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6694

Total database: 17430
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4518 (67.5%)
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3751 (56.0%)
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81 (1.2%)
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6694 (100.0%)

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Halaman 66 / 134
Idelalisib Approved DB09054
small molecule | CAS: 870281-82-6

Idelalisib is a phosphoinositide 3-kinase inhibitor indicated in the treatment of chronic lymphocytic leukemia (CLL), relapsed follicular B-cell non-Hodgkin lymphoma (FL), and relapsed small lymphocytic lymphoma (SLL). For the treatment of relapsed CLL, it is…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +47
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu ParuhThe terminal elimin…
Vol. Distribusi23 L
Klirens14.9 L/hr
Genetik -
IDM-1 DB05292
small molecule

IDM-1 is IDM’s most advanced antibody-based Cell drug for the treatment of cancer. It is comprised of MAK(Monocytes-derived Activated Killer) cells associated with MDX-210, a bispecific anti-HER-2/neu antibody developed by Medarex Inc.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
IDM-4 DB05438
biotech

IDM-4 is an immuno-designed molecule that completed phase I/II of investigation for the treatment of Leukemia. It is a monoclonal antibody-specific antigen that can selectively target cancer-affected cells by coupling with tumor cell-killing MAK cells, which …

Waktu Paruh-
Vol. Distribusi-
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Genetik -
IDN-7314 DB18073
small molecule | CAS: 254750-11-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Idoxuridine Approved DB00249
small molecule | CAS: 54-42-2

An analog of deoxyuridine that inhibits viral DNA synthesis. The drug is used as an antiviral agent.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +15
Target Protein:
DNAThymidine kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idrevloride DB18042
small molecule | CAS: 1416973-63-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idrocilamide DB13297
small molecule | CAS: 6961-46-2

Deskripsi belum tersedia.

Kategori:
AlcoholsAminesAmino Alcohols +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idronoxil DB04915
small molecule | CAS: 81267-65-4

Idronoxil is a substance that is being studied in the treatment of cancer. It belongs to the family of drugs called signal transduction inhibitors.

Kategori:
BenzopyransChromonesFlavonoids +2
Target Protein:
E3 ubiquitin-protein ligase XIAPSphingosine kinase 1Ecto-NOX disulfide-thiol exchanger 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 56472-29-8

Deskripsi belum tersedia.

Kategori:
Fatty AcidsFatty Acids, MonounsaturatedFatty Acids, Unsaturated +1
Target Protein:
Phosphatidylcholine:ceramide cholinephosphotransferase 1Phosphatidylcholine:ceramide cholinephosphotransferase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IDUA-RTB DB18612
biotech

RTB-IDUA is a fusion protein of alpha-L-iduronidase (IDUA) and ricin transport subunit B (RTB).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Idursulfase Approved DB01271
biotech | CAS: 50936-59-9

Idursulfase is a purified form of human iduronate-2-sulfatase, a lysosomal enzyme. Idursulfase is produced by recombinant DNA technology in a human cell line. Idursulfase is an enzyme that hydrolyzes the 2-sulfate esters of terminal iduronate sulfate residues…

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +4
Target Protein:
Dermatan sulfateHeparan sulfatePerilipin-3
Waktu Paruh44 ± 19 minu…
Vol. Distribusi-
Klirens* 3 mL/min/kg [Pati…
Genetik -
Ieramilimab DB16419
biotech | CAS: 2137049-37-5

Ieramilimab is under investigation in clinical trial NCT02460224 (Safety and Efficacy of LAG525 Single Agent and in Combination With PDR001 in Patients With Advanced Malignancies.).

Waktu Paruh-
Vol. Distribusi-
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Ifenprodil DB08954
small molecule | CAS: 23210-56-2

N-methyl-D-aspartate (NMDA) receptors (NMDARs) are members of the ionotropic glutamate receptor family, with key roles in brain development and neurological function.[A220118, A220128] NMDARs are heterotetramers that typically involve a dimer of dimers of bot…

Kategori:
Adrenergic AgentsAdrenergic alpha-AntagonistsAdrenergic Antagonists +12
Target Protein:
Glutamate receptor ionotropic, NMDA 2BChymotrypsin-like elastase family member 1Glutamate receptor ionotropic, NMDA 1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ifidancitinib DB16191
small molecule | CAS: 1236667-40-5

Ifidancitinib is under investigation in clinical trial NCT03585296 (A Study of ATI-502 Topical Solution for the Treatment of Atopic Dermatitis).

Kategori:
Adrenal Cortex HormonesFused-Ring CompoundsNorpregnanes +4
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase JAK1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IFx-Hu2.0 DB18396
biotech

IFx-Hu2.0 is an investigational cancer vaccine. It is composed of plasmid DNA encoding the streptococcal membrane protein, Emm55, contained within a cationic polymer.

Waktu Paruh-
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IGN101 DB06500
biotech

IGN101 is an antibody-based cancer vaccine directed against epithelial cancers. It consists of 500 ug 17-1A antibody adsorbed on aluminum hydroxide.

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Vol. Distribusi-
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Genetik -
IGN301 DB05117
biotech

IGN301 is a cancer vaccine based on an anti-idiotypic antibody which provokes an immune response to Lewis Y. Lewis Y is a carbohydrate molecule expressed on the surface of tumor cells of epithelial origin (e.g. lung, intestinal, breast, prostate or ovarian ca…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ilacirnon DB16066
small molecule | CAS: 1100318-47-5

Ilacirnon (CCX-140) is under investigation in clinical trial NCT01440257 (A Study to Evaluate the Effect of CCX140-B on Urinary Albumin Excretion in Subjects With Type 2 Diabetes and Albuminuria).

Target Protein:
C-C chemokine receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ilepcimide DB16942
small molecule | CAS: 82857-82-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ilomastat DB02255
small molecule | CAS: 142880-36-2

Ilomastat is a broad-spectrum matrix metalloproteinase inhibitor.

Kategori:
AminesAmino Acids, Peptides, and ProteinsEnzyme Inhibitors +7
Target Protein:
Interstitial collagenaseMatrix metalloproteinase-14Neutrophil collagenase +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iloperidone Approved DB04946
small molecule | CAS: 133454-47-4

Iloperidone is a benzisoxazole [A263557] and an atypical antipsychotic agent that was first approved by the FDA on May 6, 2009.[A3024] It is considered to be a second-generation antipsychotic drug [A263552] with multiple receptor binding profile, although it …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +31
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 1A +14
Waktu ParuhThe observed mean e…
Vol. DistribusiThe apparent volume…
KlirensIloperidone has an …
Genetik -
Iloprost Approved DB01088
small molecule | CAS: 78919-13-8

Iloprost is an analog of prostacyclin (PGI2; epoprostenol), an endogenous prostanoid mainly produced in the vascular endothelium. It is more stable than prostacyclin, which is short-lived.[A263326] Iloprost consists of a mixture of the 4R and 4S diastereoisom…

Kategori:
Agents Causing Muscle ToxicityAntiplatelet agentsAutacoids +16
Target Protein:
Prostacyclin receptorProstaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtype +6
Waktu ParuhThe half-life of il…
Vol. DistribusiFollowing intraveno…
KlirensClearance in normal…
Genetik -
Iluzanebart DB18275
biotech | CAS: 2733621-19-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ILY101 DB05059
small molecule

ILY101 is a metal-free, non-absorbed polymeric drug designed for the selective binding and removal of phosphate anions from the gastrointestinal tract. ILY101 is being developed for the treatment of hyperphosphatemia in CKD patients on dialysis and works by …

Waktu Paruh-
Vol. Distribusi-
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Genetik -
IMA901 DB06628
biotech

IMA901 is a vaccine consists of tumor-associated peptides (TUMAPs).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imalumab DB15558
biotech | CAS: 1430205-07-4

Imalumab is under investigation in clinical trial NCT02540356 (Phase 1/2a Two-arm Dose-escalation Study of BAX69 in Subjects With Malignant Ascites of Ovarian Cancer).

Waktu Paruh-
Vol. Distribusi-
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Imatinib Approved DB00619
small molecule | CAS: 152459-95-5

Imatinib is a small molecule kinase inhibitor that revolutionized the treatment of cancer, particularly chronic myeloid leukemia, in 2001.[A249305] It was deemed a "miracle drug" due to its clinical success, as oncologist Dr. Brian noted that "complete hemato…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +51
Target Protein:
Breakpoint cluster region proteinInduced myeloid leukemia cell differentiation protein Mcl-1Mast/stem cell growth factor receptor Kit +8
Waktu ParuhFollowing oral admi…
Vol. DistribusiPopulation pharmaco…
KlirensTypically, clearanc…
Genetik -
IMC-1C11 DB06101
biotech

IMC-1C11 is an anti-angiogenesis agent. It is a chimeric anti-kinase insert domain-containing receptor (KDR) antibody that blocks VEGFR-KDR interaction and inhibits VEGFR-induced endothelial cell proliferation. IMC-1C11 is used for treatment of patients with …

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +4
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 138660-99-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imdevimab Approved DB15940
biotech | CAS: 2415933-40-1

Imdevimab is a monoclonal antibody combined with [casirivimab] in Regeneron's antibody cocktail known as REGEN-COV2 for the treatment of COVID-19.[L23539] This drug is a combination of antibodies derived from humanized VelocImmune® mice in addition to blood …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Spike glycoprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imelasomeran Approved DB17090
biotech | CAS: 2763208-92-8

Imelasomeran was first approved in Canada on September 1, 2022, as one-half of Moderna's Spikevax Bivalent COVID-19 mRNA vaccine.[L45320] It encodes for the viral spike protein of the Omicron BA.1 variant of SARS-CoV-2, a particularly infectious variant of co…

Kategori:
COVID-19 VaccinesmRNA VaccinesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imetelstat Approved DB14909
small molecule | CAS: 868169-64-6

Imetelstat is a first-in-class 18-amino acid oligonucleotide that directly and competitively inhibits human telomerase.[A263973] It is used to treat anemia in patients with myelodysplastic syndromes (MDS), a group of hematologic disorders characterized by ine…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsEnzyme Inhibitors +6
Target Protein:
Telomerase reverse transcriptaseHuman telomerase RNA component
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
Klirens-
Genetik -
Imidacloprid DB11421
small molecule | CAS: 105827-78-9

Imidacloprid is a neonicotinoid, which is a class of neuro-active insecticides modeled after nicotine. Imidacloprid is a patented chemical, Imidacloprid is manufactured by Bayer Cropscience (part of Bayer AG) and sold under trade names Kohinor, Admire, Advant…

Kategori:
AgrochemicalsCholinergic AgentsCompounds used in a research, industrial, or household setting +4
Target Protein:
CHRNA7-FAM7A fusion protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imidafenacin DB09262
small molecule | CAS: 170105-16-5

Imidafenacin is an antispasmodic agent with anticholinergic effects. It antagonizes muscarinic receptors in the bladder to reduce the frequency of urination in the treatment of overactive bladder. It is marketed in Japan under the tradenames Staybla by Ono Ph…

Kategori:
Agents producing tachycardiaAnticholinergic AgentsCytochrome P-450 CYP3A Substrates +8
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3
Waktu ParuhThe half life of el…
Vol. DistribusiThe estimated volum…
KlirensThe estimated clear…
Genetik -
small molecule | CAS: 36364-49-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1072-84-0

Imidazole-4-carboxylic acid is under investigation in clinical trial NCT00583895 (Safety and Efficacy Study of Imcooh Cream in Patients Suffering From Moderate Atopic Dermatitis).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Imidocarb DB11521
small molecule | CAS: 27885-92-3

Imidocarb is a urea derivative used in veterinary medicine as an antiprotozoal agent for the treatment of infection with Babesia and other parasites.

Kategori:
AmidesAminesAnilides +7
Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Imiglucerase Approved DB00053
biotech | CAS: 154248-97-2

Human Beta-glucocerebrosidase or Beta-D-glucosyl-N-acylsphingosine glucohydrolase E.C. 3.2.1.45. 497 residue protein with N-linked carbohydrates, MW=59.3 kD. Alglucerase is prepared by modification of the oligosaccharide chains of human Beta-glucocerebrosidas…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +6
Target Protein:
Glucocerebroside
Waktu Paruh3.6-10.4 min
Vol. Distribusi* 0.09 to 0.15 L/kg
Klirens* 14.5 +/- 4.0 mL/m…
Genetik -
Imipenem Approved DB01598
small molecule | CAS: 64221-86-9

Imipenem is a semisynthetic thienamycin that has a wide spectrum of antibacterial activity against gram-negative and gram-positive aerobic and anaerobic bacteria, including many multiresistant strains.[label] It is stable to many beta-lactamases. Similar comp…

Kategori:
Agents that reduce seizure thresholdAmidesAnti-Bacterial Agents +12
Target Protein:
Penicillin-binding protein 2Penicillin-binding protein 1BPenicillin-binding protein 1A +3
Waktu ParuhWhen given via IV i…
Vol. DistribusiThe reported volume…
KlirensThe total clearance…
Genetik -
Imipramine Approved DB00458
small molecule | CAS: 50-49-7

Imipramine, the prototypical tricyclic antidepressant (TCA), is a dibenzazepine-derivative TCA. TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individ…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +70
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A +21
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +6
Waktu ParuhImipramine has a me…
Vol. DistribusiImipramine has a hi…
KlirensImipramine has a me…
Genetik 9 Varian
Imiquimod Approved DB00724
small molecule | CAS: 99011-02-6

Imiquimod is an immune response modifier that acts as a toll-like receptor 7 agonist. Imiquimod is commonly used topically to treat warts on the skin of the genital and anal areas. Imiquimod does not cure warts, and new warts may appear during treatment. Imiq…

Kategori:
Adjuvants, ImmunologicAminoquinolinesAntineoplastic Agents +17
Target Protein:
Toll-like receptor 7Toll-like receptor 8
Waktu Paruh20 hours (topical d…
Vol. Distribusi-
Klirens-
Genetik -
Imlifidase Approved DB15258
biotech | CAS: 1947415-68-0

Chronic kidney disease (CKD) is a progressive and irreversible disease that represents a significant burden for both the individual and healthcare system at large.[A225916] Currently available treatments for end-stage renal disease are limited to dialysis and…

Kategori:
Antineoplastic and Immunomodulating AgentsEndopeptidasesImmunosuppressive Agents +2
Target Protein:
IgG heavy chain
Waktu ParuhThe mean distributi…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Imlunestrant DB19043
small molecule | CAS: 2408840-26-4

Imlunestrant is under investigation in clinical trial NCT05514054 (A Study of Imlunestrant Versus Standard Endocrine Therapy in Participants With Early Breast Cancer).

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IMM-0306 DB19309
biotech

IMM-0306 (bispecific antibody-trap selectively targeting cd47 and cd20) is under investigation in clinical trial NCT05805943 (Study of IMM0306 in Patients With Relapsed or Refractory Cd20-positive B-cell Non-hodgkin's Lymphoma).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
IMM-101 DB15850
biotech

IMM-101 is a heat-inactivated immune-activating mycobacterial product. It has shown to be safe and well tolerated to complement conventional cancer therapy for patients with melanoma and pancreatic ductal adenocarcinoma[A220013,A220018,A220023]. Studies with …

Kategori:
Biological ProductsComplex MixturesMelanoma, therapy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IMM101 DB15851
biotech

IMM-101 is a heat-inactivated immune-activating mycobacterial product. It has shown to be safe and well tolerated to complement conventional cancer therapy for patients with melanoma and pancreatic ductal adenocarcinoma [PMID: 21930686; PMID: 30107850; PMID: …

Waktu Paruh-
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IMMU-114 DB18458
biotech

IMMU-114 is antibody-drug conjugate consisting of humanized anti-HLA-DR IgG4 monoclonal antibody specific for alpha-chain linked to SN-38 via a CL2A linker.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Immucillin-G DB02230
small molecule

Deskripsi belum tersedia.

Kategori:
Purine-Nucleoside Phosphorylase, antagonists & inhibitorsPyrimidines
Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Immucin DB17403
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IMT-288 DB19068
small molecule | CAS: 637771-94-9

IMT-288 is under investigation in clinical trial NCT01730638 (Immunotep for Patients With Medullary Thyroid Carcinoma.).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 3251–3300 dari 6694
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