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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
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15718 (100.0%)

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Halaman 70 / 315
Bebtelovimab DB16755
biotech | CAS: 2578319-11-4

Bebtelovimab (LY-COV1404, LY-3853113) is a human monoclonal antibody approved for emergency use in the treatment of COVID-19. It binds to a portion of the SARS-CoV-2 spike (S) protein's receptor-binding domain, thereby preventing spike protein interaction wit…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesApproved Treatments for COVID-19 +6
Target Protein:
Spike glycoprotein
Waktu ParuhFollowing a single …
Vol. DistribusiAt steady-state, th…
KlirensFollowing a single …
Genetik -
Becaplermin Approved DB00102
biotech | CAS: 165101-51-9

Becaplermin is produced by recombinant DNA technology by insertion of the gene for the B chain of platelet derived growth factor (PDGF) into the yeast, Saccharomyces cerevisiae. Becaplermin has a molecular weight of approximately 25 KD and is a homodimer comp…

Kategori:
AcidsAcids, NoncarboxylicAlimentary Tract and Metabolism +24
Target Protein:
Platelet-derived growth factor receptor betaPlatelet-derived growth factor receptor alphaAlpha-2-macroglobulin
Waktu Paruh-
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Becatecarin DB06362
small molecule | CAS: 119673-08-4

Becatecarin is a derivative of [rebeccamycin].

Kategori:
CarbohydratesGlycosidesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
DNA topoisomerase 1DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
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Beclabuvir DB12225
small molecule | CAS: 958002-33-0

Beclabuvir has been used in trials studying the treatment of Hepatitis C, Chronic.

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +3
Target Protein:
Genome polyprotein
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Beclamide DB09011
small molecule | CAS: 501-68-8

Beclamide (N-benzyl-B-chloropropionamide) is a no longer used drug that possesses anticonvulsant and sedative activity. It was studied in the 1950s for generalised tonic-clonic seizures but was not effective for absence seizures.

Kategori:
Acids, AcyclicAnticonvulsantsCentral Nervous System Depressants +4
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Beclanorsen DB05606
small molecule | CAS: 1072859-54-1

Deskripsi belum tersedia.

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small molecule | CAS: 5534-18-9

An ester of beclomethasone.

Kategori:
Adrenal Cortex HormonesCorticosteroidsFused-Ring Compounds +5
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Beclomethasone dipropionate Approved DB00394
small molecule | CAS: 5534-09-8

Beclomethasone dipropionate is a second-generation[A179842] synthetic corticosteroid and diester of beclomethasone, which is structurally similar to [dexamethasone].[L6871] It is a prodrug of an active metabolite beclomethasone 17-monopropionate (17-BMP)[A179…

Kategori:
Adrenal Cortex HormonesAdrenalsAgents to Treat Airway Disease +40
Target Protein:
Glucocorticoid receptor
Waktu ParuhFollowing intraveno…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Becocalcidiol DB04891
small molecule | CAS: 524067-21-8

Becocalcidiol is a vitamin D(3) analogue which has not caused hypercalcaemia or significant irritation in preclinical trials.

Kategori:
CholestanesCholestenesFused-Ring Compounds +8
Target Protein:
Mediator of RNA polymerase II transcription subunit 1Vitamin D3 receptor
Waktu Paruh-
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Becotatug DB19069
biotech | CAS: 2648260-93-7

Becotatug is under investigation in clinical trial NCT06380348 (JMT101 in Combination With Osimertinib, Versus Cisplatin-pemetrexed in Participants With Locally Advanced or Metastatic Non-small Cell Lung Cancer (NSCLC) Characterized by Epithermal Growth Facto…

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Bectumomab DB04962
biotech | CAS: 158318-63-9

Bectumomab (marketed under the trade name LymphoScan®) is a mouse monoclonal antibody and which it's used to treat non-Hodgkin's lymphoma. It has a radioisotope, technetium (99m TC) which it's added.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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Bedaquiline Approved DB08903
small molecule | CAS: 843663-66-1

Bedaquiline is a bactericidal antimycobacterial drug belonging to the class of diarylquinoline. The quinolinic central heterocyclic nucleus with alcohol and amine side chains is responsible for bedaquiline-mediated antimycobacterial activity.[A261866] Althoug…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiinfectives for Systemic Use +10
Target Protein:
ATP synthase subunit c
Waktu ParuhThe mean terminal e…
Vol. DistribusiThe volume of distr…
KlirensBedaquiline has a l…
Genetik -
Bedoradrine DB05590
small molecule | CAS: 194785-19-8

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicAmides
Target Protein:
Beta-2 adrenergic receptor
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Bee pollen DB16612
biotech

Deskripsi belum tersedia.

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Beef Approved DB10509
biotech

Beef allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Beef liver Approved DB14694
biotech

Beef liver allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Beeswax Approved DB11600
biotech | CAS: 8012-89-3

The wax obtained from the honeycomb of the bee. It consists primarily of myricyl palmitate, cerotic acid esters and some high-carbon paraffins. Beeswax is used as a stiffening agent in ointments and creams, and enables water to be incorporated to produce wate…

Kategori:
BeesLipids
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Beet Approved DB10640
biotech

Beet allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
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Befiradol DB19033
small molecule | CAS: 208110-64-9

Befiradol is under investigation in clinical trial NCT05148884 (Study to Assess the Safety, Tolerability and Preliminary Efficacy of NLX-112 Versus Placebo in L-dopa-induced Dyskinesia).

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsNeurotransmitter Agents +3
Target Protein:
5-hydroxytryptamine receptor 1A
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Befotertinib DB18844
small molecule | CAS: 1835667-63-4

Befotertinib is under investigation in clinical trial NCT05007938 (Befotertinib and Icotinib in Treatment-naive Patients With Advanced Egfr-mutant Lung Cancer).

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Befovacimab DB16188
biotech | CAS: 2156634-62-5

Deskripsi belum tersedia.

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Befunolol DB09013
small molecule | CAS: 39552-01-7

Befunolol is a beta blocker introduced in 1983 by Kakenyaku Kakko. It is currently in experimental status, and is being tested for the management of open angle glaucoma.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic Antagonists +14
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
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Begacestat DB12263
small molecule | CAS: 769169-27-9

Begacestat has been used in trials studying the treatment and basic science of Alzheimer Disease.

Kategori:
AmidesAmyloid Precursor Protein SecretasesEnzyme Inhibitors +3
Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +2
Waktu Paruh-
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Genetik -
Begelomab DB13241
biotech | CAS: 1403744-56-8

Begelomab is a murine monoclonal antibody against CD26.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntineoplastic and Immunomodulating Agents +6
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Beinaglutide DB15072
biotech | CAS: 123475-27-4

Beinaglutide is under investigation in clinical trial NCT03829891 (Study for Beinaglutide Versus Glargine Therapy in Glycemic Variability of Type 2 Diabetes Mellitus).

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +8
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Bekanamycin DB13673
small molecule | CAS: 4696-76-8

Deskripsi belum tersedia.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +9
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biotech

Deskripsi belum tersedia.

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biotech

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biotech

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Belantamab mafodotin Approved DB15719
biotech | CAS: 2050232-20-5

Belantamab mafodotin, or GSK2857916, is an afucosylated monoclonal antibody that targets B cell maturation antigen conjugated to the microtubule disrupter monomethyl auristatin-F (MMAF).[A216756] Belantamab mafodotin was granted FDA accelerated approval on…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Tumor necrosis factor receptor superfamily member 17
Waktu ParuhThe terminal half l…
Vol. DistribusiThe mean steady sta…
KlirensThe clearance of be…
Genetik -
Belapectin DB15125
small molecule | CAS: 1980787-47-0

Belapectin is under investigation in clinical trial NCT02575404 (GR-MD-02 Plus Pembrolizumab in Melanoma, Non-small Cell Lung Cancer, and Squamous Cell Head and Neck Cancer Patients).

Kategori:
Biological ProductsBiopolymersCarbohydrates +6
Waktu Paruh-
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Belatacept Approved DB06681
biotech | CAS: 706808-37-9

Belatacept is a soluble fusion protein, which links the extracellular domain of human cytotoxic T-lymphocyte-associated antigen 4 (CTLA-4) to the modified Fc (hinge, CH2, and CH3 domains) portion of human immunoglobulin G1 (IgG1). Structurally, abatacept is a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents, Immunological +15
Target Protein:
T-lymphocyte activation antigen CD86T-lymphocyte activation antigen CD80
Waktu ParuhMean terminal elimi…
Vol. DistribusiVd, steady state, t…
KlirensIncreased body weig…
Genetik -
Belcesiran DB18226
biotech | CAS: 2375562-54-0

Deskripsi belum tersedia.

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Belimumab Approved DB08879
biotech | CAS: 356547-88-1

Belimumab is a fully human recombinant IgG1? monoclonal antibody that inhibits soluble human B lymphocyte stimulator protein (BLyS, also referred to as BAFF and TNFSF13B), a B cell survival factor.[L42630] BLyS levels are often elevated in immunodeficient and…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Tumor necrosis factor ligand superfamily member 13B
Waktu ParuhFollowing administr…
Vol. DistribusiFollowing administr…
KlirensFollowing administr…
Genetik -
Belinostat Approved DB05015
small molecule | CAS: 866323-14-0

Belinostat is a novel agent that inhibits the enzyme histone deacetylase (HDAC) with a sulfonamide-hydroxamide structure. It was developed as an orphan drug to target hematological malignancies and solid tumors by TopoTarget. The safety and efficacy of belino…

Kategori:
AmidesAminesAntineoplastic Agents +31
Target Protein:
Histone deacetylase
Gen Terkait:
UGT1A1 UGT1A1
Waktu ParuhDisplays a three-co…
Vol. DistribusiThe volume of distr…
Klirens1240 mL/min
Genetik 2 Varian
Belladonna Approved DB13913
biotech

Belladonna, also known as atropa belladonna or deadly nightshade, is a perennial herbaceous plant in the nightshade family _Solanaceae_. Its roots, leaves and fruits contain [DB00424], [DB00747], and mostly, [DB00572]. These alkaloids are naturally-occurring …

Kategori:
Anticholinergic AgentsAntimuscarinics AntispasmodicsMuscarinic Antagonists
Waktu ParuhFor pharmacokinetic…
Vol. DistribusiFor pharmacokinetic…
KlirensFor pharmacokinetic…
Genetik -
Beloranib DB12671
small molecule | CAS: 251111-30-5

Beloranib has been used in trials studying the treatment of Obesity, Over-weight, Type 2 Diabetes, Craniopharyngioma, and Hypothalamic Injury, among others.

Kategori:
Acids, CarbocyclicAngiogenesis InhibitorsAngiogenesis Modulating Agents +7
Target Protein:
Methionine aminopeptidase 2
Waktu Paruh-
Vol. Distribusi-
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Belotecan DB12459
small molecule | CAS: 256411-32-2

Belotecan has been investigated for the treatment of Epithelial Ovarian Cancer.

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +4
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
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Belrestotug DB19066
biotech | CAS: 2574438-65-4

Belrestotug is under investigation in clinical trial NCT05565378 (A Platform Study of Novel Immunotherapy Combinations in Participants With Previously Untreated, Advanced/metastatic Non-small-cell Lung Cancer).

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Beludavimab DB18952
biotech | CAS: 2423016-74-2

Beludavimab is under investigation in clinical trial NCT04746183 (AGILE (Early Phase Platform Trial for COVID-19)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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Belumosudil Approved DB16703
small molecule | CAS: 911417-87-3

Belumosudil is used in the treatment of chronic graft-versus-host disease (GVHD) and has been investigated for the treatment of pulmonary arterial hypertension.[A236634] It is an inhibitor of rho-associated coiled-coil-containing protein kinases (ROCK), with …

Kategori:
AcetatesAcids, AcyclicAmides +25
Target Protein:
Rho-associated protein kinase 2Rho-associated protein kinase 1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiFollowing a single …
KlirensThe mean clearance …
Genetik -
Belvarafenib DB17568
small molecule | CAS: 1446113-23-0

Deskripsi belum tersedia.

Target Protein:
RAF proto-oncogene serine/threonine-protein kinase
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biotech | CAS: 2390462-37-8

Deskripsi belum tersedia.

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Belzutifan Approved DB15463
small molecule | CAS: 1672668-24-4

Belzutifan is an inhibitor of hypoxia-inducible factor 2? (HIF-2?) used in the treatment of von Hippel-Lindau (VHL) disease-associated cancers.[L35995] The HIF-2? protein was first identified in the 1990s by researchers at UT Southwestern Medical Center as a …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C19 Substrates +10
Target Protein:
Endothelial PAS domain-containing protein 1
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
Bemarituzumab DB16105
biotech | CAS: 1952272-74-0

Bemarituzumab is under investigation in clinical trial NCT03694522 (A Study of Bemarituzumab (FPA144) Combined With Modified FOLFOX6 (Mfolfox6) in Gastric/gastroesophageal Junction Cancer (FIGHT)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
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Bemcentinib DB12411
small molecule | CAS: 1037624-75-1

Bemcentinib has been investigated for the treatment of Non-Small Cell Lung Cancer.

Target Protein:
Spike glycoproteinTyrosine-protein kinase receptor UFO
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Bemegride DB13740
small molecule | CAS: 64-65-3

Bemegride is a CNS stimulant that is used to induce convulsions in experimental animals. It has also been used as a respiratory stimulant and in the treatment of barbiturate overdose.

Kategori:
Central Nervous System AgentsCentral Nervous System StimulantsConvulsants +3
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biotech | CAS: 2766038-73-5

Deskripsi belum tersedia.

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Bemiparin Approved DB09258
small molecule | CAS: 91449-79-5

Bemiparin is an antithrombotic and belongs to the group of drugs known as the low molecular weight heparins (LMWH). Like semuloparin, bemiparin is classified as an ultra-LMH because of its low mean molecular mass of 3600 daltons, which is a unique property of…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +6
Target Protein:
Coagulation factor XAntithrombin-IIIHeparin cofactor 2
Waktu ParuhBemiparin, when adm…
Vol. Distribusi5.1 L [A32018].
KlirensElimination occurs …
Genetik -
Bemnifosbuvir DB19050
small molecule | CAS: 1998705-64-8

Bemnifosbuvir is under investigation in clinical trial NCT05629962 (SUNRISE-3: Efficacy and Safety of Bemnifosbuvir in High-risk Outpatients With COVID-19).

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