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11793

Total database: 17430
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8607 (73.0%)
Target
6418 (54.4%)
Genomik
102 (0.9%)
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11793 (100.0%)

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Halaman 67 / 236
Ceftibuten Approved DB01415
small molecule | CAS: 97519-39-6

Ceftibuten is a third-generation cephalosporin antibiotic that is orally-administered. It is typically used to treat acute bacterial exacerbations of chronic bronchitis (ABECB), acute bacterial otitis media, pharyngitis, and tonsilitis.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 1APenicillin-binding protein 1B +1
Waktu Paruh-
Vol. Distribusi* 0.21 L/kg [adult …
Klirens-
Genetik -
Ceftiofur DB11485
small molecule | CAS: 80370-57-6

Ceftiofur is a third generation cephalosporin antibiotic, first described in 1987, and now used in veterinary medicine. It is marketed by pharmaceutical company Zoetis as Excenel, and is the active ingredient in that company's Specramast LC (lactating cow for…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceftizoxime Approved DB01332
small molecule | CAS: 68401-81-0

A semisynthetic cephalosporin antibiotic which can be administered intravenously or by suppository. The drug is highly resistant to a broad spectrum of beta-lactamases and is active against a wide range of both aerobic and anaerobic gram-positive and gram-neg…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 1BPeptidoglycan transpeptidase +1
Waktu Paruh-
Vol. DistribusiThe mean apparent v…
Klirens-
Genetik -
Ceftobiprole Approved DB04918
small molecule | CAS: 209467-52-7

Ceftobiprole is a fifth-generation semisynthetic cephalosporin antibacterial which is available commercially as the prodrug [ceftobiprole medocaril]. Ceftobiprole is a broad-spectrum agent with demonstrated activity against both Gram-positive and Gram-negativ…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
MecAPenicillin-binding protein 2xPenicillin-binding protein 2B +2
Waktu ParuhThe half-life of ac…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
Ceftobiprole medocaril Approved DB14733
small molecule | CAS: 376653-43-9

Ceftobiprole medocaril is a prodrug of [ceftobiprole], a fifth-generation semisynthetic cephalosporin antibacterial. Ceftobiprole is a broad-spectrum agent with demonstrated activity against both Gram-positive and Gram-negative bacteria, including antibiotic-…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
MecAPenicillin-binding protein 2BPenicillin-binding protein 2X
Waktu ParuhThe half-life of ac…
Vol. DistribusiThe steady-state vo…
KlirensThe mean clearance …
Genetik -
Ceftolozane Approved DB09050
small molecule | CAS: 689293-68-3

Ceftolozane is a semi-synthetic broad-spectrum fifth generation cephalosporin.[L6685] It was approved by the FDA in 2014 for use in combination with [Tazobactam] for the treatment of serious infections, such as intra-abdominal infections and complicated urina…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +8
Target Protein:
Penicillin-binding protein 1BCell division proteinPenicillin-binding protein 1C +2
Waktu Paruh2.77 hours on day 1…
Vol. Distribusi13.5 L.[L41618] Tis…
KlirensThe renal clearance…
Genetik -
Ceftriaxone Approved DB01212
small molecule | CAS: 73384-59-5

Ceftriaxone is a broad-spectrum third-generation cephalosporin antibiotic.[A215582] It has a very long half-life compared to other cephalosporins and is high penetrable into the meninges[A215582], eyes[A215647], and inner ear[A215627]. Ceftriaxone has broader…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
Penicillin-binding protein 2BSolute carrier family 22 member 11Solute carrier family 22 member 6 +2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe plasma clearanc…
Genetik -
Cefuroxime Approved DB01112
small molecule | CAS: 55268-75-2

Broad-spectrum cephalosporin antibiotic resistant to beta-lactamase. It has been proposed for infections with gram-negative and gram-positive organisms, gonorrhea, and haemophilus.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
Penicillin-binding protein 1A
Waktu ParuhApproximately 80 mi…
Vol. Distribusi-
Klirens-
Genetik -
Celastrol DB18736
small molecule | CAS: 34157-83-0

Celastrol is a pentacyclic triterpenoid isolated from the root extracts of _Tripterygium wilfordii_.[L50567]

Kategori:
TerpenesTripterygiumTriterpenes
Target Protein:
Interleukin-1 betaTumor necrosis factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Celecoxib Approved DB00482
small molecule | CAS: 169590-42-5

Celecoxib, a selective cyclooxygenase-2 (COX-2) inhibitor, is a nonsteroidal anti-inflammatory drug (NSAID) which is known for its decreased risk of causing gastrointestinal bleeding compared to other NSAIDS.[A181544] It is used to manage symptoms of various …

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +41
Target Protein:
Prostaglandin G/H synthase 2Signal transducer and activator of transcription 3Sialidase-1 +4
Gen Terkait:
CYP2C9
Waktu ParuhThe effective half-…
Vol. DistribusiThe apparent volume…
KlirensApparent clearance …
Genetik 1 Varian
Celgosivir DB06580
small molecule | CAS: 121104-96-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingIndolizines
Target Protein:
Maltase-glucoamylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Celiprolol Approved DB04846
small molecule | CAS: 56980-93-9

Celiprolol is indicated for the management of mild to moderate hypertension and effort-induced angina pectoris. It is simultaneously a selective ?1 receptor antagonist, a ?2 receptor partial agonist and a weak ?2 receptor antagonist. In 2010 a clinical trial …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic Antagonists +30
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor +3
Waktu Paruh5 hours
Vol. DistribusiThe distribution vo…
KlirensCleared by both ren…
Genetik -
Celivarone DB16012
small molecule | CAS: 401925-43-7

Celivarone is under investigation in clinical trial NCT00233441 (Placebo Controlled Double-blind Dose Ranging Study of the Efficacy and Safety of SSR149744C 50, 100, 200 or 300 Mg OD With Amiodarone as Calibrator for the Maintenance of Sinus Rhythm in Patient…

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cellobiose DB02061
small molecule | CAS: 528-50-7

A disaccharide consisting of two glucose units in beta (1-4) glycosidic linkage. Obtained from the partial hydrolysis of cellulose. [PubChem]

Kategori:
CarbohydratesCelluloseCompounds used in a research, industrial, or household setting +4
Target Protein:
Endoglucanase GEndoglucanase 5AEndoglucanase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The Cellspan Esophageal ImplantTM (CEI) composes of autologous adipose-derived mesenchymal stromal cells (Ad-MSC) seeded onto a polyurethane tubular mesh cell delivery device.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cemdisiran DB16121
biotech | CAS: 1639264-46-2

Cemdisiran is under investigation in clinical trial NCT03841448 (A Study of Cemdisiran in Adults With Immunoglobulin a Nephropathy (Igan)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cemdomespib DB18953
small molecule | CAS: 1450642-92-8

Cemdomespib is under investigation in clinical trial NCT05895552 (A Phase 2 Study of RTA 901 in Patients With Diabetic Peripheral Neuropathic Pain (CYPRESS)).

Kategori:
AminesCarbohydratesEthylamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cemiplimab Approved DB14707
biotech | CAS: 1801342-60-8

Cemiplimab is a fully human monoclonal antibody that works against programmed death receptor-1 (PD-1), which is a negative regulator of T cell function. By blocking PD-1, cemiplimab works to enhance T cell-mediated antitumour responses.[L39804] Cemiplimab …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
Programmed cell death protein 1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensCemiplimab clearanc…
Genetik -
Cemsidomide DB18400
small molecule | CAS: 2504235-67-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cendakimab DB18427
biotech

Cendakimab is a recombinant humanized anti-interleukin 13 (IL-13) monoclonal antibody.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenegermin Approved DB13926
biotech | CAS: 1772578-74-1

Cenegermin is a human beta-nerve growth factor (beta-ngf)-(1-118)- peptide (non-covalent dimer) produced in escherichia coli. It received European Union Approval in July 2017 for the treatment of moderate to severe neurotrophic keratitis. Cenegermin received …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +7
Target Protein:
High affinity nerve growth factor receptorTumor necrosis factor receptor superfamily member 16
Waktu ParuhHalf-life data spec…
Vol. DistribusiAfter eye drop admi…
KlirensAlthough the system…
Genetik -
Cenerimod DB12705
small molecule | CAS: 1262414-04-9

Cenerimod has been used in trials studying the treatment of Systemic Lupus Erythematosus.

Kategori:
AlcoholsGlycolsOxazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenersen DB15455
biotech | CAS: 415168-49-9

Cenersen is under investigation in clinical trial NCT02243124 (A Study of Aezea® (Cenersen) in Transfusion Dependent Anemia Associated With Myelodysplastic Syndrome (MDS)).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenisertib DB06347
small molecule | CAS: 871357-89-0

Cenisertib is an aurora kinase inhibitor.

Kategori:
Bridged-Ring Compounds
Target Protein:
Aurora kinase BAurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cenobamate Approved DB06119
small molecule | CAS: 913088-80-9

Cenobamate, or YKP-3089, is an antiepileptic drug developed by SK Pharmaceuticals and used to treat partial onset seizures.[A188442,L10653] The exact mechanism of action has not been described in the literature, though it positively modulates GABA<sub>A</sub>…

Kategori:
Acids, AcyclicAnticonvulsantsBenzene Derivatives +34
Target Protein:
Voltage-gated sodium channel alpha subunitGamma-aminobutyric acid receptor subunit alpha-1
Waktu ParuhThe terminal half l…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Censavudine DB12074
small molecule | CAS: 634907-30-5

Censavudine has been used in trials studying the treatment of HIV-1 Infection.

Kategori:
Anti-HIV AgentsDeoxyribonucleosidesNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Centella asiatica Approved DB14256
biotech

Centella asiatica is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Agents that reduce seizure thresholdAngiospermsApiaceae +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Centhaquine DB16122
small molecule | CAS: 57961-90-7

Centhaquine is under investigation in clinical trial NCT04045327 (Efficacy of PMZ-2010 (Centhaquine) a Resuscitative Agent for Hypovolemic Shock).

Kategori:
Adrenergic and Dopaminergic AgentsCardiac Stimulants Excl. Cardiac GlycosidesCardiac Therapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CEP-37440 DB13060
small molecule | CAS: 1391712-60-9

CEP-37440 has been used in trials studying the treatment of Solid Tumors.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Focal adhesion kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CEP-9722 DB14882
small molecule | CAS: 916574-83-9

CEP-9722 is under investigation in clinical trial NCT01345357 (Study of CEP-9722 in Combination With Gemcitabine and Cisplatin in Patients With Advanced Solid Tumors or Mantle Cell Lymphoma).

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingImides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1192706-52-7

Cepeginterferon alfa-2B is under investigation in clinical trial NCT01889433 (An Open-label Comparative Efficacy and Safety Study of Algeron (Cepeginterferon Alfa-2b) in Treatment-naive Patients With Chronic Hepatitis C).

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP1A2 Inhibitors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cephalexin Approved DB00567
small molecule | CAS: 15686-71-2

Cephalexin is the first of the first generation cephalosporins.[A179071,A179074] This antibiotic contains a beta lactam and a dihydrothiazide.[A179071] Cephalexin is used to treat a number of susceptible bacterial infections through inhibition of cell wall s…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +23
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2aPenicillin-binding protein 1b +2
Waktu ParuhThe half life of ce…
Vol. Distribusi5.2-5.8L.[A179068]
KlirensClearance from one …
Genetik -
Cephaloglycin Approved DB00689
small molecule | CAS: 3577-01-3

A cephalorsporin antibiotic that is no longer commonly used.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +7
Target Protein:
Penicillin-binding protein 1B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Agents that reduce seizure threshold
Target Protein:
D-alanyl-D-alanine carboxypeptidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cephalosporin C DB03313
small molecule | CAS: 61-24-5

Deskripsi belum tersedia.

Kategori:
Agents that reduce seizure thresholdAmidesbeta-Lactams +4
Target Protein:
Penicillin-binding protein 1bPeptidoglycan synthase FtsIPenicillin-binding protein 1A +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cepharanthine DB16824
small molecule | CAS: 481-49-2

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnalgesicsAnalgesics, Non-Narcotic +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceralasertib DB14917
small molecule | CAS: 1352226-88-0

Ceralasertib is under investigation in clinical trial NCT03682289 (Phase II Trial of AZD6738 Alone and in Combination With Olaparib).

Kategori:
AmidesHeterocyclic Compounds, Fused-RingOxazines +2
Target Protein:
Serine/threonine-protein kinase ATR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceralifimod DB16123
small molecule | CAS: 891859-12-4

Ceralifimod is under investigation in clinical trial NCT01226745 (Phase 2 Extension Trial in Patients With Relapsing-remitting Multiple Sclerosis (RRMS)).

Kategori:
AzetinesImmunologic FactorsImmunosuppressive Agents +1
Target Protein:
Sphingosine 1-phosphate receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceramide AP DB14705
small molecule | CAS: 212070-45-6

Deskripsi belum tersedia.

Kategori:
AmidesCarbohydratesGlycoconjugates +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceramide NG DB14706
small molecule | CAS: 2304-80-5

Deskripsi belum tersedia.

Kategori:
AmidesCarbohydratesGlycoconjugates +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CERC-301 DB12063
small molecule | CAS: 808732-98-1

Mk 0657 has been used in trials studying the treatment of Major Depressive Disorder.

Kategori:
Receptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Target Protein:
Glutamate receptor ionotropic, NMDA 2B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerdulatinib DB15499
small molecule | CAS: 1198300-79-6

Cerdulatinib is under investigation in clinical trial NCT04021082 (CELTIC-1: A Phase 2B Study of Cerdulatinib in Patients With Relapsed/refractory Peripheral T-cell Lymphoma (PTCL)).

Kategori:
Sulfur Compounds
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase JAK2Tyrosine-protein kinase SYK +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
CERE-120 DB05637
biotech | CAS: 1148126-35-5

CERE-120 is an investigational drug consisting of an adeno-associated virus (AAV) that was engineered to carry the human gene for neurturin, a neurotrophic (growth) factor. It was under investigation in clinical trials for the treatment of Parkinson's Disease.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerebrolysin DB16599
biotech | CAS: 12656-61-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBrainCentral Nervous System Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1509916-03-3

Cergutuzumab amunaleukin is under investigation in clinical trial NCT02004106 (A Study to Evaluate Safety, Pharmacokinetics, and Efficacy of RO6895882 in Participants With Advanced and/or Metastatic Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ceritinib Approved DB09063
small molecule | CAS: 1032900-25-6

Ceritinib is used for the treatment of adults with anaplastic lymphoma kinase (ALK)-positive metastatic non-small cell lung cancer (NSCLC) following failure (secondary to resistance or intolerance) of prior crizotinib therapy. About 4% of patients with NSCLC …

Kategori:
Anaplastic lymphoma kinase (ALK) inhibitorsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +25
Target Protein:
ALK tyrosine kinase receptor
Waktu ParuhThe terminal half l…
Vol. DistribusiThe apparent volume…
KlirensThe geometric mean …
Genetik -
Cerium dioxide DB18493
small molecule | CAS: 1306-38-3

Deskripsi belum tersedia.

Kategori:
ElementsLanthanoid Series ElementsMetals +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Cerivastatin Approved DB00439
small molecule | CAS: 145599-86-6

On August 8, 2001 the U.S. Food and Drug Administration (FDA) announced that Bayer Pharmaceutical Division voluntarily withdrew Baycol from the U.S. market, due to reports of fatal rhabdomyolysis, a severe adverse reaction from this cholesterol-lowering (lipi…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBCRP/ABCG2 Substrates +34
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh2-3 hours
Vol. Distribusi-
Klirens-
Genetik -
Cerliponase alfa Approved DB13173
biotech | CAS: 151662-36-1

Cerliponase alfa is a hydrolytic lysosomal N-terminal tripeptidyl peptidase-1 (TPP1).[L51319] On April 27, 2017, cerliponase alfa was first approved by the FDA as the first treatment for neuronal ceroid lipofuscinosis type 2 (CLN2), also known as TPP1 deficie…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsEnzymes +6
Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu ParuhFollowing intravent…
Vol. DistribusiFollowing intravent…
KlirensFollowing intravent…
Genetik -
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