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14494

Total database: 17430
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9687 (66.8%)
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7525 (51.9%)
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14494 (100.0%)

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Halaman 67 / 290
Bimagrumab DB12584
biotech | CAS: 1356922-05-8

Bimagrumab has been used in trials studying the treatment and supportive care of Sarcopenia, Skeletal Muscle, Mechanical Ventilation, Sporadic Inclusion Body Myositis, and Sporadic Inclusion Body Myositis (sIBM), among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Bimatoprost Approved DB00905
small molecule | CAS: 155206-00-1

Bimatoprost, also known as Latisse or Lumigan, belongs to a group of drugs called prostamides, which are synthetic structural analogs of prostaglandin. Bimatoprost, marketed by Allergan, is administered in both the ophthalmic solution and implant form. It has…

Kategori:
AmidesAntiglaucoma Preparations and MioticsAntihypertensive Agents +19
Target Protein:
Prostaglandin F2-alpha receptorProstaglandin E2 receptor EP1 subtypeProstaglandin E2 receptor EP3 subtype
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance was m…
Genetik -
Bimekizumab Approved DB12917
biotech | CAS: 1418205-77-2

Bimekizumab is a humanized monoclonal antibody directed towards IL-17, which was approved for use in the EU on August 20, 2021, for the treatment of plaque psoriasis.[L39665,L39680] It is the first IL-17 inhibitor to target both IL-17A and IL-17F.[A244455] It…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +11
Target Protein:
Interleukin-17AInterleukin-17F
Waktu ParuhThe mean terminal e…
Vol. DistribusiIn patients with pl…
KlirensThe median apparent…
Genetik -
Bimiralisib DB14846
small molecule | CAS: 1225037-39-7

Bimiralisib is under investigation in clinical trial NCT02723877 (PQR309 and Eribulin in Metastatic HER2 Negative and Triple-negative Breast Cancer (PIQHASSO)).

Target Protein:
Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
Waktu Paruh-
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Bimoclomol DB06258
small molecule | CAS: 130493-03-7

Bimoclomol is an investigational drug that induces stress proteins and has cytoprotective effects.

Target Protein:
Heat shock 70 kDa protein 1BHeat shock 70 kDa protein 1AHeat shock factor protein 1
Waktu Paruh-
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Bindarit DB12739
small molecule | CAS: 130641-38-2

Bindarit has been used in trials studying the prevention and treatment of Coronary Restenosis and Diabetic Nephropathy.

Kategori:
Acids, AcyclicAnti-Inflammatory AgentsEnzyme Inhibitors +6
Target Protein:
C-C motif chemokine 2
Waktu Paruh-
Vol. Distribusi-
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Binetrakin DB12182
biotech | CAS: 207137-56-2

Binetrakin has been used in trials studying the treatment of HIV Infections, Sarcoma, Kaposi, Non-Hodgkin's Lymphoma (NHL), Myelodysplastic Syndrome (MDS), and Leukemia, Acute Myelogenous (AML), among others.

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic Agents +9
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Binimetinib Approved DB11967
small molecule | CAS: 606143-89-9

Binimetinib, also known as _Mektovi_, is a potent and selective oral mitogen-activated protein kinase 1/2 (MEK 1/2) inhibitor which is combined with [Encorafenib].[A34275,L3335] On June 27, 2018, the Food and Drug Administration approved the combination of…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +16
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 2Dual specificity mitogen-activated protein kinase kinase 1
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiThe geometric mean …
KlirensThe apparent cleara…
Genetik -
Binodenoson DB04853
small molecule | CAS: 144348-08-3

Binodenoson is a pharmacologic stress agent specific to the only adenosine receptor necessary for increased cardiac blood flow, the A<sub>2A</sub> receptor. This specificity allows Binodenoson to deliver - in a single injection - a more effective dose of medi…

Kategori:
Heterocyclic Compounds, Fused-RingNeurotransmitter AgentsNucleic Acids, Nucleotides, and Nucleosides +7
Target Protein:
Adenosine receptor A2a
Waktu Paruh10 &plusmn; 4 minut…
Vol. Distribusi-
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Genetik -
Bintrafusp alfa DB15387
biotech | CAS: 1918149-01-5

Bintrafusp alfa is under investigation in clinical trial NCT03833661 (M7824 Monotherapy in Locally Advanced or Metastatic Second Line (2L) Biliary Tract Cancer (Cholangiocarcinoma and Gallbladder Cancer)).

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BIO-11006 DB14886
small molecule | CAS: 901117-03-1

BIO-11006 is under investigation in clinical trial NCT03202394 (Evaluation of Safety & Efficacy of BIO-11006 Inhalation Solution in Patients With ARDS).

Target Protein:
Myristoylated alanine-rich C-kinase substrate
Waktu Paruh-
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Bioallethrin Approved DB13746
small molecule | CAS: 584-79-2

Bioallethrin refers to a mixture of two of the allethrin isomers (1R,trans;1R and 1R,trans;1S) in an approximate ratio of 1:1, where both isomers are active ingredients. A mixture of the two same stereoisomers, but in an approximate ratio of R:S in 1:3, is ca…

Kategori:
Agents causing hyperkalemiaAgrochemicalsAntiarrhythmic agents +21
Target Protein:
Sodium channel proteinVoltage-gated sodium channel alpha subunitVoltage-dependent calcium channel +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Biochanin A DB15334
small molecule | CAS: 491-80-5

Biochanin A is under investigation in clinical trial NCT02174666 (Isoflavone Treatment for Postmenopausal Osteopenia.).

Kategori:
Anticarcinogenic AgentsAntineoplastic AgentsBenzopyrans +12
Target Protein:
Steroid hormone receptor ERR1AromataseFatty acid synthase
Waktu Paruh-
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Biomed 101 DB05851
small molecule

Biomed 101 is investigated for use/treatment in adverse effects (chemotherapy) and renal cell carcinoma. Biomed 101 is a solid. Biomed 101 binds to the leukotriene B4 receptor, but does not affect interleukin-2 antitumor activity.

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Biomodulin T DB16529
biotech

Biomodulin T is a polypeptide fraction from bovine thymus with immunomodulatory effects.

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Biopterin DB03886
small molecule

A natural product that has been considered as a growth factor for some insects. [PubChem]

Kategori:
CoenzymesEnzymes and CoenzymesHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Peptide deformylase, mitochondrialSepiapterin reductase6-pyruvoyl tetrahydrobiopterin synthase +1
Waktu Paruh-
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Genetik -
Biotin Approved DB00121
small molecule | CAS: 58-85-5

A water-soluble, enzyme co-factor present in minute amounts in every living cell. It occurs mainly bound to proteins or polypeptides and is abundant in liver, kidney, pancreas, yeast, and milk.

Kategori:
Alimentary Tract and MetabolismCoenzymesDiet, Food, and Nutrition +10
Target Protein:
Propionyl-CoA carboxylase beta chain, mitochondrialBiotin--protein ligaseMethylcrotonoyl-CoA carboxylase beta chain, mitochondrial +5
Waktu Paruh-
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Bioymifi DB17493
small molecule | CAS: 1420071-30-2

Bioymifi is a small molecule that acts as a tumor necrosis factor-related apoptosis-induced ligand (TRAIL) mimetic. Upon binding to the death receptor 5 (DR5) on cancer cells, bioymifi triggers apoptosis, possibly through a caspase-dependent pathway. Bioymifi…

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingImides +5
Target Protein:
Tumor necrosis factor receptor superfamily member 10B
Waktu Paruh-
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Biperiden Approved DB00810
small molecule | CAS: 514-65-8

A muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteriosclerotic, idiopathic, and postencephalitic parkinsonism. It has also been used to alleviate extrapyramidal symptoms induc…

Kategori:
Agents producing tachycardiaAnti-Dyskinesia AgentsAnti-Parkinson Drugs +18
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
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Genetik -
small molecule | CAS: 792-74-5

Nissel has been investigated for the treatment of Chronic Liver Disease.

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Birabresib DB15189
small molecule | CAS: 202590-98-5

Birabresib is under investigation in clinical trial NCT02698176 (A Dose Exploration Study With MK-8628 in Participants With Selected Advanced Solid Tumors (MK-8628-006)).

Kategori:
AmidesAminesAnilides +2
Target Protein:
Bromodomain-containing protein 2Bromodomain-containing protein 4
Waktu Paruh-
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Birch bark extract Approved DB16536
small molecule | CAS: 84012-15-7

Birch bark extract is rich in triterpenoids with beneficial biological and pharmacological activities. Some of the compounds identified in it include betulin, [lupeol], [betulinic acid], oleanolic acid, and erythrodiol.[A249945] Birch bark extract is obtained…

Kategori:
Anti-Inflammatory AgentsAnti-inflammatory Agents, MiscellaneousBiological Products +7
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Bird pepper Approved DB14262
biotech

Bird pepper is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Biricodar DB04851
small molecule | CAS: 159997-94-1

The pipecolinate derivative biricodar (VX-710) is a clinically applicable modulator of P-glycoprotein (Pgp) and multidrug resistance protein (MRP-1).

Kategori:
P-glycoprotein inhibitors
Target Protein:
ATP-dependent translocase ABCB1ATP-binding cassette sub-family B member 5Multidrug resistance-associated protein 1 +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Birinapant DB11782
small molecule | CAS: 1260251-31-7

Birinapant has been investigated for the treatment of Myelodysplastic Syndrome (MDS) and Chronic Myelomonocytic Leukemia (CMML).

Kategori:
Amino Acids, Peptides, and ProteinsHeterocyclic Compounds, Fused-RingOligopeptides +1
Target Protein:
E3 ubiquitin-protein ligase XIAPBaculoviral IAP repeat-containing protein 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Biropepimut-S DB14816
biotech | CAS: 911338-45-9

Biropepimut-S is under investigation in clinical trial NCT02873819 (Safety and Efficacy Study of GL-0817 (With Cyclophosphamide) for the Prevention of Recurrence of Squamous Cell Carcinoma of the Oral Cavity).

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Birtamimab DB16414
biotech | CAS: 1608108-91-3

Birtamimab is under investigation in clinical trial NCT02312206 (The VITAL Amyloidosis Study, a Global Phase 3, Efficacy and Safety Study of NEOD001 in Patients With AL Amyloidosis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Genetik -
small molecule | CAS: 1282618-49-8

Deskripsi belum tersedia.

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small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
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Genetik -
small molecule

Deskripsi belum tersedia.

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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serum amyloid P-component
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serum amyloid P-component
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin G
Waktu Paruh-
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Bisacodyl Approved DB09020
small molecule | CAS: 603-50-9

Bisacodyl, a diphenylmethane derivative, is a commonly used over the counter stimulant laxative for occasional constipation.[A233300,L13362] Both bisacodyl and [picosulfate] are metabolized to the same active metabolite bis-(p-hydroxyphenyl)-pyridyl-2-methane…

Kategori:
Alimentary Tract and MetabolismBenzene DerivativesContact Laxatives +8
Target Protein:
Aquaporin-3Sodium/Potassium Transporting ATPase
Waktu ParuhData regarding the …
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Bisantrene DB17247
small molecule | CAS: 78186-34-2

Deskripsi belum tersedia.

Kategori:
Antibiotics, AntineoplasticAntineoplastic Agents
Waktu Paruh-
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Bisegliptin DB06127
small molecule | CAS: 862501-61-9

Bisegliptin is a compound for the treatment of type 2 diabetes. It is an orally active, dipeptidyl peptidase-IV (DPPIV) inhibitor which lowers blood glucose levels by blocking the degradation of the hormone GLP-1 thereby stimulating glucose-dependent insulin …

Kategori:
Agents causing angioedemaBlood Glucose Lowering AgentsDPP-IV Inhibitors
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Bismuth cation DB14572
small molecule | CAS: 23713-46-4

Deskripsi belum tersedia.

Kategori:
AntacidsAnti-Infective AgentsAnti-Ulcer Agents +2
Waktu Paruh-
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small molecule | CAS: 5892-10-4

Deskripsi belum tersedia.

Kategori:
AlkaliesAnionsBismuth containing drugs +11
Waktu Paruh-
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Bismuth subcitrate potassium Approved DB09275
small molecule | CAS: 880149-29-1

A bismuth compound used for peptic ulcer and gastro-oesophageal reflux disease (GORD).

Kategori:
Alimentary Tract and MetabolismAnti-Infective AgentsAnti-Ulcer Agents +5
Target Protein:
ATP-dependent Clp protease ATP-binding subunit ClpX
Waktu ParuhThe elimination hal…
Vol. Distribusi-
KlirensThe rate of renal e…
Genetik -
Bismuth subgallate Approved DB13909
small molecule | CAS: 99-26-3

Bismuth subgallate is a yellow colored substance that presents as an odorless powder that undergoes discoloration when exposed to sunlight. It is a heavy metal salt of gallic acid that is highly insoluble and poorly absorbed. Possessing protective effects on …

Kategori:
Acids, CarbocyclicAntacids and AdsorbentsAnti-Infective Agents +12
Waktu ParuhThe bismuth compone…
Vol. DistribusiIn general, oral ad…
KlirensOn average, the blo…
Genetik -
Bismuth subnitrate Approved DB13209
small molecule | CAS: 1304-85-4

Bismuth subnitrate, also referred to as bismuth oxynitrate or bismuthyl nitrate, is a highly water-soluble crystalline compound that has been used as a treatment for duodenal ulcers and anti-diarrheic agent [A33012]. The use of bismuth substrate as an active …

Kategori:
Alimentary Tract and MetabolismAntacidsBismuth containing drugs +11
Waktu ParuhThe distribution ha…
Vol. DistribusiBismuth has been sh…
KlirensNo pharmacokinetic …
Genetik -
Bismuth subsalicylate Approved DB01294
small molecule | CAS: 14882-18-9

Bismuth subsalicylate is an antacid and anti-diarrheal agent. Exhibiting antibacterial and gastroprotective properties, bismuth subsalicylate is an insoluble salt of [salicylic acid] linked to trivalent [bismuth cation]. Each molecule of bismuth subsalicylate…

Kategori:
Acids, CarbocyclicAntacids and AdsorbentsAntidiarrheals +16
Waktu ParuhThe terminal half-l…
Vol. DistribusiThere is no informa…
KlirensThe renal clearance…
Genetik -
Bisoctrizole Approved DB11262
small molecule | CAS: 103597-45-1

Bisoctrizole, or methylene bis-benzotriazolyl tetramethylbutylphenol, is a broad-spectrum organic UV filter that is marketed as Tinosorb M [A19212]. It is a benzotriazole-based organic compound that absorbs, reflects, and scatters both UV-A and UV-B rays. Bis…

Kategori:
Sunscreen Agents
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Bisoprolol Approved DB00612
small molecule | CAS: 66722-44-9

Bisoprolol is a cardioselective ?1-adrenergic blocking agent used to treat high blood pressure.[A180472,L7219] It is considered a potent drug with a long-half life that can be used once daily to reduce the need for multiple doses of antihypertensive drugs.[A1…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-1 Receptor Antagonists +29
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Waktu ParuhA pharmacokinetic s…
Vol. DistribusiThe volume of distr…
KlirensTotal body clearanc…
Genetik -
Bisoxatin Approved DB09219
small molecule | CAS: 17692-24-9

Bisoxatin is a stimulant laxative which increases peristalsis and inhibits absorbtion of water and ions in the intestine [L926]. It is marketed in Belgium under the tradename Wylaxine and used for the treatment of constipation and for preparation of the colon…

Kategori:
Alimentary Tract and MetabolismContact LaxativesDrugs for Constipation +2
Waktu Paruh-
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Genetik -
small molecule | CAS: 14008-48-1

Deskripsi belum tersedia.

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Bisphenol A DB06973
small molecule | CAS: 80-05-7

Deskripsi belum tersedia.

Kategori:
Air PollutantsAir Pollutants, OccupationalAntioxidants +13
Target Protein:
Androgen receptorEstrogen receptor betaEstrogen-related receptor gamma
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Bisphenol A diglycidyl ether Approved DB14083
small molecule | CAS: 1675-54-3

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBisphenolsCarcinogens +8
Target Protein:
Cation channel sperm-associated protein 1
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Bisphenol Z DB07485
small molecule | CAS: 843-55-0

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesCycloparaffinsPhenols
Target Protein:
Estrogen-related receptor gamma
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 403717-06-6

Bisphosphocin Nu-3 is under investigation in clinical trial NCT02737722 (Topically Applied Bisphosphocin Nu-3 on Infected Diabetic Ulcers of Subjects With Type I or II Diabetes Mellitus).

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