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16749

Total database: 17430
Struktur (SMILES)
11810 (70.5%)
Target
9015 (53.8%)
Genomik
112 (0.7%)
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16749 (100.0%)

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Hasil Pencarian (16749)

Halaman 68 / 335
Anagrelide Approved DB00261
small molecule | CAS: 68475-42-3

Anagrelide is a platelet-reducing agent used to lower dangerously elevated platelet levels (i.e. to treat thrombocythemia) in patients with myeloproliferative neoplasms.[L14153] It is an oral imidazoquinazoline that was first approved for use in the US in 199…

Kategori:
Agents producing tachycardiaAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A
Waktu ParuhThe t<sub>1/2</sub>…
Vol. Distribusi-
Klirens-
Genetik -
Anakinra Approved DB00026
biotech | CAS: 143090-92-0

Anakinra is a recombinant human interleukin-1 (IL-1) receptor antagonist (IL-1Ra) composed of 153 amino acid residues. Unlike native human IL-1Ra, anakinra has an additional methionine residue at the amino terminus. This drug binds to the IL-1 receptor, compe…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +12
Target Protein:
Interleukin-1 receptor type 1
Waktu ParuhIn patients with rh…
Vol. DistribusiIn adult subjects w…
KlirensIn patients with rh…
Genetik -
Anamorelin DB06645
small molecule | CAS: 249921-19-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +2
Target Protein:
Growth hormone secretagogue receptor type 1Lysosomal alpha-glucosidaseNeutral alpha-glucosidase AB +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ananain DB18353
biotech | CAS: 119129-70-3

Deskripsi belum tersedia.

Kategori:
Cysteine ProteasesEndopeptidasesEnzymes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anaritide DB17613
biotech | CAS: 95896-08-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsDiureticsHormones +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anas platyrhynchos feather Approved DB10421
biotech

Anas platyrhynchos feather is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anastrozole Approved DB01217
small molecule | CAS: 120511-73-1

Anastrozole is a non-steroidal aromatase inhibitor (AI), similar to [letrozole], used to decrease circulating estrogen levels in the treatment of postmenopausal women with estrogen-responsive breast cancer.[L8863] Anastrozole is also related to [exemestane], …

Kategori:
Antineoplastic AgentsAntineoplastic Agents, HormonalAntineoplastic and Immunomodulating Agents +30
Target Protein:
Aromatase
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensAnastrozole's clear…
Genetik -
Anatibant DB05038
small molecule | CAS: 209733-45-9

Anatibant is a selective, very potent, small-molecule Bradykinin B2 receptor antagonist. It is developed for the for the treatment of traumatic brain injury (TBI).

Kategori:
Bradykinin Receptor AntagonistsHeterocyclic Compounds, Fused-Ring
Target Protein:
B2 bradykinin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anbenitamab DB18411
biotech | CAS: 2367012-88-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ANC-501 DB18907
small molecule | CAS: 1370444-22-6

ANC-501 is under investigation in clinical trial NCT05439603 (ANC-501 in the Treatment of Adults With Major Depressive Disorder).

Kategori:
AcetatesAcids, AcyclicAmides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ancestim Approved DB09103
biotech | CAS: 163545-26-4

Ancestim is a non-glycosylated recombinant methionyl human stem cell factor. It is a 166 amino acid protein produced by E. coli with an amino acid sequence that is identical to the natural sequence predicted from human DNA sequence analysis, except for the ad…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +8
Target Protein:
Mast/stem cell growth factor receptor Kit
Waktu ParuhIn clinical trials,…
Vol. DistribusiPreclinical reports…
KlirensThe apparent cleara…
Genetik -
Ancrod Approved DB05099
biotech | CAS: 9046-56-4

Ancrod, marketed as Viprinex, is a defibrinogenating agent derived from Malayan pit viper venom. The defribrinogenation of blood results in an anticoagulant effect. Currently, Viprinex®/ancrod is not approved or marketed in any country, but is being investiga…

Kategori:
AnticoagulantsBiological FactorsBlood and Blood Forming Organs +18
Target Protein:
Fibrinogen alpha chain
Waktu Paruh3 to 5 hours
Vol. Distribusi-
Klirens-
Genetik -
Andarine DB07423
small molecule | CAS: 401900-40-1

Andarine is a non-steroidal selective androgen receptor modulator.

Kategori:
AcetatesAcids, AcyclicAmides +4
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Andecaliximab DB17564
biotech | CAS: 1518996-49-0

Andecaliximab is a monoclonal antibody directed against matrix metallopeptidase 9 (MMP9). Andecaliximab is under investigation in clinical trial NCT03631836 (Phase I Study of Monoclonal Antibondy (GS) 5745, an Matix Metalloproteinase 9 (MMP9) Mab Inhibitor, i…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Andexanet alfa Approved DB14562
biotech | CAS: 1262449-58-0

Andexanet alfa is a recombinant human coagulation Factor Xa that promotes blood coagulation. It was developed by Portola Pharmaceuticals and was approved in in May 2018. It is marketed as Andexxa for intravenous injection or infusion and is indicated for the …

Kategori:
Amino Acids, Peptides, and ProteinsAntidotesBiological Factors +12
Target Protein:
Tissue factor pathway inhibitor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensClearance for andex…
Genetik -
Andrographolide DB05767
small molecule | CAS: 5508-58-7

Andrographolide (HMPL-004) is a botanical product extracted from a herb that occurs naturally in China. The herb has an extensive history of use in TCM for the treatment of upper respiratory tract infections and other inflammatory and infectious diseases.

Kategori:
AcanthaceaeAnalgesicsAnalgesics, Non-Narcotic +25
Target Protein:
Tumor necrosis factorInterleukin-1 betaInterleukin-6 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Androstanedione DB01561
small molecule | CAS: 846-46-8

Deskripsi belum tersedia.

Target Protein:
17-beta-hydroxysteroid dehydrogenase type 1Steroid Delta-isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Androstenediol DB01524
small molecule | CAS: 521-17-5

Androstenediol is an intermediate in [testosterone] biosynthesis, found in the testis or the adrenal glands. Androstenediol, derived from dehydroepiandrosterone by the reduction of the 17-keto group (17-hydroxysteroid dehydrogenases), is converted to testoste…

Kategori:
Anabolic AgentsAndrostanesAndrostenediols +9
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Androstenedione DB01536
small molecule | CAS: 63-05-8

A delta-4 C19 steroid that is produced not only in the testis, but also in the ovary and the adrenal cortex. Depending on the tissue type, androstenedione can serve as a precursor to testosterone as well as estrone and estradiol.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesAndrostanes +12
Target Protein:
Aromatase17-beta-hydroxysteroid dehydrogenase type 13 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Andusomeran Approved DB18227
biotech | CAS: 2918977-08-7

Andusomeran is a COVID-19 mRNA vaccine developed for use during the 2023-2024 season.[L40074,L48832,L48837] It is similar to previous mRNA vaccines developed by Moderna (e.g. [elasomeran], [imelasomeran]), but is designed to be effective against the Omicron X…

Kategori:
COVID-19 VaccinesmRNA VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ANEB-001 DB18908
small molecule | CAS: 791848-71-0

ANEB-001 is under investigation in clinical trial NCT05282797 (Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of CB1 Antagonist ANEB-001 in a THC Challenge Test).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anecortave DB12081
small molecule | CAS: 10184-70-0

Anecortave is under investigation in clinical trial NCT00691717 (Anecortave Acetate Safety in Patients With Open-Angle Glaucoma or Ocular Hypertension).

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 7753-60-8

Anecortave acetate (Retaane) is an analog of cortisol acetate; among the modifications to the steroid are the removal of the 11ß hydroxyl OH group and an addition of a 21-acetate group. As a result of these modifications, anecortave acetate lacks the typical …

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAngiogenesis Inhibitors +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anethole Approved DB15916
small molecule | CAS: 4180-23-8

Deskripsi belum tersedia.

Kategori:
AlkenesAllyl CompoundsBenzene Derivatives +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anethole trithione Approved DB13853
small molecule | CAS: 532-11-6

Anethole trithione (ATT) appears to have a broad range of unique functions, from increasing salivary secretion to help treat xerostomia [A27165, A32618, A32620, A32621], to demonstrating an ability to inhibit carcinogenesis by increasing the activity of elect…

Kategori:
Alimentary Tract and MetabolismAnisolesBenzene Derivatives +10
Target Protein:
Protein-glutamine gamma-glutamyltransferase 2
Waktu ParuhDespite the medicat…
Vol. DistribusiDespite the medicat…
KlirensDespite the medicat…
Genetik -
biotech | CAS: 1375258-01-7

Anetumab ravtansine is under investigation in clinical trial NCT03455556 (Anetumab Ravtansine and Atezolizumab in Treating Participants With Advanced Non-small Cell Lung Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibody-drug Conjugates +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anfibatide DB15094
biotech | CAS: 1622134-89-7

Anfibatide is under investigation in clinical trial NCT01585259 (Anfibatide Phase Ib-IIa Clinical Trial).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsComplex Mixtures +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Angelica archangelica root Approved DB14283
biotech

Angelica archangelica root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Angelica dahurica root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Angelica sinensis root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngelicaAngiospermsApiaceae +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Angiotensin 1-7 DB11720
small molecule | CAS: 51833-78-4

TXA127 has been investigated for the treatment of Miscellaneous Peripheral Blood Cell Abnormalities.

Kategori:
Amino Acids, Peptides, and ProteinsAngiotensinsAntihypertensive Agents +13
Target Protein:
Proto-oncogene Mas
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Angiotensin II Approved DB11842
biotech | CAS: 4474-91-3

Angiotensin II is under investigation for the treatment of Sepsis, Septic Shock, Diabetes Mellitus, and Acute Renal Failure. Angiotensin II has been investigated for the treatment, basic science, and diagnostic of Hypertension, Renin Angiotensin System, and I…

Kategori:
Amino Acids, Peptides, and ProteinsAngiotensin II, antagonists & inhibitorsAngiotensins +16
Target Protein:
Type-2 angiotensin II receptorType-1 angiotensin II receptor
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe official prescr…
KlirensThe official prescr…
Genetik -
biotech | CAS: 53-73-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAngiotensinsAutacoids +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 38390-45-3

Anhydrovinblastine has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1224-78-8

Deskripsi belum tersedia.

Kategori:
AlkenesBiological FactorsCarotenoids +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anidulafungin Approved DB00362
biotech | CAS: 166663-25-8

Anidulafungin or Eraxis is an anti-fungal drug manufactured by Pfizer that gained approval by the Food and Drug Administration (FDA) in February 21, 2006; it was previously known as LY303366. There is preliminary evidence that it has a similar safety profile …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntifungal Agents +6
Target Protein:
1,3-beta-glucan synthase component FKS11,3-beta-glucan synthase component GSC2
Waktu Paruh40-50 hours
Vol. Distribusi* 30 to 50 L
Klirens* 1 L/h
Genetik -
Anifrolumab Approved DB11976
biotech | CAS: 1326232-46-5

Anifrolumab, or MEDI-546, is a type 1 interferon receptor (IFNAR) inhibiting IgG1? monoclonal antibody indicated in the treatment of adults with moderate to severe systemic lupus erythematosus.[A237074,L34929] The standard therapy for systemic lupus erythemat…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Interferon alpha/beta receptor 1
Waktu ParuhThe serum eliminati…
Vol. DistribusiBased on population…
KlirensFollowing the admin…
Genetik -
Anileridine Approved DB00913
small molecule | CAS: 144-14-9

Anileridine is a synthetic opioid and strong analgesic medication. It is a narcotic pain reliever used to treat moderate to severe pain. Narcotic analgesics act in the central nervous system (CNS) to relieve pain. Some of their side effects are also caused by…

Kategori:
AnestheticsAnesthetics, GeneralNervous System +2
Target Protein:
Mu-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aniline DB06728
small molecule | CAS: 62-53-3

Aniline, phenylamine or aminobenzene is an organic compound with the formula C6H5NH2. Consisting of an amine attached to a benzene ring, aniline is the prototypical aromatic amine. Being a precursor to many industrial chemicals, its main use is in the manufac…

Kategori:
AminesCarcinogensCytochrome P-450 CYP2E1 Substrates +3
Target Protein:
Kallikrein-1Albumin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aniracetam DB04599
small molecule | CAS: 72432-10-1

Compound with anti-depressive properties used as a mental performance enhancer.

Kategori:
Antidepressive AgentsCentral Nervous System AgentsCentral Nervous System Depressants +6
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2AGlutamate receptor 2 +1
Waktu Paruh1-2.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Anise oil DB15776
biotech | CAS: 8007-70-3

Deskripsi belum tersedia.

Kategori:
AngiospermsApiaceaeBiological Products +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anisindione Approved DB01125
small molecule | CAS: 117-37-3

Anisindione is a synthetic anticoagulant and an indanedione derivative. Its anticoagulant action is mediated through the inhibition of the vitamin K-mediated gamma-carboxylation of precursor proteins that are critical in forming the formation of active procoa…

Kategori:
IndansIndenes
Target Protein:
Vitamin K-dependent gamma-carboxylaseProthrombin
Waktu ParuhNot Known
Vol. Distribusi-
Klirens-
Genetik -
Anisodamine DB11785
small molecule | CAS: 55869-99-3

Anisodamine has been investigated for the treatment of Intestinal Diseases.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic Antagonists +29
Target Protein:
Beta-1 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anisomycin DB07374
small molecule | CAS: 22862-76-6

Anisomycin (sometimes known as flagecidin), is an antibiotic retrieved from the bacteria _Streptomyces griseolus_. This drug acts to inhibit bacterial protein and DNA synthesis.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiparasitic Agents +5
Target Protein:
Ribosomal protein uL16-likeLarge ribosomal subunit protein uL13Large ribosomal subunit protein uL14 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anisotropine methylbromide Approved DB00517
small molecule | CAS: 80-50-2

Anisotropine methylbromide is a quaternary ammonium compound. Its use as treatment adjunct in peptic ulcer has been replaced by the use of more effective agents. Depending on the dose, anisotropine methylbromide may reduce the motility and secretory activity …

Kategori:
Agents producing tachycardiaAlkaloidsAnticholinergic Agents +5
Target Protein:
Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2 +1
Waktu ParuhNot Known
Vol. Distribusi-
Klirens-
Genetik -
Anistreplase Approved DB00029
biotech | CAS: 81669-57-0

Human tissue plasminogen activator, purified, glycosylated, 527 residues purified from CHO cells. Eminase is a lyophilized (freeze-dried) formulation of anistreplase, the p-anisoyl derivative of the primary Lys-plasminogen-streptokinase activator complex (a c…

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +15
Target Protein:
PlasminogenFibrinogen alpha chainPlasminogen activator inhibitor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Anivamersen DB16089
biotech | CAS: 959716-29-1

Anivamersen is under investigation in clinical trial NCT01848106 (A Study to Determine the Efficacy and Safety of REG1 Compared to Bivalirudin in Patients Undergoing PCI).

Kategori:
CoagulantsNucleic Acids, Nucleotides, and NucleosidesNucleotides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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