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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 66 / 282
AV608 DB05072
small molecule

AV608 is a NK-1 antagonist. It is developed for the treatment of Social anxiety disorder (SAD), irritable bowel syndrome (IBS) and overactive bladder (OAB).

Target Protein:
Substance-P receptor
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AVA-4746 DB18022
small molecule | CAS: 422268-99-3

Deskripsi belum tersedia.

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AVA-6000 DB17398
small molecule | CAS: 1841402-73-0

Deskripsi belum tersedia.

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AVAC DB05441
biotech

AVAC is derived from M. vaccae. It has been tested in uses related to asthma and in treating eczema and atopic dermatitis. [Mycobacterium vaccae] is a non-pathogenic, saprophytic bacteria whose antigens can be used to induce peripheral immune activation throu…

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Avacincaptad pegol Approved DB15165
biotech | CAS: 1613641-69-2

Avacincaptad pegol is an RNA aptamer covalently bound to a branched polyethylene glycol (PEG) molecule. It was developed to treat an advanced form of age-related macular degeneration (AMD) called geographic atrophy (GA).[L47696] AMD is the leading cause of vi…

Kategori:
Aptamers, NucleotideComplement Inactivating AgentsComplement Inactivator Proteins
Target Protein:
Complement C5
Waktu ParuhThe estimated appar…
Vol. DistribusiLimited information…
KlirensLimited information…
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Avacopan Approved DB15011
small molecule | CAS: 1346623-17-3

Anti-neutrophil cytoplasmic (auto)antibody (ANCA)-associated vasculitis (AAV) is a rare (estimated incidence of 3 cases per 100,000 per year) form of "pauci-immune" systemic small-vessel vasculitis typified by the presence of ANCAs in the serum.[A240249, A240…

Kategori:
AminesAntineoplastic and Immunomodulating AgentsComplement 5a Receptor Antagonist +22
Target Protein:
C5a anaphylatoxin chemotactic receptor 1
Waktu ParuhA single 30 mg dose…
Vol. DistribusiAvacopan has an app…
KlirensAvacopan has an est…
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Avadomide DB14857
small molecule | CAS: 1015474-32-4

Avadomide is under investigation in clinical trial NCT02031419 (Novel Combinations of CC-122, CC-223, CC-292, and Rituximab in Diffuse Large B-cell Lymphoma and Follicular Lymphoma).

Kategori:
Heterocyclic Compounds, Fused-RingPiperidinesQuinazolines
Target Protein:
Protein cereblon
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Avagacestat DB11893
small molecule | CAS: 1146699-66-2

Avagacestat has been investigated for the basic science and treatment of Alzheimer Disease.

Kategori:
AmidesAmyloid Precursor Protein Secretases, antagonists & inhibitorsEnzyme Inhibitors +4
Target Protein:
Gamma-secretase subunit APH-1ANicastrinGamma-secretase subunit APH-1B +2
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Avalglucosidase alfa Approved DB16099
biotech | CAS: 1802558-87-7

Avalglucosidase alfa, or NeoGAA, is a drug for enzyme replacement therapy specifically designed for Pompe disease, a rare inherited neuromuscular disorder caused by the deficiency of the alpha-glucosidase (GAA) enzyme. GAA is an essential enzyme that hydrolyz…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +2
Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu ParuhThe mean avalglucos…
Vol. DistribusiThe volume of distr…
KlirensThe mean avalglucos…
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biotech | CAS: 2227000-30-6

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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Avanafil Approved DB06237
small molecule | CAS: 330784-47-9

Avanafil is a phosphodiesterase-5 (PDE5) inhibitor used in the treatment of erectile dysfunction. In comparison with other drugs of the same class, it shows greater selectivity for PDE5 over PDE6 than both [sildenafil] and [vardenafil] but less selectivity th…

Kategori:
BCRP/ABCG2 InhibitorsCytochrome P-450 CYP2C9 SubstratesCytochrome P-450 CYP3A Substrates +9
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesterase
Waktu ParuhStudies have demons…
Vol. DistribusiThe apparent volume…
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Avapritinib Approved DB15233
small molecule | CAS: 1703793-34-3

Avapritinib, or BLU-285,[A189327] is a selective tyrosine kinase inhibitor of KIT and platelet derived growth factor receptor alpha indicated for the treatment of unresectable, metastatic gastrointestinal stromal tumors and advanced systemic mastocytosis.[A18…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +17
Target Protein:
Platelet-derived growth factor receptor alphaMast/stem cell growth factor receptor Kit
Waktu ParuhThe half life of av…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent o…
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Avasimibe DB06442
small molecule | CAS: 166518-60-1

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicAmides +14
Target Protein:
Liver carboxylesterase 1
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Avasopasem DB18481
small molecule

Deskripsi belum tersedia.

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small molecule | CAS: 435327-40-5

Avasopasem manganese, also known as GC4419, is a highly-selective small molecule mimetic of superoxide dismutase (SOD) being investigated for the reduction of radiation-induced severe oral mucositis.[L27246, L27256] This drug has potential application for rad…

Kategori:
AntioxidantsFree Radical Scavengers
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Avatrombopag Approved DB11995
small molecule | CAS: 570406-98-3

Avatrombopag (_Doptelet_), is an orally administered, small molecule thrombopoietin receptor (c-Mpl) agonist that increases platelet number without increasing platelet activation,[A33097,L2824] thereby decreasing the need for blood transfusions.[L2824] Patien…

Kategori:
BCRP/ABCG2 InhibitorsBlood and Blood Forming OrgansCytochrome P-450 CYP2C8 Inducers +14
Target Protein:
Thrombopoietin receptor
Waktu ParuhThe mean plasma eli…
Vol. DistribusiAvatrombopag has an…
KlirensThe mean (%CV) of t…
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AVB-001 DB18452
biotech

AVB-001 is an encapsulated, engineered human ARPE-19 cell line that constitutively expresses the native human IL-2 cytokine

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Avdoralimab DB16392
biotech | CAS: 2226393-85-5

Avdoralimab is under investigation in clinical trial NCT04333914 (Prospective Study in Patients With Advanced or Metastatic Cancer and Sars-cov-2 Infection).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Inflammatory Agents +9
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AVE-2865 DB07396
small molecule | CAS: 648917-13-9

Deskripsi belum tersedia.

Target Protein:
Glycogen phosphorylase, liver form
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Avelumab Approved DB11945
biotech | CAS: 1537032-82-8

Avelumab is a human IgG1 lambda monoclonal antibody that binds programmed cell death ligand-1 (PD-L1) to block its interaction with its receptors found on T cells and antigen-presenting cells.[A261496] Avelumab was first approved by the FDA on March 23, 2017.…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Programmed cell death 1 ligand 1
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe geometric mean …
KlirensThe total systemic …
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Avena sativa flowering top Approved DB14253
biotech

Avena sativa flowering top is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Avenciguat DB18882
small molecule | CAS: 1579514-06-9

Avenciguat is under investigation in clinical trial NCT05282121 (A Study to Test Whether BI 685509 Alone or in Combination With Empagliflozin Helps People With Liver Cirrhosis Caused by Viral Hepatitis or Non-alcoholic Steatohepatitis (NASH) Who Have High Blo…

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Avexitide DB14806
small molecule | CAS: 133514-43-9

Avexitide is under investigation in clinical trial NCT02996812 (Evaluation of Single Ascending Doses of Subcutaneous Exendin 9-39 in Patients With Post-Bariatric Hypoglycemia).

Kategori:
Amino Acids, Peptides, and ProteinsGlucagon-Like Peptide 1Peptides
Target Protein:
Glucagon-like peptide 1 receptor
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AVI-4020 DB05873
small molecule

AVI-4020 is a neugene antisense drug candidate for the treatment of patients with acute West Nile virus disease who have serious neurological impairment (WNV neuroinvasive disease).

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AVI-4065 DB05620
small molecule

AVI-4065, a phosphorodiamidate Morpholino oligomer (PMO), is an investigational antisense HCV drug. It was developed by Sarepta Therapeutics, Inc. After phase II trials it was cancelled due to lack of potency. [L2917]

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AVI-5126 DB05726
small molecule

AVI-526 is an improved formulation of [AVI-4557], developed for use on Vein Grafts before use in Heart by-Pass Graft Surgery. AVI-526 works by silencing a gene known as c-myc, a key regulatory gene involved in cardiovascular restenosis. The drug was under inv…

Kategori:
MorpholinesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
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AVI-7287 DB17799
biotech

Deskripsi belum tersedia.

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AVI-7288 DB17800
biotech

Deskripsi belum tersedia.

Kategori:
MorpholinesNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
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AVI-7537 DB15433
biotech

AVI-7537 is an antisense molecule that binds to the Ebola virus mRNA to prevent the viral replication.[L46207] AVI-7537 is under investigation in clinical trial NCT01593072 (A Study to Assess the Safety, Tolerability and Pharmacokinetics of AVI-7537 in Health…

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Avibactam Approved DB09060
small molecule | CAS: 1192500-31-4

Avibactam is a non-?-lactam ?-lactamase inhibitor that is available in combination with ceftazidime (Avycaz). This combination was approved by the FDA on February 25, 2015 for the treatment of complicated intra-abdominal infections in combination with metroni…

Kategori:
Anti-Infective AgentsAza Compoundsbeta-Lactamase Inhibitors +2
Target Protein:
Beta-lactamase TEMBeta-lactamase CTX-MBeta-lactamase +7
Waktu ParuhCeftazidime-avibact…
Vol. DistribusiThe steady state vo…
KlirensAvibactam and cefta…
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Avicin D DB17240
small molecule | CAS: 197787-20-5

Deskripsi belum tersedia.

Kategori:
CarbohydratesGlycosides
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AVID-200 DB18454
biotech | CAS: 2269485-28-9

AVID-200 is an Anti-transforming growth factor beta (TGF-?) trap fusion protein.

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Avidin DB15228
biotech | CAS: 110539-97-4

Avidin is under investigation in clinical trial NCT00345618 (Clinical Study Assessing Idrabiotaparinux Sodium Injections Once-weekly in Pulmonary Embolism Therapeutic Approach).

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsAnimal Proteins, Dietary +10
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Aviptadil DB06260
small molecule | CAS: 40077-57-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsErectile DysfunctionGastrointestinal Hormones +9
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Aviscumine DB12684
biotech | CAS: 223577-45-5

Cy 503 is under investigation in clinical trial NCT00658437 (Aviscumine for the Treatment of Malignant Melanoma Stage IV After Failure of Prior Therapy).

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsBiological Factors +12
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Avizakimab DB18842
biotech | CAS: 2229685-51-0

Avizakimab is under investigation in clinical trial NCT03371251 (Study of BOS161721 in Systemic Lupus Erythematosus (SLE) Patients on a Background of Limited Standard of Care).

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AVL-3288 DB18707
small molecule | CAS: 917837-54-8

Deskripsi belum tersedia.

Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
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Avoralstat DB12120
small molecule | CAS: 918407-35-9

Avoralstat has been used in trials studying the prevention of HAE and Hereditary Angioedema.

Kategori:
Acids, CarbocyclicAlkenesAmides +6
Target Protein:
Kallikrein-2Kininogen-1
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Avotaciclib DB16652
small molecule | CAS: 1983983-41-0

Avotaciclib is under investigation in clinical trial NCT03579836 (Evaluation of Safety and Efficacy in BEY1107 in Monotherapy Gemcitabine Combination in Patient With Pancreatic Cancer).

Target Protein:
Cyclin-dependent kinase 1
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Avotermin DB11955
biotech | CAS: 182212-66-4

Juvista has been investigated for the treatment, prevention, and basic science of Scars, Keloid, and Cicatrix.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
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AVP-21D9 DB17798
biotech

AVP-21D9 is a fully human anthrax monoclonal antibody that is being investigated as an anthrax antitoxin.[A259522]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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AVR-48 DB18294
small molecule | CAS: 3459-18-5

Deskripsi belum tersedia.

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AVR-RD-02 DB17650
biotech

AVR-RD-02 is an investigational _ex vivo_ lentiviral gene therapy developed by AVROBIO Inc. It consists of autologous CD34+ enriched hematopoietic stem cells (HSCs) that have been genetically modified _ex vivo_ with a lentiviral vector (LV) to contain a ribon…

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AVR-RD-05 DB18631
biotech

AVR-RD-05 is a gene therapy comprising genetically modified autologous stem cells transduced _ex vivo_ with a lentiviral vector encoding the human iduronate-2-sulfatase (IDS) enzyme. It is under investigation for the treatment of Hunter Syndrome (Mucopolysacc…

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AVS-100 DB18068
small molecule | CAS: 2245942-72-5

Deskripsi belum tersedia.

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Avutometinib DB15254
small molecule | CAS: 946128-88-7

Avutometinib (RO-5126766 free base) is under investigation in clinical trial NCT03875820 (Phase I Trial of VS-6063 and RO5126766.).

Kategori:
BenzopyransHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors +1
Target Protein:
Serine/threonine-protein kinase A-RafSerine/threonine-protein kinase B-rafRAF proto-oncogene serine/threonine-protein kinase
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AVX-001 DB19194
small molecule | CAS: 300553-18-8

AVX-001 is under investigation in clinical trial NCT05164393 (Phase I/iia Trial to Evaluate AVX001 Gel in Doses of 1% or 3% Compared With Vehicle Over Four Weeks of Field-directed Treatment Period in Adult Subjects With AK).

Kategori:
Dietary FatsDietary Fats, UnsaturatedFats +5
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AVXS-201 DB16997
biotech

Deskripsi belum tersedia.

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AX200 DB05093
small molecule

AX200, which has been developed for the treatment of stroke, is the most advanced drug candidate and is halfway through the process of gaining clinical approval. The expression of the endogenous AX200 protein in the brain is increased after brain damage. Thus…

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biotech

Axalimogene filolisbac is under investigation in clinical trial NCT02853604 (Study of ADXS11-001 in Subjects With High Risk Locally Advanced Cervical Cancer).

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