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14063

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10481 (74.5%)
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8038 (57.2%)
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107 (0.8%)
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14063 (100.0%)

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Halaman 65 / 282
Atoltivimab Approved DB15898
biotech | CAS: 2135632-29-8

Ebola virus (EBOV) remains an important human pathogen within the _Ebolavirus_ genus, having been responsible for at least 17 known outbreaks with an average case fatality rate of 43.92%.[A221825] Immune therapy using monoclonal antibodies (mAbs) is becoming …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +10
Target Protein:
Envelope glycoprotein
Waktu ParuhAtoltivimab adminis…
Vol. DistribusiAtoltivimab adminis…
KlirensAtoltivimab adminis…
Genetik -
Atomoxetine Approved DB00289
small molecule | CAS: 83015-26-3

Atomoxetine is a selective norepinephrine (NE) reuptake inhibitor used for the treatment of attention deficit hyperactivity disorder (ADHD). Also known as the marketed product Strattera, atomoxetine is used with other treatment modalities (psychological, educ…

Kategori:
Adrenergic AgentsAgents producing tachycardiaAgents that produce hypertension +17
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporterNMDA receptor +2
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +3
Waktu ParuhThe reported half-l…
Vol. DistribusiThe reported volume…
KlirensThe clearance rate …
Genetik 6 Varian
Atopaxar DB12046
small molecule | CAS: 751475-53-3

Atopaxar has been investigated for the treatment of Coronary Artery Disease and Acute Coronary Syndrome.

Kategori:
Receptors, Thrombin, antagonists & inhibitors
Target Protein:
Proteinase-activated receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atorvastatin Approved DB01076
small molecule | CAS: 134523-00-5

Atorvastatin (Lipitor®), is a lipid-lowering drug included in the statin class of medications. By inhibiting the endogenous production of cholesterol in the liver, statins lower abnormal cholesterol and lipid levels, and ultimately reduce the risk of cardiova…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBSEP/ABCB11 Substrates +37
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseDipeptidyl peptidase 4Aryl hydrocarbon receptor +2
Gen Terkait:
KIF6 HMGCR CYP3A4
Waktu ParuhThe half-life of at…
Vol. DistribusiThe reported volume…
KlirensThe registered tota…
Genetik 3 Varian
Atovaquone Approved DB01117
small molecule | CAS: 95233-18-4

Atovaquone is a hydroxynaphthoquinone, or an analog of ubiquinone, that has antimicrobial and antipneumocystis activity. It is being used in antimalarial protocols.

Kategori:
Anti-Infective AgentsAntibiotics for Pneumocystis PneumoniaAntimalarials +16
Target Protein:
Cytochrome bDihydroorotate dehydrogenase (quinone), mitochondrialDihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh2.2 to 3.2 days
Vol. Distribusi* 0.60 ± 0.17 L/kg
Klirens* 10.4 +/- 5.5 ml/m…
Genetik -
Atpenin A5 DB04631
small molecule | CAS: 119509-24-9

Deskripsi belum tersedia.

Kategori:
Pyridines
Target Protein:
Succinate dehydrogenase iron-sulfur subunitSuccinate dehydrogenase cytochrome b556 subunitSuccinate dehydrogenase hydrophobic membrane anchor subunit +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atractylodes japonica root Approved DB11261
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Atractylodes japonica root oil is obtained from the roots of Atractylodes japonica, which is a herb native to eastern Asia. It is present in some cosmetic products such as whitening creams as an active ingredient and lubricant for skin irritation. Atractylode…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Atracurium Approved DB13295
small molecule | CAS: 64228-79-1

Deskripsi belum tersedia.

Kategori:
Anticholinergic AgentsBenzylisoquinolinesCentral Nervous System Depressants +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atracurium besylate Approved DB00732
small molecule | CAS: 64228-81-5

A non-depolarizing neuromuscular blocking agent with short duration of action. Its lack of significant cardiovascular effects and its lack of dependence on good kidney function for elimination provide clinical advantage over alternate non-depolarizing neuromu…

Kategori:
Anticholinergic AgentsBenzylisoquinolinesCentral Nervous System Depressants +10
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Atrasentan DB06199
small molecule | CAS: 173937-91-2

Atrasentan is a substance that is being studied in the treatment of cancer. It belongs to the family of drugs called endothelin-1 protein receptor antagonists. It is a novel, selective endothelin A receptor antagonist (SERA).

Kategori:
Antineoplastic AgentsBenzodioxolesDioxoles +5
Target Protein:
Endothelin-1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atrazine DB07392
small molecule | CAS: 1912-24-9

Atrazine is a selective triazine herbicide. Inhalation hazard is low and there are no apparent skin manifestations or other toxicity in humans. Acutely poisoned sheep and cattle may show muscular spasms, fasciculations, stiff gait, increased respiratory rates…

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingHerbicides +3
Target Protein:
Photosynthetic reaction center cytochrome c subunitReaction center protein H chainReaction center protein L chain +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atreleuton DB12758
small molecule | CAS: 154355-76-7

Atreleuton has been used in trials studying the treatment of Atherosclerosis and Coronary Artery Disease.

Kategori:
AmidesEnzyme InhibitorsLipoxygenase Inhibitors
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Atropine Approved DB00572
small molecule | CAS: 51-55-8

Atropine is an alkaloid originally synthesized from Atropa belladonna. It is a racemic mixture of d-and l-hyoscyamine, of which only l-hyoscyamine is pharmacologically active.[A251670,L42835] Atropine is generally available as a sulfate salt and can be admini…

Kategori:
Adjuvants, AnesthesiaAgents producing tachycardiaAgents that produce hypertension +32
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +5
Waktu ParuhFollowing intraveno…
Vol. DistribusiAtropine is distrib…
KlirensFollowing intraveno…
Genetik -
ATSN-101 DB18327
biotech

ATSN-101 is a adeno-associated virus serotype 5 encoding human retinal guanylate cyclase 1 gene (AAV5-GUCY2D)

Waktu Paruh-
Vol. Distribusi-
Klirens-
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Attapulgite Approved DB01574
small molecule | CAS: 12174-11-7

Attapulgite is a magnesium aluminium phyllosilicate which occurs in a type of clay soil common to the Southeastern United States. When used in medicine, it physically binds to acids and toxic substances in the stomach and digestive tract. For that reason, it …

Kategori:
Alimentary Tract and MetabolismAntidiarrheals, Intestinal Antiinflammatory/antiinfective AgentsAntidotes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ATU-027 DB12171
biotech | CAS: 1415935-22-6

Atu027 has been used in trials studying the treatment of Advanced Solid Tumors.

Waktu Paruh-
Vol. Distribusi-
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Atuliflapon DB19029
small molecule | CAS: 2041075-86-7

Atuliflapon is under investigation in clinical trial NCT05251259 (Study to Assess the Efficacy and Safety of Atuliflapon in Moderate-to-severe Uncontrolled Asthma).

Waktu Paruh-
Vol. Distribusi-
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Atuzaginstat DB19030
small molecule | CAS: 2211981-76-7

Atuzaginstat is under investigation in clinical trial NCT03823404 (GAIN Trial: Phase 2/3 Study of COR388 in Subjects With Alzheimer's Disease).

Waktu Paruh-
Vol. Distribusi-
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ATX-01 DB18141
biotech

ATX-01 is an antimiR, a chemically modified antisense oligonucleotide, designed to target microRNA 23b (miR-23b).

Waktu Paruh-
Vol. Distribusi-
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ATX-201 DB05765
small molecule

ATX-201 is one of a family of novel compounds that inhibits microtubule polymerization. It is developed by Kythera Biopharmaceuticals, Inc. for the treatment of actinic keratosis. The company announced the decision to discontinue its ATX-201 clinical program…

Waktu Paruh-
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ATX-914 DB12673
small molecule

Axt914 is under investigation in clinical trial NCT00417261 (Safety, Tolerability, Pharmacodynamic and Pharmacokinetic Effects of Single and Multiple-Doses of ATF936 and AXT914 Administered Orally in Healthy Subjects.).

Kategori:
Heterocyclic Compounds, Fused-RingQuinazolines
Waktu Paruh-
Vol. Distribusi-
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ATX-F8-117 DB17712
biotech

ATX-F8-117 is an investigational peptide derived from Factor VIII. Developed by Apitope, it is being investigated for the treatment of hemophilia A.[L46163]

Waktu Paruh-
Vol. Distribusi-
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Genetik -
ATYR-1940 DB16991
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AUM-302 DB18114
small molecule | CAS: 1414455-21-2

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsProtein Kinase InhibitorsSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
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Genetik -
AUM-601 DB17382
small molecule

AUM-601 is a highly selective pan-TRK(tropomyosin receptor kinase). It is currently being investigated in clinical trials for the treatment of cancer.

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AUNP-12 DB15771
biotech | CAS: 1353563-85-5

Deskripsi belum tersedia.

Kategori:
Immune Checkpoint Inhibitors
Target Protein:
Programmed cell death 1 ligand 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Auranofin Approved DB00995
small molecule | CAS: 34031-32-8

Auranofin is a gold salt that is capable of eliciting pharmacologic actions that suppress inflammation and stimulate cell-mediated immunity. It has subsequently been listed by the World Health Organization as a member of the antirheumatic agent category. Aura…

Kategori:
Antiinflammatory and Antirheumatic ProductsAntirheumatic AgentsDrugs that are Mainly Renally Excreted +6
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Aureobasidium pullulans var. pullutans is a fungus which can provoke allergic reactions. Aureobasidium pullulans var. pullutans extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Auriclosene DB12197
small molecule | CAS: 846056-87-9

Auriclosene has been used in trials studying the treatment of Impetigo, Bacterial Conjunctivitis, Asymptomatic Bacteriuria, and Adenoviral Conjunctivitis.

Kategori:
AlkanesAlkanesulfonic AcidsHydrocarbons, Acyclic +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aurodox DB04124
small molecule | CAS: 12704-90-4

Aurodox is an antibiotic obtained from a streptomyces variant considered as possibly effective against streptococcus pyogenes infections. It may promote growth in poultry.

Kategori:
AlkenesAnti-Bacterial AgentsAnti-Infective Agents +2
Target Protein:
Elongation factor Tu-B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Aurothioglucose Approved DB09121
small molecule | CAS: 12192-57-3

Aurothioglucose, also known as gold thioglucose, was formerly used to treat rheumatoid arthritis. Contemporary research on the effect of gold salts treatment began in 1935, primarily to reduce inflammation and to slow disease progression in patients with r…

Kategori:
Antiinflammatory and Antirheumatic ProductsAntirheumatic AgentsDrugs that are Mainly Renally Excreted +5
Target Protein:
Adenylate cyclase type 1Adenylate cyclase type 2Adenylate cyclase type 5
Waktu ParuhThe biological half…
Vol. DistribusiReadily accessible …
KlirensWhen a standard wee…
Genetik -
Aurothioglycanide Approved DB19361
small molecule | CAS: 16925-51-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
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Aurotioprol DB13763
small molecule | CAS: 27279-43-2

Deskripsi belum tersedia.

Kategori:
AlcoholsAntiinflammatory and Antirheumatic ProductsAntirheumatic Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AUTO3 DB17364
biotech

AUTO3 is bicistronic chimeric antigen receptor T-cell therapy investigated for acute lymphoblastic leukemia (ALL). It is an investigational chimeric antigen receptor (CAR) T cell treatment targeting CD19 and CD22.

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Genetik -
biotech | CAS: 2365453-34-3

Autogene cevumeran is an mRNA-based cancer vaccine targeting an unspecified amount of tumour-associated antigens. It is being investigated for cancers.

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Genetik -
biotech

Deskripsi belum tersedia.

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Genetik -
biotech

Deskripsi belum tersedia.

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Genetik -
biotech

Deskripsi belum tersedia.

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biotech

Autologous DNP-conjugated tumour vaccine, or melanoma vaccine, is an investigational autologous cell vaccine technology for melanoma.[A254806]

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biotech

Autologous hematopoietic peripheral blood stem cells were tested in a clinical trial (NCT00424489) by Northwestern University for the treatment of refractory myasthenia gravis.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Autologous pancreatic islet therapy involves isolating the patient's own insulin-producing cells.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Autologous peripheral blood-derived CD34+ cells, or CLBS119 (a proprietary version being developed by Caladrius Biosciences, Inc.), are hematopoietic stem cells.[L27741] It is also a cell therapy being investigated by Caladrius Biosciences in the clinical tri…

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biotech

Deskripsi belum tersedia.

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AUY922 DB11881
small molecule | CAS: 747412-64-2

AUY922 has been used in trials studying the treatment of Lymphoma, Breast Cancer, Metastatic Disease, Advanced Solid Tumors, and Hematologic Neoplasms, among others.

Kategori:
Benzene DerivativesHSP90 Heat-Shock Proteins, antagonists & inhibitorsPhenols
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AV-0113 DB18386
biotech

AV-0113 consists of IL-12 secreting dendritic cells loaded with autologous tumor lysate.

Waktu Paruh-
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AV-101 DB12878
small molecule | CAS: 153152-32-0

AV-101 has been used in trials studying the treatment of Neuropathic Pain.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsSweetening Agents
Waktu Paruh-
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Genetik -
AV-412 DB06021
small molecule | CAS: 451493-31-5

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Epidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
AV-COVID-19 DB15802
biotech

AV-COVID-19 is a vaccine composed of autologous dendritic cells loaded with SARS-CoV-2 antigens and with or without Granulocyte-macrophage colony-stimulating factor (GM-CSF). The vaccine is created from the receiving patients’ isolated peripheral blood mon…

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Menampilkan 3201–3250 dari 14063
Sebelumnya Halaman 65 / 282 Berikutnya