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BBIBP-CorV DB15807
biotech

BBIBP-CorV vaccine contains a SARS-CoV-2 strain inactivated inside Vero Cells. Investigation shows this vaccine induces neutralizing antibodies in several mammalian species while also showing protective efficacy with SARS-CoV-2 challenge in rhesus macaques[A2…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BBM-H803 DB17700
biotech

BBM-H803 is a recombinant adeno-associated virus (AAV) based gene therapy drug for hemophilia A developed and manufactured by Belief BioMed. It consists of an adeno-associated virus vector containing an expression cassette of the human Factor VIII transgene.

Waktu Paruh-
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Genetik -
BBV152 DB15847
biotech

BBV152 is a vaccine candidate created by the Indian Council of Medical Research (ICMR). The candidate, a whole virion inactivated SARS-CoV-2 vaccine, was developed from a well-known SARS-CoV-2 strain and a vero cell platform (CCL-81) with adjuncts of either a…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BCX10013 DB18496
small molecule

BCX10013 is a small molecule inhibitor of human complement factor D.

Waktu Paruh-
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Bebtelovimab DB16755
biotech | CAS: 2578319-11-4

Bebtelovimab (LY-COV1404, LY-3853113) is a human monoclonal antibody approved for emergency use in the treatment of COVID-19. It binds to a portion of the SARS-CoV-2 spike (S) protein's receptor-binding domain, thereby preventing spike protein interaction wit…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesApproved Treatments for COVID-19 +6
Target Protein:
Spike glycoprotein
Waktu ParuhFollowing a single …
Vol. DistribusiAt steady-state, th…
KlirensFollowing a single …
Genetik -
Becotatug DB19069
biotech | CAS: 2648260-93-7

Becotatug is under investigation in clinical trial NCT06380348 (JMT101 in Combination With Osimertinib, Versus Cisplatin-pemetrexed in Participants With Locally Advanced or Metastatic Non-small Cell Lung Cancer (NSCLC) Characterized by Epithermal Growth Facto…

Waktu Paruh-
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Genetik -
Beeswax Approved DB11600
biotech | CAS: 8012-89-3

The wax obtained from the honeycomb of the bee. It consists primarily of myricyl palmitate, cerotic acid esters and some high-carbon paraffins. Beeswax is used as a stiffening agent in ointments and creams, and enables water to be incorporated to produce wate…

Kategori:
BeesLipids
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Befovacimab DB16188
biotech | CAS: 2156634-62-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Befunolol DB09013
small molecule | CAS: 39552-01-7

Befunolol is a beta blocker introduced in 1983 by Kakenyaku Kakko. It is currently in experimental status, and is being tested for the management of open angle glaucoma.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic Antagonists +14
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Belantamab mafodotin Approved DB15719
biotech | CAS: 2050232-20-5

Belantamab mafodotin, or GSK2857916, is an afucosylated monoclonal antibody that targets B cell maturation antigen conjugated to the microtubule disrupter monomethyl auristatin-F (MMAF).[A216756] Belantamab mafodotin was granted FDA accelerated approval on…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Tumor necrosis factor receptor superfamily member 17
Waktu ParuhThe terminal half l…
Vol. DistribusiThe mean steady sta…
KlirensThe clearance of be…
Genetik -
Belatacept Approved DB06681
biotech | CAS: 706808-37-9

Belatacept is a soluble fusion protein, which links the extracellular domain of human cytotoxic T-lymphocyte-associated antigen 4 (CTLA-4) to the modified Fc (hinge, CH2, and CH3 domains) portion of human immunoglobulin G1 (IgG1). Structurally, abatacept is a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents, Immunological +15
Target Protein:
T-lymphocyte activation antigen CD86T-lymphocyte activation antigen CD80
Waktu ParuhMean terminal elimi…
Vol. DistribusiVd, steady state, t…
KlirensIncreased body weig…
Genetik -
Belimumab Approved DB08879
biotech | CAS: 356547-88-1

Belimumab is a fully human recombinant IgG1? monoclonal antibody that inhibits soluble human B lymphocyte stimulator protein (BLyS, also referred to as BAFF and TNFSF13B), a B cell survival factor.[L42630] BLyS levels are often elevated in immunodeficient and…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Tumor necrosis factor ligand superfamily member 13B
Waktu ParuhFollowing administr…
Vol. DistribusiFollowing administr…
KlirensFollowing administr…
Genetik -
Belladonna Approved DB13913
biotech

Belladonna, also known as atropa belladonna or deadly nightshade, is a perennial herbaceous plant in the nightshade family _Solanaceae_. Its roots, leaves and fruits contain [DB00424], [DB00747], and mostly, [DB00572]. These alkaloids are naturally-occurring …

Kategori:
Anticholinergic AgentsAntimuscarinics AntispasmodicsMuscarinic Antagonists
Waktu ParuhFor pharmacokinetic…
Vol. DistribusiFor pharmacokinetic…
KlirensFor pharmacokinetic…
Genetik -
Belrestotug DB19066
biotech | CAS: 2574438-65-4

Belrestotug is under investigation in clinical trial NCT05565378 (A Platform Study of Novel Immunotherapy Combinations in Participants With Previously Untreated, Advanced/metastatic Non-small-cell Lung Cancer).

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Beludavimab DB18952
biotech | CAS: 2423016-74-2

Beludavimab is under investigation in clinical trial NCT04746183 (AGILE (Early Phase Platform Trial for COVID-19)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 2390462-37-8

Deskripsi belum tersedia.

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Bempedoic acid Approved DB11936
small molecule | CAS: 738606-46-7

High levels of LDL cholesterol (LDL-C) are a major risk factor for cardiovascular events. Caused by genetic mutations or lifestyle factors, hypercholesterolemia can significantly reduce quality of life and increase the risk of mortality from cardiovascular di…

Kategori:
Acids, AcyclicAdenosine Triphosphate-Citrate Lyase InhibitorAdenosine Triphosphate-Citrate Lyase Inhibitors +11
Target Protein:
ATP-citrate synthase
Waktu ParuhThe half-life of be…
Vol. DistribusiThe apparent volume…
KlirensThe clearance (CL/F…
Genetik -
Bendazac Approved DB13501
small molecule | CAS: 20187-55-7

Bendazac is an oxyacetic acid [A39863, A39869]. Despite possessing anti-inflammatory, anti-necrotic, choleretic, and anti-lipidemic characteristics, most research has revolved around studying and demonstrating the agent's principal action in inhibiting the de…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +18
Target Protein:
Free radicalsProstaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe volume of distr…
KlirensThe plasma clearanc…
Genetik -
Benfluorex DB09022
small molecule | CAS: 23602-78-0

Benfluorex is an anorectic and hypolipidemic agent that is structurally related to fenfluramine. It was patented and manufactured by a French pharmaceutical company Servier. The European Medicines Agency (EMA) recommended withdrawing all benfluorex containing…

Kategori:
Alimentary Tract and MetabolismAminesAnti-Obesity Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Benralizumab Approved DB12023
biotech | CAS: 1044511-01-4

Benralizumab is a humanized recombinant monoclonal antibody of the isotype IgG1k immunoglobulin that specifically binds to the alpha chain of the interleukin 5 receptor (IL-5R) expressed on eosinophils and basophils.[A31294] It inhibits the binding of IL-5 as…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAntibodies +13
Target Protein:
Interleukin-5 receptor subunit alphaLow affinity immunoglobulin gamma Fc region receptor III-A
Waktu ParuhThe half-life of Be…
Vol. DistribusiPharmacokinetic rep…
KlirensFor a subject weigh…
Genetik -
Benserazide Approved DB12783
small molecule | CAS: 322-35-0

When levodopa is used by itself as a therapy for treating Parkinson's disease, its ubiquitous metabolism into dopamine is responsible for a resultant increase in the levels of circulating dopamine in the blood and to various extracerebral tissues. This can re…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsAromatic L-amino Acid Decarboxylase Inhibitors +6
Target Protein:
Aromatic-L-amino-acid decarboxylase
Waktu ParuhThe half-life of be…
Vol. DistribusiReadily accessible …
KlirensReadily accessible …
Genetik -
Benzgalantamine Approved DB19353
small molecule | CAS: 224169-27-1

Benzgalantamine is a prodrug of [galantamine]. Gastrointestinal adverse effects are the most frequently reported side effects in patients undergoing treatment with cholinesterase inhibitors, including galantamine, and are often a reason for treatment disconti…

Kategori:
AlkaloidsAlzheimer Disease, drug therapyAmaryllidaceae Alkaloids +11
Target Protein:
AcetylcholinesteraseCholinesteraseNeuronal acetylcholine receptor subunit alpha-7 +1
Waktu Paruh-
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Benzhydrocodone Approved DB15465
small molecule | CAS: 1259440-61-3

Benzhydrocodone is a benzylic prodrug of hydrocodone.[L4894] It was developed in an effort to reduce parenteral bioavailability of the active metabolite as a deterrent to abuse.[A182177] Benzhydrocodone is indicated for use in the short-term management of pai…

Kategori:
Opioids
Target Protein:
Mu-type opioid receptor
Waktu ParuhThe hydrocodone met…
Vol. DistribusiThe hydrocodone met…
KlirensThe apparent cleara…
Genetik -
Benzocaine Approved DB01086
small molecule | CAS: 94-09-7

Benzocaine is an ester local anesthetic that acts by preventing transmission of impulses along nerve fibers and at nerve endings.[A231219] It is commonly used for local anesthesia in many over the counter products.[L32454,L32459,L32464] Benzocaine was first u…

Kategori:
Acids, CarbocyclicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAminobenzoates +29
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 627861-07-8

Beperminogene perplasmid is under investigation in clinical trial NCT02144610 (Efficacy and Safety of AMG0001 in Subjects With Critical Limb Ischemia).

Kategori:
Vasoprotectives
Waktu Paruh-
Vol. Distribusi-
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Bepranemab DB17945
biotech | CAS: 2244960-75-4

Bepranemab is a recombinant humanized Igg4P monoclonal antibody directed against human Tau.

Waktu Paruh-
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Berbamine DB18146
small molecule | CAS: 478-61-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnalgesicsAnalgesics, Non-Narcotic +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Berberine Approved DB04115
small molecule | CAS: 2086-83-1

An alkaloid from Hydrastis canadensis L., Berberidaceae. It is also found in many other plants. It is relatively toxic parenterally, but has been used orally for various parasitic and fungal infections and as antidiarrheal.

Kategori:
AlkaloidsBenzylisoquinolinesBerberine Alkaloids +1
Target Protein:
Telomerase reverse transcriptaseBaculoviral IAP repeat-containing protein 5HTH-type transcriptional regulator QacR
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Beremagene geperpavec Approved DB17831
biotech | CAS: 2241888-62-8

Beremagene geperpavec is a live, replication-defective herpes simplex virus type 1 (HSV-1)-based vector therapy. Developed by Krystal Biotech, it was first approved by the FDA on May 19, 2023, for the treatment of wounds associated with dystrophic epidermolys…

Kategori:
Administration, TopicalCellular and Gene TherapyCicatrizants +2
Waktu ParuhThere is no informa…
Vol. DistribusiThere is no informa…
KlirensThere is no informa…
Genetik -
Bersanlimab DB17377
biotech | CAS: 1987854-08-9

Bersanlimab is an investigational monoclonal antibody directed against intercellular adhesion molecule 1 (ICAM-1).

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Bertilimumab DB05429
biotech

Bertilimumab is a fully human anti-eotaxin monoclonal antibody with potential in the treatment of allergic disorders, has moved into pre-clinical development. It is developed by MedImmune for the treatment of Allergic Rhinitis.

Target Protein:
Eotaxin
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Besilesomab Approved DB13979
biotech | CAS: 537694-98-7

Besilesomab is a mouse monoclonal antibody labelled with the radioactive isotope technetium-99m for determining the location of inflammation/infection in peripheral bone in adults with suspected osteomyelitis [FDA Label]. Utilised only as a diagnostic agent, …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Carcinoembryonic antigen
Waktu ParuhWhole blood concent…
Vol. DistribusiIn the besilesomab …
KlirensOnce administered i…
Genetik -
beta-Mannobiose DB01687
small molecule

Deskripsi belum tersedia.

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Betaine Approved DB06756
small molecule | CAS: 107-43-7

Betaine is a methyl group donor that functions in the normal metabolic cycle of methionine. It is a naturally occurring choline derivative commonly ingested through diet, with a role in regulating cellular hydration and maintaining cell function.[A252235,A252…

Kategori:
Acid PreparationsAlimentary Tract and MetabolismAmines +12
Target Protein:
Betaine--homocysteine S-methyltransferase 1
Waktu ParuhIn healthy voluntee…
Vol. DistribusiBased on a study do…
KlirensBased on a study do…
Genetik -
Betamethasone Approved DB00443
small molecule | CAS: 378-44-9

Betamethasone is a long-acting corticosteroid with immunosuppressive and antiinflammatory properties.[A192444] It can be used topically to manage inflammatory skin conditions such as eczema, and parenterally to manage several disease states including autoimmu…

Kategori:
Adrenal Cortex HormonesAdrenalsAgents Causing Muscle Toxicity +52
Target Protein:
Glucocorticoid receptor
Waktu ParuhIn a study that inc…
Vol. DistribusiIn a study that inc…
KlirensIn a study that inc…
Genetik -
Betrixaban Approved DB12364
small molecule | CAS: 330942-05-7

Betrixaban is a non-vitamin K oral anticoagulant whose action is driven by the competitive and reversible inhibition of the factor Xa [A7708]. It was selected among all lead compounds due to its low hERG channel affinity while sustaining its factor Xa inhibit…

Kategori:
Acids, CarbocyclicAmidesAnticoagulants +11
Target Protein:
Coagulation factor X
Waktu ParuhBetrixaban presents…
Vol. DistribusiThe apparent volume…
KlirensBetrixaban presents…
Genetik -
small molecule | CAS: 8001-88-5

Betula pendula tar oil is an essential oil found in the buds of the plant with the same name. The origin plant, also known as the European white or silver birch, grows mainly in the northern hemisphere. This oil is usually obtained by using both hydrodistilla…

Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Bevacizumab Approved DB00112
biotech | CAS: 216974-75-3

There is a great deal of evidence indicating that vascular endothelial growth factor (VEGF) is important for the survival and proliferation of cancer cells.[A192939,A192837,A192891,A193275] VEGF plays an important role in angiogenesis, lymphangiogenesis, and …

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +27
Target Protein:
Vascular endothelial growth factor A, long formComplement C1q subcomponent subunit AComplement C1q subcomponent subunit B +6
Waktu ParuhThe half-life of be…
Vol. DistribusiThe volume of distr…
KlirensThe clearance (CL) …
Genetik -
Bevirimat DB06581
small molecule | CAS: 174022-42-5

Bevirimat, also known as PA-457 or YK-FH312, is investigated in clinical trials for treating HIV infection. Bevirimat is a solid. This compound belongs to the androgens and derivatives, which are hydroxylated C19 steroid hormones. They are known to favour the…

Kategori:
Acids, AcyclicAnti-HIV AgentsDicarboxylic Acids +2
Target Protein:
Gag-Pol polyprotein
Waktu Paruh56.3 to 69.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Bezlotoxumab Approved DB13140
biotech | CAS: 1246264-45-8

Bezlotoxumab is a fully humanized ImmunoglobulinG1 (IgG1) kappa monoclonal antibody that binds to _Clostridium difficile_ toxin B and neutralizes its effects.[L46976] First approved by the FDA on October 21, 2016,[A260106] bezlotoxumab is used to reduce the r…

Kategori:
Amino Acids, Peptides, and ProteinsAntibacterial monoclonal antibodiesAntibodies +11
Target Protein:
Toxin B
Waktu ParuhBased on a populati…
Vol. DistribusiBased on a populati…
KlirensBased on a populati…
Genetik -
BGT-DTDS DB18664
biotech

BGT-DTDS is an investigational gene therapy comprising an adeno-associated viral vector type 2 (AAV2) encoding the human _SLC6A3_ gene. It is under investigation for the treatment of dopamine transporter deficiency syndrome (DTDS).

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BI-1206 DB17429
biotech

BI-1206 is a fully human immunoglobulin G1 monoclonal antibody that targets CD32b.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
BI-765063 DB17482
biotech

BI-765063 is a humanized IgG4 monoclonal antibody antagonist of signal regulatory protein ? (SIRP?).

Waktu Paruh-
Vol. Distribusi-
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BI-836858 DB17267
biotech | CAS: 2206770-25-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
BI-836880 DB17484
biotech

BI-836880 is a humanized bispecific nanobody that targets VEGF and Ang2.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bi104 DB18743
biotech

Bi104 is being investigated for the treatment of Angelman syndrome.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bifenthrin DB15056
small molecule | CAS: 82657-04-3

Bifenthrin is under investigation in clinical trial NCT01560247 (Percutaneous Recanalization in Ischemic Stroke Management in Europe Observational Registry).

Kategori:
Cyclopentane MonoterpenesMonoterpenesSarcoma, Experimental, chemically induced +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bifikafusp alfa DB19185
biotech | CAS: 1957239-90-5

Bifikafusp alfa is under investigation in clinical trial NCT05329792 (L19IL2/L19TNF in Skin Cancer Patients).

Waktu Paruh-
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Genetik -
BIIB015 DB06304
biotech

BIIB015 is a humanized, IgG1 [immunoglobulin G 1], DM4-Conjugated, anti-cripto, monoclonal antibody. It has been investigated for the treatment of subjects with relapsed or refractory solid tumours.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bimekizumab Approved DB12917
biotech | CAS: 1418205-77-2

Bimekizumab is a humanized monoclonal antibody directed towards IL-17, which was approved for use in the EU on August 20, 2021, for the treatment of plaque psoriasis.[L39665,L39680] It is the first IL-17 inhibitor to target both IL-17A and IL-17F.[A244455] It…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +11
Target Protein:
Interleukin-17AInterleukin-17F
Waktu ParuhThe mean terminal e…
Vol. DistribusiIn patients with pl…
KlirensThe median apparent…
Genetik -
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