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1977

Total database: 17430
Struktur (SMILES)
1074 (54.3%)
Target
1046 (52.9%)
Genomik
39 (2.0%)
Referensi
1977 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (1977)

Halaman 7 / 40
Cantharidin Approved DB12328
small molecule | CAS: 56-25-7

Cantharidin is a naturally occurring odorless, colorless fatty substance of the terpenoid class that is produced as an oral fluid in the alimentary canal of the male blister beetle.[A32891, A32892] For its natural purpose, the male blister beetle secretes and…

Kategori:
BenzofuransCompounds used in a research, industrial, or household settingEnzyme Inhibitors +4
Target Protein:
Serine/threonine-protein phosphatase PP1-alpha catalytic subunitAryl hydrocarbon receptor
Waktu ParuhLittle pharmacodyna…
Vol. DistribusiAfter oral or IP in…
KlirensLittle pharmacodyna…
Genetik -
biotech | CAS: 400010-39-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capmatinib Approved DB11791
small molecule | CAS: 1029712-80-8

Capmatinib is a small molecule kinase inhibitor targeted against c-Met (a.k.a. hepatocyte growth factor receptor [HGFR]), a receptor tyrosine kinase that, in healthy humans, activates signaling cascades involved in organ regeneration and tissue repair.[A19912…

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +20
Target Protein:
Hepatocyte growth factor receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -
Capsicum Approved DB10897
biotech

Capsicum (Chili pepper) allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Capsicum oleoresin Approved DB11131
biotech | CAS: 8023-77-6

Capsicum oleoresin is an oily organic resin derived from the fruit of plants in the Capsicum genus, such as chilli peppers. When the plants are finely ground, capsicum oleoresin is formed after the extraction process of capsaicin using oragnic solvents such a…

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +1
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu ParuhFor pharmacokinetic…
Vol. DistribusiFor pharmacokinetic…
KlirensFor pharmacokinetic…
Genetik -
Carbamide peroxide Approved DB11129
small molecule | CAS: 124-43-6

Carbamide peroxide, also known as urea-hydrogen peroxide, is a water-soluble, white crystalline solid compound consisting of hydrogen peroxide and urea. As it is a source of hydrogen peroxide, it can be found in disinfecting and dental bleaching products. Som…

Kategori:
AmidesAnionsAnti-Infective Agents +14
Waktu ParuhNo established phar…
Vol. DistribusiNo established phar…
KlirensNo established phar…
Genetik -
Carbazochrome DB09012
small molecule | CAS: 69-81-8

Carbazochrome is a hemostatic agent that promotes clotting, preventing blood loss from open wounds. It is an oxidation product of adrenaline which enhances the microcirculatory tone [A19747]. In the future this may prevent excessive blood flow during surgical…

Kategori:
Biological FactorsBlood and Blood Forming OrgansCoagulants +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carbenicillin Approved DB00578
small molecule | CAS: 4697-36-3

Broad-spectrum semisynthetic penicillin derivative used parenterally. It is susceptible to gastric juice and penicillinase and may damage platelet function.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
Penicillin-binding proteinBeta-lactamase Toho-1
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
Cardiopet DB18913
small molecule | CAS: 855927-17-2

Cardiopet is under investigation in clinical trial NCT01826773 (Cardiopet as PET Imaging Agent to Assess Myocardial Perfusion and Fatty Acid Uptake in Known or Suspected CAD Subjects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carfentanil DB01535
small molecule | CAS: 59708-52-0

Carfentanil or carfentanyl (Wildnil) is an analogue of the popular synthetic opioid analgesic fentanyl, and is one of the most potent opioids known (also the most potent opioid used commercially). Carfentanil was first synthesized in 1974 by a team of chemist…

Kategori:
AnalgesicsCarbon RadioisotopesCentral Nervous System Agents +9
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carfilzomib Approved DB08889
small molecule | CAS: 868540-17-4

Carfilzomib is an injectable antineoplastic agent (IV only). Chemically, it is a modified tetrapeptidyl epoxide and an analog of epoxomicin. It is also a selective proteasome inhibitor. FDA approved carfilzomib in July 2012 for the treatment of adults with re…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +8
Target Protein:
Proteasome subunit beta type-5Proteasome subunit beta type-8Proteasome subunit beta type-1 +3
Waktu ParuhFollowing intraveno…
Vol. DistribusiVd, steady state, 2…
KlirensSystemic clearance …
Genetik -
Cariprazine Approved DB06016
small molecule | CAS: 839712-12-8

Cariprazine is an atypical antipsychotic agent and a piperazine derivative that was first developed in Hungary.[A247100] It works as a partial agonist at central dopamine D2, dopamine D3, and serotonin 5-HT<sub>1A</sub> receptors and as an antagonist at serot…

Kategori:
Agents that produce hypertensionAntidepressive AgentsAntipsychotic Agents +48
Target Protein:
D(3) dopamine receptorD(2) dopamine receptor5-hydroxytryptamine receptor 1A +5
Waktu ParuhCariprazine and its…
Vol. Distribusi-
Klirens-
Genetik -
Carisoprodol Approved DB00395
small molecule | CAS: 78-44-4

Originally approved by the FDA in 1959 [FDA label], carisoprodol is a centrally acting muscle relaxant used in painful musculoskeletal conditions in conjunction with physical therapy and other medications [A176047]. This drug is available by itself in an ora…

Kategori:
CarbamatesCarbamic Acid EstersCentral Nervous System Agents +7
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit gamma-2 +2
Waktu ParuhThe terminal half-l…
Vol. Distribusi0.93 to 1.3 L/kg, a…
KlirensFollowing an oral d…
Genetik -
small molecule | CAS: 401905-67-7

Carotegrast methyl is under investigation in clinical trial NCT03531892 (A Study to Evaluate the Safety and Efficacy of AJM300 in Participants With Active Ulcerative Colitis).

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carotuximab DB06322
biotech | CAS: 1268714-50-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Endoglin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carprofen Approved DB00821
small molecule | CAS: 53716-49-7

Carprofen is a non-steroidal anti-inflammatory drug (NSAID) that is used by veterinarians as a supportive treatment for the relief of arthritic symptoms in geriatric dogs. Carprofen was previously used in human medicine for over 10 years (1985-1995). It was g…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +15
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhApproximately 8 hou…
Vol. Distribusi-
Klirens-
Genetik -
Carya illinoinensis pollen Approved DB10380
biotech

Carya illinoinensis pollen allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Carya laciniosa pollen Approved DB10987
biotech

Carya laciniosa pollen allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Casdozokitug DB17513
biotech | CAS: 2643331-37-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cashew Approved DB10653
biotech

Cashew allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cashew fruit Approved DB15602
biotech

Cashew fruit extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Castor oil Approved DB11113
biotech | CAS: 8001-79-4

Castor oil is a vegetable oil obtained by pressing the seeds of the castor oil plant (_Ricinus communis_ L.) mainly cultivated in India, South America, Africa, and China. Castor oil is a rich source of [DB02955], which represents up to 90% of the total castor…

Kategori:
Alimentary Tract and MetabolismBiological ProductsComplex Mixtures +10
Target Protein:
Prostaglandin E2 receptor EP3 subtypeProstaglandin E2 receptor EP4 subtype
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Catridecacog Approved DB09310
biotech | CAS: 606138-08-3

Coagulation Factor XIII A-Subunit (Recombinant), also known as catridecacog, is a recombinant form of the Factor XIII-A2 homodimer composed of two factor XIII (FXIII) A-subunits [FDA Label]. For people with congenital deficiency or mutation of Factor XIII, a …

Kategori:
Blood and Blood Forming OrgansBlood Coagulation FactorsHemostatics
Target Protein:
Coagulation factor XIII B chain
Waktu Paruh7.1 days
Vol. Distribusi-
Klirens0.41 mL/h/kg
Genetik -
Catumaxomab Approved DB06607
biotech | CAS: 509077-98-9

Catumaxumab is a trifunctional monoclonal antibody developed for use in cancer treatment. It has affinity for T-cells, accessory immune cells, and cancer cells. Catumaxumab was initially authorized for market by the European Medicines Agency in April 2009 for…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +13
Target Protein:
Low affinity immunoglobulin gamma Fc region receptor II-aLow affinity immunoglobulin gamma Fc region receptor III-ALow affinity immunoglobulin gamma Fc region receptor III-B +3
Waktu ParuhCatumaxomab has an …
Vol. Distribusi-
Klirens-
Genetik -
CB-1158 DB15286
small molecule | CAS: 2095732-06-0

CB-1158 is under investigation in clinical trial NCT03910530 (A Study of INCMGA00012, INCB001158, and the Combination in Japanese Participants With Advanced Solid Tumors).

Kategori:
Enzyme Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CE-VST01-JC DB17190
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cedar leaf oil DB15836
biotech | CAS: 8007-20-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cedar oil Approved DB10917
biotech | CAS: 8000-27-9

Cedar oil (Juniperus virginiana) allergenic extract is used in allergenic testing.

Kategori:
Biological ProductsLipidsOils +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cedazuridine Approved DB15694
small molecule | CAS: 1141397-80-9

Myelodysplastic syndromes (MDS) are a group of hematopoietic neoplasms that give rise to variable cytopenias progressing to secondary acute myeloid leukemia (sAML), which is invariably fatal if untreated.[A215082, A215092, A215097] Hypomethylating agents such…

Kategori:
Cytidine Deaminase, antagonists & inhibitorsNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Cytidine deaminase
Waktu ParuhCedazuridine has a …
Vol. DistribusiThe apparent volume…
KlirensCedazuridine has an…
Genetik -
Cefapirin Approved DB01139
small molecule | CAS: 21593-23-7

Cefapirin (INN, also spelled cephapirin), commonly marketed under the trade name Cefadyl, is a first-generation cephalosporin antibiotic that is available in injectable formulations. Production for use in humans has been discontinued in the United States. Cef…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefminox DB09062
small molecule | CAS: 84305-41-9

Cefminox (INN) is a second generation cephalosporin antibiotic. It is approved for use in Japan.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cefovecin DB11505
small molecule

Cefovecin is a cephalosporin antibiotic used for the treatment of skin infections in cats and dogs. It is the first single-dose injectable antibiotic for dogs and cats that assures owner compliance with dosing for the animal. It is used for the treatment of s…

Kategori:
Amidesbeta-LactamsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceftazidime Approved DB00438
small molecule | CAS: 72558-82-8

Bacteria possess a cell wall comprising a glycopeptide polymer commonly known as peptidoglycan, which is synthesized and remodelled through the action of a family of enzymes known as "penicillin-binding proteins" (PBPs).[A232920] ?-lactam antibiotics, includi…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1APenicillin-binding protein 1B +2
Waktu ParuhCeftazidime has an …
Vol. DistribusiCeftazidime has a v…
KlirensThe mean renal clea…
Genetik -
Ceftolozane Approved DB09050
small molecule | CAS: 689293-68-3

Ceftolozane is a semi-synthetic broad-spectrum fifth generation cephalosporin.[L6685] It was approved by the FDA in 2014 for use in combination with [Tazobactam] for the treatment of serious infections, such as intra-abdominal infections and complicated urina…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +8
Target Protein:
Penicillin-binding protein 1BCell division proteinPenicillin-binding protein 1C +2
Waktu Paruh2.77 hours on day 1…
Vol. Distribusi13.5 L.[L41618] Tis…
KlirensThe renal clearance…
Genetik -
Cemiplimab Approved DB14707
biotech | CAS: 1801342-60-8

Cemiplimab is a fully human monoclonal antibody that works against programmed death receptor-1 (PD-1), which is a negative regulator of T cell function. By blocking PD-1, cemiplimab works to enhance T cell-mediated antitumour responses.[L39804] Cemiplimab …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Programmed cell death protein 1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensCemiplimab clearanc…
Genetik -
Cendakimab DB18427
biotech

Cendakimab is a recombinant humanized anti-interleukin 13 (IL-13) monoclonal antibody.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenegermin Approved DB13926
biotech | CAS: 1772578-74-1

Cenegermin is a human beta-nerve growth factor (beta-ngf)-(1-118)- peptide (non-covalent dimer) produced in escherichia coli. It received European Union Approval in July 2017 for the treatment of moderate to severe neurotrophic keratitis. Cenegermin received …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +7
Target Protein:
High affinity nerve growth factor receptorTumor necrosis factor receptor superfamily member 16
Waktu ParuhHalf-life data spec…
Vol. DistribusiAfter eye drop admi…
KlirensAlthough the system…
Genetik -
Centanafadine DB14841
small molecule | CAS: 924012-43-1

Centanafadine is under investigation in clinical trial NCT02827513 (A Phase 1 Study to Investigate the Safety, Tolerance, Food Effect, Pharmacokinetics and Pharmacodynamics of Single and Multiple Doses of Extended Release Formulations of Centanafadine (CTN) i…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Centella asiatica Approved DB14256
biotech

Centella asiatica is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Agents that reduce seizure thresholdAngiospermsApiaceae +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cephalexin Approved DB00567
small molecule | CAS: 15686-71-2

Cephalexin is the first of the first generation cephalosporins.[A179071,A179074] This antibiotic contains a beta lactam and a dihydrothiazide.[A179071] Cephalexin is used to treat a number of susceptible bacterial infections through inhibition of cell wall s…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +23
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2aPenicillin-binding protein 1b +2
Waktu ParuhThe half life of ce…
Vol. Distribusi5.2-5.8L.[A179068]
KlirensClearance from one …
Genetik -
Ceramide NP DB14111
small molecule | CAS: 100403-19-8

Ceramide NP is a lipid molecule included in a group of lipid molecules called ceramides. Ceramides are major lipid components in the stratum corneum of the human skin. Ceramide 3 consists of a phytosphingosine backbone N-acylated with a saturated fatty acid (…

Kategori:
AntigensAntigens, NeoplasmBiological Factors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CERC-301 DB12063
small molecule | CAS: 808732-98-1

Mk 0657 has been used in trials studying the treatment of Major Depressive Disorder.

Kategori:
Receptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Target Protein:
Glutamate receptor ionotropic, NMDA 2B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cethromycin DB06419
small molecule | CAS: 205110-48-1

Cethromycin is a 3-keto (ketolide) derivative of erythromycin A with an 11,12-carbamate group and an O-6-linked aromatic ring system.[A203369] Cethromycin represents a joint development effort by Abbott Laboratories, Taisho Pharmaceuticals, and Advanced Life …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCytochrome P-450 CYP3A Inhibitors +15
Target Protein:
23S ribosomal RNA
Waktu ParuhCethromycin given i…
Vol. DistribusiCethromycin given i…
KlirensCethromycin clearan…
Genetik -
Cetrelimab DB15421
biotech | CAS: 2050478-92-5

Cetrelimab is under investigation in clinical trial NCT03547037 (A Study to Evaluate the Safety, Pharmacokinetics, Pharmacodynamics, and Immunogenicity of JNJ-63723283, an Anti-Programmed Cell Death (PD)-1 Monoclonal Antibody, as Monotherapy or in Combination…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2166339-33-7

Cetuximab sarotalocan is under investigation in clinical trial NCT03769506 (ASP-1929 Photoimmunotherapy (PIT) Study in Recurrent Head/Neck Cancer for Patients Who Have Failed at Least Two Lines of Therapy) for the treatment of Recurrent Head/Neck Cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cevimeline Approved DB00185
small molecule | CAS: 107233-08-9

Cevimeline is a parasympathomimetic agent that act as an agonist at the muscarinic acetylcholine receptors M1 and M3. It is indicated by the Food and Drug Administration for the treatment of dry mouth associated with Sjögren's syndrome.

Kategori:
Autonomic AgentsCholinergic AgentsCholinergic Agonists +12
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1
Waktu Paruh5 &plusmn; 1 hours
Vol. Distribusi* 6 L/kg
Klirens-
Genetik -
CG0070 DB05148
small molecule

CG0070 is investigated in clinical trials for treating bladder cancer. CG0070 is a solid. CG0070 can potentially destroy cancer cells by two different mechanisms: direct cell killing by the virus and immune-mediated cell killing stimulated by GM-CSF. CG0070, …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CGI-1842 DB12744
small molecule | CAS: 900573-88-8

JI-101 has been used in trials studying the treatment of Cancer, Colon Cancer, Neuroendocrine, Ovarian Cancer, and Advanced Solid Tumors.

Kategori:
AmidesBenzene DerivativesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Receptor tyrosine-protein kinase erbB-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 301–350 dari 1977
Sebelumnya Halaman 7 / 40 Berikutnya