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14063

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10481 (74.5%)
Target
8038 (57.2%)
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107 (0.8%)
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14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 67 / 282
Axatilimab Approved DB16388
biotech | CAS: 2155851-88-8

Axatilimab is a humanized IgG4 monoclonal antibody produced in Chinese hamster ovary cells.[L51194] It is targeted against macrophage colony-stimulating factor 1 receptor (CSF-1R), causing a reduction in circulating levels of monocytes and macrophages respons…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Macrophage colony-stimulating factor 1 receptor
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe volume of distr…
KlirensThe total clearance…
Genetik -
Axelopran DB12013
small molecule | CAS: 949904-48-7

Axelopran has been used in trials studying the treatment of OIC and Opioid-induced Constipation.

Kategori:
Acids, CarbocyclicAlkaloidsAmides +5
Target Protein:
Mu-type opioid receptor
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Axicabtagene ciloleucel Approved DB13915
biotech

Axicabtagene ciloleucel is an anti-CD19 chimeric antigen receptor (CAR) T-cell therapy. The drug has a unique mechanism of action, as it utilizes the patient's own T cells, which play a central role in immune response to cancer.[A216163] Once T-cells are coll…

Kategori:
AntigensAntigens, CDAntigens, Differentiation +16
Target Protein:
B-lymphocyte antigen CD19
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Axitinib Approved DB06626
small molecule | CAS: 319460-85-0

Axitinib is a second generation tyrosine kinase inhibitor that works by selectively inhibiting vascular endothelial growth factor receptors (VEGFR-1, VEGFR-2, VEGFR-3).[L6676] Through this mechanism of action, axitinib blocks angiogenesis, tumour growth and m…

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +31
Target Protein:
Tyrosine-protein kinase ABL1Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2 +1
Waktu ParuhAxitinib has a half…
Vol. DistribusiThe volume of distr…
KlirensThe average clearan…
Genetik -
Axomadol DB16100
small molecule | CAS: 187219-99-4

Axomadol is under investigation in clinical trial NCT01043263 (Efficacy and Safety of EN3324 (Axomadol) in Subjects With Chronic Low Back Pain).

Kategori:
AlcoholsCyclohexanesCycloparaffins +3
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AXV101 DB18320
biotech

Deskripsi belum tersedia.

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AZ-3102 DB18502
small molecule

AZ-3102 is a Biphenyl-substituted L-ido configured deoxynojirimycin derivative

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Azacitidine Approved DB00928
small molecule | CAS: 320-67-2

Azacitidine is a pyrimidine nucleoside analogue with anti-neoplastic activity. It differs from cytosine by the presence of nitrogen in the C5-position, key in its hypomethylating activity.[A1406,A1413,A1415] Two main mechanisms of action have been proposed fo…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
DNA (cytosine-5)-methyltransferase 1RNADNA
Waktu ParuhThe mean half-life …
Vol. DistribusiIn patients given a…
KlirensAzacitidine has an …
Genetik -
Azadirachta indica leaf Approved DB14352
biotech

Azadirachta indica leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Azadirachtin DB19419
small molecule | CAS: 11141-17-6

Azadirachtin is under investigation in clinical trial NCT06617026 (Short-term Outcome of Medical vs. Surgical Management of Chronic Anal Fissure).

Kategori:
AgrochemicalsAzadirachtaCompounds used in a research, industrial, or household setting +5
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Azafenidin DB19031
small molecule | CAS: 68049-83-2

Azafenidin is under investigation in clinical trial NCT01726582 (Pancreas Cancer: Molecular Profiling as a Guide to Therapy Before and After Surgery ("Personalized Medicine")).

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Azanidazole DB13350
small molecule | CAS: 62973-76-6

Deskripsi belum tersedia.

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsGenito Urinary System and Sex Hormones +5
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Azapentacene DB15951
small molecule | CAS: 3863-80-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
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Azaperone DB11376
small molecule | CAS: 1649-18-9

Azaperone is a pyridinylpiperazine and butyrophenone agent that is capable of eliciting neuroleptic sedative and antiemetic effects. It is subsequently employed predominantly as a veterinary tranquilizer and mainly for pigs and elephants. At the same time, th…

Kategori:
Antipsychotic AgentsAntipsychotic Agents (First Generation [Typical])Butyrophenones +11
Target Protein:
D(3) dopamine receptorD(2) dopamine receptor
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Azapetine DB13727
small molecule | CAS: 146-36-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingPeripheral Vasodilators
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Azapropazone DB07402
small molecule | CAS: 13539-59-8

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +13
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Azaribine Approved DB19364
small molecule | CAS: 2169-64-4

Deskripsi belum tersedia.

Kategori:
Aza CompoundsDermatologicalsNucleic Acids, Nucleotides, and Nucleosides +4
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Azasetron DB16837
small molecule | CAS: 123040-69-7

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsAntiemeticsAutonomic Agents +7
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Azatadine Approved DB00719
small molecule | CAS: 3964-81-6

Antihistamines such as azatadine appear to compete with histamine for histamine H1- receptor sites on effector cells. The antihistamines antagonize those pharmacological effects of histamine which are mediated through activation of H1- receptor sites and ther…

Kategori:
Agents that reduce seizure thresholdAnticholinergic AgentsAntihistamines for Systemic Use +10
Target Protein:
Histamine H1 receptor
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Azathioprine Approved DB00993
small molecule | CAS: 446-86-6

Azathioprine is a prodrug of 6-mercaptopurine, first synthesized in 1956 by Gertrude Elion, William Lange, and George Hitchings in an attempt to produce a derivative of 6-mercaptopurine with a better therapeutic index.[A189678,A189687,A189690] Azathioprine is…

Kategori:
AntimetabolitesAntineoplastic and Immunomodulating AgentsAntirheumatic Agents +21
Target Protein:
AmidophosphoribosyltransferaseRas-related C3 botulinum toxin substrate 1
Gen Terkait:
TPMT TPMT TPMT
Waktu ParuhThe half life of az…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik 3 Varian
AZD-0328 DB12145
small molecule | CAS: 220099-91-2

AZD0328 has been used in trials studying the treatment and basic science of Schizophrenia and Alzheimer's Disease.

Kategori:
Receptors, Nicotinic
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
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AZD-0424 DB13088
small molecule | CAS: 692054-06-1

AZD0424 has been used in trials studying the treatment of Advanced Solid Tumours.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
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AZD-1236 DB11961
small molecule | CAS: 459814-89-2

AZD1236 has been used in trials studying the basic science and treatment of Cystic Fibrosis and Chronic Obstructive Pulmonary Disease.

Kategori:
AmidesImidazolesImidazolidines +2
Target Protein:
Macrophage metalloelastase
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AZD-1305 DB11766
small molecule | CAS: 872045-91-5

AZD1305 has been used in trials studying the treatment and basic science of Atrial Flutter, Atrial Fibrillation, and Left Ventricle Function.

Kategori:
Acids, AcyclicAza Compounds
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AZD-1386 DB15333
small molecule | CAS: 942937-80-6

AZD-1386 is under investigation in clinical trial NCT00945178 (Double-blind Placebo-controlled 2-part Study Assessing the Safety, Tolerability and PK of AZD1386 in Healthy Volunteers).

Kategori:
Heterocyclic Compounds, Fused-Ring
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AZD-1480 DB12588
small molecule | CAS: 935666-88-9

AZD1480 has been used in trials studying the treatment of Solid Malignancies, Post-Polycythaemia Vera, Primary Myelofibrosis (PMF), and Essential Thrombocythaemia Myelofibrosis.

Kategori:
Janus Kinase 2, antagonists & inhibitorsJanus Kinases, antagonists & inhibitors
Target Protein:
Tyrosine-protein kinase JAK2
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AZD-1656 DB14810
small molecule | CAS: 919783-22-5

AZD-1656 is under investigation in clinical trial NCT00747175 (A Study to Evaluate Safety, Tolerability and P-Glucose After Multiple Ascending Oral Doses of AZD1656 in Type 2 Diabetes).

Kategori:
AzetinesGlucokinase
Target Protein:
Hexokinase-4
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AZD-1940 DB17077
small molecule | CAS: 881413-29-2

Deskripsi belum tersedia.

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AZD-1981 DB11946
small molecule | CAS: 802904-66-1

AZD1981 has been used in trials studying the treatment and basic science of Asthma, Postmenopausal, Pharmakokinetic, Asthma Patients, and Drug Interaction, among others.

Target Protein:
Prostaglandin D2 receptor 2
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AZD-2066 DB12644
small molecule | CAS: 934282-55-0

AZD2066 has been used in trials studying the treatment and basic science of Pain, Chronic Pain, Reflux Episodes, Neuropathic Pain, and Diabetic Neuropathy, among others.

Target Protein:
Metabotropic glutamate receptor 5
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AZD-3043 DB12576
small molecule | CAS: 579494-66-9

AZD3043 has been used in trials studying the treatment and basic science of Safety, Sedation, Tolerability, and Pharmacokinetics.

Kategori:
Acids, CarbocyclicCentral Nervous System DepressantsHypnotics and Sedatives
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3
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AZD-3759 DB14795
small molecule | CAS: 1626387-80-1

AZD-3759 is under investigation in clinical trial NCT03360929 (Evaluate Safety, Tolerability, Pharmacokinetics and Anti-tumor Activity of AZD3759).

Kategori:
Heterocyclic Compounds, Fused-Ring
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AZD-3839 DB12368
small molecule | CAS: 1227163-84-9

AZD3839 has been used in trials studying the basic science of Safety, Tolerability, Alzheimer's Disease, and Blood Concentration.

Kategori:
Heterocyclic Compounds, Fused-Ring
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AZD-4017 DB14875
small molecule | CAS: 1024033-43-9

AZD-4017 is under investigation in clinical trial NCT01173471 (A Phase IIa Study to Assess the Tolerability, Safety, and Efficacy of AZD4017 for Raised Intra-ocular Pressure).

Kategori:
11-beta-Hydroxysteroid Dehydrogenase Type 1, antagonists & inhibitorsNicotinic AcidsPyridines
Target Protein:
11-beta-hydroxysteroid dehydrogenase 1
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AZD-4547 DB12247
small molecule | CAS: 1035270-39-3

AZD4547 has been used in trials studying the treatment of Cancer, LYMPHOMA, Gastric Cancer, Adenocarcinoma, and Solid Neoplasm, among others.

Target Protein:
Fibroblast growth factor receptor 1
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AZD-4818 DB12002
small molecule | CAS: 1003566-93-5

AZD4818 has been used in trials studying the treatment of Chronic Obstructive Pulmonary Disease (COPD).

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AZD-5069 DB16822
small molecule | CAS: 878385-84-3

Deskripsi belum tersedia.

Kategori:
AmidesSulfonesSulfur Compounds
Target Protein:
C-X-C chemokine receptor type 2
Waktu Paruh-
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AZD-5153 DB17018
small molecule | CAS: 1869912-39-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Bromodomain-containing protein 4
Waktu Paruh-
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AZD-5423 DB12280
small molecule | CAS: 1034148-04-3

AZD5423 has been used in trials studying the basic science and treatment of Asthma, Bioavailability and AUC, and Chronic Obstructive Pulmonary Disease (COPD).

Kategori:
AcetatesAcids, AcyclicAmides +4
Target Protein:
Glucocorticoid receptor
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AZD-5672 DB11804
small molecule | CAS: 780750-65-4

Azd5672 has been used in trials studying the basic science and treatment of Pharmacokinetics, Renal Impairment, and Rheumatoid Arthritis.

Kategori:
AcetamidesAmidesAnti-HIV Agents +5
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AZD-5991 DB14792
small molecule | CAS: 2143010-83-5

AZD-5991 is under investigation in clinical trial NCT03218683 (Study of AZD5991 in Relapsed or Refractory Haematologic Malignancies.).

Kategori:
Antineoplastic Agents
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AZD-6280 DB12210
small molecule | CAS: 942436-93-3

AZD6280 has been used in trials studying the basic science of Anxiety.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Opioid, delta, agonists
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-3
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AZD-6482 DB14980
small molecule | CAS: 1173900-33-8

AZD-6482 is under investigation in clinical trial NCT00688714 (Study to Investigate Safety and Tolerability of a Single Dose of AZD6482).

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +3
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
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AZD-7268 DB19203
small molecule | CAS: 1018988-00-5

AZD-7268 is under investigation in clinical trial NCT01020799 (AZD7268 Safety and Tolerability Study).

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Opioid, delta, agonists
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AZD-7295 DB12724
small molecule | CAS: 929890-64-2

AZD7295 has been investigated for the treatment of Hepatitis C.

Target Protein:
Genome polyprotein
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AZD-7325 DB13994
small molecule | CAS: 942437-37-8

AZD7325 is a high affinity, selective modulator of the GABAA receptor system. [L2936]

Kategori:
GABA ModulatorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-3Gamma-aminobutyric acid receptor subunit alpha-2
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AZD-7648 DB16834
small molecule | CAS: 2230820-11-6

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
DNA-dependent protein kinase catalytic subunit
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AZD-7687 DB14949
small molecule | CAS: 1166827-44-6

AZD-7687 is under investigation in clinical trial NCT01119352 (AZD7687 Multiple Ascending Dose Study).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
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AZD-7762 DB12242
small molecule | CAS: 860352-01-8

AZD7762 has been investigated for the treatment of Cancer, Solid Tumors, and Advanced Solid Malignancies.

Kategori:
AmidesSulfur Compounds
Target Protein:
Serine/threonine-protein kinase Chk1
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AZD-8055 DB12774
small molecule | CAS: 1009298-09-2

AZD8055 has been used in trials studying the treatment of Cancer, Lymphomas, Solid Tumors, MALIGNANT GLIOMA, and brainstem glioma, among others.

Kategori:
Oxazines
Target Protein:
Serine/threonine-protein kinase mTOR
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Menampilkan 3301–3350 dari 14063
Sebelumnya Halaman 67 / 282 Berikutnya