Apatorsen DB06094
biotech | CAS: 1002331-21-6

Apatorsen is a second generation antisense drug which in preclinical experiments, inhibits production of Heat Shock Protein 27 (Hsp27) a cell survival protein found at elevated levels in many human cancers including prostate, lung, breast, ovarian, bladder, r…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Heat shock protein beta-1
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Apaziquone DB12593
small molecule | CAS: 114560-48-4

Apaziquone has been investigated for the treatment of Bladder Cancer and Bladder Neoplasms.

Kategori:
Antineoplastic AgentsAzirinesHeterocyclic Compounds, Fused-Ring +2
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Apc001 DB17819
biotech

Apc001 is an aptamer developed for the treatment of osteogenesis imperfecta.

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Apc001PE DB17902
biotech

Deskripsi belum tersedia.

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APC8020 DB17228
biotech

Deskripsi belum tersedia.

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APD-209 DB18759
small molecule | CAS: 1261156-82-4

Deskripsi belum tersedia.

Target Protein:
Beta-2 adrenergic receptor
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APD668 DB05166
small molecule

APD668 is a novel, highly potent and orally active glucose-dependent insulinotropic receptor (GDIR) agonist intended to more efficiently stimulate insulin release by beta cells in response to elevated blood glucose levels, and to also avoid hypoglycemia.

Target Protein:
Glucose-dependent insulinotropic receptor
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APD791 DB05227
small molecule

APD791 is an oral anti-thrombotic drug candidate being evaluated in a Phase 1 clinical trial by Arena. APD791 is intended to lower the risk of arterial thrombosis by reducing the amplification of platelet aggregation, arterial constriction and intimal hyperpl…

Kategori:
Acids, CarbocyclicAmidesAntidepressive Agents +8
Target Protein:
5-hydroxytryptamine receptor 2A
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Apelin DB18909
biotech | CAS: 372170-33-7

Apelin is under investigation in clinical trial NCT03449251 (A Series of Pilot Studies to Evaluate the Haemodynamic and Metabolic Effects of Apelin and Relaxin).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +1
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APG-1387 DB16095
small molecule | CAS: 1570231-89-8

APG-1387 is under investigation in clinical trial NCT04568265 (A Clinical Study of APG-1387 in Combination With Entecavir in Patients With Chronic Hepatitis B).

Kategori:
AmidesSulfonesSulfur Compounds
Target Protein:
E3 ubiquitin-protein ligase XIAPBaculoviral IAP repeat-containing protein 2Baculoviral IAP repeat-containing protein 3 +3
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APG-157 DB18683
small molecule

APG-157 consists of zinflavonoids being investigated for the treatment of cancers.

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Aphidicolin DB17742
small molecule | CAS: 38966-21-1

Aphidicolin is an antimitotic and antiviral metabolite of the mould _Cephalosporium aphidicola_. It inhibits DNA polymerase alpha and blocks DNA replication.[A259157, A259162]

Kategori:
Anti-Infective AgentsAntiviral AgentsDiterpenes +2
Target Protein:
DNA polymerase catalytic subunit
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Apigenin DB07352
small molecule | CAS: 520-36-5

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavones +3
Target Protein:
Casein kinase II subunit alphaAldo-keto reductase family 1 member B1Cytochrome P450 1B1 +5
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Apinocaltamide DB16241
small molecule | CAS: 1838651-58-3

Apinocaltamide is under investigation in clinical trial NCT03239691 (A Study to Evaluate the Effect of ACT-709478 in Photosensitive Epilepsy Patients).

Kategori:
AcetatesAcids, AcyclicAmides +5
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Apiospora montagnei Approved DB10844
biotech

Apiospora montagnei is a fungus which can provoke allergic reactions. Apiospora montagnei extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Fungal Allergenic Extract
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Apis mellifera venom Approved DB10955
biotech

Apis mellifera venom is an extract of Apis mellifera venom. Apis mellifera venom is used in allergenic testing.

Kategori:
Allergenic ExtractsBee and Wasp VenomCell-mediated Immunity +4
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Apitegromab DB16096
biotech | CAS: 2278276-46-1

Apitegromab is under investigation in clinical trial NCT03921528 (An Active Treatment Study of SRK-015 in Patients With Type 2 or Type 3 Spinal Muscular Atrophy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Apitolisib DB12180
small molecule | CAS: 1032754-93-0

Apitolisib has been used in trials studying the treatment of Solid Cancers, Breast Cancer, Prostate Cancer, Renal Cell Carcinoma, and Endometrial Carcinoma, among others.

Kategori:
Phosphatidylinositol 3-Kinases, antagonists & inhibitors
Target Protein:
Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
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Apixaban Approved DB06605
small molecule | CAS: 503612-47-3

Apixaban is an oral, direct, and highly selective factor Xa (FXa) inhibitor of both free and bound FXa, as well as prothrombinase, independent of antithrombin III for the prevention and treatment of thromboembolic diseases[Label,A6897]. It is marketed under t…

Kategori:
AnticoagulantsAntithrombinsBCRP/ABCG2 Substrates +17
Target Protein:
Coagulation factor X
Waktu Paruh12.7±8.55h[Label,A1…
Vol. DistribusiApproximately 21L[L…
Klirens3.3L/h[Label] thoug…
Genetik -
APL-030 DB18735
small molecule

APL-030 is a orally-active small molecule inhibitor of GCN2.

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APL-502 DB17473
biotech | CAS: 2303884-58-2

APL 502 is a humanised immunoglobulin G1 (IgG1) monoclonal antibody targeting the programmed cell death-1 ligand-1 (PD-L1).

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APL-9 DB16460
small molecule

APL-9 is an investigational drug intended to centrally control the complement cascade at C3, potentially treating various diseases caused by excessive or uncontrolled complement activation. It shares the same mechanism of action as Apellis’ lead compound, peg…

Kategori:
Experimental Unapproved Treatments for COVID-19
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Aplaviroc DB06497
small molecule | CAS: 461443-59-4

A spiro-diketo-piperazine; a potent noncompetitive allosteric antagonist of the CCR5 receptor with concomitantly potent antiviral effects for HIV-1.

Kategori:
Acids, CarbocyclicAnti-HIV AgentsAnti-Infective Agents +6
Target Protein:
C-C chemokine receptor type 5
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Aplindore DB06620
small molecule | CAS: 189681-70-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
D(2) dopamine receptor
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Aplyronine A DB04629
small molecule

Deskripsi belum tersedia.

Kategori:
Actins, antagonists & inhibitorsLactonesPolyketides
Target Protein:
Actin, alpha skeletal muscle
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Apocynin DB12618
small molecule | CAS: 498-02-2

Acetovanillone has been used in trials studying the treatment of Bronchial Asthma and Chronic Obstructive Pulmonary Disease.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +9
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Apolizumab DB06467
biotech | CAS: 267227-08-7

Apolizumab is a humanized monoclonal antibody that is being studied as a treatment for hematologic cancers.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Apomab DB15022
biotech | CAS: 1108170-71-3

Apomab is under investigation in clinical trial NCT00851136 (A Study of PRO95780 Administered in Combination With the FOLFOX Regimen and Bevacizumab in Patients With Previously Untreated, Locally Advanced, Recurrent, and Metastatic Colorectal Cancer (APM4566g…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Apomine DB12276
small molecule | CAS: 126411-13-0

Apomine has been used in trials studying the treatment of Osteoporosis and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
OrganophosphonatesOrganophosphorus Compounds
Target Protein:
Bile acid receptor
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Apomorphine Approved DB00714
small molecule | CAS: 58-00-4

Apomorphine is a non-ergoline dopamine D2 agonist indicated to treat hypomobility associated with Parkinson's. It was first synthesized in 1845 and first used in Parkinson's disease in 1884.[A203618] Apomorphine has also been investigated as an emetic, a seda…

Kategori:
AlkaloidsAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +32
Target Protein:
D(4) dopamine receptorD(2) dopamine receptorD(3) dopamine receptor +11
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensThe clearance of a …
Genetik -
small molecule | CAS: 42337-33-7

Deskripsi belum tersedia.

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Apoptone DB06307
small molecule | CAS: 183387-50-0

Deskripsi belum tersedia.

Kategori:
AndrostanesFused-Ring CompoundsSteroids
Target Protein:
Apoptosis regulator Bcl-2
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APPD DB18603
small molecule | CAS: 2364414-26-4

Deskripsi belum tersedia.

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Apple Approved DB10501
biotech

Apple allergenic extract is used in allergenic testing.

Kategori:
Increased Histamine ReleaseNon-Standardized Food Allergenic Extract
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biotech

Deskripsi belum tersedia.

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Apple fruit oil DB14355
biotech

Apple fruit oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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APR-2020 DB18497
biotech

APR-2020 is a CD34+ cells that have been transduced in vitro with a lentiviral vector carrying a codon-optimized sequence for expressing the wild type RPS19 protein

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