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807

Total database: 17430
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608 (75.3%)
Target
525 (65.1%)
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15 (1.9%)
Referensi
807 (100.0%)

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Hasil Pencarian (807)

Halaman 7 / 17
Desipramine Approved DB01151
small molecule | CAS: 50-47-5

Desipramine hydrochloride is a dibenzazepine-derivative tricyclic antidepressant (TCA). TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individuals, de…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +52
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A +14
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +4
Waktu Paruh7-60+ hours; 70% el…
Vol. Distribusi-
Klirens-
Genetik 7 Varian
Desmeninol DB15832
small molecule | CAS: 583-91-5

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desmoteplase DB04925
biotech | CAS: 145137-38-8

Desmoteplase is a chemical in the saliva of vampire bats. It activates plasminogen to the serine protease, plasmin. Plasmin acts by breaking down fibrin blood clots. When a vampire bat bites its victim, it secretes an enzyme that prevents the blood from clott…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBlood Proteins +13
Target Protein:
Plasminogen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desoximetasone Approved DB00547
small molecule | CAS: 382-67-2

A topical anti-inflammatory glucocorticoid used in dermatoses, skin allergies, psoriasis, etc.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroid Hormone Receptor Agonists +14
Target Protein:
Estrogen-related receptor gammaGlucocorticoid receptorSteroid hormone receptor ERR2 +1
Waktu ParuhThe half-life of th…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1079043-55-2

Deudextromethorphan is under investigation in clinical trial NCT02153502 (Efficacy, Safety, and Tolerability Study of AVP-786 as an Adjunctive Therapy in Patients With Major Depressive Disorder With an Inadequate Response to Antidepressant Treatment).

Target Protein:
Sodium-dependent serotonin transporterSigma non-opioid intracellular receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2143580-11-2

Devafidugene civaparvovec is an investigational _in vivo_ genome editing product. It uses proprietary zinc finger nucleases (ZFN) that insert a functional copy of the alpha-L-iduronidase (IDUA) enzyme. Developed by Sangamo Therapeutics, Inc., devafidugene civ…

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexamethasone Approved DB01234
small molecule | CAS: 50-02-2

Dexamethasone, or MK-125, is a corticosteroid fluorinated at position 9 used to treat endocrine, rheumatic, collagen, dermatologic, allergic, ophthalmic, gastrointestinal, respiratory, hematologic, neoplastic, edematous, and other conditions.[L10701] Develope…

Kategori:
Adrenal Cortex HormonesAdrenalsAgents Causing Muscle Toxicity +74
Target Protein:
Glucocorticoid receptorNuclear receptor subfamily 0 group B member 1Annexin A1 +2
Waktu ParuhThe mean terminal h…
Vol. DistribusiA 1.5mg oral dose o…
KlirensA 20mg oral tablet …
Genetik -
Dexamethasone acetate Approved DB14649
small molecule | CAS: 1177-87-3

Commonly known as decadron, dexamethasone acetate is a glucocorticosteroid previously marketed in the USA for the treatment of inflammatory respiratory, allergic, autoimmune, and other conditions.[T797,L10695,L14348] Developed in 1957, dexamethasone is struct…

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsBCRP/ABCG2 Inhibitors +38
Target Protein:
Glucocorticoid receptorAnnexin A1Nitric oxide synthase, inducible +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14899-36-6

Dexamethasone palmitate is under investigation in clinical trial NCT05693467 (Preemptive Co-infiltration of Dexamethasone Palmitate With Ropivacaine for Postoperative Pain in Major Spinal Surgery).

Kategori:
Fused-Ring CompoundsPregnadienesPregnadienetriols +3
Target Protein:
Steroid hormone receptor ERR1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexmedetomidine Approved DB00633
small molecule | CAS: 113775-47-6

An agonist of receptors, adrenergic alpha-2 that is used in veterinary medicine for its analgesic and sedative properties. It is the racemate of dexmedetomidine.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +28
Target Protein:
Alpha-2A adrenergic receptor
Waktu Paruh2 hours
Vol. Distribusi* 118 L
Klirens* 39 L/h [Healthy v…
Genetik -
Diamorphine Approved DB01452
small molecule | CAS: 561-27-3

Diamorphine (heroin) is a narcotic analgesic that may be habit-forming. It is a controlled substance (opium derivative) listed in the U.S. Code of Federal Regulations, Title 21 Parts 329.1, 1308.11 (1987). Sale is forbidden in the United States by Federal sta…

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +16
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor +1
Waktu ParuhIn humans, administ…
Vol. DistribusiData regarding the …
KlirensSome studies have d…
Genetik -
Dienestrol Approved DB00890
small molecule | CAS: 13029-44-2

Dienestrol is a synthetic, non-steroidal estrogen. It is an estrogen receptor agonist. Estrogens work partly by increasing a normal clear discharge from the vagina and making the vulva and urethra healthy. Using or applying an estrogen relieves or lessens: dr…

Kategori:
Benzene DerivativesBenzyl CompoundsBenzylidene Compounds +12
Target Protein:
Estrogen receptorSex hormone-binding globulin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dienogest Approved DB09123
small molecule | CAS: 65928-58-7

Dienogest is an orally-active semisynthetic progestogen which also possesses the properties of 17?-hydroxyprogesterone. It is a derivative of 19-nortestosterone and has antiandrogenic properties. It is primarily used as a contraceptive in combination with eth…

Kategori:
Adrenal Cortex HormonesAntineoplastic AgentsAntineoplastic Agents, Hormonal +29
Target Protein:
Progesterone receptorAndrogen receptor
Waktu ParuhElimination half-li…
Vol. DistribusiThe apparent volume…
KlirensThe metabolic clear…
Genetik -
Diethylpropion Approved DB00937
small molecule | CAS: 90-84-6

A appetite depressant considered to produce less central nervous system disturbance than most drugs in this therapeutic category. It is also considered to be among the safest for patients with hypertension. (From AMA Drug Evaluations Annual, 1994, p2290)

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAlimentary Tract and Metabolism +14
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterSodium-dependent dopamine transporter
Waktu ParuhUsing a phosphoresc…
Vol. Distribusi-
Klirens-
Genetik -
Dihydro-alpha-ergocryptine Approved DB11274
small molecule | CAS: 25447-66-9

Alpha-dihydroergocryptine is usually referred to the mixture of the alpha and beta dihydroergocryptine. These two compounds are differentiated in the position of a methyl group. This structural difference is due to a proteinogenic amino acid replacement from …

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 Substrates
Target Protein:
5-hydroxytryptamine receptor 75-hydroxytryptamine receptor 2BD(2) dopamine receptor +2
Waktu ParuhAlpha-dihydroergocr…
Vol. DistribusiIn preclinical stud…
KlirensIn preclinical stud…
Genetik -
Dihydroergocornine Approved DB11273
small molecule | CAS: 25447-65-8

Dihydroergocornine is one of the dihydrogenated ergot compounds that present very large hypotensive effects.[A32962] It is an artificial derivative of the crude extract of ergot and later purified, ergocornine.[A32964] The formation of dihydroergocornine impl…

Kategori:
Agents that produce hypertensionAlkaloidsCytochrome P-450 CYP3A Substrates +10
Target Protein:
Serotonin ReceptorsBeta adrenergic receptorAlpha adrenergic receptor
Waktu ParuhTo know more about …
Vol. DistribusiTo know more about …
KlirensNo pharmacokinetic …
Genetik -
Dihydroergotamine Approved DB00320
small molecule | CAS: 511-12-6

A 9,10alpha-dihydro derivative of [ergotamine]. Dihydroergotamine is used as an abortive therapy for migraines.[L38469] Its use has largely been supplanted by triptans in current therapy due to the class's greater selectivity and more favourable side effect p…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +37
Target Protein:
5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1F +13
Waktu ParuhDHE exhibits a biph…
Vol. DistribusiDHE has a steady-st…
KlirensThe total clearance…
Genetik -
Dihydrostreptomycin Approved DB11512
small molecule | CAS: 128-46-1

Dihydrostreptomycin is an aminoglycoside antibiotic. In humans, the use of dihydrostreptomycin has been associated with ototoxicity. The FDA withdrew its approval for the use of all drug products containing dihydrostreptomycin sulfate.[L43942]

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dimepheptanol DB19094
small molecule | CAS: 545-90-4

Dimepheptanol is under investigation in clinical trial NCT00218127 (Treatment of Opioid/heroin Dependence: Comparison of Three Medication Dosing Regimens).

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +5
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dinoprost tromethamine Approved DB01160
small molecule | CAS: 38562-01-5

The tromethamine (THAM) salt of the naturally occurring prostaglandin F2 alpha, dinoprost tromethamine occurs as a white to off-white, very hygroscopic, crystalline powder. Dinoprost tromethamine may also be known as dinoprost trometamol, PGF2 alpha THAM, or …

Kategori:
Abortifacient AgentsAbortifacient Agents, NonsteroidalAngiography +11
Target Protein:
Prostaglandin F2-alpha receptorProstacyclin receptor
Waktu ParuhThe half-life of di…
Vol. Distribusi-
Klirens-
Genetik -
Dinoprostone Approved DB00917
small molecule | CAS: 363-24-6

Dinoprostone is a naturally occurring prostaglandin E2 (PGE2). It has important effects in labour. It also stimulates osteoblasts to release factors which stimualtes bone resorption by osteoclasts. As a prescription drug it is used as a vaginal suppository, t…

Kategori:
AutacoidsBiological FactorsDinoprostone, antagonists & inhibitors +19
Target Protein:
Prostaglandin F2-alpha receptorProstaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtype +3
Waktu ParuhLess than 5 minutes.
Vol. Distribusi-
Klirens-
Genetik -
Diphenidol Approved DB01231
small molecule | CAS: 972-02-1

Diphenidol is an antiemetic agent used in the treatment of vomiting and vertigo. Diphenidol overdose may result in serious toxicity in children.

Kategori:
Agents producing tachycardiaAnticholinergic AgentsAntiemetics +6
Target Protein:
Muscarinic acetylcholine receptor M4Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M1 +1
Waktu Paruh4 hours
Vol. Distribusi-
Klirens-
Genetik -
Disomotide DB17469
biotech | CAS: 181477-43-0

Disomotide is a synthetic peptide cancer vaccine.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Disufenton DB17298
small molecule | CAS: 168021-77-0

Deskripsi belum tersedia.

Kategori:
AntioxidantsArylsulfonatesArylsulfonic Acids +9
Target Protein:
Extracellular sulfatase Sulf-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-alpha tocopheryl acetate Approved DB14477
small molecule | CAS: 52225-20-4

Deskripsi belum tersedia.

Kategori:
Vitamin EVitaminsVitamins (Fat Soluble)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-alpha-Tocopherol Approved DB14476
small molecule | CAS: 10191-41-0

Deskripsi belum tersedia.

Kategori:
Vitamin EVitaminsVitamins (Fat Soluble)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Doconexent Approved DB03756
small molecule | CAS: 6217-54-5

A mixture of fish oil and primrose oil, doconexent is used as a high-docosahexaenoic acid (DHA) supplement. DHA is a 22 carbon chain with 6 cis double bonds with anti-inflammatory effects. It can be biosythesized from alpha-linolenic acid or commercially manu…

Kategori:
Cytochrome P-450 CYP2C9 InhibitorsCytochrome P-450 CYP2C9 Inhibitors (strength unknown)Cytochrome P-450 CYP2C9 Substrates +11
Target Protein:
Peroxisome proliferator-activated receptor alphaProstaglandin G/H synthase 1Prostaglandin G/H synthase 2 +6
Waktu ParuhApproximately 20 ho…
Vol. DistribusiDHA is the most abu…
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Retinoic acid receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dornase alfa Approved DB00003
biotech | CAS: 143831-71-4

Dornase alfa is a biosynthetic form of human deoxyribunuclease I (DNase I) enzyme. It is produced in genetically modified Chinese hamster ovary (CHO) cells using recombinant DNA technology. The 260-amino acid sequence of dornase alfa is identical to the endog…

Kategori:
Amino Acids, Peptides, and ProteinsCough and Cold PreparationsDecreased Respiratory Secretion Viscosity +10
Target Protein:
Deoxyribonuclease-1
Waktu Paruh-
Vol. DistribusiIn studies in rats …
KlirensStudies in rats ind…
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Doxazosin Approved DB00590
small molecule | CAS: 74191-85-8

Doxazosin is an alpha-1 antagonist used for the treatment of benign prostatic hypertrophy (BPH) symptoms and hypertension. Other members of this drug class include [Prazosin], [Terazosin], [Tamsulosin], and [Alfuzosin].[A180661] Because of its long-lasting e…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +22
Target Protein:
Alpha-1A adrenergic receptorAlpha-1D adrenergic receptorHERG human cardiac K+ channel +1
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of do…
Genetik -
Doxofylline DB09273
small molecule | CAS: 69975-86-6

Doxofylline is a methylxanthine derivative with the presence of a dioxolane group in position 7. As a drug used in the treatment of asthma, doxofylline has shown similar efficacy to theophylline but with significantly fewer side effects in animal and human st…

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +21
Target Protein:
Beta-2 adrenergic receptorcGMP-dependent 3',5'-cyclic phosphodiesteraseAdenosine receptor A2a
Waktu ParuhFollowing administr…
Vol. DistribusiDoxofylline demonst…
KlirensFollowing oral admi…
Genetik -
Doxycycline Approved DB00254
small molecule | CAS: 564-25-0

Doxycycline is a broad-spectrum antibiotic synthetically derived from [oxytetracycline].[L42880] It is a second-generation tetracycline that was first discovered in 1967.[A19429] Second-generation tetracyclines exhibit lesser toxicity than first-generation te…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAnti-Bacterial Agents +17
Target Protein:
30S ribosomal protein
Waktu ParuhThere is limited in…
Vol. DistribusiThere is limited in…
KlirensPopulation pharmaco…
Genetik -
Doxylamine Approved DB00366
small molecule | CAS: 469-21-6

Histamine H1 antagonist with pronounced sedative properties. It is used in allergies and as an antitussive, antiemetic, and hypnotic. Doxylamine has also been administered in veterinary applications and was formerly used in parkinsonism.

Kategori:
Agents producing tachycardiaAminoalkyl EthersAnticholinergic Agents +17
Target Protein:
Histamine H1 receptorNuclear receptor subfamily 1 group I member 3Muscarinic acetylcholine receptor
Waktu Paruh10 hours
Vol. Distribusi-
Klirens-
Genetik -
DPI-221 DB06121
small molecule | CAS: 519058-15-2

DPI-221 is an investigational drug and a selective agonist for the ?-opioid receptor.

Kategori:
Benzene DerivativesReceptors, Opioid, delta, agonists
Target Protein:
Delta-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Drostanolone DB00858
small molecule | CAS: 58-19-5

Drostanolone (also known as dromostanolone) is a potent synthetic androgenic anabolic steroid similar to testosterone. Drostanolone is indicated in postmenopausal women with recurrent breast cancer, in a combined hormone therapy.

Kategori:
AndrostanesFused-Ring CompoundsSteroids
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dupilumab Approved DB12159
biotech | CAS: 1190264-60-8

Dupilumab is a fully human monoclonal antibody of the immunoglobulin G4 subclass that binds to the interleukin-4 (IL-4) receptor, inhibiting the receptor signaling pathways.[A180478] As an interleukin-4 receptor alpha antagonist, dupilumab inhibits the signal…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmino Acids, Peptides, and ProteinsAnti-Asthmatic Agents +13
Target Protein:
Interleukin-4 receptor subunit alphaInterleukin-13Interleukin-4
Waktu ParuhThere is limited hu…
Vol. DistribusiThe estimated volum…
KlirensThere is limited da…
Genetik -
Duvoglustat DB03206
small molecule | CAS: 19130-96-2

An alpha-glucosidase inhibitor with antiviral action. Derivatives of deoxynojirimycin may have anti-HIV activity.

Kategori:
AlkaloidsAmino SugarsAnti-Infective Agents +7
Target Protein:
Maltase-glucoamylaseLysosomal alpha-glucosidaseNeutral alpha-glucosidase AB +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Efalizumab Approved DB00095
biotech | CAS: 214745-43-4

Humanized IgG1 kappa isotype monoclonal antibody that binds to human CD11a. Efalizumab has a molecular weight of approximately 150 kilodaltons and is produced in a Chinese hamster ovary mammalian cell expression system in a nutrient medium containing the anti…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Integrin alpha-XIntegrin alpha-L
Waktu Paruh5 days
Vol. Distribusi-
Klirens-
Genetik -
Efinaconazole Approved DB09040
small molecule | CAS: 164650-44-6

Efinaconazole is a 14 alpha-demethylase inhibitor indicated in the treatment of fungal infection of the nail, known as onychomycosis. It was approved for use in Canada and the USA in 2014 and is marketed by Valeant Pharmaceuticals North America LLC under the …

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +4
Target Protein:
Lanosterol 14-alpha demethylaseLanosterol 14-alpha demethylase
Waktu Paruh29.9 hours in healt…
Vol. Distribusi-
Klirens-
Genetik -
Eflornithine Approved DB06243
small molecule | CAS: 70052-12-9

Eflornithine is an irreversible ornithine decarboxylase inhibitor originally developed as a treatment for human African trypanosomiasis.[A262829] Further research has also implicated ornithine decarboxylase in other conditions like facial hirsutism and cancer…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAmino AcidsAmino Acids, Basic +15
Target Protein:
Ornithine decarboxylase
Waktu ParuhThe terminal plasma…
Vol. DistribusiEflornithine volume…
KlirensThe clearance (CL/F…
Genetik -
Efocipegtrutide DB18194
biotech | CAS: 2513399-19-2

Efocipegtrutide is a long-acting, monomeric peptide triple agonist.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1800476-36-1

Eftilagimod alfa is under investigation in clinical trial NCT02614833 (IMP321 (Eftilagimod Alpha) as Adjunctive to a Standard Chemotherapy Paclitaxel Metastatic Breast Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Differentiation +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EGT-201 DB17648
biotech

EGT-201 is an adeno-associated viral vector serotype 9 (AAV9) vector-based gene therapy consisting of the alpha-N-acetyglucosaminidase (NAGLU) transgene. Developed by Esteve Pharmaceuticals, it is being investigated for Sanfilippo syndrome type B.[L45939]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elacestrant Approved DB06374
small molecule | CAS: 722533-56-4

Elacestrant is a non-steroidal small molecule and an estrogen receptor (ER) antagonist.[A256838,L44918] In January 2023, it was approved by the FDA for the treatment of ER-positive, HER2-negative, ESR1-mutated advanced or metastatic breast cancer.[L44918,L449…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Estrogen receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiElacestrant has an …
KlirensElacestrant has an …
Genetik -
Elapegademase Approved DB14712
biotech | CAS: 1709806-75-6

Elapegademase is a PEGylated recombinant adenosine deaminase. It can be defined molecularly as a genetically modified bovine adenosine deaminase with a modification in cysteine 74 for serine and with about 13 methoxy polyethylene glycol chains bound via carbo…

Kategori:
Adenosine Deaminase InhibitorsAdjuvants, ImmunologicAmino Acids, Peptides, and Proteins +12
Target Protein:
Adenosine
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Elinzanetant DB18968
small molecule | CAS: 929046-33-3

Elinzanetant is under investigation in clinical trial NCT05099159 (A Study to Learn More About How Well Elinzanetant Works and How Safe It Is for the Treatment of Vasomotor Symptoms (Hot Flashes) That Are Caused by Hormonal Changes Over 26 Weeks in Women Who …

Target Protein:
Neuromedin-K receptorSubstance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enisoprost DB19319
small molecule | CAS: 81026-63-3

Deskripsi belum tersedia.

Kategori:
Anti-Ulcer AgentsAutacoidsBiological Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Entacapone Approved DB00494
small molecule | CAS: 130929-57-6

Entacapone is a selective, reversible catechol-O-methyl transferase (COMT) inhibitor for the treatment of Parkinson's disease. It is a member of the class of nitrocatechols. When administered concomittantly with levodopa and a decarboxylase inhibitor (e.g., c…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsBenzene Derivatives +11
Target Protein:
Catechol O-methyltransferase
Waktu Paruh0.4-0.7 hour
Vol. Distribusi* 20 L
Klirens* 850 mL/min
Genetik -
Ephedrine Approved DB01364
small molecule | CAS: 299-42-3

Ephedrine was first described in western literature in 1888, as a naturally occurring component of the ephedra plant, along with [pseudoephedrine].[A193698] Ephedrine acts as both a direct and indirect sympathomimetic. It is an alpha- and beta-adrenergic rece…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-Agonists +39
Target Protein:
D(2) dopamine receptorAlpha-1A adrenergic receptorBeta-1 adrenergic receptor +2
Waktu ParuhOral ephedrine has …
Vol. DistribusiOral ephedrine has …
KlirensOral ephedrine has …
Genetik -
Menampilkan 301–350 dari 807
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